BDBM209025 US9243038, 5a (cis olefin)::US9243038, 5b (trans olefin)

SMILES NC(=O)[C@@H]1CCCCNC(=O)[C@@H](Cc2ccc(cc2)C(=O)c2ccccc2)NC(=O)[C@H](CC2CCCCC2)NC(=O)[C@H](CC2CC2)NC(=O)\C=C\C(=O)N1

InChI Key InChIKey=FFJICIDEVUQXRQ-ZCHKFXGQSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 209025   

TargetInsulin-degrading enzyme(Homo sapiens (Human))
President and Fellows of Harvard College

US Patent
LigandPNGBDBM209025(US9243038, 5a (cis olefin) | US9243038, 5b (trans ...)
Affinity DataIC50: >1.00E+3nMAssay Description:Macrocycles were assayed for IDE inhibition by monitoring cleavage of a substrate peptide containing a fluorophore-quencher pair such that cleavage o...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInsulin-degrading enzyme(Homo sapiens (Human))
President and Fellows of Harvard College

US Patent
LigandPNGBDBM209025(US9243038, 5a (cis olefin) | US9243038, 5b (trans ...)
Affinity DataIC50: >2.00E+4nMAssay Description:Macrocycles were assayed for IDE inhibition by monitoring cleavage of a substrate peptide containing a fluorophore-quencher pair such that cleavage o...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent