11 articles for thisTarget
The following articles (labelled with PubMed ID or TBD) are for your review
PMID
Data
Article Title
Organization
Highly Potent, Water Soluble Benzimidazole Antagonist for Activated alpha(4)beta(1) Integrin.
University of California Davis
Synthesis, biological evaluation, and pharmacokinetic study of prolyl-1-piperazinylacetic acid and prolyl-4-piperidinylacetic acid derivatives as VLA-4 antagonists.
Daiichi Pharmaceutical
Synthesis and biological evaluation of benzoic acid derivatives as potent, orally active VLA-4 antagonists.
Daiichi Pharmaceutical
Selection of a 2-azabicyclo[2.2.2]octane-based alpha4beta1 integrin antagonist as an inhaled anti-asthmatic agent.
Johnson & Johnson Pharmaceutical
Pyridone derivatives as potent and selective VLA-4 integrin antagonists.
Glaxosmithkline
Pyridone derivatives as potent, orally bioavailable VLA-4 integrin antagonists.
Glaxosmithkline
Structure-activity relationship studies of a series of peptidomimetic ligands for alpha(4) beta(1) integrin on Jurkat T-leukemia cells.
University of California Davis
Aza-bicyclic amino acid carboxamides as alpha4beta1/alpha4beta7 integrin receptor antagonists.
Johnson & Johnson Pharmaceutical