BDBM3191 (+-)-2-[[2,6-Dihydroxy-4-[[[2-(N,N-dimethylamino)-3-(4-hydroxyphenyl)propyl]oxy]carbonyl]phenyl]carbonyl]-3-hydroxybenzoic Acid, trifluoroacetic acid salt::2-[(4-{[2-(dimethylamino)-3-(4-hydroxyphenyl)propoxy]carbonyl}-2,6-dihydroxyphenyl)carbonyl]-3-hydroxybenzoic acid::Acyclic Balanol Analog 15b

SMILES CN(C)C(COC(=O)c1cc(O)c(C(=O)c2c(O)cccc2C(O)=O)c(O)c1)Cc1ccc(O)cc1

InChI Key InChIKey=WQSCDMQTCWOCID-UHFFFAOYSA-N

Data  8 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 8 hits for monomerid = 3191   

TargetProtein kinase C delta type(Human)
Sphinx Laboratories

LigandChemical structure of BindingDB Monomer ID 3191BDBM3191(2-[(4-{[2-(dimethylamino)-3-(4-hydroxyphenyl)propo...)
Affinity DataIC50: 270nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2005
Entry Details Article
PubMed
TargetProtein kinase C beta type(Human)
Sphinx Laboratories

LigandChemical structure of BindingDB Monomer ID 3191BDBM3191(2-[(4-{[2-(dimethylamino)-3-(4-hydroxyphenyl)propo...)
Affinity DataIC50: 500nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2005
Entry Details Article
PubMed
TargetProtein kinase C beta type(Human)
Sphinx Laboratories

LigandChemical structure of BindingDB Monomer ID 3191BDBM3191(2-[(4-{[2-(dimethylamino)-3-(4-hydroxyphenyl)propo...)
Affinity DataIC50: 880nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2005
Entry Details Article
PubMed
TargetProtein kinase C eta type(Human)
Sphinx Laboratories

LigandChemical structure of BindingDB Monomer ID 3191BDBM3191(2-[(4-{[2-(dimethylamino)-3-(4-hydroxyphenyl)propo...)
Affinity DataIC50: 1.40E+3nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2005
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Sphinx Laboratories

LigandChemical structure of BindingDB Monomer ID 3191BDBM3191(2-[(4-{[2-(dimethylamino)-3-(4-hydroxyphenyl)propo...)
Affinity DataIC50: 4.00E+3nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2005
Entry Details Article
PubMed
TargetProtein kinase C gamma type(Human)
Sphinx Laboratories

LigandChemical structure of BindingDB Monomer ID 3191BDBM3191(2-[(4-{[2-(dimethylamino)-3-(4-hydroxyphenyl)propo...)
Affinity DataIC50: 4.20E+3nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2005
Entry Details Article
PubMed
TargetProtein kinase C epsilon type(Human)
Sphinx Laboratories

LigandChemical structure of BindingDB Monomer ID 3191BDBM3191(2-[(4-{[2-(dimethylamino)-3-(4-hydroxyphenyl)propo...)
Affinity DataIC50: 3.00E+4nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 3191BDBM3191(2-[(4-{[2-(dimethylamino)-3-(4-hydroxyphenyl)propo...)
Affinity DataIC50: 5.00E+4nMAssay Description:The activity of PKA, activated by cAMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2005
Entry Details Article
PubMed