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12 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Optimization of Novel Antagonists to the Neurokinin-3 Receptor for the Treatment of Sex-Hormone Disorders (Part II).EBI
Euroscreen
Discovery and optimization of novel antagonists to the human neurokinin-3 receptor for the treatment of sex-hormone disorders (Part I).EBI
Euroscreen
Development of novel neurokinin 3 receptor (NK3R) selective agonists with resistance to proteolytic degradation.EBI
Kyoto University
Cyclic peptides as selective tachykinin antagonists.EBI
Merck Sharp and Dohme Research Laboratories
N',2-diphenylquinoline-4-carbohydrazide based NK3 receptor antagonists.EBI
Merck Sharp & Dohme Research Laboratories
Use of a dipeptide chemical library in the development of non-peptide tachykinin NK3 receptor selective antagonists.EBI
Cambridge University Forvie Site
Design and synthesis of side-chain conformationally restricted phenylalanines and their use for structure-activity studies on tachykinin NK-1 receptor.EBI
Universit£
Conformationally constrained tachykinin analogues: potent and highly selective neurokinin NK-2 receptor agonists.EBI
Glaxo Group Research
Imidazo[4,5-b]quinoxaline cyanines as neurokinin antagonists.EBI
Rochester
Discovery of 3-aryl-5-acylpiperazinyl-pyrazoles as antagonists to the NK3 receptor.EBI
Euroscreen
 
The dipeptide neurokinin-1 receptor antagonist S19752 is a potent and long-acting inhibitor of bronchoconstriction when administered by aerosol to the guinea pig in vivoEBI
TBA
Synthesis and biological activity of NK-1 selective, N-backbone cyclic analogs of the C-terminal hexapeptide of substance P.EBI
Hebrew University of Jerusalem