BDBM50295515 CHEMBL560780::N-(4-Iodophenyl)-2-[5-(3-methoxybenzyl)-3-methyl-6-oxo-6H-pyridazin-1-yl]-acetamide

SMILES COc1cccc(Cc2cc(C)nn(CC(=O)Nc3ccc(I)cc3)c2=O)c1

InChI Key InChIKey=CRXUEUHJLRJWGE-UHFFFAOYSA-N

Data  7 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 7 hits for monomerid = 50295515   

TargetfMet-Leu-Phe receptor(Homo sapiens (Human))
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50295515(CHEMBL560780 | N-(4-Iodophenyl)-2-[5-(3-methoxyben...)
Affinity DataEC50:  3.20E+3nMAssay Description:Agonist activity at FPR1 in human neutrophiles by chemotaxis assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50295515(CHEMBL560780 | N-(4-Iodophenyl)-2-[5-(3-methoxyben...)
Affinity DataEC50:  1.80E+3nMAssay Description:Agonist activity at FPRL1 in human neutrophiles by chemotaxis assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetfMet-Leu-Phe receptor(Homo sapiens (Human))
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50295515(CHEMBL560780 | N-(4-Iodophenyl)-2-[5-(3-methoxyben...)
Affinity DataEC50:  2.80E+3nMAssay Description:Agonist activity at FPR1 expressed in human HL60 cells assessed as induction of intracellular calcium flux by FLIPR3 calcium assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 3(Homo sapiens (Human))
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50295515(CHEMBL560780 | N-(4-Iodophenyl)-2-[5-(3-methoxyben...)
Affinity DataEC50:  1.30E+4nMAssay Description:Agonist activity at FPRL2 expressed in human HL60 cells assessed as induction of intracellular calcium flux by FLIPR3 calcium assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50295515(CHEMBL560780 | N-(4-Iodophenyl)-2-[5-(3-methoxyben...)
Affinity DataEC50:  1.80E+3nMAssay Description:Agonist activity at FPRL1 in human neutrophiles assessed as induction of intracellular calcium flux by FLIPR3 calcium assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50295515(CHEMBL560780 | N-(4-Iodophenyl)-2-[5-(3-methoxyben...)
Affinity DataEC50:  6.80E+3nMAssay Description:Agonist activity at FPRL1 expressed in human HL60 cells assessed as induction of intracellular calcium flux by FLIPR3 calcium assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetfMet-Leu-Phe receptor(Homo sapiens (Human))
Universita Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50295515(CHEMBL560780 | N-(4-Iodophenyl)-2-[5-(3-methoxyben...)
Affinity DataEC50:  3.20E+3nMAssay Description:Agonist activity at FPR1 in human neutrophiles assessed as induction of intracellular calcium flux by FLIPR3 calcium assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed