BDBM50254655 CHEMBL465086::N-benzyl-7-(3,4-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide

SMILES CC1=Nc2ccnn2C(C1C(=O)NCc1ccccc1)c1ccc(Cl)c(Cl)c1

InChI Key InChIKey=LQXPLQZAVHAHQZ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50254655   

TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50254655(CHEMBL465086 | N-benzyl-7-(3,4-dichlorophenyl)-5-m...)
Affinity DataIC50:  160nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cells by EP voltage clamp techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed