BDBM50263224 CHEMBL4066795

SMILES C1C2=C(CN1)N(C(=O)NC2=O)C[C@@H](C(=O)O)N

InChI Key InChIKey=PGFCMMRTCMWFGC-UHFFFAOYSA-N

Data  4 KI

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50263224   

TargetGlutamate receptor ionotropic, kainate 1(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50263224(CHEMBL4066795)
Affinity DataKi:  869nMAssay Description:Displacement of [3H]SYM2081 from recombinant homomeric rat GluK1 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/29/2020
Entry Details Article
PubMed
TargetGlutamate receptor 2(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50263224(CHEMBL4066795)
Affinity DataKi:  2.37E+3nMAssay Description:Displacement of [3H]AMPA from recombinant homomeric rat GluA2 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/29/2020
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50263224(CHEMBL4066795)
Affinity DataKi:  1.81E+4nMAssay Description:Displacement of [3H]SYM2081 from recombinant homomeric rat GluK3 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/29/2020
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50263224(CHEMBL4066795)
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]SYM2081 from recombinant homomeric rat GluK2 receptor expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/29/2020
Entry Details Article
PubMed