BDBM50065110 CHEMBL418890::N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-phenyl]-2,4-dichloro-benzamide
SMILES Clc1ccc(C(=O)Nc2ccc(cc2)C(=O)N2Cc3cccn3Cc3ccccc23)c(Cl)c1
InChI Key InChIKey=QJUIBLKMWVDTSN-UHFFFAOYSA-N
Data 10 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 10 hits for monomerid = 50065110
Affinity DataIC50: 3.20nMAssay Description:Displacement of [3H]-AVP from human V2 receptor expressed in murine fibroblast cell line (LV2) membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Displacement of (Phe-3,4,5-H) Vasopressin from V1a recptor from rat liver membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 3.10nMAssay Description:Displacement of [3H]-AVP from vasopressin V2 receptor of rat kidney medulla.More data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Displacement of [3H]-AVP from vasopressin receptor (V1a) from human platelet membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of [3H]-AVP binding to Dawley rat kidney medullary vasopressin V2 receptor.More data for this Ligand-Target Pair
Affinity DataIC50: 3.10nMAssay Description:Binding affinity to rat V2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:In vitro binding affinity to human V1a receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:In vitro binding affinity for rat V1a receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of [3H]-AVP binding to Dawley rat hepatic vasopressin V1a receptor.More data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:In vitro binding affinity to human V2 receptorMore data for this Ligand-Target Pair