27 articles for U Holzgrabe
The following articles (labelled with PubMed ID or TBD) are for your review
PMID
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Data
Article Title
Organization
17
Oxime Ethers of (E)-11-Isonitrosostrychnine as Highly Potent Glycine Receptor Antagonists.
The German University In Cairo
27
Development, synthesis and structure-activity-relationships of inhibitors of the macrophage infectivity potentiator (Mip) proteins of Legionella pneumophila and Burkholderia pseudomallei.
University of W£Rzburg
13
Rational design of partial agonists for the muscarinic m1 acetylcholine receptor.
University of W£Rzburg
14
Semisynthetic analogues of toxiferine I and their pharmacological properties ata7 nAChRs, muscle-type nAChRs, and the allosteric binding site of muscarinic M2 receptors.
The German University In Cairo
11
Bis(ammonio)alkane-type agonists of muscarinic acetylcholine receptors: synthesis, in vitro functional characterization, and in vivo evaluation of their analgesic activity.
University of Milan
2
Design, synthesis, and action of oxotremorine-related hybrid-type allosteric modulators of muscarinic acetylcholine receptors.
University of Milan
11
Structure-activity relationships in a series of bisquaternary bisphthalimidine derivatives modulating the muscarinic M(2)-receptor allosterically.
University of W�Rzburg
14
Pipecolic acid derivatives as small-molecule inhibitors of the Legionella MIP protein.
University of Wu£Rzburg
14
Search for the pharmacophore of bispyridinium-type allosteric modulators of muscarinic receptors.
University of Bonn
10
Interaction of (benzylidene-hydrazono)-1,4-dihydropyridines with beta-amyloid, acetylcholine, and butyrylcholine esterases.
Ege University
7
A small-molecule inhibitor of Nipah virus envelope protein-mediated membrane fusion.
University of W£Rzburg
4
Structure-activity relationship and studies on the molecular mechanism of leishmanicidal N,C-coupled arylisoquinolinium salts.
University of WüRzburg
2
Structure and Dynamics of Macrophage Infectivity Potentiator Proteins from Pathogenic Bacteria and Protozoans Bound to Fluorinated Pipecolic Acid Inhibitors.
Friedrich Schiller University Jena
36
Aziridine-2,3-dicarboxylate inhibitors targeting the major cysteine protease of Trypanosoma brucei as lead trypanocidal agents.
University of Wuerzburg
2
Random chemistry as a new tool for the generation of small compound libraries: development of a new acetylcholinesterase inhibitor.
University of WüRzburg
27
C-2-Linked Dimeric Strychnine Analogues as Bivalent Ligands Targeting Glycine Receptors.
The German University In Cairo
9
Targeting Protein Folding: A Novel Approach for the Treatment of Pathogenic Bacteria.
University of W£Rzburg
1
Mechanism of action of the diazabicyclononanone-type kappa-agonists.
UniversitäT WüRzburg
9
Synthesis and opioid receptor affinity of a series of 2, 4-diaryl-substituted 3,7-diazabicylononanones.
University of WüRzburg
22
Bisquaternary ligands of the common allosteric site of M2 acetylcholine receptors: search for the minimum essential distances between the pharmacophoric elements.
University of Bonn
15
Fluorination of Photoswitchable Muscarinic Agonists Tunes Receptor Pharmacology and Photochromic Properties.
Julius Maximilian University of W£Rzburg
15
Dualsteric muscarinic antagonists--orthosteric binding pose controls allosteric subtype selectivity.
University of W£Rzburg
35
Systematic development of high affinity bis(ammonio)alkane-type allosteric enhancers of muscarinic ligand binding.
University of W£Rzburg
9
Elevation of ligand binding to muscarinic M(2) acetylcholine receptors by bis(ammonio)alkane-type allosteric modulators.
University of Bonn