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21 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Parallel fluorescent probe synthesis based on the large-scale preparation of BODIPY FL propionic acid.EBI
Takeda Pharmaceutical
Synthesis and biological evaluation of novel 4-hydroxytamoxifen analogs as estrogen-related receptor gamma inverse agonists.EBI
Daegu-Gyeongbuk Medical Innovation Foundation
Synthesis and Biological Evaluation of Cyclopentaquinoline Derivatives as Nonsteroidal Glucocorticoid Receptor Antagonists.EBI
TBA
1-Phenyl-4-benzoyl-1H-1,2,3-triazoles as orally bioavailable transcriptional function suppressors of estrogen-related receptora.EBI
Chinese Academy of Sciences
Synthesis of novel estrogen receptor antagonists using metal-catalyzed coupling reactions and characterization of their biological activity.EBI
University of Kansas Medical Center
Identification of Potent and Selective Diphenylpropanamide ROR? Inhibitors.EBI
New York University School of Medicine
Identification of diaryl ether-based ligands for estrogen-related receptora as potential antidiabetic agents.EBI
Johnson & Johnson Pharmaceutical Research and Development
ERbeta ligands. Part 6: 6H-Chromeno[4,3-b]quinolines as a new series of estrogen receptor beta-selective ligands.EBI
Wyeth Research
Identification of a selective inverse agonist for the orphan nuclear receptor estrogen-related receptor alpha.EBI
X-Ceptor Therapeutics
Discovery of a Novel Class of ERR? Agonists.EBI
Daiichi Sankyo
An orally available inverse agonist of estrogen-related receptor gamma showed expanded efficacy for the radioiodine therapy of poorly differentiated thyroid cancer.EBI
Daegu-Gyeongbuk Medical Innovation Foundation
Insights of a Lead Optimization Study and Biological Evaluation of Novel 4-Hydroxytamoxifen Analogs as Estrogen-Related Receptor ? (ERR?) Inverse Agonists.EBI
Daegu-Gyeongbuk Medical Innovation Foundation
Discovery of Potent, Selective, and Orally Bioavailable Estrogen-Related Receptor-? Inverse Agonists To Restore the Sodium Iodide Symporter Function in Anaplastic Thyroid Cancer.EBI
Daegu-Gyeongbuk Medical Innovation Foundation
Identification of New Small-Molecule Inducers of Estrogen-related Receptor ? (ERR?) Degradation.EBI
Jinan University
The discovery of novel, potent ERR-alpha inverse agonists for the treatment of triple negative breast cancer.EBI
Qilu University of Technology
Indazole-based ligands for estrogen-related receptor ? as potential anti-diabetic agents.EBI
Janssen Research and Development
Inhibitors of Src homology-2 domain containing protein tyrosine phosphatase-2 (Shp2) based on oxindole scaffolds.BDB
Moffitt Cancer Center