BDBM50387545 CHEMBL2059907

SMILES CC(=O)Nc1nc2ccc(cn2n1)-c1cncc(c1)S(C)(=O)=O

InChI Key InChIKey=RCRCKEODQLBHAY-UHFFFAOYSA-N

Data  8 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50387545   

LigandChemical structure of BindingDB Monomer ID 50387545BDBM50387545(CHEMBL2059907)
Affinity DataIC50: 79.4nMAssay Description:Inhibition of PI3Kgamma by high throughput chemoproteomics binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50387545BDBM50387545(CHEMBL2059907)
Affinity DataIC50: 79.4nMAssay Description:Inhibition of PI3Kgamma in human HL60 cell lysate by kinobead assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50387545BDBM50387545(CHEMBL2059907)
Affinity DataIC50: 3.98E+3nMAssay Description:Inhibition of PI3Kalpha in human HL60 cell lysate by kinobead assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50387545BDBM50387545(CHEMBL2059907)
Affinity DataIC50: 3.98E+3nMAssay Description:Inhibition of PI3Kalpha by high throughput chemoproteomics binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50387545BDBM50387545(CHEMBL2059907)
Affinity DataIC50: 5.01E+3nMAssay Description:Inhibition of PI3Kdelta in human HL60 cell lysate by kinobead assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50387545BDBM50387545(CHEMBL2059907)
Affinity DataIC50: 5.01E+3nMAssay Description:Inhibition of PI3Kdelta by high throughput chemoproteomics binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed