BDBM50352494 CHEMBL1824332
SMILES COc1ccc(CNC(=O)Nc2nc3ccc(cc3s2)-c2nnn[nH]2)cc1
InChI Key InChIKey=AYGDBNIQKVIIGQ-UHFFFAOYSA-N
Data 6 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50352494
TargetProtein kinase C alpha type(Homo sapiens (Human))
Technische Universit£T Darmstadt
Curated by ChEMBL
Technische Universit£T Darmstadt
Curated by ChEMBL
Affinity DataIC50: 2.42E+7nMAssay Description:Inhibition of human PKCalpha activity using Ser/Thr 7 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Technische Universit£T Darmstadt
Curated by ChEMBL
Technische Universit£T Darmstadt
Curated by ChEMBL
Affinity DataIC50: 2.64E+7nMAssay Description:Inhibition of human CDK5/p35 activity using Ser/Thr 12 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.80E+6nMAssay Description:Inhibition of human AURKA activity using Ser/Thr 1 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Technische Universit£T Darmstadt
Curated by ChEMBL
Technische Universit£T Darmstadt
Curated by ChEMBL
Affinity DataIC50: 1.30E+5nMAssay Description:Inhibition of human GSK3alpha activity using Ser/Thr 11 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Technische Universit£T Darmstadt
Curated by ChEMBL
Technische Universit£T Darmstadt
Curated by ChEMBL
Affinity DataIC50: 1.53E+7nMAssay Description:Inhibition of human CKI epsilon activity using Ser/Thr 11 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Technische Universit£T Darmstadt
Curated by ChEMBL
Technische Universit£T Darmstadt
Curated by ChEMBL
Affinity DataIC50: 1.40E+5nMAssay Description:Inhibition of human GSK3-beta activity using Ser/Thr 9 peptide as substrate by FRET assayMore data for this Ligand-Target Pair