2187 SMILES Strings for DNA-dependent protein kinase catalytic subunit

Compound Name
SMILES String
COc1cc2ncc3n(C)nc(-c4ccc(cc4)-c4ccn[nH]4)c3c2cc1-c1cn[nH]c1
Nc1ncnc2n(nc(-c3ccn4ccnc4c3)c12)C1CCCC1
COc1cc2ncc3[nH]nc(-c4ccc(cc4)C#N)c3c2cc1OC
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OC
COc1cc2ncc3n(C)nc(-c4ccc(C#N)c(Br)c4)c3c2cc1OC
COc1cc2c3c(nn(C)c3cnc2cc1O)-c1ccc(cc1)C#N
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1O
COc1cc2ncc3n(C)nc(-c4ccc(cc4F)C#N)c3c2cc1O
COc1cc2ncc3[nH]nc(-c4ccc(C#N)c(Cl)c4)c3c2cc1OC
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OC(C(N)=O)c1ccc(F)cc1
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1O[C@@H](C(N)=O)c1ccc(F)cc1 |r|
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1O[C@H](C(N)=O)c1ccc(F)cc1 |r|
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OCc1ccncc1
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OCc1cccnc1
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OCc1ccccn1
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OCc1ccccc1C#N
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OCc1ccc(F)cc1
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OC(F)F
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OC(F)(F)c1ccccc1
COC(=O)C(Oc1cc2c3c(nn(C)c3cnc2cc1OC)-c1ccc(cc1)C#N)c1ccc(F)cc1
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OC(C(O)=O)c1ccc(F)cc1
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OC(C(O)=O)c1ccccc1
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OC(C(O)=O)c1cccs1
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OC(C)(C(O)=O)c1ccccc1
COc1cc2ncc3n(C)nc(-c4ccc(cc4F)C#N)c3c2cc1OC(C(N)=O)c1ccc(F)cc1
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OS(=O)(=O)c1ccc(C)cc1
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OP(O)(=O)c1ccccc1
COc1cc2c3c(nn(C)c3cnc2cc1OC(F)F)-c1ccc(cc1)C#N
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OCc1ccc(CO)cc1
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OCc1cccc(CN2CCOCC2)c1
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OCc1ccc(nc1)-n1cccn1
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OCc1cnc2[nH]ccc2c1
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OCc1ccc(cc1)-n1cncn1
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OCc1cccc(CN)c1
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OCc1ccnc(N)c1
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OCc1cccs1
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OCc1ccsc1
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OCc1cc(Br)cs1
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OCc1cc2ccccc2s1
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OCc1ccnc(c1)C#N
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OCc1nccs1
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OCCN(C)C
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OCc1cccc(c1)N(C)C
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OCc1cscn1
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OCc1cncs1
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OCc1cccc(CN2CCN(C)CC2)c1
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OCc1cccc(c1)-c1csc(C)n1
COc1cc2c3c(nn(C)c3cnc2cc1OCCN(C)C)-c1ccc(cc1)C#N
COc1cc2c3c(nn(C)c3cnc2cc1OCC(O)CO)-c1ccc(cc1)C#N
CCN1CCN(CCNC(=O)C(Oc2cc3c4c(nn(C)c4cnc3cc2OC)-c2ccc(cc2)C#N)c2ccc(F)cc2)CC1
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OC(C(=O)NCCN(C)C)c1ccc(F)cc1
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OC(C(=O)NCCN1CCNCC1)c1ccc(F)cc1
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OC(C(=O)NOCC#N)c1ccc(F)cc1
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OC(C(=O)NCCS(N)(=O)=O)c1ccc(F)cc1
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OC(C(=O)NO)c1ccc(F)cc1
COc1cc2ncc3n(C)nc(-c4ccc(cc4)C#N)c3c2cc1OC(C(=O)NC(N)=N)c1ccc(F)cc1
COCCNC(=O)C(Oc1cc2c3c(nn(C)c3cnc2cc1OC)-c1ccc(cc1)C#N)c1ccc(F)cc1
CCn1nc(-c2ccc(cc2)C#N)c2c1cnc1cc(OC)c(OC)cc21
CCn1nc(-c2ccc(cc2F)C#N)c2c1cnc1cc(OC)c(OC)cc21
CCCCn1nc(-c2ccc(cc2)C#N)c2c1cnc1cc(OC)c(OC)cc21
CCCn1nc(-c2ccc(cc2)C#N)c2c1cnc1cc(OC)c(OC)cc21
COc1cc2ncc3n(nc(-c4ccc(cc4)C#N)c3c2cc1OC)C(C)C
COc1cc2ncc3n(CC(C)C)nc(-c4ccc(cc4)C#N)c3c2cc1OC
COc1cc2ncc3n(nc(-c4ccc(cc4)C#N)c3c2cc1OC)C1CC1
COc1cc2ncc3n(CC=C)nc(-c4ccc(cc4)C#N)c3c2cc1OC
COc1cc2ncc3n(Cc4cccnc4)nc(-c4ccc(cc4F)C#N)c3c2cc1OC
COc1cc2ncc3n(nc(-c4ccc(cc4)C#N)c3c2cc1OC)C#N
COc1cc2ncc3n(CC#N)nc(-c4ccc(cc4)C#N)c3c2cc1OC
COc1cc2ncc3n(CC(O)=O)nc(-c4ccc(cc4)C#N)c3c2cc1OC
COc1cc2ncc3n(CC(N)=O)nc(-c4ccc(cc4)C#N)c3c2cc1OC
COc1cc2ncc3n(nc(-c4ccc(cc4)C#N)c3c2cc1OC)C(F)F
COc1cc2ncc3n[nH]c(-c4ccc(C#N)c(c4)N4CCCC4)c3c2cc1OC
COCc1cc(ccc1C#N)-c1nn(C)c2cnc3cc(OC)c(OC)cc3c12
COC(=O)c1cc(ccc1C#N)-c1[nH]nc2cnc3cc(OC)c(OC)cc3c12
COc1cc2ncc3n[nH]c(-c4ccc(C#N)c(c4)C(O)=O)c3c2cc1OC
COc1cc2ncc3n[nH]c(-c4ccc(C#N)c(c4)-c4ccccc4)c3c2cc1OC
CCN1CCN(CC1)c1ccc(cc1)-c1nn(C)c2cnc3cc(OC)c(OC)cc3c12
COc1cc2ncc3n(C)nc(-c4ccccc4F)c3c2cc1OC
COc1cc2ncc3n(C)nc(-c4ccc(cc4F)C#N)c3c2cc1-c1cccnc1
COc1cc2ncc3n(C)nc(-c4ccc(cc4F)C#N)c3c2cc1-c1cnc2ccccc2c1
COc1cc2ncc3n(C)nc(-c4ccc(cc4F)C#N)c3c2cc1-c1cc[nH]c1
COc1cc2ncc3[nH]c(=O)n(-c4ccc(cc4)C#N)c3c2cc1OC
COc1cc2ncc3n(C)c(=O)n(-c4ccc(cc4)C#N)c3c2cc1OC
COc1cc2ncc3n(C)c(=O)n(-c4ccc(cc4)C#N)c3c2cc1O
COc1cc2ncc3n(C)c(=O)n(-c4ccc(cc4F)C#N)c3c2cc1O |(-5.55,.03,;-4.22,.8,;-2.89,.03,;-2.89,-1.51,;-1.55,-2.28,;-1.55,-3.82,;-.22,-4.59,;1.11,-3.82,;2.58,-4.3,;3.35,-5.63,;3.48,-3.05,;5.02,-3.05,;2.58,-1.81,;2.98,-.32,;1.89,.77,;2.29,2.26,;3.77,2.66,;4.86,1.57,;4.47,.08,;5.55,-1.01,;4.17,4.14,;4.57,5.63,;1.11,-2.28,;-.22,-1.51,;-.22,.03,;-1.55,.8,;-1.55,2.34,)|
COc1cc2ncc3n(C)c(=O)n(-c4c(F)cc(cc4F)C#N)c3c2cc1O |(-5.55,.03,;-4.22,.8,;-2.89,.03,;-2.89,-1.51,;-1.55,-2.28,;-1.55,-3.82,;-.22,-4.59,;1.11,-3.82,;2.58,-4.3,;3.35,-5.63,;3.48,-3.05,;5.02,-3.05,;2.58,-1.81,;2.98,-.32,;4.47,.08,;5.55,-1.01,;4.86,1.57,;3.77,2.66,;2.29,2.26,;1.89,.77,;.4,.37,;4.17,4.14,;4.57,5.63,;1.11,-2.28,;-.22,-1.51,;-.22,.03,;-1.55,.8,;-1.55,2.34,)|
COc1cc2ncc3[nH]c(=O)n(-c4ccc(cc4)C#N)c3c2cc1OCc1ccccc1
COc1cc2ncc3n(C)c(=O)n(-c4ccc(cc4)C#N)c3c2cc1OCc1ccccc1
COc1cc2ncc3[nH]c(=O)n(-c4ccc(cc4F)C#N)c3c2cc1OCc1ccccc1 |(-5.55,-1.54,;-4.22,-.77,;-2.89,-1.54,;-2.89,-3.08,;-1.55,-3.85,;-1.55,-5.39,;-.22,-6.16,;1.11,-5.39,;2.58,-5.87,;3.48,-4.62,;5.02,-4.62,;2.58,-3.37,;2.98,-1.89,;1.89,-.8,;2.29,.69,;3.77,1.09,;4.86,-0,;4.47,-1.49,;5.55,-2.58,;4.17,2.58,;4.57,4.06,;1.11,-3.85,;-.22,-3.08,;-.22,-1.54,;-1.55,-.77,;-1.55,.77,;-2.89,1.54,;-2.89,3.08,;-1.55,3.85,;-1.55,5.39,;-2.89,6.16,;-4.22,5.39,;-4.22,3.85,)|
COc1cc2ncc3n(C)c(=O)n(-c4ccc(cc4F)C#N)c3c2cc1OCc1ccccc1 |(-5.55,-1.02,;-4.22,-.25,;-2.89,-1.02,;-2.89,-2.56,;-1.55,-3.33,;-1.55,-4.87,;-.22,-5.64,;1.11,-4.87,;2.58,-5.35,;3.35,-6.68,;3.48,-4.1,;5.02,-4.1,;2.58,-2.85,;2.98,-1.37,;1.89,-.28,;2.29,1.21,;3.77,1.61,;4.86,.52,;4.47,-.97,;5.55,-2.06,;4.17,3.1,;4.57,4.58,;1.11,-3.33,;-.22,-2.56,;-.22,-1.02,;-1.55,-.25,;-1.55,1.29,;-2.89,2.06,;-2.89,3.6,;-1.55,4.37,;-1.55,5.91,;-2.89,6.68,;-4.22,5.91,;-4.22,4.37,)|
COc1cc2ncc3[nH]c(=O)n(-c4c(F)cc(cc4F)C#N)c3c2cc1OCc1ccccc1 |(-5.55,-1.54,;-4.22,-.77,;-2.89,-1.54,;-2.89,-3.08,;-1.55,-3.85,;-1.55,-5.39,;-.22,-6.16,;1.11,-5.39,;2.58,-5.87,;3.48,-4.62,;5.02,-4.62,;2.58,-3.37,;2.98,-1.89,;4.47,-1.49,;5.55,-2.58,;4.86,-0,;3.77,1.09,;2.29,.69,;1.89,-.8,;.4,-1.2,;4.17,2.58,;4.57,4.06,;1.11,-3.85,;-.22,-3.08,;-.22,-1.54,;-1.55,-.77,;-1.55,.77,;-2.89,1.54,;-2.89,3.08,;-1.55,3.85,;-1.55,5.39,;-2.89,6.16,;-4.22,5.39,;-4.22,3.85,)|
COc1cc2ncc3n(C)c(=O)n(-c4c(F)cc(cc4F)C#N)c3c2cc1OCc1ccccc1 |(-5.55,-1.02,;-4.22,-.25,;-2.89,-1.02,;-2.89,-2.56,;-1.55,-3.33,;-1.55,-4.87,;-.22,-5.64,;1.11,-4.87,;2.58,-5.35,;3.35,-6.68,;3.48,-4.1,;5.02,-4.1,;2.58,-2.85,;2.98,-1.37,;4.47,-.97,;5.55,-2.06,;4.86,.52,;3.77,1.61,;2.29,1.21,;1.89,-.28,;.4,-.68,;4.17,3.1,;4.57,4.58,;1.11,-3.33,;-.22,-2.56,;-.22,-1.02,;-1.55,-.25,;-1.55,1.29,;-2.89,2.06,;-2.89,3.6,;-1.55,4.37,;-1.55,5.91,;-2.89,6.68,;-4.22,5.91,;-4.22,4.37,)|
COC(=O)n1c2cnc3cc(OC)c(OCc4ccccc4)cc3c2n(-c2ccc(cc2F)C#N)c1=O |(2.29,-8.04,;1.89,-6.56,;2.98,-5.47,;4.47,-5.87,;2.58,-3.98,;1.11,-3.51,;-.22,-4.28,;-1.55,-3.51,;-1.55,-1.97,;-2.89,-1.2,;-2.89,.34,;-4.22,1.11,;-5.55,.34,;-1.55,1.11,;-1.55,2.65,;-2.89,3.42,;-2.89,4.96,;-1.55,5.73,;-1.55,7.27,;-2.89,8.04,;-4.22,7.27,;-4.22,5.73,;-.22,.34,;-.22,-1.2,;1.11,-1.97,;2.58,-1.49,;2.98,-0,;1.89,1.09,;2.29,2.57,;3.77,2.97,;4.86,1.88,;4.47,.4,;5.55,-.69,;4.17,4.46,;4.57,5.95,;3.48,-2.74,;5.02,-2.74,)|
COc1cc2ncc3n(C)c(=O)n(-c4ccc(cc4F)C#N)c3c2cc1OCc1ccsc1 |(-5.55,-.67,;-4.22,.1,;-2.89,-.67,;-2.89,-2.21,;-1.55,-2.98,;-1.55,-4.52,;-.22,-5.29,;1.11,-4.52,;2.58,-4.99,;3.35,-6.32,;3.48,-3.75,;5.02,-3.75,;2.58,-2.5,;2.98,-1.01,;1.89,.08,;2.29,1.56,;3.77,1.96,;4.86,.87,;4.47,-.61,;5.55,-1.7,;4.17,3.45,;4.57,4.94,;1.11,-2.98,;-.22,-2.21,;-.22,-.67,;-1.55,.1,;-1.55,1.64,;-2.89,2.41,;-2.89,3.95,;-4.13,4.86,;-3.66,6.32,;-2.12,6.32,;-1.64,4.86,)|
COc1cc2ncc3n(C)c(=O)n(-c4ccc(cc4F)C#N)c3c2cc1OCc1cccs1 |(-5.55,-.67,;-4.22,.1,;-2.89,-.67,;-2.89,-2.21,;-1.55,-2.98,;-1.55,-4.52,;-.22,-5.29,;1.11,-4.52,;2.58,-4.99,;3.35,-6.32,;3.48,-3.75,;5.02,-3.75,;2.58,-2.5,;2.98,-1.01,;1.89,.08,;2.29,1.56,;3.77,1.96,;4.86,.87,;4.47,-.61,;5.55,-1.7,;4.17,3.45,;4.57,4.94,;1.11,-2.98,;-.22,-2.21,;-.22,-.67,;-1.55,.1,;-1.55,1.64,;-2.89,2.41,;-2.89,3.95,;-4.13,4.86,;-3.66,6.32,;-2.12,6.32,;-1.64,4.86,)|
COc1cc2ncc3n(C)c(=O)n(-c4ccc(cc4F)C#N)c3c2cc1OC(C(N)=O)c1ccc(F)cc1 |(-5.55,-1.66,;-4.22,-.89,;-2.89,-1.66,;-2.89,-3.2,;-1.55,-3.97,;-1.55,-5.51,;-.22,-6.28,;1.11,-5.51,;2.58,-5.99,;3.35,-7.32,;3.48,-4.74,;5.02,-4.74,;2.58,-3.49,;2.98,-2.01,;1.89,-.92,;2.29,.57,;3.77,.97,;4.86,-.12,;4.47,-1.61,;5.55,-2.7,;4.17,2.46,;4.57,3.94,;1.11,-3.97,;-.22,-3.2,;-.22,-1.66,;-1.55,-.89,;-1.55,.65,;-2.32,1.98,;-3.86,1.98,;-4.63,3.32,;-4.63,.65,;-1.55,3.32,;-.01,3.32,;.76,4.65,;-.01,5.99,;.76,7.32,;-1.55,5.99,;-2.32,4.65,)|
COCCNC(=O)C(Oc1cc2c3n(-c4ccc(cc4F)C#N)c(=O)n(C)c3cnc2cc1OC)c1ccc(F)cc1 |(-7.4,5.99,;-6.63,4.65,;-5.09,4.65,;-4.32,3.32,;-2.78,3.32,;-2.01,1.98,;-2.78,.65,;-.47,1.98,;.3,.65,;.3,-.89,;1.63,-1.66,;1.63,-3.2,;2.96,-3.97,;4.43,-3.49,;4.83,-2.01,;3.74,-.92,;4.14,.57,;5.62,.97,;6.71,-.12,;6.31,-1.61,;7.4,-2.7,;6.02,2.46,;6.42,3.94,;5.33,-4.74,;6.87,-4.74,;4.43,-5.99,;5.2,-7.32,;2.96,-5.51,;1.63,-6.28,;.3,-5.51,;.3,-3.97,;-1.04,-3.2,;-1.04,-1.66,;-2.37,-.89,;-3.7,-1.66,;.3,3.32,;1.84,3.32,;2.61,4.65,;1.84,5.99,;2.61,7.32,;.3,5.99,;-.47,4.65,)|
COc1cc2ncc3n(C)c(=O)n(-c4ccc(cc4F)C#N)c3c2cc1OCc1ccc(F)cc1 |(-5.55,-1.79,;-4.22,-1.02,;-2.89,-1.79,;-2.89,-3.33,;-1.55,-4.1,;-1.55,-5.64,;-.22,-6.41,;1.11,-5.64,;2.58,-6.12,;3.35,-7.45,;3.48,-4.87,;5.02,-4.87,;2.58,-3.62,;2.98,-2.14,;1.89,-1.05,;2.29,.44,;3.77,.84,;4.86,-.25,;4.47,-1.74,;5.55,-2.83,;4.17,2.33,;4.57,3.81,;1.11,-4.1,;-.22,-3.33,;-.22,-1.79,;-1.55,-1.02,;-1.55,.52,;-2.89,1.29,;-2.89,2.83,;-1.55,3.6,;-1.55,5.14,;-2.89,5.91,;-2.89,7.45,;-4.22,5.14,;-4.22,3.6,)|
COc1cc2ncc3n(C)c(=O)n(-c4ccc(cc4F)C#N)c3c2cc1OC(C(N)=O)c1ccccc1 |(-5.55,-.99,;-4.22,-.22,;-2.89,-.99,;-2.89,-2.53,;-1.55,-3.3,;-1.55,-4.84,;-.22,-5.61,;1.11,-4.84,;2.58,-5.32,;3.35,-6.65,;3.48,-4.07,;5.02,-4.07,;2.58,-2.83,;2.98,-1.34,;1.89,-.25,;2.29,1.24,;3.77,1.64,;4.86,.55,;4.47,-.94,;5.55,-2.03,;4.17,3.12,;4.57,4.61,;1.11,-3.3,;-.22,-2.53,;-.22,-.99,;-1.55,-.22,;-1.55,1.32,;-2.32,2.65,;-3.86,2.65,;-4.63,3.98,;-4.63,1.32,;-1.55,3.98,;-.01,3.98,;.76,5.32,;-.01,6.65,;-1.55,6.65,;-2.32,5.32,)|
COc1cc2ncc3n(C)c(=O)n(-c4ccc(cc4F)C#N)c3c2cc1OCc1sccc1S(=O)(=O)N1CCOCC1 |(-3.29,-.67,;-1.96,.1,;-.62,-.67,;-.62,-2.21,;.71,-2.98,;.71,-4.52,;2.04,-5.29,;3.38,-4.52,;4.84,-4.99,;5.61,-6.32,;5.75,-3.75,;7.29,-3.75,;4.84,-2.5,;5.24,-1.01,;4.15,.08,;4.55,1.56,;6.04,1.96,;7.13,.87,;6.73,-.61,;7.82,-1.7,;6.44,3.45,;6.84,4.94,;3.38,-2.98,;2.04,-2.21,;2.04,-.67,;.71,.1,;.71,1.64,;-.62,2.41,;-.62,3.95,;.62,4.86,;.15,6.32,;-1.39,6.32,;-1.87,4.86,;-3.36,4.46,;-3.75,5.95,;-2.96,2.97,;-4.84,4.06,;-5.93,5.15,;-7.42,4.75,;-7.82,3.27,;-6.73,2.18,;-5.24,2.58,)|
COc1cc2ncc3n(C)c(=O)n(-c4ccc(cc4F)C#N)c3c2cc1OCc1ccncc1 |(-5.55,-1.02,;-4.22,-.25,;-2.89,-1.02,;-2.89,-2.56,;-1.55,-3.33,;-1.55,-4.87,;-.22,-5.64,;1.11,-4.87,;2.58,-5.35,;3.35,-6.68,;3.48,-4.1,;5.02,-4.1,;2.58,-2.85,;2.98,-1.37,;1.89,-.28,;2.29,1.21,;3.77,1.61,;4.86,.52,;4.47,-.97,;5.55,-2.06,;4.17,3.1,;4.57,4.58,;1.11,-3.33,;-.22,-2.56,;-.22,-1.02,;-1.55,-.25,;-1.55,1.29,;-2.89,2.06,;-2.89,3.6,;-1.55,4.37,;-1.55,5.91,;-2.89,6.68,;-4.22,5.91,;-4.22,4.37,)|
COc1cc2ncc3n(C)c(=O)n(-c4ccc(cc4F)C#N)c3c2cc1OCc1ccccc1Br |(-5.55,-1.02,;-4.22,-.25,;-2.89,-1.02,;-2.89,-2.56,;-1.55,-3.33,;-1.55,-4.87,;-.22,-5.64,;1.11,-4.87,;2.58,-5.35,;3.35,-6.68,;3.48,-4.1,;5.02,-4.1,;2.58,-2.85,;2.98,-1.37,;1.89,-.28,;2.29,1.21,;3.77,1.61,;4.86,.52,;4.47,-.97,;5.55,-2.06,;4.17,3.1,;4.57,4.58,;1.11,-3.33,;-.22,-2.56,;-.22,-1.02,;-1.55,-.25,;-1.55,1.29,;-2.89,2.06,;-2.89,3.6,;-4.22,4.37,;-4.22,5.91,;-2.89,6.68,;-1.55,5.91,;-1.55,4.37,;-.22,3.6,)|
COc1cc2ncc3n(C)c(=O)n(-c4ccc(cc4F)C#N)c3c2cc1OCc1ccc(F)cc1Br |(-5.55,-1.79,;-4.22,-1.02,;-2.89,-1.79,;-2.89,-3.33,;-1.55,-4.1,;-1.55,-5.64,;-.22,-6.41,;1.11,-5.64,;2.58,-6.12,;3.35,-7.45,;3.48,-4.87,;5.02,-4.87,;2.58,-3.62,;2.98,-2.14,;1.89,-1.05,;2.29,.44,;3.77,.84,;4.86,-.25,;4.47,-1.74,;5.55,-2.83,;4.17,2.33,;4.57,3.81,;1.11,-4.1,;-.22,-3.33,;-.22,-1.79,;-1.55,-1.02,;-1.55,.52,;-2.89,1.29,;-2.89,2.83,;-4.22,3.6,;-4.22,5.14,;-2.89,5.91,;-2.89,7.45,;-1.55,5.14,;-1.55,3.6,;-.22,2.83,)|
COc1cc2ncc3n(C)c(=O)n(-c4ccc(cc4F)C#N)c3c2cc1OCc1ccc(F)cc1Cl |(-5.55,-1.79,;-4.22,-1.02,;-2.89,-1.79,;-2.89,-3.33,;-1.55,-4.1,;-1.55,-5.64,;-.22,-6.41,;1.11,-5.64,;2.58,-6.12,;3.35,-7.45,;3.48,-4.87,;5.02,-4.87,;2.58,-3.62,;2.98,-2.14,;1.89,-1.05,;2.29,.44,;3.77,.84,;4.86,-.25,;4.47,-1.74,;5.55,-2.83,;4.17,2.33,;4.57,3.81,;1.11,-4.1,;-.22,-3.33,;-.22,-1.79,;-1.55,-1.02,;-1.55,.52,;-2.89,1.29,;-2.89,2.83,;-4.22,3.6,;-4.22,5.14,;-2.89,5.91,;-2.89,7.45,;-1.55,5.14,;-1.55,3.6,;-.22,2.83,)|
COc1cc2ncc3n(C)c(=O)n(-c4ccc(cc4F)C#N)c3c2cc1OCc1ccc(F)c(Cl)c1 |(-5.55,-1.79,;-4.22,-1.02,;-2.89,-1.79,;-2.89,-3.33,;-1.55,-4.1,;-1.55,-5.64,;-.22,-6.41,;1.11,-5.64,;2.58,-6.12,;3.35,-7.45,;3.48,-4.87,;5.02,-4.87,;2.58,-3.62,;2.98,-2.14,;1.89,-1.05,;2.29,.44,;3.77,.84,;4.86,-.25,;4.47,-1.74,;5.55,-2.83,;4.17,2.33,;4.57,3.81,;1.11,-4.1,;-.22,-3.33,;-.22,-1.79,;-1.55,-1.02,;-1.55,.52,;-2.89,1.29,;-2.89,2.83,;-4.22,3.6,;-4.22,5.14,;-2.89,5.91,;-2.89,7.45,;-1.55,5.14,;-.22,5.91,;-1.55,3.6,)|
COc1cc2ncc3n(C)c(=O)n(-c4c(F)cc(cc4F)C#N)c3c2cc1OC(C(N)=O)c1ccc(F)cc1 |(-5.55,-1.66,;-4.22,-.89,;-2.89,-1.66,;-2.89,-3.2,;-1.55,-3.97,;-1.55,-5.51,;-.22,-6.28,;1.11,-5.51,;2.58,-5.99,;3.35,-7.32,;3.48,-4.74,;5.02,-4.74,;2.58,-3.49,;2.98,-2.01,;4.47,-1.61,;5.55,-2.7,;4.86,-.12,;3.77,.97,;2.29,.57,;1.89,-.92,;.4,-1.32,;4.17,2.46,;4.57,3.94,;1.11,-3.97,;-.22,-3.2,;-.22,-1.66,;-1.55,-.89,;-1.55,.65,;-2.32,1.98,;-3.86,1.98,;-4.63,3.32,;-4.63,.65,;-1.55,3.32,;-.01,3.32,;.76,4.65,;-.01,5.99,;.76,7.32,;-1.55,5.99,;-2.32,4.65,)|
COc1cc2ncc3n(C)c(=O)n(-c4c(F)cc(cc4F)C#N)c3c2cc1OCc1ccsc1 |(-5.55,-.67,;-4.22,.1,;-2.89,-.67,;-2.89,-2.21,;-1.55,-2.98,;-1.55,-4.52,;-.22,-5.29,;1.11,-4.52,;2.58,-4.99,;3.35,-6.32,;3.48,-3.75,;5.02,-3.75,;2.58,-2.5,;2.98,-1.01,;4.47,-.61,;5.55,-1.7,;4.86,.87,;3.77,1.96,;2.29,1.56,;1.89,.08,;.4,-.32,;4.17,3.45,;4.57,4.94,;1.11,-2.98,;-.22,-2.21,;-.22,-.67,;-1.55,.1,;-1.55,1.64,;-2.89,2.41,;-2.89,3.95,;-4.13,4.86,;-3.66,6.32,;-2.12,6.32,;-1.64,4.86,)|
COc1cc2ncc3n(C)c(=O)n(-c4c(F)cc(cc4F)C#N)c3c2cc1OCc1ccc(F)cc1 |(-5.55,-1.79,;-4.22,-1.02,;-2.89,-1.79,;-2.89,-3.33,;-1.55,-4.1,;-1.55,-5.64,;-.22,-6.41,;1.11,-5.64,;2.58,-6.12,;3.35,-7.45,;3.48,-4.87,;5.02,-4.87,;2.58,-3.62,;2.98,-2.14,;4.47,-1.74,;5.55,-2.83,;4.86,-.25,;3.77,.84,;2.29,.44,;1.89,-1.05,;.4,-1.45,;4.17,2.33,;4.57,3.81,;1.11,-4.1,;-.22,-3.33,;-.22,-1.79,;-1.55,-1.02,;-1.55,.52,;-2.89,1.29,;-2.89,2.83,;-1.55,3.6,;-1.55,5.14,;-2.89,5.91,;-2.89,7.45,;-4.22,5.14,;-4.22,3.6,)|
COc1cc2ncc3n(C)c(=O)n(-c4c(F)cc(cc4F)C#N)c3c2cc1OCc1cccs1 |(-5.55,-.67,;-4.22,.1,;-2.89,-.67,;-2.89,-2.21,;-1.55,-2.98,;-1.55,-4.52,;-.22,-5.29,;1.11,-4.52,;2.58,-4.99,;3.35,-6.32,;3.48,-3.75,;5.02,-3.75,;2.58,-2.5,;2.98,-1.01,;4.47,-.61,;5.55,-1.7,;4.86,.87,;3.77,1.96,;2.29,1.56,;1.89,.08,;.4,-.32,;4.17,3.45,;4.57,4.94,;1.11,-2.98,;-.22,-2.21,;-.22,-.67,;-1.55,.1,;-1.55,1.64,;-2.89,2.41,;-2.89,3.95,;-4.13,4.86,;-3.66,6.32,;-2.12,6.32,;-1.64,4.86,)|
COc1cc2ncc3n(C)c(=O)n(-c4ccc(cc4)C#N)c3c2cc1OCc1cccs1
COc1cc2ncc3n(C)c(=O)n(-c4ccc(cc4F)C#N)c3c2cc1OCc1cncs1 |(-5.55,-.67,;-4.22,.1,;-2.89,-.67,;-2.89,-2.21,;-1.55,-2.98,;-1.55,-4.52,;-.22,-5.29,;1.11,-4.52,;2.58,-4.99,;3.35,-6.32,;3.48,-3.75,;5.02,-3.75,;2.58,-2.5,;2.98,-1.01,;1.89,.08,;2.29,1.56,;3.77,1.96,;4.86,.87,;4.47,-.61,;5.55,-1.7,;4.17,3.45,;4.57,4.94,;1.11,-2.98,;-.22,-2.21,;-.22,-.67,;-1.55,.1,;-1.55,1.64,;-2.89,2.41,;-2.89,3.95,;-4.13,4.86,;-3.66,6.32,;-2.12,6.32,;-1.64,4.86,)|
COc1cc2ncc3n(C)c(=O)n(-c4ccc(cc4F)C#N)c3c2cc1OC(CN)c1cccs1 |(-5.55,-.49,;-4.22,.28,;-2.89,-.49,;-2.89,-2.03,;-1.55,-2.8,;-1.55,-4.34,;-.22,-5.11,;1.11,-4.34,;2.58,-4.81,;3.35,-6.15,;3.48,-3.57,;5.02,-3.57,;2.58,-2.32,;2.98,-.83,;1.89,.25,;2.29,1.74,;3.77,2.14,;4.86,1.05,;4.47,-.44,;5.55,-1.53,;4.17,3.63,;4.57,5.12,;1.11,-2.8,;-.22,-2.03,;-.22,-.49,;-1.55,.28,;-1.55,1.82,;-1.55,3.36,;-2.89,4.13,;-4.22,3.36,;-.22,4.13,;-.22,5.67,;1.25,6.15,;2.15,4.9,;1.25,3.66,)|
COc1cc2ncc3n(C)c(=O)n(-c4ccc(cc4F)C#N)c3c2cc1OC(CN)c1ccc(F)cc1 |(-5.55,-.64,;-4.22,.13,;-2.89,-.64,;-2.89,-2.18,;-1.55,-2.95,;-1.55,-4.49,;-.22,-5.26,;1.11,-4.49,;2.58,-4.96,;3.35,-6.29,;3.48,-3.72,;5.02,-3.72,;2.58,-2.47,;2.98,-.98,;1.89,.11,;2.29,1.59,;3.77,1.99,;4.86,.9,;4.47,-.58,;5.55,-1.67,;4.17,3.48,;4.57,4.97,;1.11,-2.95,;-.22,-2.18,;-.22,-.64,;-1.55,.13,;-1.55,1.67,;-1.55,3.21,;-2.89,3.98,;-4.22,3.21,;-.22,3.98,;1.11,3.21,;2.45,3.98,;2.45,5.52,;3.78,6.29,;1.11,6.29,;-.22,5.52,)|
COc1cc2ncc3n(C)c(=O)n(-c4ccc(cc4F)C#N)c3c2cc1-c1cccnc1 |(-5.55,.03,;-4.22,.8,;-2.89,.03,;-2.89,-1.51,;-1.55,-2.28,;-1.55,-3.82,;-.22,-4.59,;1.11,-3.82,;2.58,-4.3,;3.35,-5.63,;3.48,-3.05,;5.02,-3.05,;2.58,-1.81,;2.98,-.32,;1.89,.77,;2.29,2.26,;3.77,2.66,;4.86,1.57,;4.47,.08,;5.55,-1.01,;4.17,4.14,;4.57,5.63,;1.11,-2.28,;-.22,-1.51,;-.22,.03,;-1.55,.8,;-1.55,2.34,;-2.89,3.11,;-2.89,4.65,;-1.55,5.42,;-.22,4.65,;-.22,3.11,)|
