BDBM50247673 2-[1'-Phenyl-3'-(4-methoxyphenyl)-2'-propenylidene]hydrazine-3-methyl-4(3H)-quinazolinone::CHEMBL454379

SMILES COc1ccc(CC=C(N=Nc2nc3ccccc3c(=O)n2C)c2ccccc2)cc1

InChI Key InChIKey=KDCHQCSIQQEGPS-UHFFFAOYSA-N

Data  2 KI  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50247673   

TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50247673(2-[1'-Phenyl-3'-(4-methoxyphenyl)-2'-propenylidene...)
Affinity DataKi:  1.15E+3nMAssay Description:Inhibition of MAO-A in rat liver homogenate after 60 mins by Lineweaver-Burk plotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50247673(2-[1'-Phenyl-3'-(4-methoxyphenyl)-2'-propenylidene...)
Affinity DataKi:  1.06E+4nMAssay Description:Inhibition of MAO-B in rat liver homogenate after 60 mins by Lineweaver-Burk plotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50247673(2-[1'-Phenyl-3'-(4-methoxyphenyl)-2'-propenylidene...)
Affinity DataIC50:  9.05E+3nMAssay Description:Inhibition of MAO-A in rat liver homogenate after 60 mins by residual activity plotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50247673(2-[1'-Phenyl-3'-(4-methoxyphenyl)-2'-propenylidene...)
Affinity DataIC50:  3.99E+5nMAssay Description:Inhibition of MAO-B in rat liver homogenate after 60 mins by residual activity plotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed