BDBM50185366 CHEMBL2371911::CHEMBL436499::Sub[-Trp-Arg-Nva-Arg-Tyr-NH2]2
SMILES CCC[C@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](N)CCCC[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCC)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccc(O)cc1)C(N)=O)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccc(O)cc1)C(N)=O
InChI Key InChIKey=OWXAFDOATMPIJT-YCMBARDJSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 9 hits for monomerid = 50185366
Affinity DataKi: 2nMAssay Description:Reduced farnesylation of H-ras transformed NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of [3H]-FPP incorporation into biotin-linked K-ras decapeptide (CVIM) by bovine farnesyltransferaseMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:In vitro inhibitory activity against Factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:In vitro inhibitory activity against Factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 390nMAssay Description:Displacement of [125I]NPY from human NPY2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 530nMAssay Description:In vitro inhibitory activity against Factor XaMore data for this Ligand-Target Pair
Affinity DataEC50: 430nMAssay Description:Agonist activity at human NPY4 receptor in HEK293 cells by inhibition of forskolin-stimulated cAMP synthesisMore data for this Ligand-Target Pair
Affinity DataEC50: 1.41E+3nMAssay Description:Agonist activity at human NPY1 receptor in CHO cells by inhibition of forskolin-stimulated cAMP synthesisMore data for this Ligand-Target Pair
Affinity DataEC50: 370nMAssay Description:Inhibition of [3H]-FPP incorporation into biotin-linked K-ras decapeptide (CVIM) by bovine farnesyltransferaseMore data for this Ligand-Target Pair