COc1ccc(cn1)-c1cc2c3n(-c4ccc(cc4F)C#N)c(=O)n(C)c3cnc2cc1OC |(-.22,6.68,;-1.55,5.91,;-1.55,4.37,;-2.89,3.6,;-2.89,2.06,;-1.55,1.29,;-.22,2.06,;-.22,3.6,;-1.55,-.25,;-.22,-1.02,;-.22,-2.56,;1.11,-3.33,;2.58,-2.85,;2.98,-1.37,;1.89,-.28,;2.29,1.21,;3.77,1.61,;4.86,.52,;4.47,-.97,;5.55,-2.06,;4.17,3.1,;4.57,4.58,;3.48,-4.1,;5.02,-4.1,;2.58,-5.35,;3.35,-6.68,;1.11,-4.87,;-.22,-5.64,;-1.55,-4.87,;-1.55,-3.33,;-2.89,-2.56,;-2.89,-1.02,;-4.22,-.25,;-5.55,-1.02,)|
COc1cc2ncc3n(C)c(=O)n(-c4ccc(cc4F)C#N)c3c2cc1-c1cnc2ccccc2c1 |(-5.55,-1.02,;-4.22,-.25,;-2.89,-1.02,;-2.89,-2.56,;-1.55,-3.33,;-1.55,-4.87,;-.22,-5.64,;1.11,-4.87,;2.58,-5.35,;3.35,-6.68,;3.48,-4.1,;5.02,-4.1,;2.58,-2.85,;2.98,-1.37,;1.89,-.28,;2.29,1.21,;3.77,1.61,;4.86,.52,;4.47,-.97,;5.55,-2.06,;4.17,3.1,;4.57,4.58,;1.11,-3.33,;-.22,-2.56,;-.22,-1.02,;-1.55,-.25,;-1.55,1.29,;-.22,2.06,;-.22,3.6,;-1.55,4.37,;-1.55,5.91,;-2.89,6.68,;-4.22,5.91,;-4.22,4.37,;-2.89,3.6,;-2.89,2.06,)|
COc1cc2ncc3n(C)c(=O)n(-c4ccc(cc4F)C#N)c3c2cc1-c1cnn(C)c1 |(-5.55,-.18,;-4.22,.59,;-2.89,-.18,;-2.89,-1.72,;-1.55,-2.49,;-1.55,-4.03,;-.22,-4.8,;1.11,-4.03,;2.58,-4.5,;3.35,-5.84,;3.48,-3.26,;5.02,-3.26,;2.58,-2.01,;2.98,-.52,;1.89,.57,;2.29,2.05,;3.77,2.45,;4.86,1.36,;4.47,-.12,;5.55,-1.21,;4.17,3.94,;4.57,5.43,;1.11,-2.49,;-.22,-1.72,;-.22,-.18,;-1.55,.59,;-1.55,2.13,;-.31,3.04,;-.78,4.5,;-2.32,4.5,;-3.09,5.84,;-2.8,3.04,)|
COc1cc2ncc3n(C)c(=O)n(-c4ccc(cc4F)C#N)c3c2cc1-c1cn[nH]c1 |(-5.55,.03,;-4.22,.8,;-2.89,.03,;-2.89,-1.51,;-1.55,-2.28,;-1.55,-3.82,;-.22,-4.59,;1.11,-3.82,;2.58,-4.3,;3.35,-5.63,;3.48,-3.05,;5.02,-3.05,;2.58,-1.81,;2.98,-.32,;1.89,.77,;2.29,2.26,;3.77,2.66,;4.86,1.57,;4.47,.08,;5.55,-1.01,;4.17,4.14,;4.57,5.63,;1.11,-2.28,;-.22,-1.51,;-.22,.03,;-1.55,.8,;-1.55,2.34,;-.31,3.24,;-.78,4.71,;-2.32,4.71,;-2.8,3.24,)|
COc1cc2ncc3n(C)c(=O)n(-c4ccc(cc4F)C#N)c3c2cc1-c1ccnn1C |(-5.55,.03,;-4.22,.8,;-2.89,.03,;-2.89,-1.51,;-1.55,-2.28,;-1.55,-3.82,;-.22,-4.59,;1.11,-3.82,;2.58,-4.3,;3.35,-5.63,;3.48,-3.05,;5.02,-3.05,;2.58,-1.81,;2.98,-.32,;1.89,.77,;2.29,2.26,;3.77,2.66,;4.86,1.57,;4.47,.08,;5.55,-1.01,;4.17,4.14,;4.57,5.63,;1.11,-2.28,;-.22,-1.51,;-.22,.03,;-1.55,.8,;-1.55,2.34,;-.31,3.24,;-.78,4.71,;-2.32,4.71,;-2.8,3.24,;-4.13,2.47,)|
COc1cc2ncc3n(C)c(=O)n(-c4ccc(cc4F)C#N)c3c2cc1-c1ccn[nH]1 |(-5.55,.03,;-4.22,.8,;-2.89,.03,;-2.89,-1.51,;-1.55,-2.28,;-1.55,-3.82,;-.22,-4.59,;1.11,-3.82,;2.58,-4.3,;3.35,-5.63,;3.48,-3.05,;5.02,-3.05,;2.58,-1.81,;2.98,-.32,;1.89,.77,;2.29,2.26,;3.77,2.66,;4.86,1.57,;4.47,.08,;5.55,-1.01,;4.17,4.14,;4.57,5.63,;1.11,-2.28,;-.22,-1.51,;-.22,.03,;-1.55,.8,;-1.55,2.34,;-.31,3.24,;-.78,4.71,;-2.32,4.71,;-2.8,3.24,)|
COc1cc2ncc3n(C)c(=O)n(-c4ccc(cc4F)C#N)c3c2cc1-c1cc(nn1C)C(F)(F)F |(-5.55,-.84,;-4.22,-.07,;-2.89,-.84,;-2.89,-2.38,;-1.55,-3.15,;-1.55,-4.69,;-.22,-5.46,;1.11,-4.69,;2.58,-5.17,;3.35,-6.5,;3.48,-3.92,;5.02,-3.92,;2.58,-2.68,;2.98,-1.19,;1.89,-.1,;2.29,1.39,;3.77,1.78,;4.86,.7,;4.47,-.79,;5.55,-1.88,;4.17,3.27,;4.57,4.76,;1.11,-3.15,;-.22,-2.38,;-.22,-.84,;-1.55,-.07,;-1.55,1.47,;-.31,2.37,;-.78,3.84,;-2.32,3.84,;-2.8,2.37,;-4.13,1.6,;-.01,5.17,;-.78,6.5,;1.32,5.94,;1.32,4.4,)|
COc1cc2ncc3n(C)c(=O)n(-c4ccc(cc4F)C#N)c3c2cc1\C=C\c1ccsc1 |(-5.55,-.67,;-4.22,.1,;-2.89,-.67,;-2.89,-2.21,;-1.55,-2.98,;-1.55,-4.52,;-.22,-5.29,;1.11,-4.52,;2.58,-4.99,;3.35,-6.32,;3.48,-3.75,;5.02,-3.75,;2.58,-2.5,;2.98,-1.01,;1.89,.08,;2.29,1.56,;3.77,1.96,;4.86,.87,;4.47,-.61,;5.55,-1.7,;4.17,3.45,;4.57,4.94,;1.11,-2.98,;-.22,-2.21,;-.22,-.67,;-1.55,.1,;-1.55,1.64,;-2.89,2.41,;-2.89,3.95,;-1.64,4.86,;-2.12,6.32,;-3.66,6.32,;-4.13,4.86,)|
COc1cc2ncc3n(C)c(=O)n(-c4ccc(cc4F)C#N)c3c2cc1CCc1ccsc1 |(-5.55,-.67,;-4.22,.1,;-2.89,-.67,;-2.89,-2.21,;-1.55,-2.98,;-1.55,-4.52,;-.22,-5.29,;1.11,-4.52,;2.58,-4.99,;3.35,-6.32,;3.48,-3.75,;5.02,-3.75,;2.58,-2.5,;2.98,-1.01,;1.89,.08,;2.29,1.56,;3.77,1.96,;4.86,.87,;4.47,-.61,;5.55,-1.7,;4.17,3.45,;4.57,4.94,;1.11,-2.98,;-.22,-2.21,;-.22,-.67,;-1.55,.1,;-1.55,1.64,;-2.89,2.41,;-2.89,3.95,;-1.64,4.86,;-2.12,6.32,;-3.66,6.32,;-4.13,4.86,)|
COc1cc2ncc3n(C)c(=O)n(-c4ccc(cc4F)C#N)c3c2cc1\C=C\c1ccccc1 |(-5.55,-1.02,;-4.22,-.25,;-2.89,-1.02,;-2.89,-2.56,;-1.55,-3.33,;-1.55,-4.87,;-.22,-5.64,;1.11,-4.87,;2.58,-5.35,;3.35,-6.68,;3.48,-4.1,;5.02,-4.1,;2.58,-2.85,;2.98,-1.37,;1.89,-.28,;2.29,1.21,;3.77,1.61,;4.86,.52,;4.47,-.97,;5.55,-2.06,;4.17,3.1,;4.57,4.58,;1.11,-3.33,;-.22,-2.56,;-.22,-1.02,;-1.55,-.25,;-1.55,1.29,;-2.89,2.06,;-2.89,3.6,;-1.55,4.37,;-1.55,5.91,;-2.89,6.68,;-4.22,5.91,;-4.22,4.37,)|
C1CCN(CC1)c1ncnc2cc(ccc12)N1CCOCC1
Clc1nc(N2CCCCC2)c2ccc(cc2n1)N1CCOCC1
COc1ccc(cc1)C1CCCN(C1)c1ncnc2cc(ccc12)N1CCOCC1
C1CC(CN(C1)c1ncnc2cc(ccc12)N1CCOCC1)c1ccccc1
C1C[C@H](CN(C1)c1ncnc2cc(ccc12)N1CCOCC1)c1ccccc1 |r|
C1C[C@@H](CN(C1)c1ncnc2cc(ccc12)N1CCOCC1)c1ccccc1 |r|
C1CCN(C1)c1ncnc2cc(ccc12)N1CCOCC1
C1CN(CCO1)c1ccc2c(ncnc2c1)N1CCCCCC1
Fc1ccc2[nH]cc(C3CCCN(C3)c3ncnc4cc(ccc34)N3CCOCC3)c2c1
C(C1CCCCC1)C1CCCN(C1)c1ncnc2cc(ccc12)N1CCOCC1
C([C@@H]1CCCN(C1)c1ncnc2cc(ccc12)N1CCOCC1)c1ccccc1 |r|
CC1CCCN(C1)c1ncnc2cc(ccc12)N1CCOCC1
C(C1CCCN(C1)c1ncnc2cc(ccc12)N1CCOCC1)n1cccc1
C1CC(CN(C1)c1ncnc2cc(ccc12)N1CCOCC1)c1nc2ccccc2s1
OC1(CCCN(C1)c1ncnc2cc(ccc12)N1CCOCC1)c1ccccc1
Fc1ccc(cc1)C(=O)C1CCCN(C1)c1ncnc2cc(ccc12)N1CCOCC1
NC(=O)C1CCCN(C1)c1ncnc2cc(ccc12)N1CCOCC1
CCOCC1CCCN(C1)c1ncnc2cc(ccc12)N1CCOCC1
Cc1noc(n1)C1CCCN(C1)c1ncnc2cc(ccc12)N1CCOCC1
O=C(C1CCCN(C1)c1ncnc2cc(ccc12)N1CCOCC1)N1CCCCC1
C(C1CCCN(C1)c1ncnc2cc(ccc12)N1CCOCC1)N1CCOCC1
COc1cccc(c1)C1CCCN(C1)c1ncnc2cc(ccc12)N1CCOCC1
C(C1CCCN(C1)c1ncnc2cc(ccc12)N1CCOCC1)n1ccnc1
C1CC(CN(C1)c1ncnc2cc(ccc12)N1CCOCC1)c1nc2ccccc2[nH]1
Clc1nc(N2CCCC(Cn3ccnc3)C2)c2ccc(cc2n1)N1CCOCC1
C1CC(CN(C1)c1ncnc2cc(ccc12)N1CCOCC1)c1nc2ccccc2o1
Cc1cccc(c1)C1CCCN(C1)c1ncnc2cc(ccc12)N1CCOCC1
FC(F)(F)c1cccc(c1)C1CCCN(C1)c1ncnc2cc(ccc12)N1CCOCC1
Cn1ccnc1CC1CCCN(C1)c1ncnc2cc(ccc12)N1CCOCC1
Clc1nc(N2CCCC(Cn3cccc3)C2)c2ccc(cc2n1)N1CCOCC1
C(C1CCCN(C1)c1ncnc2cc(ccc12)N1CCOCC1)c1ncccn1
C(C1CCCN(C1)c1ncnc2cc(ccc12)N1CCOCC1)c1nccs1
C(C1CCCN(C1)c1ncnc2cc(ccc12)N1CCOCC1)c1cccs1
Cc1nc(N2CCCCC2)c2ccc(cc2n1)N1CCOCC1
C(C1CCCN(C1)c1ncnc2cc(ccc12)N1CCOCC1)c1cc2ccccc2s1
Clc1nc(N2CCCC(Cc3nccs3)C2)c2ccc(cc2n1)N1CCOCC1
C1CN(CCO1)c1ccc2c(ncnc2c1)N1CCC=C(C1)c1cccs1 |c:22|
COc1cccc(c1)C(O)C1CCCN(C1)c1ncnc2cc(ccc12)N1CCOCC1
COc1nc(N2CCCCC2)c2ccc(cc2n1)N1CCOCC1
C1CC(CN(C1)c1ncnc2cc(ccc12)N1CCOCC1)c1cccs1
COc1cccc(CC2CCCN(C2)c2ncnc3cc(ccc23)N2CCOCC2)c1
COc1ccc(CC2CCCN(C2)c2ncnc3cc(ccc23)N2CCOCC2)cc1OC
C(C1CCCN(C1)c1ncnc2cc(ccc12)N1CCOCC1)c1nc2ccccc2s1
C(C1CCCN(C1)c1ncnc2cc(ccc12)N1CCOCC1)c1ccsc1
OC(C1CCCN(C1)c1ncnc2cc(ccc12)N1CCOCC1)c1ccsc1
OC(C1CCCN(C1)c1ncnc2cc(ccc12)N1CCOCC1)c1nccs1
Cc1cnc(s1)C(O)C1CCCN(C1)c1ncnc2cc(ccc12)N1CCOCC1
Cc1nc(sc1C)C(O)C1CCCN(C1)c1ncnc2cc(ccc12)N1CCOCC1
Cc1csc(n1)C(O)C1CCCN(C1)c1ncnc2cc(ccc12)N1CCOCC1
O=C(C1CCCN(C1)c1ncnc2cc(ccc12)N1CCOCC1)c1nccs1
Cc1cnc(CC2CCCN(C2)c2ncnc3cc(ccc23)N2CCOCC2)s1
Cc1nc(CC2CCCN(C2)c2ncnc3cc(ccc23)N2CCOCC2)sc1C
OC(C1CCCN(C1)c1ncnc2cc(ccc12)N1CCOCC1)c1ncco1
Oc1nc(N2CCCCC2)c2ccc(cc2n1)N1CCOCC1
Cn1ccnc1C(O)C1CCCN(C1)c1ncnc2cc(ccc12)N1CCOCC1
Cc1csc(CC2CCCN(C2)c2ncnc3cc(ccc23)N2CCOCC2)n1
Nc1nc(N2CCCCC2)c2ccc(cc2n1)N1CCOCC1
N#Cc1nc(N2CCCCC2)c2ccc(cc2n1)N1CCOCC1
Clc1nc(N2CCCC(C2)NC(=O)c2cncs2)c2ccc(cc2n1)N1CCOCC1
Clc1nc(N2CCCC(C2)NC(=O)c2nccs2)c2ccc(cc2n1)N1CCOCC1
Clc1nc(N2CCCC(C2)NC(=O)c2cscn2)c2ccc(cc2n1)N1CCOCC1
CN(C1CCCN(C1)c1nc(Cl)nc2cc(ccc12)N1CCOCC1)C(=O)c1nccs1
CN(C1CCCN(C1)c1nc(Cl)nc2cc(ccc12)N1CCOCC1)C(=O)c1cncs1
Clc1nc(N2CCCC(C2)NC(=O)c2cccs2)c2ccc(cc2n1)N1CCOCC1
O[C@H](C1CCCN(C1)c1ncnc2cc(ccc12)N1CCOCC1)c1nccs1 |r|
O[C@@H](C1CCCN(C1)c1ncnc2cc(ccc12)N1CCOCC1)c1nccs1 |r|
Clc1nc(N2CCCC(C2)NS(=O)(=O)c2cccs2)c2ccc(cc2n1)N1CCOCC1
O[C@H](C1CCCN(C1)c1nnnc2cc(ccc12)N1CCOCC1)c1nccs1 |r|
O[C@@H](C1CCCN(C1)c1nnnc2cc(ccc12)N1CCOCC1)c1nccs1 |r|
Cc1csc(n1)[C@@H](O)C1CCCN(C1)c1nnnc2cc(ccc12)N1CCOCC1 |r|
Cc1csc(n1)[C@H](O)C1CCCN(C1)c1nnnc2cc(ccc12)N1CCOCC1 |r|
C[C@@](O)(C1CCCN(C1)c1nnnc2cc(ccc12)N1CCOCC1)c1nccs1 |r|
C[C@](O)(C1CCCN(C1)c1nnnc2cc(ccc12)N1CCOCC1)c1nccs1 |r|
Cc1nc(sc1C)[C@H](O)C1CCCN(C1)c1nnnc2cc(ccc12)N1CCOCC1 |r|
Cc1nc(sc1C)[C@@H](O)C1CCCN(C1)c1nnnc2cc(ccc12)N1CCOCC1 |r|
Cc1cnc(s1)[C@@H](O)C1CCCN(C1)c1nnnc2cc(ccc12)N1CCOCC1 |r|
Cc1cnc(s1)[C@H](O)C1CCCN(C1)c1nnnc2cc(ccc12)N1CCOCC1 |r|
COc1ccc(nn1)[C@@H](O)C1CCCN(C1)c1nnnc2cc(ccc12)N1CCOCC1 |r|
COc1ccc(nn1)[C@H](O)C1CCCN(C1)c1nnnc2cc(ccc12)N1CCOCC1 |r|
COc1ccc(cn1)[C@@H](O)C1CCCN(C1)c1nnnc2cc(ccc12)N1CCOCC1 |r|
COc1ccc(cn1)[C@H](O)C1CCCN(C1)c1nnnc2cc(ccc12)N1CCOCC1 |r|
CC(C)n1cc(cn1)[C@@H](O)C1CCCN(C1)c1nnnc2cc(ccc12)N1CCOCC1 |r|
CC(C)(C)n1cc(cn1)[C@@H](O)C1CCCN(C1)c1nnnc2cc(ccc12)N1CCOCC1 |r|
CCn1cc(cn1)[C@@H](O)C1CCCN(C1)c1nnnc2cc(ccc12)N1CCOCC1 |r|
C[C@H](Nc1ncnc2[nH]cnc12)c1nc2ccc(F)cc2c(=O)n1-c1ccccc1 |r|
Cc1c(OCC(=O)Nc2ccc(cc2)S(N)(=O)=O)ccc2c1oc(nc2=O)N1CCOCC1
CC(=O)NS(=O)(=O)c1ccc(NC(=O)COc2ccc3c(oc(nc3=O)N3CCOCC3)c2C)cc1
Cc1c(OCC(=O)Nc2ccc(cc2)S(=O)(=O)Nc2ccccn2)ccc2c1oc(nc2=O)N1CCOCC1
Cc1c(OCC(=O)Nc2ccc(cc2)S(=O)(=O)Nc2nccs2)ccc2c1oc(nc2=O)N1CCOCC1
Cc1c(OCC(=O)Nc2ccc(cc2)S(=O)(=O)NC(N)=N)ccc2c1oc(nc2=O)N1CCOCC1
Cc1noc(NS(=O)(=O)c2ccc(NC(=O)COc3ccc4c(oc(nc4=O)N4CCOCC4)c3C)cc2)c1C
Cc1c(OCC(=O)NCc2ccccc2)ccc2c1oc(nc2=O)N1CCOCC1
COc1ccc(CNC(=O)COc2ccc3c(oc(nc3=O)N3CCOCC3)c2C)cc1
Cc1ccc(CNC(=O)COc2ccc3c(oc(nc3=O)N3CCOCC3)c2C)cc1
Cc1c(OCC(=O)NCc2ccc(Cl)cc2)ccc2c1oc(nc2=O)N1CCOCC1
Cc1c(OCC(=O)NCc2ccc(F)cc2)ccc2c1oc(nc2=O)N1CCOCC1
Cc1c(OCC(=O)NCc2ccc(O)cc2)ccc2c1oc(nc2=O)N1CCOCC1
C[C@H](NC(=O)COc1ccc2c(oc(nc2=O)N2CCOCC2)c1C)C(O)=O |r|
CCC(C)C(NC(=O)COc1ccc2c(oc(nc2=O)N2CCOCC2)c1C)C(O)=O
Cc1c(OCC(=O)N[C@@H](Cc2ccccc2)C(O)=O)ccc2c1oc(nc2=O)N1CCOCC1 |r|
CC(C)(c1nc(nc2N3CCOCC3COc12)-c1cccc2[nH]ccc12)S(C)(=O)=O
CS(=O)(=O)C1(CCOCC1)c1nc(nc2N3CCOCC3COc12)-c1cccc2[nH]ccc12
CS(=O)(=O)C1(CCOCC1)c1nc(nc2N3CCOC[C@H]3COc12)-c1cccc2[nH]ccc12 |r|
CC(C)(c1nc(nc2N3CCOCC3COc12)-c1cccc2[nH]ccc12)S(=O)(=O)C1CC1
FC(F)(F)S(=O)(=O)Cc1nc(nc2N3CCOCC3COc12)-c1cccc2[nH]ccc12
CS(=O)(=O)C1(CC1)c1nc(nc2N3CCOC[C@H]3COc12)-c1cccc2[nH]ccc12 |r|
CS(=O)(=O)Cc1nc(nc2N3CCOCC3COc12)-c1cccc2[nH]ccc12
CNc1nc2ccccc2n1-c1nc2N3CCOCC3COc2c(n1)C(C)(C)S(C)(=O)=O
CS(=O)(=O)C1(CCOCC1)c1nc(nc2N3CCOCC3COc12)-c1cncc2[nH]ccc12
CS(=O)(=O)C1(CCOCC1)c1nc(nc2N3CCOC[C@@H]3COc12)-c1cccc2[nH]ccc12 |r|
CNc1nc2ccccc2n1-c1nc2N3CCOC[C@H]3COc2c(n1)C(C)(C)S(C)(=O)=O |r|
CNc1nc2ccccc2n1-c1nc2N3CCOCC3COc2c(n1)C1(CCOCC1)S(C)(=O)=O
CS(=O)(=O)C1(CCOCC1)c1nc(nc2N3CCOCC3COc12)-c1c(F)ccc2[nH]ccc12
CC(C)(c1nc(nc2N3CCOCC3COc12)-c1c(F)ccc2[nH]ccc12)S(C)(=O)=O
CC(C)(c1nc(nc2N3CCOC[C@@H]3COc12)-c1cccc2[nH]ccc12)S(C)(=O)=O |r|
CC(C)(c1nc(nc2N3CCOCC3COc12)-c1ccnc2[nH]ccc12)S(C)(=O)=O
CS(=O)(=O)C1(CCOCC1)c1nc(nc2N3CCOCC3COc12)-c1cc(F)cc2[nH]ccc12
CS(=O)(=O)C1(CCOCC1)c1nc(nc2N3CCOCC3COc12)-c1ccnc2[nH]ccc12
COc1cc(-c2nc3N4CCOCC4COc3c(n2)C2(CCOCC2)S(C)(=O)=O)c2cc[nH]c2c1
Cc1cc2c(cccc2[nH]1)-c1nc2N3CCOCC3COc2c(n1)C1(CCOCC1)S(C)(=O)=O
CC(C)(c1nc(nc2N3CCOC[C@@H]3COc12)-c1cccc2[nH]ncc12)S(C)(=O)=O |r|
CS(=O)(=O)C1(CCOCC1)c1nc(nc2N3CCOC[C@H]3CCOc12)-c1cccc2[nH]ccc12 |r|
CS(=O)(=O)C1(CCOCC1)c1nc(nc2N3CCOC[C@@H]3CCOc12)-c1cccc2[nH]ccc12 |r|
CC(C)(c1nc(nc2N3CCOC[C@@H]3CCOc12)-c1cccc2[nH]ccc12)S(C)(=O)=O |r|
CC(C)(c1nc(nc2N3CCOC[C@H]3CCOc12)-c1cccc2[nH]ccc12)S(C)(=O)=O |r|
CC(C)(c1nc(nc2N3CCOC[C@@H]3COc12)-c1c(F)ccc2[nH]ccc12)S(C)(=O)=O |r|
CS(=O)(=O)C1(CC1)c1nc(nc2N3CCOCC3COc12)-c1cccc2[nH]ccc12
CS(=O)(=O)C1(CCOCC1)c1nc(nc2N3CCOC[C@H]3COc12)-c1cc(F)cc2[nH]ccc12 |r|
COc1cc(-c2nc3N4CCOC[C@H]4COc3c(n2)C2(CCOCC2)S(C)(=O)=O)c2cc[nH]c2c1 |r|
CS(=O)(=O)C1(CCOCC1)c1nc(nc2N3CCOC[C@H]3COc12)-c1ccnc2[nH]ccc12 |r|
CNc1nc2ccccc2n1-c1nc2N3CCOCC3CCOc2c(n1)C(C)(C)S(C)(=O)=O |@:14,@@:26|
CNc1nc2ccccc2n1-c1nc2N3CCOCC3CCOc2c(n1)C1(CCOCC1)S(C)(=O)=O |@:14|
CS(=O)(=O)C1(CCOCC1)c1nc(nc2N3CCOCC3CCOc12)-c1cc(F)cc2[nH]ccc12 |@:15|
COc1cc(-c2nc3N4CCOCC4CCOc3c(n2)C2(CCOCC2)S(C)(=O)=O)c2cc[nH]c2c1 |@:8|
CS(=O)(=O)Nc1nc(nc2N3CCOCC3COc12)-c1cccc2[nH]ccc12
CN1CCC(CC1)(c1nc(nc2N3CCOCC3COc12)-c1cccc2[nH]ccc12)S(C)(=O)=O
COc1ccc(-c2nc3N4CCOCC4COc3c(n2)C2(CCOCC2)S(C)(=O)=O)c2cc[nH]c12
CC(C)(O)c1nc(nc2N3CCOCC3COc12)-c1cccc2[nH]ccc12
CNc1nc2ccccc2n1-c1nc2N3CCOCC3COc2c(n1)C(C)(C)O
CC(C)(C#N)c1nc(nc2N3CCOCC3COc12)-c1cccc2[nH]ccc12
CC1(CCCS1(=O)=O)c1nc(nc2N3CCOCC3COc12)-c1cccc2[nH]ccc12
C1CN2C(CO1)COc1c2nc(nc1-c1cccc2[nH]ccc12)-c1cccc2[nH]ccc12
CS(=O)(=O)c1cccc(c1)-c1nc(nc2N3CCOCC3COc12)-c1cccc2[nH]ccc12
CC(C)(O)c1nc(nc2N3CCOC[C@H]3COc12)-c1cccc2[nH]ccc12 |r|
CC(C)(O)c1nc(nc2N3CCOC[C@H]3COc12)-c1cc(F)cc2[nH]ccc12 |r|
COc1cc(-c2nc3N4CCOC[C@H]4COc3c(n2)C(C)(C)O)c2cc[nH]c2c1 |r|
CC(C)(c1nc(nc2N3CCOC[C@H]3COc12)-c1cccc2[nH]ccc12)S(=O)(=O)C1CC1 |r|
CNc1nc2ccccc2n1-c1nc2N3CCOC[C@H]3CCOc2c(n1)C(C)(C)S(C)(=O)=O |r|
CC(C)Nc1nc2ccccc2n1-c1nc2N3CCOC[C@H]3COc2c(n1)C(C)(C)S(C)(=O)=O |r|
CCNc1nc2ccccc2n1-c1nc2N3CCOC[C@H]3COc2c(n1)C(C)(C)S(C)(=O)=O |r|
CCCNc1nc2ccccc2n1-c1nc2N3CCOC[C@H]3COc2c(n1)C(C)(C)S(C)(=O)=O |r|
CNc1nc2ccccc2n1-c1nc2N3CCOC[C@H]3COc2c(n1)C1(CC1)S(C)(=O)=O |r|
CS(=O)(=O)C1(CCC1)c1nc(nc2N3CCOC[C@H]3COc12)-c1cccc2[nH]ccc12 |r|
CCOC(=O)N1CCC(CC1)(c1nc(nc2N3CCOC[C@H]3COc12)-c1cccc2[nH]ccc12)S(C)(=O)=O |r|
CS(=O)(=O)C1(CCNCC1)c1nc(nc2N3CCOC[C@H]3COc12)-c1cccc2[nH]ccc12 |r|
CC(C)(c3nc(n2c(N)nc1ccccc12)nc4c3OC[C@@H]5COCCN45)S(C)(=O)=O
CC(C)(c1nc(nc2N3CCOC[C@H]3COc12)-c1cc(F)cc2[nH]ccc12)S(C)(=O)=O |r|
COc1cc(-c2nc3N4CCOC[C@H]4COc3c(n2)C(C)(C)S(C)(=O)=O)c2cc[nH]c2c1 |r|
CC(C)(c4nc(n3c(N1CCOCC1)nc2ccccc23)nc5c4OC[C@@H]6COCCN56)S(C)(=O)=O
CS(=O)(=O)C1(CC1)c1nc(nc2N3CCOC[C@H]3COc12)-c1cc(F)cc2[nH]ccc12 |r|
COc1cc(-c2nc3N4CCOC[C@H]4COc3c(n2)C2(CC2)S(C)(=O)=O)c2cc[nH]c2c1 |r|
CS(=O)(=O)C1(CCC1)c1nc(nc2N3CCOC[C@H]3COc12)-c1ccc(F)c2[nH]ccc12 |r|
CS(=O)(=O)C1(CCC1)c1nc(nc2N3CCOC[C@H]3COc12)-c1cc(F)cc2[nH]ccc12 |r|
CN(C)c1nc2ccccc2n1-c1nc2N3CCOC[C@H]3COc2c(n1)C(C)(C)S(C)(=O)=O |r|
CNc1nc2cc(Cl)ccc2n1-c1nc2N3CCOC[C@H]3COc2c(n1)C(C)(C)S(C)(=O)=O |r|
CNc1nc2ccc(Cl)cc2n1-c1nc2N3CCOC[C@H]3COc2c(n1)C(C)(C)S(C)(=O)=O |r|
CNc1nc2cc(F)ccc2n1-c1nc2N3CCOC[C@H]3COc2c(n1)C(C)(C)S(C)(=O)=O |r|
CNc1nc2ccc(F)cc2n1-c1nc2N3CCOC[C@H]3COc2c(n1)C(C)(C)S(C)(=O)=O |r|
CNc1nc2cc(Cl)ccc2n1-c1nc2N3CCOC[C@H]3COc2c(n1)C1(CC1)S(C)(=O)=O |r|
CNc1nc2ccc(Cl)cc2n1-c1nc2N3CCOC[C@H]3COc2c(n1)C1(CC1)S(C)(=O)=O |r|
CNc1nc2ccccc2n1-c1nc2N3CCOC[C@H]3COc2c(n1)C1(CCC1)S(C)(=O)=O |r|
Cc1cc2c(cccc2[nH]1)-c1nc2N3CCOC[C@H]3COc2c(n1)C1(CCC1)S(C)(=O)=O |r|
CNc1nc2cc(Cl)ccc2n1-c1nc2N3CCOC[C@H]3COc2c(n1)C1(CCC1)S(C)(=O)=O |r|
CNc1nc2ccc(Cl)cc2n1-c1nc2N3CCOC[C@H]3COc2c(n1)C1(CCC1)S(C)(=O)=O |r|
CNc1nc2cc(F)ccc2n1-c1nc2N3CCOC[C@H]3COc2c(n1)C1(CCC1)S(C)(=O)=O |r|
CNc1nc2ccc(F)cc2n1-c1nc2N3CCOC[C@H]3COc2c(n1)C1(CCC1)S(C)(=O)=O |r|
CC(C)(c1nc(nc2N3CCOC[C@H]3COc12)-c1cc(cc2[nH]ccc12)C(F)(F)F)S(C)(=O)=O |r|
CC(C)(c1nc(nc2N3CCOC[C@H]3COc12)-c1ccc(F)c2[nH]ccc12)S(C)(=O)=O |r|
Cc1cc2c(cccc2[nH]1)-c1nc2N3CCOC[C@H]3COc2c(n1)C(C)(C)S(C)(=O)=O |r|
CS(=O)(=O)C1(CCOCC1)c1nc(nc2N3CCOC[C@H]3COc12)-c1cc(cc2[nH]ccc12)C(F)(F)F |r|
CS(=O)(=O)C1(CCOCC1)c1nc(nc2N3CCOC[C@H]3COc12)-c1ccc(F)c2[nH]ccc12 |r|
CS(=O)(=O)C1(CC1)c1nc(nc2N3CCOC[C@H]3COc12)-c1cc(cc2[nH]ccc12)C(F)(F)F |r|
Cc1cc2c(cccc2[nH]1)-c1nc2N3CCOC[C@H]3COc2c(n1)C1(CC1)S(C)(=O)=O |r|
CS(=O)(=O)C1(CC1)c1nc(nc2N3CCOC[C@H]3COc12)-c1ccc(F)c2[nH]ccc12 |r|
CS(=O)(=O)C1(CCC1)c1nc(nc2N3CCOC[C@H]3COc12)-c1cc(cc2[nH]ccc12)C(F)(F)F |r|
CNc1nc2ccc(cc2n1-c1nc2N3CCOC[C@H]3COc2c(n1)C(C)(C)S(C)(=O)=O)C#N |r|
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1c(F)cncc1F
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1cncc(F)c1Cl
COc1ccnnc1C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
COc1nnccc1C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncc[nH]c1=O
COc1nnc(Cl)cc1C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
COc1cc(C(O)c2ccc(F)c(c2)-c2ncnc3cc(ccc23)N2CCOCC2)c(Cl)nn1
COc1cc(Cl)nnc1C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
COc1nnc(Cl)cc1C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
COc1cc(Cl)nnc1C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
COc1nnccc1C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
CC(C)(C)Oc1nccnc1C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1nccnc1N1CCCC1
COc1nccnc1C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1c(Cl)cncc1Cl
COc1ccnnc1C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1ccc2nccn2n1)c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1
COc1cnc(Cl)c(c1)C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1ccc(F)c(c1)-c1ncnc2cc(sc12)N1CCOCC1)c1nccnc1Cl
COc1ncc(Cl)nc1C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
COc1cnc(Cl)c(n1)C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1nccnc1Cl
OC(c1cccnn1)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
COc1cnc(C(O)c2ccc(F)c(c2)-c2ncnc3cc(ccc23)N2CCOCC2)c(Cl)c1
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1nccnc1OC1COC1
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1cnccn1
OC(c1cnccn1)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1nc(Cl)cnc1Cl
OC(c1ccnnc1)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1ccn2nccc2n1)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
COc1nnc(C(O)c2cc(c(F)cc2Cl)-c2ncnc3cc(ccc23)N2CCOCC2)c2ccncc12
OC(c1ccc(Cl)nn1)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncccc1Cl
CNC(=O)c1ccc(nn1)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
Cn1nc(ccc1=O)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
Cc1cnnc(c1)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1cccnn1)c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1ccc(Cl)nn1)c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1
CN(C)C(=O)c1ccc(nn1)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
COc1cnc(cn1)C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1ccc(nn1)C(O)=O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1ccc2nccn2n1)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
COC(=O)c1ccc(nn1)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
COc1cnc(cn1)C(O)c1ccc(OC)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
NC(=O)c1ccc(nn1)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1)c1nccnc1Cl
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1cccnn1
COc1cnc(nc1)C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
