BDBM578574 3-(5-fluoro-5'- (methylsulfonyl)- [3,3'-bipyridin]- 2-yl)-3-methoxy- 5,5-dimethyl-6- oxocyclohex-1- ene-1- carbonitrile::US11479539, Compound 235::US11479539, Compound 96
SMILES COC1(CC(C)(C)C(=O)C(=C1)C#N)c1ncc(F)cc1-c1cncc(c1)S(C)(=O)=O
InChI Key InChIKey=UKSQFPLHWJYMNO-UHFFFAOYSA-N
Data 2 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 578574
Affinity DataEC50: 7nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Affinity DataEC50: 79nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair