BDBM50369624 CHEMBL1790730
SMILES OC[C@H]1O[C@H](C[C@@H]1O)n1cnc2c(NC3CCCCC3)ncnc12
InChI Key InChIKey=YYOYZRBZIVNMFY-YNEHKIRRSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50369624
Affinity DataKi: 412nMAssay Description:Binding affinity for adenosine A1 receptor, was assessed from the ability to displace [3H]-DPCPX (without GTP) from rat cortical membranes.More data for this Ligand-Target Pair
Affinity DataKi: 8.94E+3nMAssay Description:Affinity for the Adenosine A1 receptor in the absence of GTP (A1-GTP) by using [3H]DPCPX as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.67E+4nMAssay Description:Binding affinity for adenosine A1 receptor, was assessed from the ability to displace [3H]DPCPX (with 1 mM GTP) from rat cortical membranes.More data for this Ligand-Target Pair
Affinity DataKi: 2.28E+4nMAssay Description:Affinity for the Adenosine A1 receptor in the presence of GTP (A1+GTP) by using [3H]-DPCPX as radioligandMore data for this Ligand-Target Pair
Affinity DataEC50: 9.64E+3nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding to rat brain membranes by adenosine A1 receptor activationMore data for this Ligand-Target Pair