CN(C)c1ccc(nn1)C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
Cc1ccc(nn1)C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
COc1ccc(nn1)[C@H](O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1 |r|
COc1ccc(nn1)[C@@H](O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1 |r|
COC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1ccc(OC)nn1
COc1ccc(nn1)C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1C2CCC1COC2)c1ccc(=O)[nH]n1
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1ccc(=O)[nH]n1
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1c(F)cncc1Cl
Cc1nccnc1C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
CCOc1cnnc(c1)C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncccc1C(F)(F)F
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncccc1OC(F)F
Cc1nccnc1[C@@H](O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1 |r|
Cc1nccnc1[C@H](O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1 |r|
Cc1nccnc1[C@H](O)c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1 |r|
Cc1nccnc1C(O)c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1
COc1cncnc1C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
Cc1cnc(C)c(n1)C(O)c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1cc(ccc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncnc2ccsc12
OC(c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncnc2sccc12
Cn1c(cccc1=O)C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1ccc(=O)[nH]n1)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
CCn1nc(ccc1=O)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
NCCn1nc(ccc1=O)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1ccc(=O)n(n1)C1CC1)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
NC(=O)Cn1nc(ccc1=O)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
OCCn1nc(ccc1=O)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1ccc(OC2COC2)nn1)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
CC(Oc1ccc(nn1)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1)C#N
OCCOc1nccnc1C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
OCCNc1nccnc1C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1ccc(OCCC#N)nn1)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
CSc1ccc(nn1)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
COc1cc(C)c(nn1)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
COc1nnc(cc1C)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
NC(=O)COc1ccc(nn1)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
COCCOc1ccc(nn1)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1ccc(OCC(O)=O)nn1)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
COC(=O)COc1ccc(nn1)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1ccc(OCC(F)(F)F)nn1)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
OCCOc1ccc(nn1)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
Nc1nccnc1C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1ccc(nn1)C#N)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1ccc(OCC#N)nn1)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
COc1ccc(cc1)C(O)c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1ccc(OC(F)F)nn1
COc1ccc(nn1)C(O)(C#C)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
COc1ccc(nn1)C(O)(C(F)F)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
COc1ccc(C(O)c2cc(c(F)cc2F)-c2ncnc3cc(ccc23)N2CCOCC2)c(F)c1
COc1ccc(nn1)C(C)(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
COc1ccc(nn1)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(sc12)N1CCOCC1
COc1ccc(nn1)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
COc1ccc(nn1)C(O)c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1
COc1ccc(nn1)C(O)c1cc(c(F)cc1Cl)-c1nc(Cl)nc2cc(ccc12)N1CCOCC1
CN(C)CCOc1ccc(nn1)C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
CCOc1ccc(nn1)C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
COc1ccc(nn1)[C@H](O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1 |r|
COc1ccc(nn1)[C@@H](O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1 |r|
CC(O)(c1nccs1)c1cncc(c1)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1nccs1)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)C1=CCOCC1 |t:28|
OC(c1nccs1)c1ccc(F)c(c1)-c1ncnc2cc(ncc12)N1CCOCC1
OCc1csc(n1)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ncc12)N1CCOCC1
OCc1csc(n1)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
CNCc1csc(n1)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1nccs1)c1ccc(F)c(c1)-c1ncnc2cc(sc12)N1CCOCC1
OC(c1ccc(s1)-c1ncnc2cc(ccc12)N1CCOCC1)c1nccs1
OC(c1nccs1)c1cccc(c1)-c1ncnc2cc(ccc12)N1CCOCC1
CC(O)(c1nccs1)c1cc(ccn1)-c1ncnc2cc(ccc12)N1CCOCC1
CC(O)(c1nccs1)c1cccc(c1)-c1ncnc2cc(ccc12)N1CCOCC1
Cc1ccc(cc1-c1ncnc2cc(ccc12)N1CCOCC1)C(C)(O)c1nccs1
CC(O)(c1cc(cs1)-c1ncnc2cc(ccc12)N1CCOCC1)c1nccs1
OC(c1nccs1)(c1cccc(c1)-c1ncnc2cc(ccc12)N1CCOCC1)C(F)(F)F
CC(O)(c1nccs1)c1cccc(c1F)-c1ncnc2cc(ccc12)N1CCOCC1
CC(O)(c1nccs1)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1csc(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1nccs1
OC(c1nccs1)c1cc(F)cc(c1)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1nccs1)c1cc(ccc1F)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1nccs1)c1cc(F)c(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1nccs1)c1cncc(c1)-c1ncnc2cc(ccc12)N1CCOCC1
COC(c1nccs1)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1nccs1)c1cnc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
Cc1csc(n1)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1nccs1)c1cccc(c1)-c1ncnc2cc(sc12)N1CCOCC1
OCc1csc(n1)[C@@H](O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1 |r|
OCc1csc(n1)[C@H](O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1 |r|
OCc1csc(n1)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1C2CCC1COC2
CCNCc1csc(n1)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
Cn1cc(cn1)C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
Cc1nc(sc1C)C(O)c1cc(cnc1F)-c1ncnc2cc(ncc12)N1CCOCC1
Cc1nc(sc1C)C(O)c1cc(cnc1F)-c1ncnc2cc(ccc12)N1CCOCC1
Cc1csc(n1)C(O)c1cnc(F)c(c1)-c1ncnc2cc(ncc12)N1CCOCC1
Cc1nc(sc1C)C(O)c1cnc(F)c(c1)-c1ncnc2cc(ncc12)N1CCOCC1
CC(C)n1cc(cn1)C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
CC(C)(C)n1cc(cn1)C(O)c1cc(cnc1F)-c1ncnc2cc(ccc12)N1CCOCC1
FC(F)OC(c1nccs1)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
Cc1nc(sc1CO)C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
CC(O)c1csc(n1)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
CCn1cc(cn1)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
Cc1cc(F)c(cc1C(O)c1nccs1)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1nccs1)c1ccc(F)c(c1)-c1nc(nc2cc(ccc12)N1CCOCC1)C#C
OC(c1nccs1)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
Cn1nccc1C(O)c1ccc(F)c(c1)-c1nc(Cl)nc2cc(ccc12)N1CCOCC1
OC(c1cccnc1)c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1ccccn1)c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1
Cn1nc(ccc1=O)C(O)c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1
Cn1nc(ccc1=O)C(O)c1ccc(F)c(c1F)-c1ncnc2cc(ccc12)N1CCOCC1 |(-2.67,-.39,;-2.67,1.15,;-1.33,1.93,;-1.33,3.47,;-2.67,4.23,;-4,3.47,;-4,1.93,;-5.33,1.16,;,4.23,;,5.78,;1.33,3.47,;2.67,4.23,;4,3.47,;4,1.93,;5.33,1.15,;2.67,1.15,;1.33,1.93,;,1.15,;2.67,-.38,;4,-1.15,;4,-2.69,;2.67,-3.47,;1.33,-2.69,;,-3.47,;-1.33,-2.69,;-1.33,-1.15,;,-.38,;1.33,-1.15,;-2.67,-3.47,;-4,-2.69,;-5.33,-3.47,;-5.33,-5,;-4,-5.78,;-2.67,-5,)|
COc1ccc(cn1)C(O)c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1ccc2ncnn2c1)c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1cn2ccnc2cn1)c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1
COc1ccc(nc1)C(O)c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1
COc1ccc(nn1)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(cnc12)N1CCOCC1
CNC(=O)C(c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1)c1nccnc1OC
CNC(=O)C(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncccc1Cl
COc1nccnc1C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(cnc12)N1CCOCC1
Cc1nccnc1[C@@H](O)c1ccc(F)c(c1)-c1ncnc2cc(cnc12)N1CCOCC1 |r|
Cc1nccnc1[C@H](O)c1ccc(F)c(c1)-c1ncnc2cc(cnc12)N1CCOCC1 |r|
Fc1cc(Cl)c(Cc2ccc3nccn3n2)cc1-c1ncnc2cc(ccc12)N1CCOCC1
CNC(=O)C(c1ccc2nccn2n1)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
Cc1nccnc1C(O)c1ccc(F)c(c1)-c1ncnc2cc(cnc12)N1CCOCC1
Cc1nccnc1C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(cnc12)N1CCOCC1
COc1nccnc1C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
Cc1nccnc1C(O)c1ccc(F)c(c1)-c1ncnc2cc(sc12)N1CCOCC1
Cc1nccnc1[C@H](O)c1ccc(F)c(c1)-c1ncnc2cc(cc(F)c12)N1CCOCC1 |r|
COc1nccnc1C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(cc(F)c12)N1CCOCC1
Cc1nccnc1[C@@H](O)c1ccc(F)c(c1)-c1ncnc2cc(cc(F)c12)N1CCOCC1 |r|
COc1nccnc1C(O)c1ccc(F)c(c1)-c1ncnc2cc(cc(F)c12)N1CCOCC1
CNC(=O)C(c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1)c1nccnc1C
COc1ccc(nn1)C(O)c1ccc(F)c(c1)-c1ncnc2cc(cc(F)c12)N1CCOCC1
COc1nccnc1C(C(N)=O)c1cc(c(F)cc1Cl)-c1ncnc2cc(cc(F)c12)N1CCOCC1
COc1ccc(nn1)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(cc(F)c12)N1CCOCC1
Cc1nccnc1C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(sc12)N1CCOCC1
Cc1nccnc1C(O)c1ccc(F)c(c1)-c1ncnc2cc(cc(F)c12)N1CCOCC1
Cc1nccnc1C(C(N)=O)c1cc(c(F)cc1Cl)-c1ncnc2cc(sc12)N1CCOCC1
Cc1nccnc1C(C(N)=O)c1ccc(F)c(c1)-c1ncnc2cc(sc12)N1CCOCC1
COc1ccc(nn1)C(C(N)=O)c1cc(c(F)cc1Cl)-c1ncnc2cc(sc12)N1CCOCC1
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1nccn2ncnc12
NC(=O)C(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1nccn2ncnc12
COc1ccc(nn1)C(O)c1ccc(F)c(c1)-c1ncnc2cc(N3CCOCC3)c(F)cc12
Cc1nccnc1C(O)c1ccc(F)c(c1)-c1ncnc2cc(N3CCOCC3)c(F)cc12
NC(=O)C(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1nncc2ccsc12
NC(=O)C(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1nncc2sccc12
CN1N=C(CCC1=O)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1 |c:2|
NC(=O)C(c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncccc1Cl
NC(=O)C(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1nnc(Cl)c2ccsc12
NC(=O)C(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1nnc(Cl)c2sccc12
NC(=O)C(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1cncc(n1)C(N)=O
NC(=O)C(c1cccnc1)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
NC(=O)C(c1cccnc1)c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1
NC(=O)C(c1cccnc1)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
Cc1cncc(n1)C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
NC(=O)C(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1cncc(Cl)c1
NC(=O)C(c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1)c1cccc2nncn12
NC(=O)C(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncnn2cccc12
NC(=O)C(c1cccnn1)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
Cc1cnc(C(C(N)=O)c2cc(c(F)cc2Cl)-c2ncnc3cc(ccc23)N2CCOCC2)c(C)n1
Nc1cncc(n1)C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
Cc1nccnc1C(C(N)=O)c1cc(ccc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
COc1nccnc1C(C(N)=O)c1cc(ccc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
COc1nccnc1C(C(N)=O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
COc1ccc(nn1)C(C(N)=O)c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1
COc1nnccc1C(C(N)=O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
COc1ccc(nn1)C(C(N)=O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
NC(=O)C(c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncnn2cccc12
COc1ccc(nn1)C(C(N)=O)c1cc(ccc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
Cn1nc(ccc1=O)C(C(N)=O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
Cn1c(cccc1=O)C(C(N)=O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
NC(=O)C(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncccc1Cl
Cc1ncc(nc1C)C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
NC(=O)C(c1cc(ccc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1)c1nccnc1Cl
COc1nccnc1C(C(N)=O)c1cc(ccc1F)-c1ncnc2cc(ccc12)N1CCOCC1
Cn1nc(ccc1=O)C(C(N)=O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
Cc1cnc(C(C(N)=O)c2ccc(F)c(c2)-c2ncnc3cc(ccc23)N2CCOCC2)c(C)n1
COc1nccnc1C(C(N)=O)c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1
COc1nccnc1C(C(N)=O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
NC(=O)C(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1c(F)cncc1F
NC(=O)C(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1cncc(F)c1Cl
NC(=O)C(c1ccc2nccn2n1)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
Cc1nccnc1C(C(N)=O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
COc1ccc(nn1)C(C(N)=O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
Cn1nc(ccc1=O)C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
Cc1nccnc1C(C(N)=O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1nccc2ccoc12
Cc1nccnc1C(C(N)=O)c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1cc(ccc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncnc(O)c1Cl
Cc1nccnc1\C(C(O)=O)=C1\C=CC(=O)C(=C1)c1ncnc2cc(ccc12)N1CCOCC1 |c:13,17|
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1nncc2ccsc12
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1nncc2sccc12
Cc1cc(C(C(N)=O)c2cc(c(F)cc2Cl)-c2ncnc3cc(ccc23)N2CCOCC2)n(C)c(=O)c1
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1nncc2ccoc12
OC(c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1)c1nncc2ccoc12
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1n[nH]c(=O)c2ccsc12
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1n[nH]c(=O)c2sccc12
Cc1cc(C(O)c2cc(c(F)cc2Cl)-c2ncnc3cc(ccc23)N2CCOCC2)n(C)c(=O)c1
Cc1cc(C(O)c2ccc(F)c(c2)-c2ncnc3cc(ccc23)N2CCOCC2)n(C)c(=O)c1
OC(c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1)c1nncc2sccc12
OC(c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1)c1nncc2ccsc12
OC(c1nnc2ccccn12)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncnn2cccc12
Cn1cnc2c(ncnc12)C(O)c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1
NC(=O)C(c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1)c1nncn2cccc12
Cc1nccnc1Cc1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1)c1cccc2nncn12
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1nccn2cnnc12
COC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1nccnc1C
Cc1cnc(C(O)c2ccc(F)c(c2)-c2ncnc3cc(ccc23)N2CCOCC2)c(C)n1
Cc1cnc(C(O)c2cc(c(F)cc2F)-c2ncnc3cc(ccc23)N2CCOCC2)c(C)n1
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1nccn2cccc12
COc1ccc(nn1)C(O)c1cc(ccc1F)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1)c1nccn2cccc12
OC(c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1)c1nccn2cccc12
Cn1c(nccc1=O)C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1cc(ccc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1)c1nccn2cccc12
OC(c1cc(ccc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncnn2cccc12
Cn1c(cccc1=O)C(O)c1cc(ccc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
Cn1c(cccc1=O)C(O)c1cc(ccc1F)-c1ncnc2cc(ccc12)N1CCOCC1
Cn1c(nccc1=O)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1cc(ccc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1)c1nccn2ccnc12
Cn1cnc2c(ncnc12)C(O)c1cc(ccc1F)-c1ncnc2cc(ccc12)N1CCOCC1
Cn1cnc2c(ncnc12)C(O)c1cc(ccc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1cc(ccc1F)-c1ncnc2cc(ccc12)N1CCOCC1)c1nccn2ccnc12
OC(c1cc(ccc1F)-c1ncnc2cc(ccc12)N1CCOCC1)c1cccc2nncn12
OC(c1cc(ccc1F)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncnc2ccoc12
Cc1cncnc1C(C(N)=O)c1cc(ccc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1nnc2ccccn12)c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1
Cn1c(cccc1=O)C(O)c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1
Cn1c(cccc1=O)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
Cn1cnc2ncnc(C(O)c3cc(c(F)cc3F)-c3ncnc4cc(ccc34)N3CCOCC3)c12
Cn1ncc2c(ncnc12)C(O)c1cc(ccc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncnc2CNCCc12
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncnc2CNCCc12
OC(c1cc(ccc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncncc1F
Cn1ncc2c(ncnc12)C(O)c1cc(ccc1F)-c1ncnc2cc(ccc12)N1CCOCC1
Cc1cncnc1C(O)c1cc(ccc1F)-c1ncnc2cc(ccc12)N1CCOCC1
Cc1nccnc1C(O)c1cc(ccc1F)-c1ncnc2cc(ccc12)N1CCOCC1
COc1nccnc1C(O)c1cc(ccc1F)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1)c1nccn2ccnc12
CCn1c(cccc1=O)C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
Cn1ncc2c(ncnc12)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
Cn1ncc2c(ncnc12)C(O)c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1
Cn1ncc2c(ncnc12)C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1cc(ccc1F)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncnc2ccsc12
OC(c1cc(ccc1F)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncnc2sccc12
COc1cncnc1C(O)c1cc(ccc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
COc1nccnc1C(O)c1cc(ccc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1cc(ccc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncnc2ccoc12
OC(c1cc(ccc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncnc2occc12
Cc1cncnc1C(O)c1cc(ccc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
Cn1cnc2c(ncnc12)C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
Cn1cnc2ncnc(C(O)c3cc(c(F)cc3Cl)-c3ncnc4cc(ccc34)N3CCOCC3)c12
CN1CCN(C1=O)c1nccnc1C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1nccnc1N1CCCC1=O
Cc1nccnc1C(O)c1cc(ccc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncnc2sccc12
OC(c1cc(ccc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncnc2sccc12
Cn1cnc2ncnc(C(O)c3ccc(F)c(c3)-c3ncnc4cc(ccc34)N3CCOCC3)c12
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncnc2occc12
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncnc2sccc12
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncnc2ccsc12
OC(c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncnc2ccsc12
OC(c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncnc2ccoc12
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncnc2ccoc12
OC(c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncnc2ccoc12
COc1cncnc1C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
COc1cncnc1C(O)c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1)c1nccnc1OC(F)F
COc1nccnc1C(O)c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1
COc1nccnc1[C@H](O)c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1 |r|
