BDBM50254697 (7-(3,4-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)(pyrrolidin-1-yl)methanone::CHEMBL465276

SMILES CC1=Nc2ccnn2C(C1C(=O)N1CCCC1)c1ccc(Cl)c(Cl)c1

InChI Key InChIKey=MWOOFQXRXCRPCL-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50254697   

TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50254697((7-(3,4-dichlorophenyl)-5-methyl-4,7-dihydropyrazo...)
Affinity DataIC50:  660nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50254697((7-(3,4-dichlorophenyl)-5-methyl-4,7-dihydropyrazo...)
Affinity DataIC50:  660nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cells by EP voltage clamp techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed