BDBM50246881 CHEMBL4076292

SMILES OC(=O)c1ccc(cc1)S(=O)(=O)Nc1ccc(Oc2ccc(Cl)c(c2)C(F)(F)F)c(c1)C#N

InChI Key InChIKey=DJDKMQCYTRHYFU-UHFFFAOYSA-N

Data  1 IC50

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50246881   

TargetPlatelet-activating factor acetylhydrolase(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50246881(CHEMBL4076292)
Affinity DataIC50:  5nMAssay Description:Inhibition of human recombinant GST-tagged Lp-PLA2 (47 to 429 residues) expressed in Escherichia coli Rosetta(DE3) pLysS using 2-thio-PAF as substrat...More data for this Ligand-Target Pair