BDBM3196 (+-)-2-[[2,6-Dihydroxy-4-[[2-(4-hydroxyphenyl)-2-[(phenylsulfonyl)amino]ethoxy]carbonyl]phenyl]carbonyl]-3-hydroxybenzoic Acid::2-[(4-{[2-benzenesulfonamido-2-(4-hydroxyphenyl)ethoxy]carbonyl}-2,6-dihydroxyphenyl)carbonyl]-3-hydroxybenzoic acid::Acyclic Balanol Analog 13b

SMILES OC(=O)c1cccc(O)c1C(=O)c1c(O)cc(cc1O)C(=O)OCC(NS(=O)(=O)c1ccccc1)c1ccc(O)cc1

InChI Key InChIKey=VMKYWYSMWRGVAG-UHFFFAOYSA-N

Data  8 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 8 hits for monomerid = 3196   

TargetProtein kinase C delta type(Human)
Sphinx Laboratories

LigandChemical structure of BindingDB Monomer ID 3196BDBM3196(2-[(4-{[2-benzenesulfonamido-2-(4-hydroxyphenyl)et...)
Affinity DataIC50: 1.90E+3nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2005
Entry Details Article
PubMed
TargetProtein kinase C beta type(Human)
Sphinx Laboratories

LigandChemical structure of BindingDB Monomer ID 3196BDBM3196(2-[(4-{[2-benzenesulfonamido-2-(4-hydroxyphenyl)et...)
Affinity DataIC50: 2.80E+3nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2005
Entry Details Article
PubMed
TargetProtein kinase C eta type(Human)
Sphinx Laboratories

LigandChemical structure of BindingDB Monomer ID 3196BDBM3196(2-[(4-{[2-benzenesulfonamido-2-(4-hydroxyphenyl)et...)
Affinity DataIC50: 3.30E+3nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2005
Entry Details Article
PubMed
TargetProtein kinase C gamma type(Human)
Sphinx Laboratories

LigandChemical structure of BindingDB Monomer ID 3196BDBM3196(2-[(4-{[2-benzenesulfonamido-2-(4-hydroxyphenyl)et...)
Affinity DataIC50: 4.80E+3nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2005
Entry Details Article
PubMed
TargetProtein kinase C beta type(Human)
Sphinx Laboratories

LigandChemical structure of BindingDB Monomer ID 3196BDBM3196(2-[(4-{[2-benzenesulfonamido-2-(4-hydroxyphenyl)et...)
Affinity DataIC50: 1.10E+4nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 3196BDBM3196(2-[(4-{[2-benzenesulfonamido-2-(4-hydroxyphenyl)et...)
Affinity DataIC50: 5.00E+4nMAssay Description:The activity of PKA, activated by cAMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2005
Entry Details Article
PubMed
TargetProtein kinase C epsilon type(Human)
Sphinx Laboratories

LigandChemical structure of BindingDB Monomer ID 3196BDBM3196(2-[(4-{[2-benzenesulfonamido-2-(4-hydroxyphenyl)et...)
Affinity DataIC50: 5.00E+4nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2005
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Sphinx Laboratories

LigandChemical structure of BindingDB Monomer ID 3196BDBM3196(2-[(4-{[2-benzenesulfonamido-2-(4-hydroxyphenyl)et...)
Affinity DataIC50: 5.00E+4nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2005
Entry Details Article
PubMed