Binding Database

The following articles (labelled with PubMed ID or TBD) are for your review

PMID

Data

Article Title

Organization

Synthesis and Evaluation of Macrocyclic Peptide Aldehydes as Potent and Selective Inhibitors of the 20S Proteasome.

Whitman College

Protease inhibitors: current status and future prospects.

University of Queensland

D-amino acid containing, high-affinity inhibitors of recombinant human calpain I.

Cephalon

Peptidyl aldehyde derivatives as potent and selective inhibitors of cathepsin L

TBA

Molecular modeling: a search for a calpain inhibitor as a new treatment for cataractogenesis.

University of Canterbury

Discovery of Fluoromethylketone-Based Peptidomimetics as Covalent ATG4B (Autophagin-1) Inhibitors.

Roche Pharma Research and Early Development

The role of N-terminal heterocycles in hydrogen bonding to ?-chymotrypsin.

The University of Adelaide

Novel peptidyl alpha-keto amide inhibitors of calpains and other cysteine proteases.

Georgia Institute of Technology

Peptide alpha-keto ester, alpha-keto amide, and alpha-keto acid inhibitors of calpains and other cysteine proteases.

Georgia Institute of Technology

Stereospecific synthesis of peptidyl alpha-keto amides as inhibitors of calpain.

Alkermes

Phosphorylation of Capsaicinoid Derivatives Provides Highly Potent and Selective Inhibitors of the Transcription Factor STAT5b.

University of Leipzig