COc1nccnc1[C@@H](O)c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1 |r|
Cc1nccnc1C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
COc1ccc(nn1)C(O)c1cc(ccc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
Cn1cnc2ccnc(C(O)c3ccc(F)c(c3)-c3ncnc4cc(ccc34)N3CCOCC3)c12
CCc1nccnc1C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
CCOc1cccnc1C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1nccnc1OC(F)F
OC(c1cccnn1)c1cc(ccc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
Cc1cccnc1C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
COc1cnc(C(O)c2ccc(F)c(c2)-c2ncnc3cc(ccc23)N2CCOCC2)c(Br)c1
OC(c1cn2ccsc2n1)c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncccc1OC(F)(F)F
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1nccnc1C(F)(F)F
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncccc1Br
O[C@H](c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1nccnc1Cl |r|
O[C@@H](c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1nccnc1Cl |r|
Cn1ccnc1C(O)c1ccc(F)c(c1)-c1nc(Cl)nc2cc(ccc12)N1CCOCC1
COc1ccc(cc1)C(O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
NC(=O)C(c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1)c1nccn2cccc12
COc1nccnc1[C@H](O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1 |r|
COc1nccnc1[C@@H](O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1 |r|
Cc1cc2ncnn2cc1Nc1ncc2c(n1)n(C13CCC(O)(CC1)C3)c(=O)n2C
Cc1cc2c(cc1Nc1ncc3c(n1)n(C14CCC(O)(CC1)C4)c(=O)n3C)OCO2
Cc1cc2nsnc2cc1Nc1ncc2c(n1)n(C13CCC(O)(CC1)C3)c(=O)n2C
Cc1cc2nccnc2cc1Nc1ncc2c(n1)n(C13CCC(O)(CC1)C3)c(=O)n2C
Cc1cc2c(cc1Nc1ncc3c(n1)n(C14CCC(O)(CC1)C4)c(=O)n3C)OCCO2
COC12CCC(n3c(=O)n(C)c4cnc(Nc5cn6ncnc6cc5C)nc43)(CC1)C2
COC12CCC(n3c(=O)n(C)c4cnc(Nc5cc6c(cc5C)OCO6)nc43)(CC1)C2
COC12CCC(n3c(=O)n(C)c4cnc(Nc5cc6nsnc6cc5C)nc43)(CC1)C2
COC12CCC(n3c(=O)n(C)c4cnc(Nc5cc6nccnc6cc5C)nc43)(CC1)C2
COC12CCC(n3c(=O)n(C)c4cnc(Nc5cc6c(cc5C)OCCO6)nc43)(CC1)C2
Cc1cc2ncccc2cc1Nc1ncc2c(n1)n(C13CC(F)(C1)C3)c(=O)n2C
Cc1cc2ncnn2cc1Nc1ncc2c(n1)n(C13CC(F)(C1)C3)c(=O)n2C
Cc1cc2c(cc1Nc1ncc3c(n1)n(C14CC(F)(C1)C4)c(=O)n3C)OCO2
Cc1cc2nsnc2cc1Nc1ncc2c(n1)n(C13CC(F)(C1)C3)c(=O)n2C
Cc1cc2nccnc2cc1Nc1ncc2c(n1)n(C13CC(F)(C1)C3)c(=O)n2C
Cc1cc2c(cc1Nc1ncc3c(n1)n(C14CC(F)(C1)C4)c(=O)n3C)OCCO2
Cc1cc2c(cc1Nc1ncc3c(n1)n(C14CC(C#N)(C1)C4)c(=O)n3C)OCO2
Cc1cc2ncnn2cc1Nc1ncc2c(n1)n(C13CC(C(F)(F)F)(C1)C3)c(=O)n2C
Cc1cc2c(cc1Nc1ncc3c(n1)n(C14CC(C(F)(F)F)(C1)C4)c(=O)n3C)OCO2
COCC12CC(n3c(=O)n(C)c4cnc(Nc5cn6ncnc6cc5C)nc43)(C1)C2
COCC12CC(n3c(=O)n(C)c4cnc(Nc5cc6c(cc5C)OCO6)nc43)(C1)C2
Cc1cc2ncnn2cc1Nc1ncc2c(n1)n(C13CC(CC#N)(C1)C3)c(=O)n2C
Cc1cc2c(cc1Nc1ncc3c(n1)n(C14CC(CC#N)(C1)C4)c(=O)n3C)OCO2
Cc1cc2c(cc1Nc1ncc3c(n1)n(C14CCC(C#N)(CC1)CC4)c(=O)n3C)OCO2
COC12CCC(n3c(=O)n(C)c4cnc(Nc5cn6ncnc6cc5C)nc43)(CC1)CC2
COC12CCC(n3c(=O)n(C)c4cnc(Nc5cc6c(cc5C)OCO6)nc43)(CC1)CC2
Cc1cc2c(cc1Nc1ncc3c(n1)n(C14CCC(O)(CC1)CC4)c(=O)n3C)OCO2
COC12CCC(n3c(=O)n(C)c4cnc(Nc5cc6c(cc5C)OCO6)nc43)(C1)C2
COC12CCC(n3c(=O)n(C)c4cnc(Nc5cn6ncnc6cc5C)nc43)(C1)C2
COC12CCC(n3c(=O)n(C)c4cnc(Nc5cc6nsnc6cc5C)nc43)(C1)C2
Cc1cc2ncnn2cc1Nc1ncc2c(n1)n(C13CCC(O)(CC1)C3)c(=S)n2C
Cc1cc2c(cc1Nc1ncc3c(n1)n(C14CCC(O)(CC1)C4)c(=S)n3C)OCO2
Cc1cc2nccnc2cc1Nc1ncc2c(n1)n(C13CCC(O)(CC1)C3)c(=S)n2C
Cc1cc2ncnn2cc1Nc1ncc2c(n1)n(C13CC(F)(C1)C3)c(=S)n2C
Cc1cc2c(cc1Nc1ncc3c(n1)n(C14CC(F)(C1)C4)c(=S)n3C)OCO2
Cc1cc(-c2cnco2)c(F)cc1Nc1ncc2c(n1)n(C13CCC(O)(CC1)C3)c(=O)n2C
Cc1cc(-c2cnn(C)c2)c(F)cc1Nc1ncc2c(n1)n(C13CCC(O)(CC1)C3)c(=O)n2C
Cc1cc(-c2cnn(C)c2)c(F)cc1Nc1ncc2c(n1)n(C13CC(F)(C1)C3)c(=O)n2C
COC12CCC(n3c(=O)n(C)c4cnc(Nc5cc(F)c(-c6cnn(C)c6)cc5C)nc43)(C1)C2
COC12CCC(n3c(=O)n(C)c4cnc(Nc5cc(F)c(C(N)=O)cc5C)nc43)(C1)C2
COC12CCC(n3c(=O)n(C)c4cnc(Nc5cc(F)c(-c6cnco6)cc5C)nc43)(C1)C2
Cc1cc2ncnn2cc1Nc1ncc2c(n1)n(C1CC3CCC1CC3)c(=O)n2C
Cc1cc2c(cc1Nc1ncc3c(n1)n(C1CC4CCC1CC4)c(=O)n3C)OCO2
Cc1cc2ncccc2cc1Nc1ncc2c(n1)n([C@H]1C[C@@H]3CC[C@H]1C3)c(=O)n2C
Cc1cc2ncnn2cc1Nc1ncc2c(n1)n([C@H]1C[C@@H]3CC[C@H]1C3)c(=O)n2C
Cc1cc2c(cc1Nc1ncc3c(n1)n([C@H]1C[C@@H]4CC[C@H]1C4)c(=O)n3C)OCO2
Cc1cc2ncnn2cc1Nc1ncc2c(C)nn(C34CC(C3)C4)c2n1
Cc1cc2c(cc1Nc1ncc3c(C)nn(C45CC(C4)C5)c3n1)OCO2
Cc1cc2nccnc2cc1Nc1ncc2c(C)nn(C34CC(C3)C4)c2n1
Cc1cc2nsnc2cc1Nc1ncc2c(C)nn(C34CC(C3)C4)c2n1
Cc1cc2ncnn2cc1Nc1ncc2c(n1)N(C13CCC(O)(CC1)C3)CC(=O)N2C
Cc1cc2c(cc1Nc1ncc3c(n1)N(C14CCC(O)(CC1)C4)CC(=O)N3C)OCO2
Cc1cc2ncccc2cc1Nc1ncc2c(n1)N(C13CCC(O)(CC1)C3)CC(=O)N2C
Cc1cc2ncnn2cc1Nc1ncc2c(n1)N(C13CC(F)(C1)C3)CC(=O)N2C
Cc1cc2nsnc2cc1Nc1ncc2c(n1)N(C13CCC(O)(CC1)C3)CC(=O)N2C
Cc1cc2c(cc1Nc1ncc3c(n1)N(C14CC(F)(C1)C4)CC(=O)N3C)OCO2
Cc1cc2ncccc2cc1Nc1ncc2c(n1)N(C13CC(F)(C1)C3)CC(=O)N2C
Cc1cc2nsnc2cc1Nc1ncc2c(n1)N(C13CC(F)(C1)C3)CC(=O)N2C
Cc1cc2nccnc2cc1Nc1ncc2c(n1)N(C13CCC(O)(CC1)C3)CC(=O)N2C
Cc1cc2nonc2cc1Nc1ncc2c(n1)N(C13CCC(O)(CC1)C3)CC(=O)N2C
Cc1cc2nnccc2cc1Nc1ncc2c(n1)N(C13CCC(O)(CC1)C3)CC(=O)N2C
COC12CCC(N3CC(=O)N(C)c4cnc(Nc5cn6ncnc6cc5C)nc43)(CC1)C2
COC12CCC(N3CC(=O)N(C)c4cnc(Nc5cc6c(cc5C)OCO6)nc43)(CC1)C2
COC12CCC(N3CC(=O)N(C)c4cnc(Nc5cc6nsnc6cc5C)nc43)(CC1)C2
COC12CCC(N3CC(=O)N(C)c4cnc(Nc5cc6cccnc6cc5C)nc43)(CC1)C2
Cc1cc2ncnn2cc1Nc1ncc2c(n1)N(C13CCC(O)(CC1)C3)C(=O)C21CC1
Cc1cc2nccnc2cc1Nc1ncc2c(n1)N(C13CCC(O)(CC1)C3)C(=O)C21CC1
Cc1cc2c(cc1Nc1ncc3c(n1)N(C14CCC(O)(CC1)C4)C(=O)C31CC1)OCO2
Cc1cc2nsnc2cc1Nc1ncc2c(n1)N(C13CCC(O)(CC1)C3)C(=O)C21CC1
Cc1cc2ncnn2cc1Nc1ncc2c(n1)N(C13CC(F)(C1)C3)C(=O)C21CC1
Cc1cc2ncccc2cc1Nc1ncc2c(n1)N(C13CC(F)(C1)C3)C(=O)C21CC1
Cc1cc2nccnc2cc1Nc1ncc2c(n1)N(C13CC(F)(C1)C3)C(=O)C21CC1
Cc1cc2nsnc2cc1Nc1ncc2c(n1)N(C13CC(F)(C1)C3)C(=O)C21CC1
Cc1cc(-c2cnco2)ncc1Nc1ncc2c(n1)N(C13CC(F)(C1)C3)C(=O)C21CC1
Cc1cc(-c2cnn(C)c2)ncc1Nc1ncc2c(n1)N(C13CC(F)(C1)C3)C(=O)C21CC1
Cc1cc2c(cc1Nc1ncc3c(n1)N(C14CC(F)(C1)C4)C(=O)C31CC1)OCO2
[2H]C([2H])([2H])n1c(=O)n(C23CCC(O)(CC2)C3)c2nc(Nc3cn4ncnc4cc3C)ncc21
Cc1cc2ncnn2cc1Nc1ncc2c(n1)n(C13CCC(O)(CC1)CC3)c(=O)n2C
CC(C)NCCOC1=NCC(C2=CC3C4=C(C=NC3CC2F)N(C)C(=O)C42CCC2)C=C1NS(=O)(=O)C(C)C
CC(C)NCCOc1ncc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CCC2)cc1NS(C)(=O)=O
CCS(=O)(=O)NC1=CC(C2=CC3C4=C(C=NC3CC2F)N(C)C(=O)C42CCC2)CN=C1OCCNC(C)C
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(N4CC(N(C)C)C4)c(NS(C)(=O)=O)c3)cc21
CNC(=O)C(c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncccc1Cl
NC(=O)C(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1nccc2ccsc12
NC(=O)C(c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1)c1cncc2nncn12
COc1cc(C)c(nn1)C(C(N)=O)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1)c1nccc2nncn12
Cn1cnc2cccc(C(O)c3cc(c(F)cc3F)-c3ncnc4cc(ccc34)N3CCOCC3)c12
Cn1ncc2c(cccc12)C(O)c1cc(ccc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
OC(c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1)c1cccc2CNCCc12
OC(c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1)c1cccc2CNCCc12
Cn1cnc2cccc(C(O)c3cc(c(F)cc3Cl)-c3ncnc4cc(ccc34)N3CCOCC3)c12
OC(c1cc(c(F)cc1F)-c1ncnc2cc(ccc12)N1CCOCC1)c1ncncc1OC(F)F
Cc1cncnc1C(O)c1ccc(F)c(c1)-c1ncnc2cc(ccc12)N1CCOCC1
Cc1cc2ncnn2cc1Nc1ncc2n(C)c(=O)n([C@H]3CC[C@H](O)CC3)c2n1 |r,wU:23.25,wD:20.21,(-.77,3.78,;-2.1,3.01,;-3.44,3.78,;-4.77,3.01,;-6.24,3.49,;-7.14,2.24,;-6.24,1,;-4.77,1.47,;-3.44,.7,;-2.1,1.47,;-.77,.7,;.56,1.47,;.56,3.01,;1.9,3.78,;3.23,3.01,;4.7,3.49,;5.17,4.95,;5.6,2.24,;7.14,2.24,;4.7,1,;5.09,-.49,;4.01,-1.58,;4.4,-3.07,;5.89,-3.47,;6.29,-4.95,;6.98,-2.38,;6.58,-.89,;3.23,1.47,;1.9,.7,)|
Cc1cc2ncnn2cc1Nc1ncc2n(C)c(=O)n([C@@H]3CC[C@H](O)CC3)c2n1 |r,wU:20.21,23.25,(-.77,3.78,;-2.1,3.01,;-3.44,3.78,;-4.77,3.01,;-6.24,3.49,;-7.14,2.24,;-6.24,1,;-4.77,1.47,;-3.44,.7,;-2.1,1.47,;-.77,.7,;.56,1.47,;.56,3.01,;1.9,3.78,;3.23,3.01,;4.7,3.49,;5.17,4.95,;5.6,2.24,;7.14,2.24,;4.7,1,;5.09,-.49,;4.01,-1.58,;4.4,-3.07,;5.89,-3.47,;6.29,-4.95,;6.98,-2.38,;6.58,-.89,;3.23,1.47,;1.9,.7,)|
Cc1cc2ncnn2cc1Nc3ncc4c(n3)N(C(=O)N4C)C5CCOCC5
Cc1nc2cc(C)c(Nc3ncc4n(C)c(=O)n(C5CCOCC5)c4n3)cn2n1
CO[C@H]1CC[C@H](CC1)n1c2nc(Nc3cn4ncnc4cc3C)ncc2n(C)c1=O |r,wU:5.8,2.1,(7.49,-4.96,;5.95,-4.96,;5.55,-3.48,;4.06,-3.08,;3.66,-1.59,;4.75,-.5,;6.24,-.9,;6.64,-2.39,;4.35,.99,;2.89,1.46,;1.55,.69,;.22,1.46,;-1.11,.69,;-2.45,1.46,;-3.78,.69,;-5.12,1.46,;-6.58,.99,;-7.49,2.23,;-6.58,3.48,;-5.12,3,;-3.78,3.77,;-2.45,3,;-1.11,3.77,;.22,3,;1.55,3.77,;2.89,3,;4.35,3.48,;4.75,4.96,;5.26,2.23,;6.8,2.23,)|
CO[C@H]1CC[C@@H](CC1)n1c2nc(Nc3cn4ncnc4cc3C)ncc2n(C)c1=O |r,wU:2.1,wD:5.8,(7.49,-4.89,;5.95,-4.89,;5.55,-3.4,;4.06,-3,;3.66,-1.51,;4.75,-.43,;6.24,-.82,;6.64,-2.31,;4.35,1.06,;2.89,1.54,;1.55,.77,;.22,1.54,;-1.11,.77,;-2.45,1.54,;-3.78,.77,;-5.12,1.54,;-6.58,1.06,;-7.49,2.31,;-6.58,3.55,;-5.12,3.08,;-3.78,3.85,;-2.45,3.08,;-1.11,3.85,;.22,3.08,;1.55,3.85,;2.89,3.08,;4.35,3.55,;5.12,4.89,;5.26,2.31,;6.8,2.31,)|
Cc1cc2ncnn2cc1Nc1ncc2n(C)c(=O)n([C@H]3CCCOC3)c2n1 |r|
Cc1cc2ncnn2cc1Nc1ncc2n(C)c(=O)n([C@@H]3CCCOC3)c2n1 |r|
Cc1cc2ncnn2cc1Nc1ncc2n(C)c(=O)n([C@H]3CC[C@](C)(O)CC3)c2n1 |r,wU:20.21,23.25,wD:23.26,(3.5,1.28,;3.5,2.82,;4.83,3.59,;4.83,5.13,;5.97,6.16,;5.35,7.57,;3.82,7.41,;3.5,5.9,;2.16,5.13,;2.16,3.59,;.83,2.82,;-.51,3.59,;-1.84,2.82,;-3.17,3.59,;-3.17,5.13,;-4.32,6.16,;-5.8,5.76,;-3.69,7.57,;-4.46,8.9,;-2.16,7.41,;-1.07,8.5,;-1.47,9.99,;-.38,11.07,;1.11,10.68,;2.59,11.07,;1.11,12.22,;1.51,9.19,;.42,8.1,;-1.84,5.9,;-.51,5.13,)|
Cc1cc2ncnn2cc1Nc1ncc2n(C)c(=O)n([C@H]3CC[C@@](C)(O)CC3)c2n1 |r,wU:20.21,23.26,wD:23.25,(3.5,1.28,;3.5,2.82,;4.83,3.59,;4.83,5.13,;5.97,6.16,;5.35,7.57,;3.82,7.41,;3.5,5.9,;2.16,5.13,;2.16,3.59,;.83,2.82,;-.51,3.59,;-1.84,2.82,;-3.17,3.59,;-3.17,5.13,;-4.32,6.16,;-5.8,5.76,;-3.69,7.57,;-4.46,8.9,;-2.16,7.41,;-1.07,8.5,;-1.47,9.99,;-.38,11.07,;1.11,10.68,;1.11,12.22,;2.59,11.07,;1.51,9.19,;.42,8.1,;-1.84,5.9,;-.51,5.13,)|
Cc1cc2ncnn2cc1Nc1ncc2n(C)c(=O)n([C@H]3CCOC3)c2n1 |r|
Cc1cc2ncnn2cc1Nc1ncc2n(C)c(=O)n(c2n1)[C@]1(C)CC[C@H](O)CC1 |r,wU:26.30,wD:22.26,(3.41,-5.24,;3.41,-3.7,;4.74,-2.93,;4.74,-1.39,;5.89,-.36,;5.26,1.05,;3.73,.89,;3.41,-.62,;2.08,-1.39,;2.08,-2.93,;.74,-3.7,;-.59,-2.93,;-1.92,-3.7,;-3.26,-2.93,;-3.26,-1.39,;-4.4,-.36,;-5.89,-.76,;-3.78,1.05,;-4.17,2.53,;-2.24,.89,;-1.92,-.62,;-.59,-1.39,;-1.15,1.97,;-2.64,2.37,;.33,1.58,;1.42,2.66,;1.02,4.15,;2.11,5.24,;-.46,4.55,;-1.55,3.46,)|
Cc1cc2ncnn2cc1Nc1ncc2n(C)c(=O)n(C3CCCCC3)c2n1
C[C@H](Nc1ccccc1C(O)=O)c1cc(C)cc2c1oc(cc2=O)N1Cc2ccccc2C1 |r|
CC(Nc1ccccc1C(O)=O)c1cc(C)cc2c1oc(cc2=O)N1CCC(C)(C)CC1
CS(=O)(=O)Nc1cc(cnc1Cl)-c1ccc2ncnc(NCc3ccccc3)c2c1
CS(=O)(=O)Nc1cc(cnc1Cl)-c1ccc2ncnc(Nc3ccc(F)c(Cl)c3)c2c1
C[C@@H](Nc1ncnc2ccc(cc12)-c1cnc(Cl)c(NS(C)(=O)=O)c1)c1ccccc1 |r|
C[C@H](Nc1ncnc2ccc(cc12)-c1cnc(Cl)c(NS(C)(=O)=O)c1)c1ccccc1 |r|
COc1cc(cnc1OC)-c1ccc2ncnc(NC(C)c3ccccc3)c2c1
C[C@H](Nc1c(cnc2ccc(cc12)-c1cnc(Cl)c(NS(C)(=O)=O)c1)C#N)c1ccccc1 |r|
CC(Nc1c(cnc2ccc(cc12)-c1cnc(N)nc1)C#N)c1ccccc1
C[C@@H](Nc1c(cnc2ccc(cc12)-c1cnc(N)nc1)C#N)c1ccccc1 |r|
CC(Nc1c(cnc2ccc(cc12)-c1cnc2[nH]ncc2c1)C#N)c1ccccc1
CC(Nc1c(cnc2ccc(cc12)-c1cnc(Cl)c(NS(C)(=O)=O)c1)C#N)c1ccc(F)cc1
C[C@H](Nc1ncnc2ccc(cc12)-c1cnc(Cl)c(NS(C)(=O)=O)c1)c1ccc(F)cc1 |r|
CC(Nc1ncnc2ccc(cc12)-c1cnc(N)nc1)c1ccc(F)cc1
CC(Nc1c(cnc2ccc(cc12)-c1cncc(c1)-c1n[nH]c(=O)o1)C#N)c1ccccc1
C[C@@H]1COCCN1c1cc(-c2c(C)nn(c2C)-c2cncc(F)c2)n2ncc(-c3ccn[nH]3)c2n1 |wD:1.0,(6.26,6.69,;7.59,5.92,;8.92,6.69,;10.26,5.92,;10.26,4.38,;8.92,3.61,;7.59,4.38,;6.26,3.61,;6.26,2.07,;4.92,1.3,;4.92,-.24,;6.17,-1.14,;7.63,-.67,;5.69,-2.61,;4.15,-2.61,;3.68,-1.14,;2.21,-.67,;3.25,-3.85,;3.88,-5.26,;2.97,-6.51,;1.44,-6.34,;.81,-4.94,;-.72,-4.78,;1.72,-3.69,;3.59,2.07,;2.13,1.6,;1.22,2.84,;2.13,4.09,;1.65,5.55,;.18,6.03,;.18,7.57,;1.65,8.04,;2.55,6.8,;3.59,3.61,;4.92,4.38,)|
C[C@@H]1COCCN1c1cc(-c2c(C)nn(c2C)-c2cncc(c2)C(F)F)n2ncc(-c3ccn[nH]3)c2n1 |wD:1.0,(6.26,6.69,;7.59,5.92,;8.92,6.69,;10.26,5.92,;10.26,4.38,;8.92,3.61,;7.59,4.38,;6.26,3.61,;6.26,2.07,;4.92,1.3,;4.92,-.24,;6.17,-1.14,;7.63,-.67,;5.69,-2.61,;4.15,-2.61,;3.68,-1.14,;2.21,-.67,;3.25,-3.85,;3.88,-5.26,;2.97,-6.51,;1.44,-6.34,;.81,-4.94,;1.72,-3.69,;-.72,-4.78,;-1.62,-6.02,;-1.35,-3.37,;3.59,2.07,;2.13,1.6,;1.22,2.84,;2.13,4.09,;1.65,5.55,;.18,6.03,;.18,7.57,;1.65,8.04,;2.55,6.8,;3.59,3.61,;4.92,4.38,)|
CC(=O)N1CCC(CC1)n1c2nc(Nc3cc4ccnnc4cc3C)ncc2n(C)c1=O
CC(=O)N1CCC(CC1)n1c2nc(Nc3cc4nccnc4cc3C)ncc2n(C)c1=O
CC(=O)N1CCC(CC1)n1c2nc(Nc3cc4cncnc4cc3C)ncc2n(C)c1=O
CC(=O)N1CCC(CC1)n1c2nc(Nc3cc4ncc(C)nc4cc3C)ncc2n(C)c1=O
CC(=O)N1CCC(CC1)n1c2nc(Nc3cc4nc(C)cnc4cc3C)ncc2n(C)c1=O
Cc1cc2ncccc2cc1Nc1ncc2n(C)c(=O)n([C@H]3CC[C@H](O)CC3)c2n1 |r,wU:24.26,wD:21.22,(3.34,-5.73,;3.34,-4.19,;4.68,-3.42,;4.68,-1.88,;6.01,-1.11,;6.01,.43,;4.68,1.2,;3.34,.43,;3.34,-1.11,;2.01,-1.88,;2.01,-3.42,;.68,-4.19,;-.66,-3.42,;-1.99,-4.19,;-3.33,-3.42,;-3.33,-1.88,;-4.47,-.85,;-6.01,-.85,;-3.84,.56,;-4.61,1.89,;-2.31,.4,;-1.54,1.73,;-0,1.73,;.77,3.06,;-0,4.4,;.77,5.73,;-1.54,4.4,;-2.31,3.06,;-1.99,-1.11,;-.66,-1.88,)|
Cc1cc2nnccc2cc1Nc1ncc2n(C)c(=O)n([C@H]3CC[C@H](O)CC3)c2n1 |r,wU:24.26,wD:21.22,(3.34,-5.73,;3.34,-4.19,;4.68,-3.42,;4.68,-1.88,;6.01,-1.11,;6.01,.43,;4.68,1.2,;3.34,.43,;3.34,-1.11,;2.01,-1.88,;2.01,-3.42,;.68,-4.19,;-.66,-3.42,;-1.99,-4.19,;-3.33,-3.42,;-3.33,-1.88,;-4.47,-.85,;-6.01,-.85,;-3.84,.56,;-4.61,1.89,;-2.31,.4,;-1.54,1.73,;-0,1.73,;.77,3.06,;-0,4.4,;.77,5.73,;-1.54,4.4,;-2.31,3.06,;-1.99,-1.11,;-.66,-1.88,)|
Cc1cc2nccc(C)c2cc1Nc1ncc2n(C)c(=O)n(C3CCC(O)CC3)c2n1 |(2.53,5.92,;3.86,6.69,;5.2,5.92,;6.53,6.69,;7.87,5.92,;9.2,6.69,;9.2,8.23,;7.87,9,;7.87,10.54,;6.53,8.23,;5.2,9,;3.86,8.23,;2.53,9,;1.2,8.23,;1.2,6.69,;-.14,5.92,;-1.47,6.69,;-2.94,6.22,;-3.41,4.75,;-3.84,7.46,;-5.38,7.46,;-2.94,8.71,;-3.41,10.17,;-4.92,10.49,;-5.39,11.96,;-4.36,13.1,;-4.84,14.57,;-2.86,12.78,;-2.38,11.32,;-1.47,8.23,;-.14,9,)|
COc1ccnc2cc(C)c(Nc3ncc4n(C)c(=O)n([C@H]5CC[C@H](O)CC5)c4n3)cc12 |r,wU:24.24,wD:21.20,(2.01,2.74,;2.01,1.2,;3.34,.43,;4.68,1.2,;6.01,.43,;6.01,-1.11,;4.68,-1.88,;4.68,-3.42,;3.34,-4.19,;3.34,-5.73,;2.01,-3.42,;.68,-4.19,;-.66,-3.42,;-1.99,-4.19,;-3.33,-3.42,;-3.33,-1.88,;-4.47,-.85,;-6.01,-.85,;-3.84,.56,;-4.61,1.89,;-2.31,.4,;-1.54,1.73,;-0,1.73,;.77,3.06,;-0,4.4,;.77,5.73,;-1.54,4.4,;-2.31,3.06,;-1.99,-1.11,;-.66,-1.88,;2.01,-1.88,;3.34,-1.11,)|
Cc1cc2nccnc2cc1Nc1ncc2n(C)c(=O)n(C3CCC(O)CC3)c2n1 |(,-3.08,;1.33,-2.31,;2.67,-3.08,;4,-2.31,;5.33,-3.08,;6.67,-2.31,;6.67,-.77,;5.33,,;4,-.77,;2.67,,;1.33,-.77,;;-1.33,-.77,;-1.33,-2.31,;-2.67,-3.08,;-4,-2.31,;-5.47,-2.79,;-5.94,-4.25,;-6.37,-1.54,;-7.91,-1.54,;-5.47,-.29,;-5.94,1.17,;-4.91,2.32,;-5.39,3.78,;-6.89,4.1,;-7.37,5.56,;-7.92,2.96,;-7.45,1.49,;-4,-.77,;-2.67,,)|
Cc1cc2ncccc2cc1Nc1ncc2n(C)c(=O)n(C3CCC(O)CC3)c2n1 |(,-3.08,;1.33,-2.31,;2.67,-3.08,;4,-2.31,;5.33,-3.08,;6.67,-2.31,;6.67,-.77,;5.33,,;4,-.77,;2.67,,;1.33,-.77,;;-1.33,-.77,;-1.33,-2.31,;-2.67,-3.08,;-4,-2.31,;-5.47,-2.79,;-5.94,-4.25,;-6.37,-1.54,;-7.91,-1.54,;-5.47,-.29,;-5.94,1.17,;-4.91,2.32,;-5.39,3.78,;-6.89,4.1,;-7.37,5.56,;-7.92,2.96,;-7.45,1.49,;-4,-.77,;-2.67,,)|
Cc1cc2nnccc2cc1Nc1ncc2n(C)c(=O)n([C@@H]3CC[C@H](O)CC3)c2n1 |r,wU:21.22,24.26,(3.34,-5.24,;3.34,-3.7,;4.68,-2.93,;4.68,-1.39,;6.01,-.62,;6.01,.92,;4.68,1.69,;3.34,.92,;3.34,-.62,;2.01,-1.39,;2.01,-2.93,;.68,-3.7,;-.66,-2.93,;-1.99,-3.7,;-3.33,-2.93,;-3.33,-1.39,;-4.47,-.36,;-6.01,-.36,;-3.84,1.05,;-4.61,2.38,;-2.31,.89,;-1.22,1.97,;.26,1.58,;1.35,2.66,;.95,4.15,;2.04,5.24,;-.53,4.55,;-1.62,3.46,;-1.99,-.62,;-.66,-1.39,)|
Cc1cc2ncccc2cc1Nc1ncc2n(C)c(=O)n([C@H]3CC[C@@](C)(O)CC3)c2n1 |r,wU:24.26,wD:21.22,24.27,(3.32,3.93,;3.32,5.47,;4.65,6.24,;4.65,7.78,;5.98,8.55,;5.98,10.09,;4.65,10.86,;3.32,10.09,;3.32,8.55,;1.98,7.78,;1.98,6.24,;.65,5.47,;-.68,6.24,;-2.02,5.47,;-3.35,6.24,;-3.35,7.78,;-4.5,8.81,;-5.98,8.41,;-3.87,10.22,;-4.64,11.55,;-2.34,10.06,;-1.25,11.14,;.24,10.75,;1.33,11.83,;.93,13.32,;.93,14.86,;2.47,13.32,;-.56,13.72,;-1.65,12.63,;-2.02,8.55,;-.68,7.78,)|
Cc1cc2ncccc2cc1Nc1ncc2n(C)c(=O)n([C@H]3CC[C@](C)(O)CC3)c2n1 |r,wU:24.27,wD:21.22,24.26,(3.32,3.93,;3.32,5.47,;4.65,6.24,;4.65,7.78,;5.98,8.55,;5.98,10.09,;4.65,10.86,;3.32,10.09,;3.32,8.55,;1.98,7.78,;1.98,6.24,;.65,5.47,;-.68,6.24,;-2.02,5.47,;-3.35,6.24,;-3.35,7.78,;-4.5,8.81,;-5.98,8.41,;-3.87,10.22,;-4.64,11.55,;-2.34,10.06,;-1.25,11.14,;.24,10.75,;1.33,11.83,;.93,13.32,;.93,14.86,;2.47,13.32,;-.56,13.72,;-1.65,12.63,;-2.02,8.55,;-.68,7.78,)|
Cc1cc2nnccc2cc1Nc1ncc2n(C)c(=O)n([C@H]3CC[C@@](C)(O)CC3)c2n1 |r,wU:24.26,wD:21.22,24.27,(3.32,3.93,;3.32,5.47,;4.65,6.24,;4.65,7.78,;5.98,8.55,;5.98,10.09,;4.65,10.86,;3.32,10.09,;3.32,8.55,;1.98,7.78,;1.98,6.24,;.65,5.47,;-.68,6.24,;-2.02,5.47,;-3.35,6.24,;-3.35,7.78,;-4.5,8.81,;-5.98,8.41,;-3.87,10.22,;-4.64,11.55,;-2.34,10.06,;-1.25,11.14,;.24,10.75,;1.33,11.83,;.93,13.32,;.93,14.86,;2.47,13.32,;-.56,13.72,;-1.65,12.63,;-2.02,8.55,;-.68,7.78,)|
Cc1cc2nnccc2cc1Nc1ncc2n(C)c(=O)n([C@H]3CC[C@](C)(O)CC3)c2n1 |r,wU:24.27,wD:21.22,24.26,(3.32,3.93,;3.32,5.47,;4.65,6.24,;4.65,7.78,;5.98,8.55,;5.98,10.09,;4.65,10.86,;3.32,10.09,;3.32,8.55,;1.98,7.78,;1.98,6.24,;.65,5.47,;-.68,6.24,;-2.02,5.47,;-3.35,6.24,;-3.35,7.78,;-4.5,8.81,;-5.98,8.41,;-3.87,10.22,;-4.64,11.55,;-2.34,10.06,;-1.25,11.14,;.24,10.75,;1.33,11.83,;.93,13.32,;.93,14.86,;2.47,13.32,;-.56,13.72,;-1.65,12.63,;-2.02,8.55,;-.68,7.78,)|
Cc1cc2nccnc2cc1Nc1ncc2n(C)c(=O)n(C3CC[C@@](C)(O)CC3)c2n1 |r,wU:24.26,wD:24.27,(,-3.08,;1.33,-2.31,;2.67,-3.08,;4,-2.31,;5.33,-3.08,;6.67,-2.31,;6.67,-.77,;5.33,,;4,-.77,;2.67,,;1.33,-.77,;;-1.33,-.77,;-1.33,-2.31,;-2.67,-3.08,;-4,-2.31,;-5.47,-2.79,;-5.94,-4.25,;-6.37,-1.54,;-7.91,-1.54,;-5.47,-.29,;-5.94,1.17,;-4.91,2.32,;-5.39,3.78,;-6.89,4.1,;-6.32,5.53,;-8.2,4.92,;-7.92,2.96,;-7.45,1.49,;-4,-.77,;-2.67,,)|
Cc1cc2nccnc2cc1Nc1ncc2n(C)c(=O)n(C3CC[C@@](C)(O)CC3)c2n1 |r,wU:24.27,wD:24.26,(,-3.08,;1.33,-2.31,;2.67,-3.08,;4,-2.31,;5.33,-3.08,;6.67,-2.31,;6.67,-.77,;5.33,,;4,-.77,;2.67,,;1.33,-.77,;;-1.33,-.77,;-1.33,-2.31,;-2.67,-3.08,;-4,-2.31,;-5.47,-2.79,;-5.94,-4.25,;-6.37,-1.54,;-7.91,-1.54,;-5.47,-.29,;-5.94,1.17,;-7.45,1.49,;-7.92,2.96,;-6.89,4.1,;-6.32,5.53,;-8.2,4.92,;-5.39,3.78,;-4.91,2.32,;-4,-.77,;-2.67,,)|
Cc1cc2nccnc2cc1Nc1ncc2n(C)c(=O)n(c2n1)[C@]1(C)CC[C@H](O)CC1 |r,wU:27.31,wD:23.27,(3.32,-5.24,;3.32,-3.7,;4.65,-2.93,;4.65,-1.39,;5.98,-.62,;5.98,.92,;4.65,1.69,;3.32,.92,;3.32,-.62,;1.98,-1.39,;1.98,-2.93,;.65,-3.7,;-.68,-2.93,;-2.02,-3.7,;-3.35,-2.93,;-3.35,-1.39,;-4.5,-.36,;-5.98,-.76,;-3.87,1.05,;-4.64,2.38,;-2.34,.89,;-2.02,-.62,;-.68,-1.39,;-1.25,1.97,;-2.74,2.37,;.24,1.58,;1.33,2.66,;.93,4.15,;2.02,5.24,;-.56,4.55,;-1.65,3.46,)|
