BDBM50036733 1-(4-Fluoro-phenyl)-4-(4-pyridin-2-yl-piperazin-1-yl)-butan-1-one(Azaperone)::Azaperone::CHEMBL340211

SMILES Fc1ccc(cc1)C(=O)CCCN1CCN(CC1)c1ccccn1

InChI Key InChIKey=XTKDAFGWCDAMPY-UHFFFAOYSA-N

Data  38 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50036733   

Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50036733(1-(4-Fluoro-phenyl)-4-(4-pyridin-2-yl-piperazin-1-...)
Affinity DataKi:  62.7nMAssay Description:Displacement of [3H]-ketanserin from human 5HT2A receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50036733(1-(4-Fluoro-phenyl)-4-(4-pyridin-2-yl-piperazin-1-...)
Affinity DataKi:  62.7nMAssay Description:Displacement of [3H]-Ketanserin from human 5-HT2A receptor incubated for 1 hr by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50036733(1-(4-Fluoro-phenyl)-4-(4-pyridin-2-yl-piperazin-1-...)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]-Ketanserin from human 5-HT2A receptor incubated for 1 hr by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50036733(1-(4-Fluoro-phenyl)-4-(4-pyridin-2-yl-piperazin-1-...)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]-ketanserin from human 5HT2A receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed