BDBM81924 (R)-3-(1-Propyl-piperidin-3-yl)-phenol::3PPP(+/-)::CAS_85976-54-1::CHEMBL276500::NSC_202477::PPP, R(+)-3::PPP, S(-)-3
SMILES CCCN1CCCC(C1)c1cccc(O)c1
InChI Key InChIKey=HTSNFXAICLXZMA-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 38 hits for monomerid = 81924
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Janssen Research Foundation
Curated by PDSP Ki Database
Janssen Research Foundation
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 3A(GUINEA PIG)
Syntex Discovery Research
Curated by PDSP Ki Database
Syntex Discovery Research
Curated by PDSP Ki Database
Affinity DataKi: 32nMAssay Description:Binding towards Dopamine receptor D2 expressed in CHO-K1 cells using [3H]-U-86,170More data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Binding towards Dopamine receptor D2 using [3H]-spiperone from rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Binding towards Dopamine receptor D2 expressed in CHO-K1 cells using [3H]-U-86,170More data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Evaluated for binding towards Dopamine receptor D2 using [3H]-N-0437 as radioligand from rat striatal membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Virginia Commonwealth University
Curated by ChEMBL
Virginia Commonwealth University
Curated by ChEMBL
Affinity DataKi: 79nMAssay Description:Opioid activity in terms of inhibition of [3H]dihydromorphine binding to opioid receptor mu in rat brain membrane.More data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Binding towards dopamine receptor D4 expressed in CHO-K1 cells using [3H]spiperone More data for this Ligand-Target Pair
Affinity DataKi: 132nMAssay Description:Compound was measured for its ability to compete with [3H]spiperone binding to the human Dopamine receptor D3 transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 217nMAssay Description:Binding towards Dopamine receptor D2 expressed in CHO-K1 cells using [3H]-U-86,170More data for this Ligand-Target Pair
Affinity DataKi: 217nMAssay Description:Binding towards Dopamine receptor D3 expressed in CHO-K1 cells using [3H]spiperone More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A(GUINEA PIG)
Syntex Discovery Research
Curated by PDSP Ki Database
Syntex Discovery Research
Curated by PDSP Ki Database
Affinity DataKi: 700nMAssay Description:Binding towards dopamine receptor D4 expressed in CHO-K1 cells using [3H]spiperone More data for this Ligand-Target Pair
Affinity DataKi: 700nMAssay Description:Evaluated for binding towards Dopamine receptor D2 using [3H]-spiperone as radioligand, in cloned mammalian receptors expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 776nMAssay Description:Evaluated for binding towards Dopamine receptor D2 using [3H]-spiperone as radioligand, in cloned mammalian receptors expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 776nMAssay Description:Evaluated for binding towards Dopamine receptor D2 using [3H]-spiperone as radioligand, in cloned mammalian receptors expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding towards Dopamine receptor D2 expressed in CHO-K1 cells using [3H]-U-86,170More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Sri International
Curated by PDSP Ki Database
Sri International
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Mus musculus (Mouse))
Medical Research Service
Curated by PDSP Ki Database
Medical Research Service
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sri International
Curated by PDSP Ki Database
Sri International
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Sri International
Curated by PDSP Ki Database
Sri International
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
Sri International
Curated by PDSP Ki Database
Sri International
Curated by PDSP Ki Database
Affinity DataIC50: 430nMAssay Description:Evaluated for binding towards Dopamine receptor D2 using [3H]-spiperone as radioligand, in cloned mammalian receptors expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 183nMAssay Description:Inhibition of [3H]N-propylnorapomorphine binding to Dopamine receptor D2 of rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.28E+3nMAssay Description:Binding affinity towards dopamine receptor D2 in rat striatal membrane using [3H]spiperoneMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro binding affinity towards dopamine receptor D1 in rat striatal membrane using [3H]-SCH- 23390More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of binding of [3H]SCH-23390 to Dopamine receptor D1 was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 930nMAssay Description:Inhibition of [3H]haloperidol binding for Dopamine receptor D2 in rat striatal membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 590nMAssay Description:Inhibition of [3H]haloperidol binding for Dopamine receptor D2 in rat striatal membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 430nMAssay Description:Binding effinity for sigma receptor using 2 nM of [3H]-DTG as radioligand, in membranes from brain minus cerebellumMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Virginia Commonwealth University
Curated by ChEMBL
Virginia Commonwealth University
Curated by ChEMBL
Affinity DataIC50: 76nMAssay Description:Displacement of [3H]-DTG from sigma opioid receptor of homogenized guinea pig whole brainMore data for this Ligand-Target Pair
Affinity DataIC50: 184nMAssay Description:Inhibition of [3H]haloperidol binding for Dopamine receptor D2 in rat striatal membranes.More data for this Ligand-Target Pair