Cc1cc2nnccc2cc1Nc1ncc2n(C)c(=O)n([C@H]3CCOC3)c2n1 |r|
Cc1cc2nccnc2cc1Nc1ncc2n(C)c(=O)n([C@H]3CCOC3)c2n1 |r|
Cc1cc2nnccc2cc1Nc1ncc2n(C)c(=O)n([C@@H]3CCOC3)c2n1 |r|
Cc1cc2nccnc2cc1Nc1ncc2n(C)c(=O)n([C@@H]3CCOC3)c2n1 |r|
Cc1cc2nnccc2cc1Nc1ncc2n(C)c(=O)n(C3CCCOC3)c2n1
Cc1cc2nccnc2cc1Nc1ncc2n(C)c(=O)n(C3CCCOC3)c2n1
Cc1cc2nnccc2cc1Nc1ncc2n(C)c(=O)n([C@H]3CCCOC3)c2n1 |r|
Cc1cc2nccnc2cc1Nc1ncc2n(C)c(=O)n([C@H]3CCCOC3)c2n1 |r|
Cc1cc2nnccc2cc1Nc1ncc2n(C)c(=O)n(C3CCOCC3)c2n1
Cc1cc2ncccc2cc1Nc1ncc2n(C)c(=O)n(C3CCOCC3)c2n1
Cc1cc2nccnc2cc1Nc1ncc2n(C)c(=O)n(C3CCOCC3)c2n1
Cc1cc2ncncc2cc1Nc1ncc2n(C)c(=O)n(C3CCOCC3)c2n1
Cc1cnc2cc(C)c(Nc3ncc4n(C)c(=O)n(C5CCOCC5)c4n3)cc2n1
Cc1cnc2cc(Nc3ncc4n(C)c(=O)n(C5CCOCC5)c4n3)c(C)cc2n1
Cc1cc2ncccc2cc1Nc1ncc2n(C)c(=O)n(C3CCS(=O)(=O)CC3)c2n1
Cc1cc2ncccc2cc1Nc1ncc2n(C)c(=O)n(C3COC3)c2n1
Cc1cc2ncccc2cc1Nc1ncc2n(C)c(=O)n(C3CCNCC3)c2n1
Cc1cc2ncccc2cc1Nc1ncc2n(C)c(=O)n([C@@H]3CCNC[C@@H]3F)c2n1 |r|
Cc1cc2ncccc2cc1Nc1ncc2n(C)c(=O)n(C3CC[C@@](C)(N)CC3)c2n1 |r,wU:24.27,wD:24.26,(,-3.08,;1.33,-2.31,;2.67,-3.08,;4,-2.31,;5.33,-3.08,;6.67,-2.31,;6.67,-.77,;5.33,,;4,-.77,;2.67,,;1.33,-.77,;;-1.33,-.77,;-1.33,-2.31,;-2.67,-3.08,;-4,-2.31,;-5.47,-2.79,;-5.94,-4.25,;-6.37,-1.54,;-7.91,-1.54,;-5.47,-.29,;-5.94,1.17,;-7.45,1.49,;-7.92,2.96,;-6.89,4.1,;-6.32,5.53,;-8.2,4.92,;-5.39,3.78,;-4.91,2.32,;-4,-.77,;-2.67,,)|
Cc1cc2ncccc2cc1Nc1ncc2n(C)c(=O)n(C3CC[C@@](C)(N)CC3)c2n1 |r,wU:24.26,wD:24.27,(,-3.08,;1.33,-2.31,;2.67,-3.08,;4,-2.31,;5.33,-3.08,;6.67,-2.31,;6.67,-.77,;5.33,,;4,-.77,;2.67,,;1.33,-.77,;;-1.33,-.77,;-1.33,-2.31,;-2.67,-3.08,;-4,-2.31,;-5.47,-2.79,;-5.94,-4.25,;-6.37,-1.54,;-7.91,-1.54,;-5.47,-.29,;-5.94,1.17,;-4.91,2.32,;-5.39,3.78,;-6.89,4.1,;-6.32,5.53,;-8.2,4.92,;-7.92,2.96,;-7.45,1.49,;-4,-.77,;-2.67,,)|
CN1CC[C@H](C1)n1c2nc(Nc3cc4cccnc4cc3C)ncc2n(C)c1=O |r|
CN1CC[C@@H](C1)n1c2nc(Nc3cc4cccnc4cc3C)ncc2n(C)c1=O |r|
CN1CCC(CC1)n1c2nc(Nc3cc4ccnnc4cc3C)ncc2n(C)c1=O
CN1CCC(CC1)n1c2nc(Nc3cc4cccnc4cc3C)ncc2n(C)c1=O
CN1CCC(CC1)n1c2nc(Nc3cc4nccnc4cc3C)ncc2n(C)c1=O
CN1CC[C@H]([C@@H](F)C1)n1c2nc(Nc3cc4cccnc4cc3C)ncc2n(C)c1=O |r|
Cc1cc2ncccc2cc1Nc1ncc2n(C)c(=O)n(C3CCN(CC3)C3COC3)c2n1
Cc1cc2ncccc2cc1Nc1ncc2n(C)c(=O)n(C3CCN(CCO)CC3)c2n1
COCCN1CCC(CC1)n1c2nc(Nc3cc4cccnc4cc3C)ncc2n(C)c1=O
CCN1CCC(CC1)n1c2nc(Nc3cc4cccnc4cc3C)ncc2n(C)c1=O
CC(=O)N1CCC(CC1)n1c2nc(Nc3cc4cccnc4cc3C)ncc2n(C)c1=O
Cc1cc2c(cccn2)cc1Nc3ncc4c(n3)N(C(=O)N4C)[C@@H]5CNC[C@H]5F
CN1C2=NCC3(CCOCC3)N2c2nc(Nc3cn4ncnc4cc3C)ncc12 |t:2|
CN1CC2(CCOCC2)n2c1nc1cnc(Nc3cn4ncnc4cc3C)nc21
Cc1cc2ncnn2cc1Nc1ncc2nc3NCC4(CCOCC4)n3c2n1
CN1C2=NCC3(CCCCC3)N2c2nc(Nc3cn4ncnc4cc3C)ncc12 |t:2|
CN1C2=NCC3(CCC(F)(F)CC3)N2c2nc(Nc3cn4ncnc4cc3C)ncc12 |t:2|
CN1C2=NCC3(CCC(=O)CC3)N2c2nc(Nc3cn4ncnc4cc3C)ncc12 |t:2|
CN1C2=NCC3(CC[C@H](O)CC3)N2c2nc(Nc3cn4ncnc4cc3C)ncc12 |r,wU:8.8,t:2,(3.76,4.72,;3.76,3.18,;5.01,2.27,;6.55,2.27,;7.02,.81,;5.78,-.1,;4.44,-.87,;4.44,-2.41,;5.78,-3.18,;5.78,-4.72,;7.11,-2.41,;7.11,-.87,;4.53,.81,;2.99,.81,;1.96,-.34,;.45,-.02,;-.58,-1.16,;-2.08,-.84,;-3.11,-1.99,;-4.62,-1.67,;-5.87,-2.57,;-7.11,-1.67,;-6.64,-.2,;-5.1,-.2,;-4.06,.94,;-2.56,.62,;-1.53,1.77,;-.02,1.45,;1.01,2.59,;2.52,2.27,)|
CN1C2=NCC3(CC[C@H](O)CC3)N2c2nc(Nc3cn4ncnc4cc3C)ncc12 |r,wD:8.8,t:2,(3.76,4.72,;3.76,3.18,;5.01,2.27,;6.55,2.27,;7.02,.81,;5.78,-.1,;7.11,-.87,;7.11,-2.41,;5.78,-3.18,;5.78,-4.72,;4.44,-2.41,;4.44,-.87,;4.53,.81,;2.99,.81,;1.96,-.34,;.45,-.02,;-.58,-1.16,;-2.08,-.84,;-3.11,-1.99,;-4.62,-1.67,;-5.87,-2.57,;-7.11,-1.67,;-6.64,-.2,;-5.1,-.2,;-4.06,.94,;-2.56,.62,;-1.53,1.77,;-.02,1.45,;1.01,2.59,;2.52,2.27,)|
CN1C2=NCC3(CCSCC3)N2c2nc(Nc3cn4ncnc4cc3C)ncc12 |t:2|
CN1C2=NCC3(CCS(=O)(=O)CC3)N2c2nc(Nc3cn4ncnc4cc3C)ncc12 |t:2|
COC1(C)CCC2(CN=C3N(C)c4cnc(Nc5cn6ncnc6cc5C)nc4N23)CC1 |w:2.2,t:8,(7,-4.73,;5.46,-4.73,;4.69,-3.4,;3.35,-4.17,;3.66,-2.25,;4.13,-.79,;5.64,-.47,;7.1,.01,;7.1,1.55,;5.64,2.02,;4.73,3.27,;5.21,4.73,;3.27,2.79,;1.93,3.56,;.6,2.79,;.6,1.25,;-.73,.48,;-2.07,1.25,;-3.4,.48,;-4.73,1.25,;-6.2,.78,;-7.1,2.02,;-6.2,3.27,;-4.73,2.79,;-3.4,3.56,;-2.07,2.79,;-.73,3.56,;1.93,.48,;3.27,1.25,;4.73,.78,;6.67,-1.61,;6.19,-3.08,)|
CO[C@H]1CCC2(CN=C3N(C)c4cnc(Nc5cn6ncnc6cc5C)nc4N23)CC1 |r,wU:2.1,t:7,(4.53,-4.85,;5.78,-3.95,;5.78,-2.41,;4.44,-1.64,;4.44,-.1,;5.78,.67,;7.02,1.58,;6.55,3.04,;5.01,3.04,;3.76,3.95,;3.76,5.49,;2.52,3.04,;1.01,3.36,;-.02,2.22,;.45,.75,;-.58,-.39,;-2.08,-.07,;-3.11,-1.22,;-4.62,-.9,;-5.87,-1.8,;-7.11,-.9,;-6.64,.57,;-5.1,.57,;-4.06,1.71,;-2.56,1.39,;-1.53,2.54,;1.96,.43,;2.99,1.58,;4.53,1.58,;7.11,-.1,;7.11,-1.64,)|
CO[C@H]1CCC2(CN=C3N(C)c4cnc(Nc5cn6ncnc6cc5C)nc4N23)CC1 |r,wD:2.1,t:7,(4.37,-4.57,;5.78,-3.95,;5.78,-2.41,;7.11,-1.64,;7.11,-.1,;5.78,.67,;7.02,1.58,;6.55,3.04,;5.01,3.04,;3.76,3.95,;3.76,5.49,;2.52,3.04,;1.01,3.36,;-.02,2.22,;.45,.75,;-.58,-.39,;-2.08,-.07,;-3.11,-1.22,;-4.62,-.9,;-5.87,-1.8,;-7.11,-.9,;-6.64,.57,;-5.1,.57,;-4.06,1.71,;-2.56,1.39,;-1.53,2.54,;1.96,.43,;2.99,1.58,;4.53,1.58,;4.44,-.1,;4.44,-1.64,)|
CN1C2=NCC(C)(CCO)N2c2nc(Nc3cn4ncnc4cc3C)ncc12 |t:2|
CN1C2=NCC3(CCOC3)N2c2nc(Nc3cn4ncnc4cc3C)ncc12 |t:2|
CN1C2=NCC3(CCCOCC3)N2c2nc(Nc3cn4ncnc4cc3C)ncc12 |t:2|
CN1C2=NC[C@@]3(CCCOCC3)N2c2nc(Nc3cn4ncnc4cc3C)ncc12 |r,t:2|
CN1C2=NC[C@]3(CCCOCC3)N2c2nc(Nc3cn4ncnc4cc3C)ncc12 |r,t:2|
CN1C2=NCC3(CCS(=O)CC3)N2c2nc(Nc3cn4ncnc4cc3C)ncc12 |t:2|
CC(C)n1c2c(nnc3ccc(cc23)-c2ccc(COCCN3CCC(C)(C)CC3)nc2)n(C)c1=O
CC(C)n1c2c(nnc3ccc(cc23)-c2ccc(nc2)[C@@H](C)OCC(=O)N2CCC3(CC3)C2)n(C)c1=O |r|
COC1CCN(CCO[C@H](C)c2ccc(cn2)-c2ccc3nnc4n(C)c(=O)n(C(C)C)c4c3c2)CC1 |r|
CC(C)n1c2c(nnc3ccc(cc23)-c2ccc(nc2)[C@@H](C)OCCN2CCCC2)n(C)c1=O |r|
CC(C)n1c2c(nnc3ccc(cc23)-c2ccc(nc2)[C@@H](C)OCCN2CCC(C2)OC2CC2)n(C)c1=O |r|
CC(C)n1c2c(nnc3ccc(cc23)-c2ccc(nc2)[C@@H](C)OCCN2CC[C@@H](C)C2)n(C)c1=O |r|
C[C@@H](OCCN1CCC2(CC2)C1)c1ccc2nnc3n(C)c(=O)n(C4CCOCC4)c3c2c1 |r|
C[C@@H](OCCN1CCC2(CC2)CC1)c1ccc(cn1)-c1ccc2nnc3n(C)c(=O)n(C4CCOCC4)c3c2c1 |r|
CO[C@@H]1CCN(CCO[C@H](C)c2ccc(cn2)-c2ccc3nnc4n(C)c(=O)n(C5CCOCC5)c4c3c2)C1 |r|
CO[C@H]1C[C@@H](C1)n1c2c(nnc3ccc(cc23)-c2ccc(nc2)[C@@H](C)OCCN2CCCC2)n(C)c1=O |r,wU:2.1,wD:4.6,23.27,(3.84,4.98,;3.36,3.51,;4.39,2.37,;5.93,2.29,;5.85,.75,;4.31,.83,;6.88,-.39,;6.56,-1.9,;7.9,-2.67,;7.9,-4.21,;6.56,-4.98,;5.23,-4.21,;3.89,-4.98,;2.56,-4.21,;2.56,-2.67,;3.89,-1.9,;5.23,-2.67,;1.23,-1.9,;1.23,-.36,;-.11,.41,;-1.44,-.36,;-1.44,-1.9,;-.11,-2.67,;-2.77,.41,;-2.77,1.95,;-4.11,-.36,;-5.44,.41,;-6.78,-.36,;-8.11,.41,;-8.27,1.94,;-9.78,2.26,;-10.55,.93,;-9.52,-.22,;9.04,-1.64,;10.55,-1.96,;8.41,-.23,;9.18,1.1,)|
CC(C)n1c2c(nnc3ccc(cc23)-c2ccc(nc2)[C@H](OCCN2CCCC2)C(F)(F)F)n(C)c1=O |r|
CC(C)n1c2c(nnc3ccc(cc23)-c2ccc(nc2)[C@@H](OCCN2CCCC2)C(F)(F)F)n(C)c1=O |r|
Cn1c2cnc3cc(F)c(-c4ccc(OCCCN5CCCCC5)nc4)c4OC5CCCCC5n(c2c34)c1=O
CC[C@@H]1COc2c(c(F)cc3ncc4n(C)c(=O)n1c4c23)-c1ccc(OCCCN2CCCCC2)nc1 |r|
CN(C)CCCOc1ccc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cn1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCCC2)C(=O)N4C)cc1NS(=O)(=O)c1ccccc1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCCCC2)C(=O)N4C)cc1NS(=O)(=O)c1ccccc1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(=O)(=O)c1ccccc1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(=O)(=O)c1ccccc1
CN(C)CCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCCC2)C(=O)N4C)cc1NS(=O)(=O)c1ccccc1
COc1ncc(-c2ccc3ncc4c(c3c2)C2(COC2)C(=O)N4C)cc1NS(=O)(=O)c1ccccc1
COc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(=O)(=O)c1cccc(Cl)c1
CN(C)c1ncc(-c2ccc3ncc4c(c3c2)C2(COC2)C(=O)N4C)cc1NS(=O)(=O)c1ccccc1
COc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(=O)(=O)c1ccc([N+](=O)[O-])cc1
COc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(=O)(=O)c1cccc(C(C)=O)c1
COc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(=O)(=O)c1ccccc1
CN1C(=O)C2(CC2)c2c1cnc1ccc(-c3cnc(Cl)c(NS(=O)(=O)c4ccccc4)c3)cc21
COc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(=O)(=O)c1cccc(C(C)O)c1
COc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4)cc1NS(=O)(=O)c1ccccc1
COc1ncc(Br)cc1N(COCC[Si](C)(C)C)S(=O)(=O)c1ccccc1
CN1C(=O)C2(CC2)c2c1cnc1ccc(-c3ccc4ncccc4c3)cc21
Cc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(=O)(=O)c1ccccc1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(=O)(=O)C1CC1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4Cc2cn[nH]c2)cc1NS(=O)(=O)c1ccccc1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(COC2)C(=O)N4C)cc1NS(=O)(=O)c1ccccc1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCOCC2)C(=O)N4C)cc1NS(=O)(=O)c1ccccc1
CN(C)CCCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(=O)(=O)c1ccccc1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4CC2COC2)cc1NS(=O)(=O)c1ccccc1
CCN1C(=O)C2(CC2)c2c1cnc1ccc(-c3cnc(OCCCN(C)C)c(NS(=O)(=O)c4ccccc4)c3)cc21
CNCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(=O)(=O)c1ccccc1
CC(C#N)c1cccc(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3)C3(CC3)C(=O)N5C)cnc2OCCCN(C)C)c1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(COC2)C(=O)N4C)cc1NS(=O)(=O)C1CC1
CN1C(=O)C2(CC2)c2c1cnc1ccc(-c3cnc(N)nc3)cc21
CN1CCN(c2ncc(-c3ccc4ncc5c(c4c3)C3(CC3)C(=O)N5C)cc2NS(=O)(=O)c2ccccc2)CC1
CN1CCCN(c2ncc(-c3ccc4ncc5c(c4c3)C3(CC3)C(=O)N5C)cc2NS(=O)(=O)c2ccccc2)CC1
COc1cc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cnc1OCCCN(C)C
CN(C)CCCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(=O)(=O)C1CC1
Cc1cc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cnc1OCCCN(C)C
CN1C(=O)C2(CC2)c2c1cnc1ccc(-c3cnc(OCCCN4CCCC4)c(NS(=O)(=O)c4ccccc4)c3)cc21
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1OCc1ccccc1
CN1C(=O)C2(CC2)c2c1cnc1ccc(-c3cnc(OCCCN4CCCC4)c(NS(=O)(=O)C4CC4)c3)cc21
CCS(=O)(=O)Nc1cc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cnc1OCCCN(C)C
CN1C(=O)C2(CC2)c2c1cnc1ccc(-c3cnc4ncccc4c3)cc21
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(=O)(=O)c1ccccc1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(C)(=O)=O
CN(C)CCCOc1ncc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CC2)cc1NS(=O)(=O)c1ccccc1
CN(C)CCCOc1ncc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CC2)cc1NS(=O)(=O)C1CC1
CN1C(=O)C2(CC2)c2c1cnc1ccc(-c3cnc(OCCCN4CCCCC4)c(NS(=O)(=O)c4ccccc4)c3)cc21
CN1C(=O)C2(CC2)c2c1cnc1ccc(-c3cnc(OCCCN4CCCCC4)c(NS(=O)(=O)C4CC4)c3)cc21
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(=O)(=O)C1CCC1
CN(C)CCCNc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cn1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cn1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)CC2(CCC2)C(=O)N4C)cc1NS(=O)(=O)c1ccccc1
CNCCCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(=O)(=O)c1ccccc1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(=O)(=O)C1COC1
CCCS(=O)(=O)Nc1cc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cnc1OCCCN(C)C
CN1C(=O)C2(CC2)c2c1cnc1ccc(-c3cnc(OCCC4CCCN4C)c(NS(=O)(=O)c4ccccc4)c3)cc21
CN1C(=O)C2(CC2)c2c1cnc1ccc(-c3cnc(OCCC4CCCN4C)c(NS(=O)(=O)C4CC4)c3)cc21
CN1C(=O)C2(CC2)c2c1cnc1ccc(-c3cnc(OCCC4CCCCN4C)c(NS(=O)(=O)C4CC4)c3)cc21
CN1C(=O)C2(CC2)c2c1cnc1ccc(-c3cnc(OCCC4CCCCN4C)c(NS(=O)(=O)c4ccccc4)c3)cc21
COc1cc2ncc3c(c2cc1-c1cnc(OCCCN(C)C)c(NS(=O)(=O)c2ccccc2)c1)C1(CC1)C(=O)N3C
COCCS(=O)(=O)Nc1cc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cnc1OCCCN(C)C
CN1CCCC(COc2ncc(-c3ccc4ncc5c(c4c3)C3(CC3)C(=O)N5C)cc2NS(=O)(=O)c2ccccc2)C1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(=O)(=O)c1cccnc1
CN1CCCC(COc2ncc(-c3ccc4ncc5c(c4c3)C3(CC3)C(=O)N5C)cc2NS(=O)(=O)C2CC2)C1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(=O)(=O)c1ccc(F)cc1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(=O)(=O)N1CCCC1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(=O)(=O)c1cccc(F)c1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(=O)(=O)c1cnn(C)c1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(=O)(=O)c1ccsc1
COc1ccc(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3)C3(CC3)C(=O)N5C)cnc2OCCCN(C)C)cc1
N#Cc1cccc(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3)C3(CC3)C(=O)N5C)cnc2OCCCN(C)C)c1
CN(C)CCCOc1c(F)cc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(=O)(=O)c1ccccc1
CN(C)CCCOc1ccc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(=O)(=O)c1cccc(Cl)c1
Cc1ccc(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3)C3(CC3)C(=O)N5C)cnc2OCCCN(C)C)cc1
CN1C(=O)C2(CC2)c2c1cnc1ccc(-c3cnc(OC4CC(N(C)C)C4)c(NS(=O)(=O)c4ccccc4)c3)cc21
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(=O)(=O)Cc1ccccc1
COc6cccc(S(=O)(=O)Nc5cc(c2ccc1ncc4c(c1c2)C3(CC3)C(=O)N4C)cnc5OCCCN(C)C)c6
CN(C)CCCOc5ncc(c2ccc1ncc4c(c1c2)C3(CC3)C(=O)N4C)cc5NS(=O)(=O)c6cccc(C(F)(F)F)c6
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(=O)(=O)c1ccccc1F
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(=O)(=O)c1ccc(C(F)(F)F)cc1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(=O)(=O)N(C)C
CN(C)CCCOc5ncc(c2ccc1ncc4c(c1c2)C3(CC3)C(=O)N4C)cc5NS(=O)(=O)c6ccc(F)c(C#N)c6
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(=O)(=O)c1ccn(C)n1
CN1C(=O)C2(CC2)c2c1cnc1ccc(-c3cnc(N4CCC(N(C)C)CC4)c(NS(=O)(=O)C4CC4)c3)cc21
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CN(c3ccccc3)C2)C(=O)N4C)cc1NS(=O)(=O)c1ccccc1
CN(C)CC1CCN(c2ncc(-c3ccc4ncc5c(c4c3)C3(CC3)C(=O)N5C)cc2NS(=O)(=O)C2CC2)CC1
CN(C)CCCOc5ncc(c2ccc1ncc4c(c1c2)C3(CC3)C(=O)N4C)cc5NS(=O)(=O)c6ccccc6OC(F)(F)F
CN1CCN(c2ncc(-c3cc4c5c(cnc4cc3F)N(C)C(=O)C53CC3)cc2NS(=O)(=O)c2ccccc2)CC1
CN1C(=O)C2(CC2)c2c1cnc1cc(F)c(-c3cnc(OCCCN4CCCCC4)c(NS(=O)(=O)c4ccccc4)c3)cc21
COc1ccc(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3)C3(CC3)C(=O)N5C)cnc2OCCCN2CCCCC2)cc1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(=O)(=O)c1cccs1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(=O)(=O)c1ccc(OC(F)(F)F)cc1
CN(C)CCCOc1ncc(-c2ccc3c(c2)c2c(c[n+]3[O-])N(C)C(=O)C23CC3)cc1NS(=O)(=O)c1ccccc1
CN1C(=O)C2(CC2)c2c1cnc1cc(F)c(-c3cnc(OCCCN4CCCC4)c(NS(=O)(=O)c4ccccc4)c3)cc21
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(=O)(=O)c1cc(Cl)cc(Cl)c1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(=O)(=O)c1ccc(OC(F)F)cc1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(=O)(=O)c1ccc(C(C)(C)C)cc1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cc1NS(=O)(=O)c1ccc(Cl)cc1
CN(C)CCCOc1ncc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CC2)cc1NS(=O)(=O)c1ccc(Cl)cc1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(=O)(=O)c1cncc(Cl)c1
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(OCCCN4CCOCC4)c(NS(=O)(=O)c4ccccc4)c3)cc21
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(OCCCN4CCCCC4)c(NS(=O)(=O)c4ccccc4)c3)cc21
COc1ccc(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cnc2OCCCN(C)C)cn1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(=O)(=O)c1ccc(S(F)(F)(F)(F)F)cc1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(=O)(=O)N1CCOCC1
Cc1ccc(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cnc2OCCCN(C)C)cn1
Cc1cncc(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cnc2OCCCN(C)C)c1
Cc1ccc(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cnc2OCCCN2CCCCC2)cn1
COc1ccc(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cnc2OCCCN(C)C)cc1
Cc1ccc(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cnc2OCCCN(C)C)cc1
Cc1ccc(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cnc2OCCCN(C)C)cn1
N#Cc1ccc(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cnc2OCCCN(C)C)cn1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(=O)(=O)c1ccccn1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(=O)(=O)N(C)C
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(=O)(=O)c1cccc(C(F)(F)F)c1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(=O)(=O)c1cc(F)cc(F)c1
Cc1cc(Cl)cc(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cnc2OCCCN(C)C)c1
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(N4CCC(N5CCCCC5)CC4)c(NS(=O)(=O)c4ccccc4)c3)cc21
Cc1cc(F)cc(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cnc2OCCCN(C)C)c1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(=O)(=O)c1cc(Cl)cc(Cl)c1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(=O)(=O)c1ccc(F)cc1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(=O)(=O)c1ccc(F)c(C#N)c1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(=O)(=O)c1cscn1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(=O)(=O)N1CCN(C)CC1
CCN(C)S(=O)(=O)Nc1cc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cnc1OCCCN(C)C
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(=O)(=O)N1CCC1
CC1CCN(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cnc2OCCCN(C)C)CC1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(=O)(=O)c1cnn(C)c1
Cc1ccc(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cnc2N2CCC(N3CCOCC3)CC2)cc1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(=O)(=O)c1ccccc1F
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(=O)(=O)c1cncs1
Cc1cc(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cnc2OCCCN(C)C)sn1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(=O)(=O)c1cc(F)cc(Cl)c1
CC1CCCN1S(=O)(=O)Nc1cc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cnc1OCCCN(C)C
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(N4CCC(N(C)C)CC4)c(NS(=O)(=O)C4CC4)c3)cc21
CC1CCCN(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cnc2OCCCN(C)C)C1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(=O)(=O)N1CCNCC1
Cc1ccc(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cnc2N2CCC(N(C)C)CC2)cc1
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(OCCCN4CCCCC4)c(NS(=O)(=O)N(C)C)c3)cc21
COCCC(CCOC)S(=O)(=O)Nc1cc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cnc1OCCCN(C)C
CCN(CC)S(=O)(=O)Nc1cc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cnc1OCCCN(C)C
CC1CN(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cnc2OCCCN(C)C)CC(C)O1
Cc1ccc(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cnc2N2CCC(N(C)C)CC2)cn1
Cc1ccc(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cnc2OCCCN(C)C)cc1
COC1CCN(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cnc2OCCCN(C)C)CC1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(=O)(=O)c1ccns1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(C)(=O)=O
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(=O)(=O)C1CC1
Cc1ccc(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cnc2N2CCC(N3CCCCC3)CC2)nc1
