BDBM88566 US9695132, I-8

SMILES CCC(=O)Nc1cccc(CN2C(=O)N(Cc3cnc(NC4CCCCC4NC(=O)C=C)nc23)c2c(Cl)c(OC)cc(OC)c2Cl)c1

InChI Key InChIKey=ZACWLHRJLJNYCZ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 88566   

TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Celgene Car

US Patent
LigandPNGBDBM88566(US9695132, I-8)
Affinity DataIC50: <100nMpH: 7.5Assay Description:Omnia Assay Protocol for Potency Assessment Against FGFR 4 Enzyme. b) [FGFR4-WT]=2.5 nM, [ATP]=250 uM, [Y10-Sox]=10 uM (ATP KMapp 250 uM): A 10x stoc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent