BDBM27960 (2R,3S)-1-[(7-methyl-2,3-dihydro-1H-inden-4-yl)oxy]-3-(propan-2-ylamino)butan-2-ol::CHEMBL198059::ICI118551
SMILES CC(C)N[C@@H](C)[C@@H](O)COc1ccc(C)c2CCCc12
InChI Key InChIKey=VFIDUCMKNJIJTO-BBRMVZONSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 27960
Affinity DataKi: 1nM ΔG°: -12.1kcal/mole IC50: 3nMpH: 7.4 T: 2°CAssay Description:In the binding assays, the results were expressed as percent inhibition of the control radioligand specific binding. The IC50 values (concentration c...More data for this Ligand-Target Pair
Affinity DataKd: 182nMAssay Description:Displacement of [3H](-)CGP12177 from human beta1-AR expressed in CHOK1 cells after 2 hrs by TopCount microscintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKd: 0.245nMAssay Description:Displacement of [3H](-)CGP12177 from human beta2-AR expressed in CHOK1 cells after 2 hrs by TopCount microscintillation counting methodMore data for this Ligand-Target Pair
Affinity DataIC50: 0.740nMAssay Description:Displacement of [3H]CGP 12177 from human recombinant beta2 adrenergic receptor expressed in CHO cells measured after 120 mins by scintillation counti...More data for this Ligand-Target Pair