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(OCCCN4CCCCC4)c(NS(=O)(=O)c4cscn4)c3)cc21
Cc1cc(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cnc2OCCCN2CCCCC2)sn1
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(OCCCN4CCCCC4)c(NS(=O)(=O)c4ccccc4F)c3)cc21
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(OCCCN4CCCCC4)c(NS(=O)(=O)c4cc(F)cc(Cl)c4)c3)cc21
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(OCCCN4CCCCC4)c(NS(=O)(=O)C4CC4)c3)cc21
Cc1ccc(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cnc2N2CCC(N3CCCCC3)CC2)cn1
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(OCCCN4CCCCC4)c(NS(=O)(=O)c4cncs4)c3)cc21
CN1CCN(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cnc2OCCCN2CCCCC2)CC1
Cc1ccc(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cnc2N2CCN(C)CC2)cn1
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(OCCCN4CCCCC4)c(NS(=O)(=O)N4CCNCC4)c3)cc21
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(N4CCC(N5CCCCC5)CC4)c(NS(=O)(=O)c4ccccc4F)c3)cc21
Cc1ccc(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3F)C3(CCC3)C(=O)N5C)cnc2OCCCN(C)C)cc1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(=O)(=O)C1COC1
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(N4CCC(N5CCCCC5)CC4)c(NS(=O)(=O)c4ccc(F)cc4F)c3)cc21
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(N4CCC(N5CCCCC5)CC4)c(NS(=O)(=O)C4CC4)c3)cc21
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(N4CCC(N5CCCCC5)CC4)c(NS(=O)(=O)N(C)C)c3)cc21
CCN(C)S(=O)(=O)Nc1cc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cnc1N1CCC(N2CCCCC2)CC1
CN1C(=O)C2(CC2)c2c1cnc1ccc(-c3cnc(N4CCC(N5CCCCC5)CC4)c(NS(=O)(=O)c4ccccc4)c3)cc21
CCN(C)S(=O)(=O)Nc1cc(-c2ccc3ncc4c(c3c2)C2(CC2)C(=O)N4C)cnc1N1CCC(N2CCCCC2)CC1
Cc1ccc(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3F)C3(CC3)C(=O)N5C)cnc2OCCCN(C)C)cc1
Cc1ccc(S(=O)(=O)n2c(CCN3CCCCC3)cc3ncc(-c4ccc5ncc6c(c5c4)C4(CCC4)C(=O)N6C)cc32)cn1
Cc1ccc(S(=O)(=O)Nc2cc(-c3cc4c5c(cnc4cc3F)N(C)C(=O)C53CCC3)cnc2OCCCN2CCCCC2)cn1
Cc1ccc(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3)C3(CC3)C(=O)N5C)cnc2N2CCC(N3CCCCC3)CC2)cn1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(=O)(=O)c1ccc(O)cc1
[2H]C1([2H])N(CCCOc2ncc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cc2NS(=O)(=O)c2ccc(C)nc2)C([2H])([2H])C([2H])([2H])C([2H])([2H])C1([2H])[2H]
CCN(C)S(=O)(=O)Nc1cc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cnc1OCCCN1CCCCC1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(=O)(=O)CCN1C(=O)c2ccccc2C1=O
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(N4CCC(N(C)C)CC4)c(NS(C)(=O)=O)c3)cc21
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(OCCCN4CCCCC4)c(NS(C)(=O)=O)c3)cc21
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(N4CCC(N(C)C)CC4)c(NS(=O)(=O)N(C)C)c3)cc21
CN1CCN(c2ncc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cc2NS(=O)(=O)C2CC2)CC1
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(N4CCC(N5CCCCC5)CC4)c(NS(C)(=O)=O)c3)cc21
CN1CCN(c2ncc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cc2NS(C)(=O)=O)CC1
CN1CCN(c2ncc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cc2NS(=O)(=O)N(C)C)CC1
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(OCCCN4CCCC4)c(NS(=O)(=O)c4ccccc4)c3)cc21
Cc1cc(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cnc2N2CCC(N(C)C)CC2)sn1
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(OCCCN4CCCC4)c(NS(=O)(=O)C4CC4)c3)cc21
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(OCCCN4CCCC4)c(NS(C)(=O)=O)c3)cc21
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4)cc1NS(C)(=O)=O
CCS(=O)(=O)Nc1cc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cnc1OCCCN(C)C
CN(C)CCCOc5ncc(c2ccc1ncc4c(c1c2)C3(CCC3)C(=O)N4C)cc5NS(=O)(=O)C(F)(F)F
CNCCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(C)(=O)=O
CCCS(=O)(=O)Nc1cc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cnc1OCCCN(C)C
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(OCCCN4CCCC4)c(NS(=O)(=O)N(C)C)c3)cc21
CN1CCN(c2ncc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cc2NS(=O)(=O)c2ccccc2)CC1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(=O)(=O)N1CCCC1
CCc1ncc(s1)S(=O)(=O)Nc1cc(cnc1OCCCN(C)C)-c1ccc2ncc3N(C)C(=O)C4(CCC4)c3c2c1
Cc1cc(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cnc2N2CCN(C)CC2)sn1
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(=O)(=O)C(F)F
CCNCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(C)(=O)=O
CNCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(C)(=O)=O
CNCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(=O)(=O)c1ccccc1
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(N4CCC(N5CCCC(F)(F)C5)CC4)c(NS(C)(=O)=O)c3)cc21
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(OCCCN4CCCCC4)c(NS(=O)(=O)c4cccnc4)c3)cc21
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(=O)(=O)C1CCC1
CC(C)NCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCCC2)C2=NCCN24)cc1NS(C)(=O)=O
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CC(F)C2)C(=O)N4C)cc1NS(C)(=O)=O
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(=O)(=O)CCN1C(=O)c2ccccc2C1=O
COCCS(=O)(=O)Nc1cc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cnc1OCCCN(C)C
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2F)C2(CCC2)C(=O)N4C)cc1NS(C)(=O)=O
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(OCCCN4CCCC(O)C4)c(NS(C)(=O)=O)c3)cc21
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(=O)(=O)c1ccsc1
CN(C)CCOCc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(=O)(=O)CC#N
CN1CC=C(c2ncc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cc2NS(C)(=O)=O)CC1
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(N4CC(N5CCCC5)C4)c(NS(C)(=O)=O)c3)cc21
COCCN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(C)(=O)=O
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(OCCCN4CCC(F)C4)c(NS(C)(=O)=O)c3)cc21
COC1CCCN(CCCOc2ncc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cc2NS(C)(=O)=O)C1
CC(C)NCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(C)(=O)=O
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(OCCCN4CCCC(F)C4)c(NS(C)(=O)=O)c3)cc21
COC1CCN(CCCOc2ncc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cc2NS(C)(=O)=O)C1
CN1CC=C(c2ncc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cc2NS(C)(=O)=O)CC1
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(OCCCN4CCC(F)CC4)c(NS(C)(=O)=O)c3)cc21
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(OCC(O)CN4CCCCC4)c(NS(C)(=O)=O)c3)cc21
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(N4CC(N(C)C)C4)c(NS(=O)(=O)N(C)C)c3)cc21
Cc1ncc(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cnc2OCCCN(C)C)s1
CN(C)CCCOc1ncc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CCC2)cc1NS(=O)(=O)N(C)C
CN(C)CCCOc1ncc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CCC2)cc1NS(C)(=O)=O
CN(CCC#N)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cc1NS(C)(=O)=O
COCCN(C)CCCOc1ncc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CCC2)cc1NS(=O)(=O)N1CCOCC1
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(OCC(CO)N(C)C)c(NS(C)(=O)=O)c3)cc21
CN1C(=O)C2(CCC2)c2c1cnc1cc(F)c(-c3cnc(OCCCN4CCC(F)CC4)c(NS(C)(=O)=O)c3)cc21
CN1CCN(CCCOc2ncc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cc2NS(C)(=O)=O)CC1
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(OCCCN4CCCCC4)c(NS(=O)(=O)C(F)F)c3)cc21
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(OCCCN4CCOCC4)c(NS(=O)(=O)N(C)C)c3)cc21
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(OCCCN4CCOCC4)c(NS(C)(=O)=O)c3)cc21
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(OCCCN4CCOCC4)c(NS(=O)(=O)C4CC4)c3)cc21
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(OCCNC(C)(C)C)c(NS(C)(=O)=O)c3)cc21
COC1CN(S(=O)(=O)Nc2cc(-c3cc4c5c(cnc4cc3F)N(C)C(=O)C53CCC3)cnc2N2CC(N(C)C)C2)C1
CN1C(=O)C2(CCC2)c2c1cnc1cc(F)c(-c3cnc(N4CC(N(C)C)C4)c(NS(=O)(=O)c4ccc(F)cc4F)c3)cc21
CN1C(=O)C2(CCC2)c2c1cnc1cc(F)c(-c3cnc(N4CC(N(C)C)C4)c(NS(=O)(=O)N(C)C)c3)cc21
CN1C(=O)C2(CCC2)c2c1cnc1cc(F)c(-c3cnc(N4CC(N(C)C)C4)c(NS(C)(=O)=O)c3)cc21
CCS(=O)(=O)Nc1cc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cnc1N1CC(N(C)C)C1
CN1C(=O)C2(CCC2)c2c1cnc1cc(F)c(-c3cnc(N4CC(N(C)C)C4)c(NS(=O)(=O)C4CC4)c3)cc21
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(N4CC(N(C)C)C4)c(NS(=O)(=O)C4CC4)c3)cc21
Cc1ccc(S(=O)(=O)Nc2cc(-c3cc4c5c(cnc4cc3F)N(C)C(=O)C53CCC3)cnc2N2CC(N(C)C)C2)cc1
CN1C(=O)C2(CCC2)c2c1cnc1cc(F)c(-c3cnc(N4CC(N(C)C)C4)c(NS(=O)(=O)c4ccccc4)c3)cc21
CC1CCC12C(=O)N(C)c1cnc3ccc(-c4cnc(N5CC(N(C)C)C5)c(NS(C)(=O)=O)c4)cc3c12
CCN(C)C1CN(c2ncc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cc2NS(C)(=O)=O)C1
CNC1CN(c2ncc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cc2NS(C)(=O)=O)C1
CNC1CN(c2ncc(-c3cc4c5c(cnc4cc3F)N(C)C(=O)C53CCC3)cc2NS(C)(=O)=O)C1
CCNC1CN(c2ncc(-c3cc4c5c(cnc4cc3F)N(C)C(=O)C53CCC3)cc2NS(C)(=O)=O)C1
CNC1CN(c2ncc(-c3cc4c5c(cnc4cc3F)N(C)C(=O)C53CCC3)cc2NS(=O)(=O)N(C)C)C1
CNC1CN(c2ncc(-c3cc4c5c(cnc4cc3F)N(C)C(=O)C53CCC3)cc2NS(=O)(=O)C2CC2)C1
CCS(=O)(=O)Nc1cc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CCC2)cnc1N1CC(NC)C1
Cc1ncc(S(=O)(=O)Nc2cc(-c3ccc4ncc5c(c4c3)C3(CCC3)C(=O)N5C)cnc2N2CC(N(C)C)C2)s1
CCN(C)S(=O)(=O)Nc1cc(-c2ccc3ncc4c(c3c2)C2(CCC2)C(=O)N4C)cnc1N1CC(N(C)C)C1
CCS(=O)(=O)Nc1cc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CCC2)cnc1N1CC(N(C)C)C1
CN1CC2CN(c3ncc(-c4ccc5ncc6c(c5c4)C4(CCC4)C(=O)N6C)cc3NS(C)(=O)=O)CC2C1
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(N4CCC(N(C)C)C4)c(NS(C)(=O)=O)c3)cc21
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(N4CCC(N5CCCCC5)C4)c(NS(C)(=O)=O)c3)cc21
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(N4CCC(N5CCOCC5)CC4)c(NS(=O)(=O)N(C)C)c3)cc21
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(N4CCC(N5CCOCC5)CC4)c(NS(=O)(=O)C4CC4)c3)cc21
CN1C(=O)C2(CCC2)c2c1cnc1ccc(-c3cnc(N4CCC(N5CCOCC5)CC4)c(NS(C)(=O)=O)c3)cc21
CN1C(=O)C2(CCC2)c2c1cnc1cc(F)c(-c3cnc(N4CCC(N5CCCCC5)CC4)c(NS(C)(=O)=O)c3)cc21
CC(C)NCCN(C)c1ncc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CCC2)cc1NS(=O)(=O)C1CC1
CC(C)NCCOc1ncc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CCC2)cc1NS(=O)(=O)C(C)(C)C
CC(C)NCCOc1ncc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CCC2)cc1NS(=O)(=O)C1(C)CC1
CC(C)NCCOc1ncc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CCC2)cc1NS(=O)(=O)N(C)C
CC(C)NCCOc1ncc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CCC2)cc1NS(=O)(=O)N1CCC1
CC(C)NCCOc1ncc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CCC2)cc1NS(=O)(=O)N1CC(F)C1
CC(C)NCCOc1ncc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CCC2)cc1NS(=O)(=O)N1CCOCC1
CC(C)NCCOc1ncc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CCC2)cc1NS(=O)(=O)CCN(C)C
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)[C@]2(C[C@@H](O)C2)C(=O)N4C)cc1NS(C)(=O)=O
CO[C@H]1C[C@@]2(C1)C(=O)N(C)c1cnc3ccc(-c4cnc(OCCNC(C)C)c(NS(C)(=O)=O)c4)cc3c12
CO[C@H]1C[C@]2(C1)C(=O)N(C)c1cnc3cc(F)c(-c4cnc(OCCNC(C)C)c(NS(C)(=O)=O)c4)cc3c12
CO[C@H]1C[C@]2(C1)C(=O)N(C)c1cnc3cc(F)c(-c4cnc(OCCNC(C)C)c(NS(=O)(=O)C5CC5)c4)cc3c12
CO[C@H]1C[C@@]2(C1)C(=O)N(C)c1cnc3cc(F)c(-c4cnc(OCCNC(C)C)c(NS(=O)(=O)C5CC5)c4)cc3c12
CO[C@H]1C[C@]2(C1)C(=O)N(C)c1cnc3cc(F)c(-c4cnc(OCCNC(C)C)c(NS(=O)(=O)N(C)C)c4)cc3c12
CO[C@H]1C[C@@]2(C1)C(=O)N(C)c1cnc3cc(F)c(-c4cnc(OCCNC(C)C)c(NS(=O)(=O)N(C)C)c4)cc3c12
CO[C@H]1C[C@]2(C1)C(=O)N(C)c1cnc3cc(F)c(-c4cnc(N5CCC(N6CCCCC6)CC5)c(NS(C)(=O)=O)c4)cc3c12
CO[C@H]1C[C@@]2(C1)C(=O)N(C)c1cnc3cc(F)c(-c4cnc(N5CCC(N6CCCCC6)CC5)c(NS(C)(=O)=O)c4)cc3c12
CCO[C@H]1C[C@]2(C1)C(=O)N(C)c1cnc3cc(F)c(-c4cnc(OCCNC(C)C)c(NS(C)(=O)=O)c4)cc3c12
CC(C)NCCOc1ncc(-c2cc3c(cc2F)ncc2c3[C@]3(C[C@H](OC(C)C)C3)C(=O)N2C)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c(cc2F)ncc2c3[C@]3(C[C@H](OC(C)c4ccccc4)C3)C(=O)N2C)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c(cc2F)ncc2c3[C@]3(C[C@H](Oc4ccccc4)C3)C(=O)N2C)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c(cc2F)ncc2c3[C@]3(C[C@H](Oc4ccccc4)C3)C(=O)N2C)cc1NS(=O)(=O)N(C)C
CCO[C@H]1C[C@]2(C1)C(=O)N(C)c1cnc3cc(F)c(-c4cnc(OCCNC(C)C)c(NS(C)(=O)=O)c4)cc3c12
CCCO[C@H]1C[C@]2(C1)C(=O)N(C)c1cnc3cc(F)c(-c4cnc(OCCNC(C)C)c(NS(C)(=O)=O)c4)cc3c12
CC(C)NCCOc1ncc(-c2cc3c(cc2F)ncc2c3[C@]3(C[C@H](COc4ccccc4)C3)C(=O)N2C)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c(cc2F)ncc2c3[C@]3(C[C@H](COC(C)C)C3)C(=O)N2C)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c(cc2F)ncc2c3[C@]3(C[C@H](COC(C)C)C3)C(=O)N2C)cc1NS(=O)(=O)C(C)C
CC(C)NCCOc1ncc(-c2cc3c(cc2F)ncc2c3[C@]3(C[C@H](c4ccccc4)C3)C(=O)N2C)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c(cc2F)ncc2c3[C@]3(C[C@@H](c4ccccc4)C3)C(=O)N2C)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c(cc2F)ncc2c3[C@]3(C[C@H](c4ccc(Cl)cc4)C3)C(=O)N2C)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c(cc2F)ncc2c3[C@]3(C[C@@H](c4ccc(Cl)cc4)C3)C(=O)N2C)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c(cc2F)ncc2c3[C@]3(C[C@H](c4cccc(Cl)c4)C3)C(=O)N2C)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c(cc2F)ncc2c3[C@]3(C[C@@H](c4cccc(Cl)c4)C3)C(=O)N2C)cc1NS(C)(=O)=O
COc1ccc([C@H]2C[C@]3(C2)C(=O)N(C)c2cnc4cc(F)c(-c5cnc(OCCNC(C)C)c(NS(C)(=O)=O)c5)cc4c23)cc1
COc1ccc([C@H]2C[C@@]3(C2)C(=O)N(C)c2cnc4cc(F)c(-c5cnc(OCCNC(C)C)c(NS(C)(=O)=O)c5)cc4c23)cc1
CC(C)NCCOc1ncc(-c2cc3c(cc2F)ncc2c3[C@]3(C[C@@H](c4ccc(F)cc4)C3)C(=O)N2C)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c(cc2F)ncc2c3[C@]3(C[C@H](c4ccc(F)cc4)C3)C(=O)N2C)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c(cc2F)ncc2c3[C@]3(C[C@@H](c4cccc(F)c4)C3)C(=O)N2C)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c(cc2F)ncc2c3[C@]3(C[C@H](c4ccccc4F)C3)C(=O)N2C)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c(cc2F)ncc2c3[C@]3(C[C@@H](c4ccccc4F)C3)C(=O)N2C)cc1NS(C)(=O)=O
COc1cccc([C@H]2C[C@]3(C2)C(=O)N(C)c2cnc4cc(F)c(-c5cnc(OCCNC(C)C)c(NS(C)(=O)=O)c5)cc4c23)n1
COc1cccc([C@H]2C[C@@]3(C2)C(=O)N(C)c2cnc4cc(F)c(-c5cnc(OCCNC(C)C)c(NS(C)(=O)=O)c5)cc4c23)n1
COc1ccc([C@H]2C[C@]3(C2)C(=O)N(C)c2cnc4cc(F)c(-c5cnc(OCCNC(C)C)c(NS(C)(=O)=O)c5)cc4c23)cn1
COc1ccc([C@H]2C[C@@]3(C2)C(=O)N(C)c2cnc4cc(F)c(-c5cnc(OCCNC(C)C)c(NS(C)(=O)=O)c5)cc4c23)cn1
COc1cc([C@H]2C[C@]3(C2)C(=O)N(C)c2cnc4cc(F)c(-c5cnc(OCCNC(C)C)c(NS(C)(=O)=O)c5)cc4c23)ccn1
COc1cc([C@H]2C[C@@]3(C2)C(=O)N(C)c2cnc4cc(F)c(-c5cnc(OCCNC(C)C)c(NS(C)(=O)=O)c5)cc4c23)ccn1
CC(C)NCCOc1ncc(-c2cc3c(cc2F)ncc2c3[C@]3(C[C@H](c4ccccn4)C3)C(=O)N2C)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c(cc2F)ncc2c3[C@]3(C[C@@H](c4ccccn4)C3)C(=O)N2C)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c(cc2F)ncc2c3[C@]3(C[C@H](c4cccnc4)C3)C(=O)N2C)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c(cc2F)ncc2c3[C@]3(C[C@@H](c4cccnc4)C3)C(=O)N2C)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c(cc2F)ncc2c3[C@]3(C[C@H](c4ccncc4)C3)C(=O)N2C)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c(cc2F)ncc2c3[C@]3(C[C@@H](c4ccncc4)C3)C(=O)N2C)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c(cc2F)ncc2c3[C@]3(C[C@H](c4cccc(=O)[nH]4)C3)C(=O)N2C)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CC(C)(C)C2)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c(cc2F)ncc2c3[C@]3(C[C@H](C)C3)C(=O)N2C)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c(cc2F)ncc2c3[C@]3(C[C@H](Cc4ccccc4)C3)C(=O)N2C)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c(cc2F)ncc2c3[C@]3(C[C@H](C(C)(C)O)C3)C(=O)N2C)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c(cc2F)ncc2c3[C@]3(C[C@H](Nc4ccccc4)C3)C(=O)N2C)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c(cc2F)ncc2c3[C@]3(C[C@@H](Nc4ccccc4)C3)C(=O)N2C)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c(cc2F)ncc2c3[C@]3(C[C@H](Nc4ccc(Cl)cc4)C3)C(=O)N2C)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c(cc2F)ncc2c3[C@]3(C[C@H](N(C)c4ccccc4)C3)C(=O)N2C)cc1NS(C)(=O)=O
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CN(C)C2)C(=O)N4C)cc1NS(C)(=O)=O
CCS(=O)(=O)Nc1cc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CN(C(C)C)C2)cnc1OCCNC(C)C
CC(C)NCCOc1ncc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CN(C(C)C)C2)cc1NS(=O)(=O)C1CC1
CC(C)NCCOc1ncc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CN(C(C)C)C2)cc1NS(=O)(=O)C(C)C
CC(C)N1CC2(C1)C(=O)N(C)c1cnc3cc(F)c(-c4cnc(N5CCC(N6CCCCC6)CC5)c(NS(C)(=O)=O)c4)cc3c12
CC(C)NCCOc1ncc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CN(C3CCC3)C2)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CN(C3CCCC3)C2)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CN(c3ccccc3)C2)cc1NS(C)(=O)=O
Cc1ncc(S(=O)(=O)Nc2cc(-c3cc4c5c(cnc4cc3F)N(C)C(=O)C53CN(c4ccccc4)C3)cnc2OCCNC(C)C)s1
CCS(=O)(=O)Nc1cc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CN(c3ccccc3)C2)cnc1OCCNC(C)C
CC(C)NCCOc1ncc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CN(c3ccc(Cl)cc3)C2)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CN(c3cccc(Cl)c3)C2)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CN(c3ccccc3Cl)C2)cc1NS(C)(=O)=O
Cc1ccc(N2CC3(C2)C(=O)N(C)c2cnc4cc(F)c(-c5cnc(OCCNC(C)C)c(NS(C)(=O)=O)c5)cc4c23)cc1
Cc1cccc(N2CC3(C2)C(=O)N(C)c2cnc4cc(F)c(-c5cnc(OCCNC(C)C)c(NS(C)(=O)=O)c5)cc4c23)c1
Cc1ccccc1N1CC2(C1)C(=O)N(C)c1cnc3cc(F)c(-c4cnc(OCCNC(C)C)c(NS(C)(=O)=O)c4)cc3c12
CCc1ccc(N2CC3(C2)C(=O)N(C)c2cnc4cc(F)c(-c5cnc(OCCNC(C)C)c(NS(C)(=O)=O)c5)cc4c23)cc1
CC(C)NCCOc1ncc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CN(c3ccc(C(C)C)cc3)C2)cc1NS(C)(=O)=O
COCc1ccc(N2CC3(C2)C(=O)N(C)c2cnc4cc(F)c(-c5cnc(OCCNC(C)C)c(NS(C)(=O)=O)c5)cc4c23)cc1
COc1ccc(N2CC3(C2)C(=O)N(C)c2cnc4cc(F)c(-c5cnc(OCCNC(C)C)c(NS(C)(=O)=O)c5)cc4c23)cc1
COc1ccccc1N1CC2(C1)C(=O)N(C)c1cnc3cc(F)c(-c4cnc(OCCNC(C)C)c(NS(C)(=O)=O)c4)cc3c12
Cc1ccc(N2CC3(C2)C(=O)N(C)c2cnc4cc(F)c(-c5cnc(OCCNC(C)C)c(NS(C)(=O)=O)c5)cc4c23)cc1
CC(C)NCCOc1ncc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CN(c3ccc(F)cc3)C2)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CN(c3cccc(F)c3)C2)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CN(c3ccccc3F)C2)cc1NS(C)(=O)=O
CC(C)NCCOc6ncc(c2cc1c3c(cnc1cc2F)N(C)C(=O)C35CN(c4ccc(OC(F)(F)F)cc4)C5)cc6NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CN(c3ccc(-c4ccccc4)cc3)C2)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CN(c3ccc4c(c3)OCO4)C2)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2cc3c4c(cnc3cc2F)N(C)C(=O)C42CN(c3ccc4c(c3)OCCO4)C2)cc1NS(C)(=O)=O
