BDBM50316777 2-[5-(4-Hydroxyphenethoxy)-1H-indole-3-yl]ethanamine hydrochloride::CHEMBL1095957

SMILES NCCc1c[nH]c2ccc(OCCc3ccc(O)cc3)cc12

InChI Key InChIKey=FVMIAPQLQLJTFD-UHFFFAOYSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50316777   

TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50316777(2-[5-(4-Hydroxyphenethoxy)-1H-indole-3-yl]ethanami...)
Affinity DataIC50:  2.64E+3nMAssay Description:Inhibition of VEGFR3 after 30 mins by chemiluminescence ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50316777(2-[5-(4-Hydroxyphenethoxy)-1H-indole-3-yl]ethanami...)
Affinity DataIC50:  2.02E+3nMAssay Description:Noncompetitive inhibition of VEGFR2 after 30 mins by chemiluminescence ELISA in presence of 25 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50316777(2-[5-(4-Hydroxyphenethoxy)-1H-indole-3-yl]ethanami...)
Affinity DataIC50:  1.78E+3nMAssay Description:Noncompetitive inhibition of IGF1R after 30 mins by chemiluminescence ELISA in presence of 50 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50316777(2-[5-(4-Hydroxyphenethoxy)-1H-indole-3-yl]ethanami...)
Affinity DataIC50:  2.07E+3nMAssay Description:Inhibition of EGFR after 30 mins by chemiluminescence ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed