BDBM50525957 CHEMBL4461515

SMILES CC(C)C[C@H](NC(=O)c1cc2ccccc2s1)C(=O)N1CCN(CC1)C(=O)[C@H](CO)NS(=O)(=O)c1ccc(Cl)cc1Cl

InChI Key InChIKey=IVYQPSHHYIAUFO-VXKWHMMOSA-N

Data  1 EC50

PDB links: 4 PDB IDs match this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50525957   

TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Asahi Kasei Medical

Curated by ChEMBL
LigandPNGBDBM50525957(CHEMBL4461515)
Affinity DataEC50:  49nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair