BDBM50267296 CHEMBL4104658
SMILES COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cn2CCCc3cccc1c23
InChI Key InChIKey=CLXOEYRLLVMPJB-UHFFFAOYSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50267296
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Nanjing Normal University
Curated by ChEMBL
Nanjing Normal University
Curated by ChEMBL
Affinity DataIC50: 8.46E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells by lonWorks Quattro analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 405nMAssay Description:Inhibition of EGR-induced EGFR phosphorylation in human A549 cells pretreated for 2 hrs followed by EGF stimulation by immune assayMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of human recombinant cytoplasmic GST-tagged EGFR (668 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubated fo...More data for this Ligand-Target Pair