CN(C)CCCOc1ncc(-c2ccc3ncc4c(c3c2)C2(CC(F)(F)C2)C(=O)N4C)cc1NS(C)(=O)=O
CC(C)NCCOc1ncc(-c2ccc3ncc4c(c3c2F)C2(CCC2)C(=O)N4C)cc1NS(C)(=O)=O
Cc1nn(-c2cccnc2)c(C)c1-c1cc(N2CC3CCC(C2)O3)nc2c(-c3ccn[nH]3)cnn12
Cc1nn(-c2cccnc2)c(C)c1-c1cc([C@]23CCOC[C@H]2C3)nc2c(-c3ccn[nH]3)cnn12
Cn1c(=O)cnc2cc(N3CCOCC3)cc(O[C@H]3CC[C@@H](Nc4ncccn4)CC3)c21
Cn1c(=O)cnc2cc(N3CCOCC3)cc(O[C@H]3CC[C@@H](Oc4ncccn4)CC3)c21
Cc1nccc(O[C@H]2CC[C@@H](Oc3cc(N4CCOCC4)cc4ncc(=O)n(C)c34)CC2)n1
COc1cnc(O[C@H]2CC[C@@H](Oc3cc(N4CCOCC4)cc4ncc(=O)n(C)c34)CC2)nc1
COc1cnc(N[C@H]2CC[C@@H](Oc3cc(N4CCOCC4)cc4ncc(=O)n(C)c34)CC2)nc1
Cc1cnc(O[C@H]2CC[C@@H](Oc3cc(N4CCOCC4)cc4ncc(=O)n(C)c34)CC2)nc1
Cc1nc2cc(N3CCOCC3)cc(O[C@H]3CC[C@@H](Nc4ncccn4)CC3)c2n(C)c1=O
CCn1c(=O)cnc2cc(N3CCOCC3)cc(O[C@H]3CC[C@@H](Nc4ncccn4)CC3)c21
Cn1c(=O)cnc2cc(Br)cc(O[C@H]3CC[C@@H](Nc4ncccn4)CC3)c21
Cn1c(=O)cnc2cc(N3CCOCC3)cc(O[C@H]3CC[C@@H](NC(=O)OC(C)(C)C)CC3)c21
Cc1cnc(N[C@H]2CC[C@@H](Oc3cc(N4CCOCC4)cc4ncc(=O)n(C)c34)CC2)nc1
Cc1nccc(N[C@H]2CC[C@@H](Oc3cc(N4CCOCC4)cc4ncc(=O)n(C)c34)CC2)n1
CCc1ncnc(N[C@H]2CC[C@@H](Oc3cc(N4CCOCC4)cc4ncc(=O)n(C)c34)CC2)c1F
Cn1c(=O)cnc2cc(N3CCOCC3)cc(O[C@H]3CC[C@@H](NC(=O)OCc4ccccc4)CC3)c21
CNC(=O)c1ccnc(N[C@H]2CC[C@@H](Oc3cc(N4CCOCC4)cc4ncc(=O)n(C)c34)CC2)n1
COC(=O)N[C@H]1CC[C@@H](Oc2cc(N3CCOCC3)cc3ncc(=O)n(C)c23)CC1
CCOC(=O)N[C@H]1CC[C@@H](Oc2cc(N3CCOCC3)cc3ncc(=O)n(C)c23)CC1
COc1cnc(O[C@H]2CC[C@@H](Oc3cc(N4CC5CC(C4)O5)cc4ncc(=O)n(C)c34)CC2)nc1
Cc1cnc(O[C@H]2CC[C@@H](Oc3cc(N4CC5CC(C4)O5)cc4ncc(=O)n(C)c34)CC2)nc1
Cc1nccc(O[C@H]2CC[C@@H](Oc3cc(N4CC5CC(C4)O5)cc4ncc(=O)n(C)c34)CC2)n1
Cc1nc2c(c(N[C@H]3CC[C@@H](Oc4cc(N5CCOCC5)cc5ncc(=O)n(C)c45)CC3)n1)OCC2
Cc1nccc(O[C@H]2CC[C@@H](Oc3cc(C4=CCOCC4)cc4ncc(=O)n(C)c34)CC2)n1
Cc1cnc(O[C@H]2CC[C@@H](Oc3cc(C4=CCOCC4)cc4ncc(=O)n(C)c34)CC2)nc1
COc1cnc(O[C@H]2CC[C@@H](Oc3cc(C4=CCOCC4)cc4ncc(=O)n(C)c34)CC2)nc1
Cc1nccc(N[C@H]2CC[C@@H](Oc3cc(C4=CCOCC4)cc4ncc(=O)n(C)c34)CC2)n1
Cc1cnc(N[C@H]2CC[C@@H](Oc3cc(C4=CCOCC4)cc4ncc(=O)n(C)c34)CC2)nc1
COc1cnc(N[C@H]2CC[C@@H](Oc3cc(C4=CCOCC4)cc4ncc(=O)n(C)c34)CC2)nc1
CCc1ncnc(N[C@H]2CC[C@@H](Oc3cc(C4=CCOCC4)cc4ncc(=O)n(C)c34)CC2)c1F
Cn1c(=O)cnc2cc(N3CC4CC(C3)O4)cc(O[C@H]3CC[C@@H](Nc4ncccn4)CC3)c21
Cn1c(=O)cnc2cc(C3=CCOCC3)cc(O[C@H]3CC[C@@H](Nc4ncccn4)CC3)c21
Cn1c(=O)cnc2cc(N3CC4CCC(C3)O4)cc(O[C@H]3CC[C@@H](Nc4ncccn4)CC3)c21
Cn1c(=O)cnc2cc(N3CC4CC(C3)O4)cc(O[C@H]3CC[C@@H](Oc4ncccn4)CC3)c21
Cn1c(=O)cnc2cc(C3=CCOCC3)cc(O[C@H]3CC[C@@H](Oc4ncccn4)CC3)c21
Cn1c(=O)cnc2cc(N3CC4CCC(C3)O4)cc(O[C@H]3CC[C@@H](Oc4ncccn4)CC3)c21
COc1cnc(O[C@H]2CC[C@@H](Oc3cc(N4CC5CCC(C4)O5)cc4ncc(=O)n(C)c34)CC2)nc1
Cc1cnc(O[C@H]2CC[C@@H](Oc3cc(N4CC5CCC(C4)O5)cc4ncc(=O)n(C)c34)CC2)nc1
Cc1nccc(O[C@H]2CC[C@@H](Oc3cc(N4CC5CCC(C4)O5)cc4ncc(=O)n(C)c34)CC2)n1
N=NCc1[nH]c(=O)c(cc1-c1ccncc1)C#N
COc1ccc(COCc2[nH]c(=O)c(cc2-c2ccncc2)C#N)cc1
O=c1cc(oc2c(cccc12)-c1ccccc1)N1CCOCC1
OCc1[nH]c(=O)c(cc1-c1cc[nH+]cc1)C#N
CO[C@H]1C[C@H](C)Cc2c(O)c(NC(=O)C(C)=CC=C[C@H](OC)[C@@H](OC(N)=O)\C(C)=C\[C@H](C)[C@H]1O)cc(O)c2N=CC#Cc1cccc2c1oc(cc2=O)N1CCOCC1 |w:39.41,16.16,t:28|
CO[C@H]1C[C@H](C)Cc2c(O)c(NC(=O)C(C)=CC=C[C@H](OC)[C@@H](OC(N)=O)\C(C)=C\[C@H](C)[C@H]1O)cc(O)c2N=CCCC#Cc1cccc2c1oc(cc2=O)N1CCOCC1 |w:16.16,39.41,t:28|
O=c1cc(oc2ccccc12)N1CCOCC1
CO[C@H]1C[C@H](C)Cc2c(O)c(NC(=O)C(C)=CC=C[C@H](OC)[C@@H](OC(N)=O)\C(C)=C\[C@H](C)[C@H]1O)cc(O)c2N=CCOCCOc1ccc2c(oc(cc2=O)N2CCOCC2)c1C |w:16.16,39.41,t:28|
CO[C@H]1C[C@H](C)Cc2c(O)c(NC(=O)C(C)=CC=C[C@H](OC)[C@@H](OC(N)=O)\C(C)=C\[C@H](C)[C@H]1O)cc(O)c2N=CCCCOc1ccc2c(c1)oc(cc2=O)N1CCOCC1 |w:16.16,39.41,t:28|
CO[C@H]1C[C@H](C)Cc2c(O)c(NC(=O)C(C)=CC=C[C@H](OC)[C@@H](OC(N)=O)\C(C)=C\[C@H](C)[C@H]1O)cc(O)c2N=CCCOc1ccc2c(c1)oc(cc2=O)N1CCOCC1 |w:16.16,39.41,t:28|
COC[C@H]1OC(=O)c2coc3c2[C@@]1(C)C1=C(C2CCC(=O)[C@@]2(C)C[C@H]1C(=O)OC)C3=O |t:16|
CO[C@H]1C[C@H](C)Cc2c(O)c(NC(=O)C(C)=CC=C[C@H](OC)[C@@H](OC(N)=O)\C(C)=C\[C@H](C)[C@H]1O)cc(O)c2N=CCCCCCCOc1ccc2c(oc(cc2=O)N2CCOCC2)c1C |w:16.16,39.41,t:28|
CO[C@H]1C[C@H](C)Cc2c(O)c(NC(=O)C(C)=CC=C[C@H](OC)[C@@H](OC(N)=O)\C(C)=C\[C@H](C)[C@H]1O)cc(O)c2N=CCOCCOc1ccc2c(c1)oc(cc2=O)N1CCOCC1 |w:16.16,39.41,t:28|
CO[C@H]1C[C@H](C)Cc2c(O)c(NC(=O)C(C)=CC=C[C@H](OC)[C@@H](OC(N)=O)\C(C)=C\[C@H](C)[C@H]1O)cc(O)c2N=CCCCCCCCOc1ccc2c(oc(cc2=O)N2CCOCC2)c1C |w:16.16,39.41,t:28|
CO[C@H]1C[C@H](C)Cc2c(O)c(NC(=O)C(C)=CC=C[C@H](OC)[C@@H](OC(N)=O)\C(C)=C\[C@H](C)[C@H]1O)cc(O)c2N=CCCCCOc1ccc2c(c1)oc(cc2=O)N1CCOCC1 |w:16.16,39.41,t:28|
CO[C@H]1C[C@H](C)Cc2c(O)c(NC(=O)C(C)=CC=C[C@H](OC)[C@@H](OC(N)=O)\C(C)=C\[C@H](C)[C@H]1O)cc(O)c2N=CCCCCCOc1ccc2c(c1)oc(cc2=O)N1CCOCC1 |w:16.16,39.41,t:28|
CO[C@H]1C[C@H](C)Cc2c(O)c(NC(=O)C(C)=CC=C[C@H](OC)[C@@H](OC(N)=O)\C(C)=C\[C@H](C)[C@H]1O)cc(O)c2N=CC=C |r,w:16.16,38.39,t:28|
COc1ccc(cc1)-c1cc(=O)cc(o1)N1CCOCC1
CC(C)(C)c1ccc(cc1)-c1cc(=O)cc(o1)N1CCOCC1
COc1cccc(c1)-c1cc(=O)cc(o1)N1CCOCC1
COC(=O)\C=C\c1ccccc1-c1cccc(c1)-c1cc(=O)cc(s1)N1CCOCC1
O=c1cc(sc(c1)-c1ccccc1)N1CCOCC1
Cc1ccc(-c2ccc(cc2)-c2cc(=O)cc(s2)N2CCOCC2)c2ccccc12
O=c1cc(oc2c3ccccc3ccc12)N1CCOCC1
Oc1ccc(cc1)-c1cccc(c1)-c1cc(=O)cc(s1)N1CCOCC1
COc1ccccc1-c1cc(=O)cc(o1)N1CCOCC1
Fc1cccc(c1)-c1cc(=O)cc(o1)N1CCOCC1
O=c1cc(sc(c1)-c1ccc(cc1)-c1csc2ccccc12)N1CCOCC1
Brc1cccc(c1)-c1cc(=O)cc(s1)N1CCOCC1
Clc1ccc(cc1)-c1cc(=O)cc(s1)N1CCOCC1
COc1ccc(cc1)-c1cc(=O)cc(s1)N1CCOCC1
Brc1ccc(cc1)-c1cc(=O)cc(s1)N1CCOCC1
Oc1cccc(c1)-c1cccc(c1)-c1cc(=O)cc(s1)N1CCOCC1
Fc1ccc(cc1)-c1cc(=O)cc(o1)N1CCOCC1
CC(C)(C)c1ccc(cc1)-c1cc(=O)cc(s1)N1CCOCC1
O=c1cc(oc(c1)-c1ccccc1)N1CCOCC1
Clc1ccc(cc1)-c1cc(=O)cc(o1)N1CCOCC1
O=c1cc(sc(c1)-c1ccc(cc1)-c1cccc2ccccc12)N1CCOCC1
O=c1cc(oc2c(cccc12)-c1ccnc(c1)-c1ccc2cc[nH]c2c1)N1CCCCC1
Cn1ccnc1-c1cccc(c1)-c1cccc2c1oc(cc2=O)N1CCOCC1
Cn1cncc1-c1cccc(c1)-c1cccc2c1oc(cc2=O)N1CCOCC1
O=c1cc(oc2c(cccc12)-c1cccc(c1)-c1cc[nH]c1)N1CCOCC1
O=c1cc(oc2c(cccc12)-c1cccc(c1)-c1nccs1)N1CCOCC1
O=c1cc(oc2c(cccc12)-c1cccc(c1)-c1ccsc1)N1CCOCC1
Cc1ccc(s1)-c1cccc(c1)-c1cccc2c1oc(cc2=O)N1CCOCC1
O=c1cc(oc2c(cccc12)-c1ncc(s1)-c1ccsc1)N1CCCCC1
COC(=O)c1cc(N)cc(c1)-c1cccc(c1)-c1cccc2c1oc(cc2=O)N1CCOCC1
O=c1cc(oc2c(cccc12)-c1ncc(s1)-c1ccncc1)N1CCCCC1
O=c1cc(oc2c(cccc12)-c1cccc(c1)-c1cccs1)N1CCOCC1
O=c1cc(oc2c(cccc12)-c1ccnc(c1)-c1cccc2cnccc12)N1CCCCC1
O=c1cc(oc2c(cccc12)-c1ncc(s1)-c1ccccc1)N1CCCCC1
O=c1cc(oc2c(cccc12)-c1ncc(s1)-c1cccs1)N1CCCCC1
O=c1cc(oc2c(cccc12)-c1ccc(s1)-c1ccccc1)N1CCCCC1
O=c1cc(oc2c(cccc12)-c1cc(cs1)-c1ccccc1)N1CCCCC1
O=c1cc(oc2c(cccc12)-c1ncc(s1)-c1cccnc1)N1CCCCC1
O=c1cc(oc2c(cccc12)-c1ncc(s1)-c1ccoc1)N1CCCCC1
O=c1cc(oc2c(cccc12)-c1cccc2c3ccccc3sc12)N1CCOCC1
O=c1cc(oc2c(cccc12)-c1cccc(c1)-c1ccc(cc1)C#N)N1CCOCC1
Oc1ccc(cc1)-c1cccc(c1)-c1cccc2c1oc(cc2=O)N1CCOCC1
COc1ccc(cc1)-c1cccc(c1)-c1cccc2c1oc(cc2=O)N1CCOCC1
O=c1cc(oc2c(cccc12)-c1cccc(c1)-c1ccccc1)N1CCOCC1
O=c1cc(oc2c(cccc12)-c1cccc(c1)-c1ccncc1)N1CCOCC1
Nc1cc(cc(c1)-c1cccc(c1)-c1cccc2c1oc(cc2=O)N1CCOCC1)C(O)=O
O=c1cc(oc2c(cccc12)-c1cc(cs1)-c1ccsc1)N1CCCCC1
O=c1cc(oc2c(cccc12)-c1cccc(c1)-c1ncccn1)N1CCOCC1
OCc1ccc(cc1)-c1cccc(c1)-c1cccc2c1oc(cc2=O)N1CCOCC1
NCc1ccc(cc1)-c1cccc(c1)-c1cccc2c1oc(cc2=O)N1CCOCC1
O=c1cc(oc2c(cccc12)-c1cc(ccn1)-c1cncnc1)N1CCCCC1
O=c1cc(oc2c(cccc12)-c1ccnc(c1)-c1ccncc1)N1CCCCC1
O=Cc1ccc(cc1)-c1cccc(c1)-c1cccc2c1oc(cc2=O)N1CCOCC1
O=c1cc(oc2c(cccc12)-c1ccc(s1)-c1cccc2cnccc12)N1CCCCC1
O=c1cc(oc2c(cccc12)-c1ccc(s1)-c1cccc2ccccc12)N1CCCCC1
O=c1cc(oc2c(cccc12)-c1cccc(c1)-c1cncnc1)N1CCOCC1
O=c1cc(oc2c(cccc12)-c1ccc(s1)-c1ccc2[nH]ccc2c1)N1CCCCC1
O=c1cc(oc2c(cccc12)-c1cccc(c1)-c1ccccn1)N1CCOCC1
O=c1cc(oc2c(cccc12)-c1cccc(c1)-c1ccco1)N1CCOCC1
O=c1cc(oc2c(cccc12)-c1cccc(c1)-c1ccoc1)N1CCOCC1
Cc1cc(cs1)-c1cccc(c1)-c1cccc2c1oc(cc2=O)N1CCOCC1
Cc1cscc1-c1cccc(c1)-c1cccc2c1oc(cc2=O)N1CCOCC1
O=c1cc(oc2c(cccc12)-c1cc(ccn1)-c1cccs1)N1CCCCC1
O=c1cc(oc2c(cccc12)-c1cc(ccn1)-c1ccccc1)N1CCCCC1
Cc1ccsc1-c1cccc(c1)-c1cccc2c1oc(cc2=O)N1CCOCC1
O=c1cc(oc2c(cccc12)-c1cc(ccn1)-c1cccnc1)N1CCCCC1
O=c1cc(oc2c(cccc12)-c1ccnc(c1)-c1ccccc1)N1CCCCC1
O=c1cc(oc2c(cccc12)-c1cc(ccn1)-c1ccsc1)N1CCCCC1
O=c1cc(oc2c(cccc12)-c1cc(ccn1)-c1ccoc1)N1CCCCC1
CN1CCN(CC1)CCCN2c3ccccc3Sc4c2cc(cc4)C(F)(F)F
Nc1ncc(nc1C(=O)Nc1ccccc1)-c1ccccc1
CC(CN(C)C)S(=O)(=O)c1ccc(cc1)-c1cnc(N)c(n1)C(=O)Nc1ccccc1
CS(=O)(=O)c1ccc(cc1)-c1cnc(N)c(n1)C(=O)Nc1ccccc1
CCc1[nH]c(\C=C2/C(=O)Nc3ccc(cc23)S(=O)(=O)Nc2ccccc2)c(CC)c1CCC(O)=O
CO[C@@H]1C[C@H](C)Cc2c(O)c(NC(=O)C(C)=CC=C[C@@H](OC)[C@H](OC(N)=O)\C(C)=C\[C@@H](C)[C@@H]1O)cc(O)c2N=CCCCCCOc1ccc2c(c1)oc(cc2=O)N1CCOCC1 |r,w:17.16,14.14,38.39,t:28|
COc1cc(ccc1O)C=O
Cc1ccc2c3ccccc3sc2c1-c1cccc2c1oc(cc2=O)N1CCOCC1 |(19.79,-10.3,;18.46,-9.52,;18.46,-7.98,;17.12,-7.21,;15.77,-7.99,;14.3,-7.52,;13.67,-6.13,;12.14,-5.98,;11.25,-7.24,;11.89,-8.63,;13.41,-8.77,;14.32,-10.01,;15.78,-9.53,;17.12,-10.29,;17.12,-11.83,;15.78,-12.6,;15.79,-14.15,;17.12,-14.91,;18.45,-14.14,;18.45,-12.6,;19.78,-11.83,;21.12,-12.59,;21.12,-14.14,;19.79,-14.91,;19.79,-16.46,;22.44,-11.81,;23.78,-12.58,;25.11,-11.8,;25.11,-10.26,;23.76,-9.49,;22.43,-10.28,)|
CCN1CCN(CC(=O)Nc2ccc(-c3cccc4c3oc(cc4=O)N3CCOCC3)c3sc4ccccc4c23)CC1
COc1cc(C=O)c(cc1OC)[N+]([O-])=O
COc1cc(Br)c(C=O)cc1OC
COc1ccc(cc1)-c1cc(O)cc(n1)N1CCOCC1
Oc1cc(ccc1C=O)N1CCOCC1
COC[C@H]1OC(=O)c2coc3c2[C@@]1(C)C1=C([C@@H]2CCC(=O)[C@@]2(C)C[C@H]1OC(C)=O)C3=O |r,t:16|
COc1ccc(cc1)-c1cccc2c1oc(cc2=O)N1CCOCC1
O=c1cc(oc2c(cccc12)-c1cccc2c1oc1ccccc21)N1CCOCC1
OCc1ccc(cc1)-c1cccc2c1oc(cc2=O)N1CCOCC1
CC(=O)c1ccc(s1)-c1cccc2c1oc(cc2=O)N1CCOCC1
O=c1cc(oc2c(cccc12)-c1cccs1)N1CCOCC1
O=c1cc(oc2c(cccc12)-c1cc2ccccc2s1)N1CCOCC1
O=c1cc(oc2c(cccc12)-c1ccsc1)N1CCOCC1
CC1CN(CCO1)c1cc(=O)c2ccc3ccccc3c2o1
CCC1CN(CCO1)c1cc(=O)n2ccc3ccccc3c2n1
O=c1cc(oc2c3ccccc3ccc12)N1C[C@H]2C[C@@H]1CO2
Clc1ccc2oc(=O)cc(N3CCOCC3)c2c1
O=c1cc(oc2ccc(cc12)-c1ccccc1)N1CCOCC1
O=c1cc(oc2c(cccc12)-c1ccccc1)N1CCCCC1
OCC1CN(CCO1)c1cc(=O)n2ccc3ccccc3c2n1
COc1cccc2c(cc(=O)oc12)N1CCOCC1
Brc1ccccc1OCCNc1cc(=O)c2ccc3ccccc3c2o1
Clc1ccccc1-c1cc(=O)c2ccc3ccccc3c2o1
CC1CCC(C)N(C1)c1cc(=O)n2ccc3ccccc3c2n1
CN(CC(O)c1ccccc1)c1cc(=O)n2ccc3ccccc3c2n1
O=c1cc(nc2ccccn12)N1CCOCC1
OC(CNc1cc(=O)n2ccc3ccccc3c2n1)c1cccc(O)c1
CN(CCC#C)c1cc(=O)n2ccc3ccccc3c2n1
Cc1cccc2c(cc(=O)oc12)N1CCOCC1
OCCNc1cc(=O)n2ccc3ccccc3c2n1
S=c1cc(oc2c3ccccc3ccc12)N1CCOCC1
COc1cccc2oc(=O)cc(N3CCOCC3)c12
CC(O)CNc1cc(=O)n2ccc3ccccc3c2n1
OCC(O)CNc1cc(=O)n2ccc3ccccc3c2n1
O=c1cc(oc2cc3ccccc3cc12)N1CCOCC1
CN(CCc1cccs1)c1cc(=O)n2ccc3ccccc3c2n1
CC1CN(CC(C)O1)c1cc(=O)c2ccc3ccccc3c2o1
COc1cccc2c1oc(cc2=O)N1CCOCC1
CC1(C)CN(CCO1)c1cc(=O)n2ccc3ccccc3c2n1
OCCOCCNc1cc(=O)c2ccc3ccccc3c2o1
Fc1cccc(c1)-c1cc(=O)c2ccc3ccccc3c2o1
CN1CCN(CC1)c1cc(=O)n2ccc3ccccc3c2n1
O=c1cc(oc2c3CCCCc3ccc12)N1CCOCC1
CC1(C)CN(CCO1)c1cc(=O)c2ccc3ccccc3c2o1
[O-][N+](=O)c1ccc(cc1)-c1cc(=O)c2ccc3ccccc3c2o1
Fc1ccc(cc1)-c1cc(=O)c2ccc3ccccc3c2o1
CN1CCN(CC1)c1cc(=O)c2ccc3ccccc3c2o1
CC(C)(C)c1ccc(cc1)-c1cc(=O)c2ccc3ccccc3c2o1
O=c1cc(N2CCOCC2)c2ccccc2o1
O=c1cc(NCC2CCCO2)oc2c3ccccc3ccc12
O=c1cc(N2CCSCC2)c2cc3ccccc3cc2o1
Nc1ccc(cc1)-c1cc(=O)c2ccc3ccccc3c2o1
O=c1cc(N2CCOCC2)c2ccc3ccccc3c2o1
O=c1cc(nc2c3ccccc3ccn12)N1CCOCC1
O=c1cc(N2CCOCC2)c2c(ccc3ccccc23)o1
Clc1ccc(cc1)-c1cc(=O)c2ccc3ccccc3c2o1
O=c1cc(oc2c3ccccc3ccc12)N1CCCC1
Fc1ccccc1-c1cc(=O)c2ccc3ccccc3c2o1
c1ccc(cc1)C2=CC(=O)c3ccccc3O2
COc1ccc2oc(=O)cc(N3CCOCC3)c2c1
COc1ccc2c(c1)oc(cc2=O)N1CCOCC1
O=c1cc(oc2c3ccccc3ccc12)N1CCOc2ccccc12
O=c1cc(nc2c3ccccc3ccn12)N1CCSCC1
O=c1cc(oc2c3ccccc3ccc12)N1CCCCC1
Cc1ccc2oc(=O)cc(N3CCOCC3)c2c1
Nc1ccccc1-c1cc(=O)c2ccc3ccccc3c2o1
Nc1cccc(c1)-c1cc(=O)c2ccc3ccccc3c2o1
OCCN(Cc1ccccc1)c1cc(=O)n2ccc3ccccc3c2n1
O=c1cc(N2CCOCC2)c2cc3ccccc3cc2o1
CN(CCO)c1cc(=O)n2ccc3ccccc3c2n1
Cc1cccc2c1oc(cc2=O)N1CCOCC1
O=c1cc(oc2ccc3ccccc3c12)N1CCOCC1
O=c1cc(nc2c3ccccc3ccn12)N1CCCC1
C[C@H]1CN(C[C@@H](C)O1)c1cc(=O)n2ccc3ccccc3c2n1
O=c1cc(oc2c3ccccc3ccc12)N1CCNCC1
COc1ccc2c(cc(=O)oc2c1)N1CCOCC1
O=c1cc(N2CCCCC2)c2ccccc2o1
OC1CCN(C1)c1cc(=O)c2ccc3ccccc3c2o1
[O-][N+](=O)c1ccccc1-c1cc(=O)c2ccc3ccccc3c2o1
O=c1cc(NCC2CCCO2)nc2c3ccccc3ccn12
[O-][N+](=O)c1cccc(c1)-c1cc(=O)c2ccc3ccccc3c2o1
Clc1cccc(c1)-c1cc(=O)c2ccc3ccccc3c2o1
O=c1cc(oc2c3ccccc3ccc12)N1CCSCC1
c1ccc(cc1)C2=CC(=O)c3ccc4ccccc4c3O2
OCCN(CCO)c1cc(=O)n2ccc3ccccc3c2n1
O=c1cc(oc2c3ccccc3ccc12)-c1cccnc1
O[C@@H]1CCN(C1)c1cc(=O)n2ccc3ccccc3c2n1
O=c1cc(oc2c3ccccc3ccc12)N1CCCOCC1
O=S1CCN(CC1)c1cc(=O)c2cccc(-c3ccccc3)c2o1
O=c1cc(oc2c(cccc12)-c1ccccc1)N1CCSCC1
O=c1cc(oc2c3ccccc3ccc12)-c1ccncc1
O=c1cc(nc2c3ccccc3ccn12)N1CC=CC1 |c:20|
OC[C@H]1CCCN(C1)c1cc(=O)c2ccc3ccccc3c2o1 |r|
Clc1ccc(cc1)-c1cccc2c1oc(cc2=O)N1CCOCC1
Fc1cccc(COc2ccc3c(c2)oc(cc3=O)N2CCOCC2)c1
CCCCN(CCCC)c1cc(=O)c2ccc3ccccc3c2o1
CCC(CO)Nc1cc(=O)c2ccc3ccccc3c2o1
OCc1ccccc1-c1cccc2c1oc(cc2=O)N1CCOCC1
COC(=O)c1cccc(COc2ccc3c(c2)oc(cc3=O)N2CCOCC2)c1
Cc1cccc(COc2ccc3c(c2)oc(cc3=O)N2CCOCC2)c1
OCc1cccc(c1)-c1cccc2c1oc(cc2=O)N1CCOCC1
O=C1N(CCCOc2ccc3c(c2)oc(cc3=O)N2CCOCC2)C(=O)c2ccccc12
CC(=O)c1ccc(cc1)-c1cccc2c1oc(cc2=O)N1CCOCC1
COC(=O)c1ccc(COc2ccc3c(c2)oc(cc3=O)N2CCOCC2)cc1
[O-][N+](=O)c1cccc(COc2ccc3c(c2)oc(cc3=O)N2CCOCC2)c1
CC(C)(C)c1ccc(CCOc2ccc3c(c2)oc(cc3=O)N2CCOCC2)cc1
O=C(OCc1ccccc1)c1ccc(cc1)-c1cccc2c1oc(cc2=O)N1CCOCC1
Fc1ccc(COc2ccc3c(c2)oc(cc3=O)N2CCOCC2)cc1
O=c1cc(oc2cc(OCc3ccc(cc3)C#N)ccc12)N1CCOCC1
O=c1cc(oc2cc(OCc3ccc4ccccc4c3)ccc12)N1CCOCC1
O=C(Oc1ccc2c(c1)oc(cc2=O)N1CCOCC1)c1ccccc1
O=c1cc(oc2c(cccc12)-c1cccc(OCc2ccccc2)c1)N1CCOCC1
COC(=O)c1ccccc1-c1cccc2c1oc(cc2=O)N1CCOCC1
O=c1cc(oc2c(cccc12)-c1ccccc1OCc1ccccc1)N1CCOCC1
CCOC(=O)c1cccc(c1)-c1cccc2c1oc(cc2=O)N1CCOCC1
O=c1cc(oc2cc(OCCc3ccccc3)ccc12)N1CCOCC1
O=C1N(COc2ccc3oc(cc(=O)c3c2)N2CCOCC2)C(=O)c2ccccc12
Clc1ccccc1OCCOc1ccc2c(c1)oc(cc2=O)N1CCOCC1
O=c1cc(oc2c(cccc12)-c1ccccc1-c1ccccc1)N1CCOCC1
Oc1ccc2c(c1)oc(cc2=O)N1CCOCC1
Oc1cccc(c1)-c1cccc2c1oc(cc2=O)N1CCOCC1
Clc1ccc(OCCOc2ccc3c(c2)oc(cc3=O)N2CCOCC2)cc1
CC(=O)Nc1ccc(cc1)-c1cccc2c1oc(cc2=O)N1CCOCC1
CC(C)(C)c1ccc(COc2ccc3c(c2)oc(cc3=O)N2CCOCC2)cc1
COc1cccc(COc2ccc3c(c2)oc(cc3=O)N2CCOCC2)c1
O=c1cc(oc2c(cccc12)-c1cccc2c3CCCCc3sc12)N1CCOCC1
O=c1cc(oc2c(cccc12)-c1ccc(OCc2ccccc2)cc1)N1CCOCC1
O=c1cc(oc2c(cccc12)-c1cccc2Sc3ccccc3Oc12)N1CCOCC1
[O-][n+]1cccc(COc2ccc3c(c2)oc(cc3=O)N2CCOCC2)c1
OC(CNc1cc(=O)c2ccc3ccccc3c2o1)c1ccccc1
COc1ccc(CCOc2ccc3c(c2)oc(cc3=O)N2CCOCC2)cc1
O=c1cc(oc2c(cccc12)-c1ccc2[nH]ccc2c1)N1CCOCC1
Oc1ccc(cc1)-c1cccc2c1oc(cc2=O)N1CCOCC1
CCOCCOc1ccc2c(c1)oc(cc2=O)N1CCOCC1
Cc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2ccccc12
O=c1cc(oc2c(cccc12)-c1ccco1)N1CCOCC1
O=c1cc(oc2c3ccccc3ccc12)N1CCSC1
CN(CC(O)c1ccccc1)c1cc(=O)c2ccc3ccccc3c2o1
O=c1cc(oc2cc(OCC3CCCCC3)ccc12)N1CCOCC1
O=c1cc(oc2cc(OCCOc3ccc4ccccc4c3)ccc12)N1CCOCC1
CN(CCO)c1cc(=O)c2ccc3ccccc3c2o1
Fc1ccc(\C=C\c2cccc3c2oc(cc3=O)N2CCOCC2)cc1
CC(C)(C)c1ccccc1-c1cccc2c1oc(cc2=O)N1CCOCC1
CC(O)CNc1cc(=O)c2ccc3ccccc3c2o1
O=c1cc(oc2cc(OCCOc3ccccc3)ccc12)N1CCOCC1
O=c1cc(oc2c(cccc12)-c1ccc2ncccc2c1)N1CCOCC1
OCC1CCN(CC1)c1cc(=O)c2ccc3ccccc3c2o1
COC(=O)\C=C\c1cccc(c1)-c1cccc2c1oc(cc2=O)N1CCOCC1
FC(F)(F)c1cc(cc(c1)C(F)(F)F)-c1cccc2c1oc(cc2=O)N1CCOCC1
O=C1N(CCOc2ccc3c(c2)oc(cc3=O)N2CCOCC2)C(=O)c2ccccc12
CC(C)Nc1cc(=O)c2ccc3ccccc3c2o1
O=c1cc(oc2c(cccc12)-c1cccc2ccccc12)N1CCOCC1
COCCNc1cc(=O)c2ccc3ccccc3c2o1
COC(=O)\C=C\c1ccccc1-c1cccc2c1oc(cc2=O)N1CCOCC1
CSc1ccc(COc2ccc3c(c2)oc(cc3=O)N2CCOCC2)cc1
O=c1cc(oc2c(cccc12)-c1ccc(cc1)C#N)N1CCOCC1
O=c1cc(oc2cc(OCc3ccccc3)ccc12)N1CCOCC1
Cc1ccc(COc2ccc3c(c2)oc(cc3=O)N2CCOCC2)cc1
O=c1cc(oc2c(cccc12)-c1ccc2ccccc2c1)N1CCOCC1
FC(F)(F)Oc1ccc(cc1)-c1cccc2c1oc(cc2=O)N1CCOCC1
Fc1ccc(COc2ccc3c(c2)oc(cc3=O)N2CCOCC2)cc1F
O=c1cc(oc2cc(OCCS(=O)(=O)c3ccccc3)ccc12)N1CCOCC1
O=C1N(Cc2cccc(c2)-c2cccc3c2oc(cc3=O)N2CCOCC2)C(=O)c2ccccc12
CCCOc1ccc2c(c1)oc(cc2=O)N1CCOCC1
OC[C@@H]1CCCN1c1cc(=O)c2ccc3ccccc3c2o1
CCN(CC)CCCNc1cc(=O)c2ccc3ccccc3c2o1
CC(C)(C)Oc1cccc(c1)-c1cccc2c1oc(cc2=O)N1CCOCC1
Brc1cccc(COc2ccc3c(c2)oc(cc3=O)N2CCOCC2)c1
Brc1ccc(CCOc2ccc3c(c2)oc(cc3=O)N2CCOCC2)cc1
CC(=O)Nc1ccccc1-c1cccc2c1oc(cc2=O)N1CCOCC1
CC(=O)c1ccccc1-c1cccc2c1oc(cc2=O)N1CCOCC1
CCS(=O)(=O)CCOc1ccc2c(c1)oc(cc2=O)N1CCOCC1
Clc1cccc(COc2ccc3c(c2)oc(cc3=O)N2CCOCC2)c1
COC(CNc1cc(=O)c2ccc3ccccc3c2o1)OC
O=c1cc(NC2CCCC2)oc2c3ccccc3ccc12
[O-][n+]1ccc(COc2ccc3c(c2)oc(cc3=O)N2CCOCC2)cc1
O=c1cc(NC2CCN(Cc3ccccc3)CC2)oc2c3ccccc3ccc12
[O-]c1cc(oc2cc(OCCc3cc[n+]([O-])cc3)ccc12)=[N+]1CCOCC1 |(3.53,-20.8,;3.53,-19.26,;4.87,-18.49,;4.87,-16.95,;3.53,-16.19,;2.2,-16.96,;.87,-16.19,;-.46,-16.96,;-1.81,-16.19,;-3.14,-16.96,;-4.48,-16.2,;-5.82,-16.99,;-7.14,-16.22,;-8.48,-16.98,;-8.47,-18.52,;-9.82,-19.31,;-7.14,-19.29,;-5.81,-18.53,;-.46,-18.5,;.88,-19.26,;2.21,-18.49,;6.21,-16.19,;7.53,-16.96,;8.87,-16.18,;8.87,-14.64,;7.53,-13.87,;6.2,-14.64,)|
O=c1cc(oc2cc(OCCS(=O)(=O)Cc3ccccc3)ccc12)N1CCOCC1
COCCCNc1cc(=O)c2ccc3ccccc3c2o1
O=c1cc(oc2c(\C=C\c3ccccc3)cccc12)N1CCOCC1
CC(=O)Nc1cccc(c1)-c1cccc2c1oc(cc2=O)N1CCOCC1
[O-][n+]1ccccc1COc1ccc2c(c1)oc(cc2=O)N1CCOCC1
Clc1ccccc1COc1ccc2c(c1)oc(cc2=O)N1CCOCC1
[OH+]=c1cc(nc2c3ccccc3ccn12)N1CCOCC1
Brc1ccc(COc2ccc3c(c2)oc(cc3=O)N2CCOCC2)cc1
O=c1cc(oc2cc(OCc3ccc(cc3)-c3ccccc3)ccc12)N1CCOCC1
CCCCNc1cc(=O)c2ccc3ccccc3c2o1
O=c1cc(oc2ccc(OCc3ccc(cc3)C#N)cc12)N1CCOCC1
Clc1ccc(COc2ccc3c(c2)oc(cc3=O)N2CCOCC2)cc1
OCCCNc1cc(=O)c2ccc3ccccc3c2o1
FC(F)(F)c1ccccc1CNc1cc(=O)c2ccc3ccccc3c2o1
O=c1cc(oc2c(cccc12)-c1csc2ccccc12)N1CCOCC1
O=c1cc(oc(c1)-c1ccc(cc1)-c1ccccc1)N1CCOCC1
O=c1cc(sc(c1)-c1cccc2Sc3ccccc3Sc12)N1CCOCC1
CCOc1cc(nc(c1)-c1ccc(Cl)cc1)N1CCOCC1
Cc1c(oc(cc1=O)-c1ccc(Cl)cc1)N1CCOCC1
COc1ccc(cc1)-c1cc(OC)cc(n1)N1CCOCC1
Cc1c(oc(cc1=O)-c1ccccc1)N1CCOCC1
O=c1cc(oc(c1)-c1ccc2[nH]ccc2c1)N1CCOCC1
O=C(OCc1ccccc1)c1ccc(cc1)-c1cc(=O)cc(o1)N1CCOCC1
O=Cc1sccc1-c1cc(=O)cc(o1)N1CCOCC1
c1ccc2c(c1)Sc3cccc(c3S2)C4=CC(=O)C=C(O4)N5CCOCC5
O=c1cc(oc(c1)-c1cccc2c1oc1ccccc21)N1CCOCC1
FC(F)(F)Oc1cccc(c1)-c1cc(=O)cc(o1)N1CCOCC1
O=c1cc(oc(c1)-c1ccc(cc1)C#N)N1CCOCC1
O=c1cc(oc(c1)-c1cccc(c1)C#N)N1CCOCC1
O=c1cc(oc(c1)-c1csc2ccccc12)N1CCOCC1
O=c1cc(oc(c1)-c1ccccc1OCc1ccccc1)N1CCOCC1
FC(F)(F)Oc1ccc(cc1)-c1cc(=O)cc(o1)N1CCOCC1
O=c1cc(sc(c1)-c1ccc(cc1)N1CCOCC1)N1CCOCC1
O=c1cc(sc(c1)-c1ccc(cc1)C#N)N1CCOCC1
Cc1cc(=O)cc(OCC(F)(F)F)s1
O=C(\C=C\N1CCOCC1)/C=C/c1ccccc1
CC(=O)OCc1cccc(c1)-c1cc(=O)cc(o1)N1CCOCC1
COC(=O)c1ccc(c(N)c1)-c1cc(=O)cc(o1)N1CCOCC1
O=C1CC(CC(=C1)N1CCOCC1)c1ccccc1 |c:5|
O=c1cc(oc(c1)-c1cc2ccccc2o1)N1CCOCC1
O=c1cc(occ1-c1ccccc1)N1CCOCC1
O=c1cc(oc(c1)-c1cc2ccccc2s1)N1CCOCC1
O=c1cc(oc(c1)-c1cccc(OCc2ccccc2)c1)N1CCOCC1
