BDBM209025 US9243038, 5a (cis olefin)::US9243038, 5b (trans olefin)
SMILES NC(=O)[C@@H]1CCCCNC(=O)[C@@H](Cc2ccc(cc2)C(=O)c2ccccc2)NC(=O)[C@H](CC2CCCCC2)NC(=O)[C@H](CC2CC2)NC(=O)\C=C\C(=O)N1
InChI Key InChIKey=FFJICIDEVUQXRQ-ZCHKFXGQSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 209025
TargetInsulin-degrading enzyme(Homo sapiens (Human))
President and Fellows of Harvard College
US Patent
President and Fellows of Harvard College
US Patent
Affinity DataIC50: >1.00E+3nMAssay Description:Macrocycles were assayed for IDE inhibition by monitoring cleavage of a substrate peptide containing a fluorophore-quencher pair such that cleavage o...More data for this Ligand-Target Pair
TargetInsulin-degrading enzyme(Homo sapiens (Human))
President and Fellows of Harvard College
US Patent
President and Fellows of Harvard College
US Patent
Affinity DataIC50: >2.00E+4nMAssay Description:Macrocycles were assayed for IDE inhibition by monitoring cleavage of a substrate peptide containing a fluorophore-quencher pair such that cleavage o...More data for this Ligand-Target Pair