O=c1cc(cc(o1)-c1ccccc1)N1CCOCC1
COc1ccc(cc1)-c1cc(cc(=O)o1)N1CCOCC1
COC(=O)\C=C\c1cccc(c1)-c1cc(=O)cc(o1)N1CCOCC1
CC(=O)Nc1cccc(c1)-c1cccc(c1)-c1cc(=O)cc(s1)N1CCOCC1
O=C1N(Cc2ccc(cc2)-c2cc(=O)cc(o2)N2CCOCC2)C(=O)c2ccccc12
Cc1cc(=O)cc(s1)N1CCOCC1
Cc1cc(=O)cc(s1)N1CCCC1
O=C1N(Cc2cccc(c2)-c2cc(=O)cc(o2)N2CCOCC2)C(=O)c2ccccc12
CC(C)(C)c1ccc(cc1)-c1cc(cc(=O)o1)N1CCOCC1
O=c1cc(oc(c1)-c1ccc(OCc2ccccc2)cc1)N1CCOCC1
Clc1c(sc(cc1=O)-c1ccc(Br)cc1)N1CCOCC1
Clc1ccc(cc1)-c1cc(=O)c(Br)c(s1)N1CCOCC1
O=c1cc(sc2CCCCc12)N1CCOCC1
Clc1ccc(cc1)-c1cc(cc(=O)o1)N1CCOCC1
O=c1cc(\C=C\c2ccccc2)oc(c1)N1CCOCC1
O=Cc1cccc(c1)-c1cc(=O)cc(o1)N1CCOCC1
Cc1ccc(-c2cc(=O)cc(o2)N2CCOCC2)c2ccccc12
CC(=O)c1cccc(c1)-c1cc(=O)cc(o1)N1CCOCC1
O=c1cc(oc(c1)-c1ccc2ccccc2c1)N1CCOCC1
Cc1cc(=O)cc(s1)N1CCSCC1
O=c1cc(oc(c1)-c1cccc2ccccc12)N1CCOCC1
Cc1cc(=O)cc(NCc2ccccc2)s1
COc1cc(nc(c1)-c1ccc(Cl)cc1)N1CCOCC1
Oc1cc(nc(c1)-c1ccc(Cl)cc1)N1CCOCC1
COC(=O)c1cccc(c1)-c1cc(=O)cc(o1)N1CCOCC1
O=Cc1ccc(-c2cc(=O)cc(o2)N2CCOCC2)c2ccccc12
COC(=O)c1ccccc1-c1cc(=O)cc(o1)N1CCOCC1
Nc1ccccc1-c1cc(=O)cc(o1)N1CCOCC1
O=c1cc(oc(c1)-c1ccco1)N1CCOCC1
OC(=O)c1cccc(c1)-c1cc(=O)cc(o1)N1CCOCC1
O=c1cc(oc(c1)-c1ccsc1)N1CCOCC1
FC(F)(F)c1ccccc1-c1cc(=O)cc(o1)N1CCOCC1
O=c1cc(oc(c1)-c1cccs1)N1CCOCC1
Fc1ccccc1-c1cc(=O)cc(o1)N1CCOCC1
CC(C)(C)c1cc(=O)cc(s1)N1CCOCC1
CC(C)c1cc(=O)cc(s1)N1CCOCC1
O=c1cc(oc(c1)-c1cccc2cccnc12)N1CCOCC1
O=C(Nc1ccc(cc1)-c1cc(=O)cc(o1)N1CCOCC1)OCc1ccccc1
CC(C)(C)OC(=O)Nc1ccc(cc1)-c1cc(=O)cc(o1)N1CCOCC1
Oc1cc(ccc1C(=O)c1ccccc1)N1CCOCC1
COc1ccc(cc1CO)-c1ccc2c(nc(nc2n1)N1C[C@H](C)O[C@H](C)C1)N1CCOCC1 |r|
O=c1cc(N2CCOCC2)c2ccc(cc2o1)-c1ccccc1
O=c1cc(N2CCOCC2)c2cc(ccc2o1)-c1cccc2c1oc1ccccc21
O=c1cc(N2CCOCC2)c2cc(ccc2o1)-c1cccc2c3ccccc3sc12
O=c1oc(cc2c(cccc12)-c1ccccc1)N1CCOCC1
O=c1cc(N2CCOCC2)c2cc(ccc2o1)-c1cccc(c1)-c1ccccc1
O=c1cc(N2CCOCC2)c2cc(ccc2o1)-c1cc2ccccc2s1
O=c1oc(cc2c(cccc12)-c1cccc2c1oc1ccccc21)N1CCOCC1
O=c1oc(cc2c(cccc12)-c1cccc(c1)-c1ccccc1)N1CCOCC1
O=c1oc(cc2c(cccc12)-c1cccc2c3ccccc3sc12)N1CCOCC1
O=c1cc(N2CCOCC2)c2ccc(cc2o1)-c1cc2ccccc2s1
O=c1cc(N2CCOCC2)c2ccc(cc2o1)-c1cccc2c3ccccc3sc12
O=c1cc(N2CCOCC2)c2cc(ccc2o1)-c1cccs1
O=c1oc(cc2ccccc12)N1CCOCC1
O=c1cc(N2CCOCC2)c2cc(ccc2o1)-c1ccccc1
COc1cccc2c1cc(oc2=O)N1CCOCC1
O=c1cc(N2CCOCC2)c2ccc(cc2o1)-c1cccc2c1oc1ccccc21
O=c1cc(N2CCOCC2)c2ccc(cc2o1)-c1cccs1
O=c1cc(N2CCOCC2)c2ccc(cc2o1)-c1cccc(c1)-c1ccccc1
Cn1ncc2c(Oc3ccc(cc3)S(C)(=O)=O)cc(nc12)-c1cccc2[nH]ncc12
CCC(=O)N1CCN(CC1)c1ccc(cc1C(F)(F)F)-n1c2c(ccc1=O)cnc1ccc(cc21)-c1cnc2ccccc2c1
CC1(COc2cc(ccc2NC(=O)CN2CCOCC2)-c2cccc3c2oc(cc3=O)N2CCOCC2)COC1
O=C(CN1CCOCC1)Nc1ccc(cc1OCCC1CC1)-c1cccc2c1oc(cc2=O)N1CCOCC1
Oc1cc(ccc1NC(=O)CN1CCOCC1)-c1cccc2c1oc(cc2=O)N1CCOCC1
OCCOc1cc(ccc1NC(=O)CN1CCOCC1)-c1cccc2c1oc(cc2=O)N1CCOCC1
COc1cc(ccc1NC(=O)CN1CCOCC1)-c1cccc2c1oc(cc2=O)N1CCOCC1
CC1(COc2cc(ccc2NC(=O)CN2CCOCC2)-c2cccc3c2oc(cc3=O)N2CCOCC2)CCC1
COCCOc1cc(ccc1NC(=O)CN1CCOCC1)-c1cccc2c1oc(cc2=O)N1CCOCC1
NC(=O)COc1cc(ccc1NC(=O)CN1CCOCC1)-c1cccc2c1oc(cc2=O)N1CCOCC1
O=C(CN1CCOCC1)Nc1ccc(cc1OCC1CCC1)-c1cccc2c1oc(cc2=O)N1CCOCC1
O=C(CN1CCOCC1)Nc1ccc(cc1OCC1CC1)-c1cccc2c1oc(cc2=O)N1CCOCC1
O=C(CN1CCOCC1)Nc1ccc(cc1OCCN1CCCC1)-c1cccc2c1oc(cc2=O)N1CCOCC1
CC(C)Oc1cc(ccc1NC(=O)CN1CCOCC1)-c1cccc2c1oc(cc2=O)N1CCOCC1
CCOc1cc(ccc1NC(=O)CN1CCOCC1)-c1cccc2c1oc(cc2=O)N1CCOCC1
NCCOc1cc(ccc1NC(=O)CN1CCOCC1)-c1cccc2c1oc(cc2=O)N1CCOCC1
C=CCOc1cc(ccc1NC(=O)CN1CCOCC1)-c1cccc2c1oc(cc2=O)N1CCOCC1
CC(C)COc1cc(ccc1NC(=O)CN1CCOCC1)-c1cccc2c1oc(cc2=O)N1CCOCC1
O=C(CN1CCOCC1)Nc1ccc(cc1-c1ccccc1)-c1cccc2c1oc(cc2=O)N1CCOCC1
Nc1ccc(cn1)-c1ccc2ncc3ccc(=O)n(-c4cccc(c4)C(F)(F)F)c3c2c1
Cc1ccc(cc1)-c1cnc(N)c(n1)C(=O)Nc1ccccc1
CN(C)C(=O)c1ccc(cc1)-c1cnc(N)c(n1)C(=O)Nc1ccccc1
Nc1ncc(nc1C(=O)Nc1ccccc1)-c1ccc(cc1)C(=O)N1CCC1
CNC(=O)c1ccc(cc1)-c1cnc(N)c(n1)C(=O)Nc1ccccc1
NC(=O)c1ccc(cc1)-c1cnc(N)c(n1)C(=O)Nc1ccccc1
Nc1ncc(nc1C(=O)Nc1ccccc1)-c1ccc(O)cc1
Nc1ncc(nc1C(=O)Nc1ccccc1)-c1ccc(cc1)C#N
Cc1cccc(c1)-c1cnc(N)c(n1)C(=O)Nc1ccccc1
Nc1ncc(nc1C(=O)Nc1ccccc1)-c1ccc(Cl)cc1
COc1ccc(cc1)-c1cnc(N)c(n1)C(=O)Nc1ccccc1
Nc1ncc(nc1C(=O)Nc1ccccc1)-c1cccc(Cl)c1
COc1cccc(c1)-c1cnc(N)c(n1)C(=O)Nc1ccccc1
Nc1ncc(nc1C(=O)Nc1ccccc1)-c1cccc(O)c1
CS(=O)(=O)c1cccc(c1)-c1cnc(N)c(n1)C(=O)Nc1ccccc1
COc1ccccc1-c1cnc(N)c(n1)C(=O)Nc1ccccc1
Nc1ncc(nc1C(=O)Nc1ccccc1)-c1ccccc1O
CS(=O)(=O)c1ccccc1-c1cnc(N)c(n1)C(=O)Nc1ccccc1
CS(=O)c1ccccc1-c1cnc(N)c(n1)C(=O)Nc1ccccc1
Nc1ncc(nc1C(=O)Nc1ccccc1)-c1cccc(c1)C#N
Cc1ccccc1-c1cnc(N)c(n1)C(=O)Nc1ccccc1
Nc1ncc(nc1C(=O)Nc1ccccc1)-c1ccccc1Cl
CS(=O)(=O)c1ccc(cc1)-c1cnc(N)c(n1)-c1cc2ccccc2[nH]1
CS(=O)(=O)c1ccc(cc1)-c1cnc(N)c(n1)-c1nc2ccccc2s1
Nc1ncc(nc1C(=O)Nc1ccccc1)-c1ccccc1C#N
Nc1ncc(nc1C(=O)Nc1ccccc1)-c1ccncc1
COc1cc2CC(C)C(C)Cc3cc4OCOc4c(OC)c3-c2c(OC)c1OC
Nc1ncc(nc1C(=O)Nc1ccccc1)-c1cccnc1
CS(=O)(=O)c1ccc(cc1)-c1cnc(N)c(n1)-c1nc2ccccc2o1
CS(=O)(=O)c1ccc(cc1)-c1cnc(N)c(n1)-c1nc2ccccc2[nH]1
CS(=O)(=O)c1ccc(cc1)-c1cnc(N)c(n1)C(=O)NC1CCCCC1
Nc1ncc(nc1C(=O)Nc1ccccc1)-c1ccc(cc1)S(=O)(=O)[C@@H]1CCOC1 |r|
Nc1ncc(nc1C(=O)Nc1ccccc1)C1CCCCC1
CCCS(=O)(=O)c1ccc(cc1)-c1cnc(N)c(n1)C(=O)Nc1ccccc1
Nc1ncc(Br)nc1C(=O)Nc1ccccc1
CC(C)S(=O)(=O)c1ccc(cc1)-c1cnc(N)c(n1)C(=O)Nc1ccccc1
Nc1nccnc1C(=O)Nc1ccccc1
CC(CCO)S(=O)(=O)c1ccc(cc1)-c1cnc(N)c(n1)C(=O)Nc1ccccc1
CC(C)(C)S(=O)(=O)c1ccc(cc1)-c1cnc(N)c(n1)C(=O)Nc1ccccc1
Nc1ncc(nc1C(=O)Nc1ccccc1)C1=CCCCC1 |t:18|
CCC(C)S(=O)(=O)c1ccc(cc1)-c1cnc(N)c(n1)C(=O)Nc1ccccc1
Cn1cnc2c1C(=O)N(C(=O)N2C)C
CS(=O)c1ccc(cc1)-c1cnc(N)c(n1)C(=O)Nc1ccccc1
CN(C)C(=O)c1ccc(cc1Cl)-c1cnc(N)c(n1)C(=O)Nc1ccccc1
Nc1ncc(nc1C(=O)Nc1ccccc1)-c1ccc(cc1)C(=O)N1CCCCC1
Nc1ncc(nc1C(=O)Nc1ccccc1)-c1ccc(cc1)C(=O)N1CCCC1
CCS(=O)(=O)c1ccc(cc1)-c1cnc(N)c(n1)C(=O)Nc1ccccc1
CC(=O)Nc1nc2ccc(cc2s1)-c1cnc(Cl)c(NS(=O)(=O)c2ccc(F)cc2)c1
CNC(=O)c1ccc2-c3sc(cc3CCOc2c1)C(=O)N(C)c1ccc(cc1Cl)C(=O)N(C)C
O=c1nc(oc2cc3ccc(OCc4cccnc4)cc3cc12)N1CCOCC1
O=c1nc(oc2cc3c(OCc4cccnc4)cccc3cc12)N1CCOCC1
O=c1nc(oc2cc3c(OCc4ccccn4)cccc3cc12)N1CCOCC1
O=c1nc(oc2c3ccccc3c(OCc3ccccn3)cc12)N1CCOCC1
O=c1nc(oc2cc3ccccc3cc12)N1CCOCC1
O=c1nc(oc2cc3ccc(OCc4ccccn4)cc3cc12)N1CCOCC1
O=c1nc(oc2c3ccccc3c(OCc3cccnc3)cc12)N1CCOCC1
CN1CCN(CCOc2ccc3cc4oc(nc(=O)c4cc3c2)N2CCOCC2)CC1
CN1CCN(CCOc2cc3c(oc(nc3=O)N3CCOCC3)c3ccccc23)CC1
O=c1nc(oc2c3ccccc3ccc12)N1CCOCC1
CN1CCN(CCOc2cccc3cc4c(cc23)oc(nc4=O)N2CCOCC2)CC1
O=c1nc(oc2ccc3ccccc3c12)N1CCOCC1
Fc1ccc(cc1)S(=O)(=O)Nc1cc(cnc1Cl)-c1ccc2nccc(N3CCOCC3)c2c1
Fc1ccc(cc1)S(=O)(=O)Nc1cc(cnc1Cl)-c1ccc2ncc(nc2c1)N1CCOCC1
Cc1ccc(cc1NC(=O)c2cccc(c2)NC(=O)Nc3cccc(c3)C(=O)Nc4cc(ccc4C)C(=O)Nc5ccc(c6c5c(cc(c6)S(=O)(=O)O)S(=O)(=O)O)S(=O)(=O)O)C(=O)Nc7ccc(c8c7c(cc(c8)S(=O)(=O)O)S(=O)(=O)O)S(=O)(=O)O
Cc1nc(NC(=O)N2CCC[C@H]2C(N)=O)sc1-c1ccc(cc1)-n1cccn1 |r|
CCn1nnc(CCNC(=O)Nc2nc(C)c(s2)-c2ccc(c(F)c2)S(C)(=O)=O)n1
Cc1c(sc(n1)NC(=O)NCCC(=O)NC(C)(C)C)c2ccc(cc2)C(=O)C
Cc1cc(NC(=O)CCNC(=O)Nc2nc(C)c(s2)-c2ccc(cc2)-n2cccn2)no1
Cc1nc(nc(n1)N)c2cc(cnc2Nc3ccc(nc3)OC)CN4CCN(CC4)S(=O)(=O)C
O=c1nc(oc2c(cccc12)-c1ccccc1)N1CCOCC1
O=c1nc(oc2cc(OCc3ccccn3)ccc12)N1CCOCC1
Cc1cccc2c1oc(nc2=O)N(Cc1ccccn1)c1cccnc1
O=c1nc(oc2c(OCc3ccccn3)cccc12)N1CCOCC1
Cc1c(OCc2cccnc2)ccc2c1oc(=O)n(Cc1cccnc1)c2=O
CN1CCN(CCOc2ccc3c(c2)oc(nc3=O)N2CCOCC2)CC1
CN1CCN(CCOc2ccc3c(oc(nc3=O)N3CCOCC3)c2C)CC1
Cc1c(OCc2ccncc2)ccc2c1oc(nc2=O)N1CCOCC1
CN1CCN(CCOc2cccc3c2oc(nc3=O)N2CCOCC2)CC1
O=c1nc(oc2c(OCc3ccncc3)cccc12)N1CCOCC1
O=c1nc(oc2cc(OCc3ccncc3)ccc12)N1CCOCC1
Cc1c(OCc2cccnc2)ccc2c1oc(nc2=O)N(Cc1cccnc1)c1cccnc1
O=c1nc(oc2c(OCc3cccnc3)cccc12)N(Cc1cccnc1)c1cccnc1
O=c1nc(oc2c(OCc3ccccn3)cccc12)N(Cc1ccccn1)c1cccnc1
O=c1nc(oc2cc(OCc3cccnc3)ccc12)N(Cc1cccnc1)c1cccnc1
O=c1nc(oc2cc(OCc3ccccn3)ccc12)N(Cc1ccccn1)c1cccnc1
Cc1c(OCc2ccccn2)ccc2c1oc(nc2=O)N1CCOCC1
Cc1c(OCc2cccnc2)ccc2c1oc(nc2=O)N1CCOCC1
O=c1nc(oc2c(OCc3cccnc3)cccc12)N1CCOCC1
O=c1nc(oc2cc(OCc3cccnc3)ccc12)N1CCOCC1
CS(=O)(=O)Cc1cc(nc(n1)-c1cccc2[nH]ccc12)N1CCOCC1
C[C@@H]1COCCN1c1cc(nc(n1)-c1cccc2[nH]ccc12)C1(CC1)S(C)(=O)=O |r|
Cc1c(F)c(ccc1C(=O)N1CCOc2ccc(cc2C1)-c1ccc(N)nc1)S(C)(=O)=O
CC(C)n1nc(C)nc1-c1cn2CCOc3cc(ccc3-c2n1)-c1cnn(c1)C(C)(C)C(N)=O
Cc1c(sc(n1)NC(=O)N2CCC[C@H]2C(=O)N)c3ccnc(c3)C(C)(C)C(F)(F)F
CC(C)N1CCN(CCOc2ccc(-c3cccc4c3oc(cc4=O)N3CCOCC3)c3sc4ccccc4c23)CC1
O=C(COc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12)N1CCCCC1
CN1CCN(CC1)C(=O)COc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
COC(=O)[C@H](CO)NCCOc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12 |r|
CN(CCOc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12)CC(N)=O
C[C@H]1CN(C[C@@H](C)O1)C(=O)COc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12 |r|
CN1CCCN(CC1)C(=O)COc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
CN(C)CCN(C)C(=O)COc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
CC(C)N1CCN(CC1)C(=O)COc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
COC(=O)[C@H](CO)NC(=O)COc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12 |r|
CC(=O)N1CCN(CC1)C(=O)COc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
O=C(COc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12)NCc1ccncc1
COCCN(CCOC)CC(=O)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
OCCNCC(=O)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
CN1CCN(CC(=O)Nc2ccc(-c3cccc4c3oc(cc4=O)N3CCOCC3)c3sc4ccccc4c23)CC1
OCCN(CCO)CC(=O)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
OCCOCCN1CCN(CCC(=O)Nc2ccc(-c3cccc4c3oc(cc4=O)N3CCOCC3)c3sc4ccccc4c23)CC1
CCN1CCN(CCC(=O)Nc2ccc(-c3cccc4c3oc(cc4=O)N3CCOCC3)c3sc4ccccc4c23)CC1
CN(CC(N)=O)C(=O)COc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
COCCN1CCN(CCC(=O)Nc2ccc(-c3cccc4c3oc(cc4=O)N3CCOCC3)c3sc4ccccc4c23)CC1
O=C(CN1CCNCC1)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
O=C(CCN1CCN(CC1)c1ccccn1)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
Fc1ccc(cc1)N1CCN(CCC(=O)Nc2ccc(-c3cccc4c3oc(cc4=O)N3CCOCC3)c3sc4ccccc4c23)CC1
O=C(CCN1CCN(CC1)c1ncccn1)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
OCCN1CCN(CCC(=O)Nc2ccc(-c3cccc4c3oc(cc4=O)N3CCOCC3)c3sc4ccccc4c23)CC1
OCCN1CCCN(CCC(=O)Nc2ccc(-c3cccc4c3oc(cc4=O)N3CCOCC3)c3sc4ccccc4c23)CC1
CN(C)CCN1CCN(CCC(=O)Nc2ccc(-c3cccc4c3oc(cc4=O)N3CCOCC3)c3sc4ccccc4c23)CC1
CCN1CCCC1CNCCC(=O)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
CN(C)CCN(C)CC(=O)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
O=C(CCN1CCNCC1)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
CN1CCN(CCC(=O)Nc2ccc(-c3cccc4c3oc(cc4=O)N3CCOCC3)c3sc4ccccc4c23)CC1
O=C(CCN1CCOCC1)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
O=C(CNCC1CCCO1)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
OCCN1CCN(CC(=O)Nc2ccc(-c3cccc4c3oc(cc4=O)N3CCOCC3)c3sc4ccccc4c23)CC1
O=C(CNCCN1CCCCC1)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
O=C(CCN1CCCCC1)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
CN1CCCN(CC(=O)Nc2ccc(-c3cccc4c3oc(cc4=O)N3CCOCC3)c3sc4ccccc4c23)CC1
CC(C)N1CCN(CCC(=O)Nc2ccc(-c3cccc4c3oc(cc4=O)N3CCOCC3)c3sc4ccccc4c23)CC1
OCCN1CCCN(CC(=O)Nc2ccc(-c3cccc4c3oc(cc4=O)N3CCOCC3)c3sc4ccccc4c23)CC1
O=c1cc(oc2c(cccc12)-c1ccc(OCCN2CCOCC2)c2c3ccccc3sc12)N1CCOCC1
O=C(CN1CCCCCC1)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
O=C(CNCCCN1CCOCC1)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
O=C(CCNCCCN1CCOCC1)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
NCCNCC(=O)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
O=C(CCNCc1ccncc1)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
O=C(CNCc1ccncc1)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
NCC(=O)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
CC(C)N1CCN(CC(=O)Nc2ccc(-c3cccc4c3oc(cc4=O)N3CCOCC3)c3sc4ccccc4c23)CC1
O=C(CNCCN1CCOCC1)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
COc1ccc(CNCC(=O)Nc2ccc(-c3cccc4c3oc(cc4=O)N3CCOCC3)c3sc4ccccc4c23)cc1
O=C(CN1CCCNCC1)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
O=c1cc(oc2c(cccc12)-c1ccc(OCCN2CCCCC2)c2c3ccccc3sc12)N1CCOCC1
CCN(CC)CC(=O)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
CN(C)CC(=O)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
CN1CCN(CCOc2ccc(-c3cccc4c3oc(cc4=O)N3CCOCC3)c3sc4ccccc4c23)CC1
CN1CCCN(CCOc2ccc(-c3cccc4c3oc(cc4=O)N3CCOCC3)c3sc4ccccc4c23)CC1
CN(C)CCN(C)CCOc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
C[C@H]1CN(CCOc2ccc(-c3cccc4c3oc(cc4=O)N3CCOCC3)c3sc4ccccc4c23)C[C@@H](C)O1 |r|
CCN(CC)CCOc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
O=c1cc(oc2c(cccc12)-c1ccc(OCCNCCN2CCOCC2)c2c3ccccc3sc12)N1CCOCC1
O=C(CNCCN1CCNC1=O)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
O=c1cc(oc2c(cccc12)-c1ccc(OCCNc2cccnc2)c2c3ccccc3sc12)N1CCOCC1
OCCNCCC(=O)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
CN1CCCC1CCNCC(=O)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
CN1CCCN(CCC(=O)Nc2ccc(-c3cccc4c3oc(cc4=O)N3CCOCC3)c3sc4ccccc4c23)CC1
NCCNCCC(=O)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
C[C@H]1CN(CC(=O)Nc2ccc(-c3cccc4c3oc(cc4=O)N3CCOCC3)c3sc4ccccc4c23)C[C@@H](C)O1 |r|
CC(=O)N1CCN(CCOc2ccc(-c3cccc4c3oc(cc4=O)N3CCOCC3)c3sc4ccccc4c23)CC1
CCN(CC(=O)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12)Cc1ccncc1
CN(C)CCOc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
OCCN(CCO)CCC(=O)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
COCCN1CCN(CC(=O)Nc2ccc(-c3cccc4c3oc(cc4=O)N3CCOCC3)c3sc4ccccc4c23)CC1
OCCOCCN1CCN(CC(=O)Nc2ccc(-c3cccc4c3oc(cc4=O)N3CCOCC3)c3sc4ccccc4c23)CC1
COCCNCC(=O)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
O=C(CN1CCOCC1)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
CC(=O)N1CCN(CC(=O)Nc2ccc(-c3cccc4c3oc(cc4=O)N3CCOCC3)c3sc4ccccc4c23)CC1
O=C(CN1CCCCC1)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
COc1ccc(CNCCC(=O)Nc2ccc(-c3cccc4c3oc(cc4=O)N3CCOCC3)c3sc4ccccc4c23)cc1
CCN(CC)CCC(=O)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
O=C(CCN1CCCCCC1)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
O=C(CCNCC1CCCO1)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
O=C(CCNCCN1CCCCC1)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
NCCC(=O)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
O=C(CCNCCN1CCOCC1)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
CCN(CCC(=O)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12)Cc1ccncc1
CN(C)CCN(C)CCC(=O)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
C[C@H]1CN(CCC(=O)Nc2ccc(-c3cccc4c3oc(cc4=O)N3CCOCC3)c3sc4ccccc4c23)C[C@@H](C)O1 |r|
COCCNCCC(=O)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
CC(=O)N1CCN(CCC(=O)Nc2ccc(-c3cccc4c3oc(cc4=O)N3CCOCC3)c3sc4ccccc4c23)CC1
O=C(CCNCCN1CCNC1=O)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
CN1CCCC1CCNCCC(=O)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
CC(C)NCC(=O)CN1CCN(CC(=O)Nc2ccc(-c3cccc4c3oc(cc4=O)N3CCOCC3)c3sc4ccccc4c23)CC1
CN(C)CCN1CCN(CC(=O)Nc2ccc(-c3cccc4c3oc(cc4=O)N3CCOCC3)c3sc4ccccc4c23)CC1
O=C(CN1CCN(CC1)c1ccccn1)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
Fc1ccc(cc1)N1CCN(CC(=O)Nc2ccc(-c3cccc4c3oc(cc4=O)N3CCOCC3)c3sc4ccccc4c23)CC1
CCN1CCCC1CNCC(=O)Nc1ccc(-c2cccc3c2oc(cc3=O)N2CCOCC2)c2sc3ccccc3c12
Oc1cccc(c1)-c1nc(N2CCOCC2)c2oc3ncccc3c2n1
COc1ccc2C3=NCCN3C(NC(=O)c3cccnc3)=Nc2c1OC |c:22,t:6|
Fc1ccc(CN2C(=O)COc3ccc(\C=C4\SC(=S)NC4=O)cc23)cc1Cl
CC1=C(SC(=NC(=O)C)N1)c2ccc(c(c2)S(=O)(=O)NCCO)Cl
CC[C@@H](C1=Nc2cccc(c2C(=O)N1c3ccccc3)F)Nc4c5c(nc[nH]5)ncn4
C[C@@H]1Cn2ncc(c2CN1c1ccnc2[nH]ccc12)-c1ccc(cc1)S(C)(=O)=O |r|
C[C@@H]1Cn2ncc(C3CCN(CC3)S(C)(=O)=O)c2CN1c1ccnc2[nH]ccc12 |r|
C[C@@H]1Cn2ncc(C3CCN(CC3)S(C)(=O)=O)c2CN1c1cc(Cl)nc2[nH]ccc12 |r|
C[C@@H]1COCCN1c1nc(cc2n(C)cnc12)-c1nncc2[nH]ccc12 |r|
CC(C)(C#N)c1ccc(cc1)N1C(=O)OCc2cnc3ccc(cc3c12)-c1cnc2ccccc2c1
O=c1cc(nc2c(cccn12)-c1cccc2c3ccccc3sc12)N1CCOCC1
Cc1ccc2c(oc(cc2=O)N2CCOCC2)c1-c1cccc2c3ccccc3sc12 |(-5,-3.04,;-3.93,-3.66,;-3.94,-5.2,;-2.6,-5.98,;-1.26,-5.22,;-1.25,-3.68,;.09,-2.92,;1.42,-3.7,;1.41,-5.24,;.07,-6,;.06,-7.23,;2.76,-2.93,;2.77,-1.39,;4.12,-.63,;5.45,-1.41,;5.43,-2.96,;4.09,-3.72,;-2.58,-2.9,;-2.56,-1.36,;-1.31,-.65,;-1.28,.82,;-2.51,1.58,;-3.82,.87,;-6.35,.92,;-7.61,1.68,;-8.93,.97,;-8.96,-.5,;-7.67,-1.26,;-6.37,-.55,;-5.13,-1.31,;-3.85,-.6,)|
CC(=O)c1ccc(cc1O)N1CCOCC1
Oc1ccc(cc1)C(=O)c1ccc(cc1O)N1CCOCC1
Oc1cc(cc2oc(cc(=O)c12)-c1ccccc1)N1CCOCC1
CCN1C(=O)CNc2ncc(nc12)-c1ccc(nc1C)-c1nc[nH]n1
COc1cc(cnc1Cl)N1CCc2nc(NC(=O)NCCc3cn(CC(F)F)cn3)sc2C1
COc1cncc(n1)N1CCc2nc(NC(=O)NCCc3cn(CC(F)F)cn3)sc2C1
O=c1nc(oc2c(cccc12)-c1cccc2c1oc1ccccc21)N1CCOCC1
O=c1nc(oc2c(cccc12)-c1cccc2c3ccccc3sc12)N1CCOCC1
O=c1nc(oc2c(cccc12)-c1cc2ccccc2s1)N1CCOCC1
COc1ccc(cc1)-c1cc(Cl)cc2c1oc(nc2=O)N1CCOCC1
Clc1cc(-c2cccs2)c2oc(nc(=O)c2c1)N1CCOCC1
Clc1cc(-c2cc3ccccc3s2)c2oc(nc(=O)c2c1)N1CCOCC1
Clc1cc(-c2cccc3c4ccccc4sc23)c2oc(nc(=O)c2c1)N1CCOCC1
O=c1nc(oc2c(cccc12)-c1cccs1)N1CCOCC1
O=c1nc(oc2c(cccc12)-c1cccnc1)N1CCOCC1
O=c1nc(oc2c(cccc12)-c1cccc2ccccc12)N1CCOCC1
COc1ccc(cc1)-c1cccc2c1oc(nc2=O)N1CCOCC1
O=c1nc(oc2c(cccc12)-c1ccsc1)N1CCOCC1
NC(=O)c1ccc(cc1)-c1cccc2c1oc(nc2=O)N1CCOCC1
Nc1cccc(c1)-c1cccc2c1oc(nc2=O)N1CCOCC1
OCc1ccc(cc1)-c1cccc2c1oc(nc2=O)N1CCOCC1
Clc1ccc(cc1)-c1cccc2c1oc(nc2=O)N1CCOCC1
Fc1ccc(CN2C(=O)COc3ccc(\C=C4/SC(=S)NC4=O)cc23)cc1Cl
COc1ccc(Cl)c(Nc2nc3ccccc3nc2NS(=O)(=O)c2cccc(NC(=O)C(C)(C)N)c2)c1
Oc1cccc(c1)-c1cc2c3cccnc3oc2c(n1)N1CCOCC1
Cc1c(sc2c1nc(nc2N3CCOCC3)c4cnc(nc4)N)CN5CCN(CC5)C(=O)[C@H](C)O
CS(=O)(=O)N1CCN(Cc2cc3nc(nc(N4CCOCC4)c3s2)-c2cccc3[nH]ncc23)CC1
CN(C)C1CCN(CC1)C(=O)c1ccc(NC(=O)Nc2ccc(cc2)-c2nc(nc(n2)N2CCOCC2)N2CCOCC2)cc1
Nc1ncc(-c2nc(nc(n2)N2CCOCC2)N2CCOCC2)c(n1)C(F)(F)F
Nc1cc(c(cn1)-c1nc(nc(n1)N1CCOCC1)N1CCOCC1)C(F)(F)F
Nc1cc(c(cn1)-c1cc(nc(n1)N1CCOCC1)N1CCOCC1)C(F)(F)F
Nc1ccc(cn1)-c1ccc2ncc3ncc(=O)n(C4CCN(CC#N)CC4)c3c2c1
Cc1ccc2c(oc(nc2=O)N2CCOCC2)c1-c1cccc2c3ccccc3sc12 |(49.53,-8.74,;50.86,-9.51,;50.86,-11.06,;52.2,-11.83,;53.53,-11.05,;53.53,-9.5,;54.87,-8.73,;56.21,-9.51,;56.2,-11.06,;54.86,-11.82,;54.86,-13.37,;57.54,-8.74,;58.87,-9.52,;60.21,-8.76,;60.22,-7.22,;58.89,-6.44,;57.54,-7.2,;52.19,-8.74,;52.19,-7.2,;53.53,-6.42,;53.52,-4.88,;52.18,-4.13,;50.85,-4.9,;49.39,-4.44,;48.76,-3.04,;47.24,-2.89,;46.34,-4.14,;46.97,-5.53,;48.49,-5.68,;49.4,-6.92,;50.86,-6.44,)|
O=C1NC(=O)c2c1c1cncn1c1[nH]c3ccccc3c21
COc1cc(cnc1OC)-c1ccc2C(=O)N([C@H](C)c2n1)c1cnn(CC(F)(F)F)c1 |r|
Oc1cc(N2CCOCC2)c(-c2ccccc2)c2oc(cc(=O)c12)-c1ccccc1
CCC(=O)N1CC[C@@H](C1)Nc2c3c(ncn2)CCN(C3)c4cc(c(nc4)OC)C(F)(F)F
C[C@H]1Cc2ccccc2N1C(=O)CC3=NC(=CC(=O)N3)N4CCOCC4
CNC(=O)c1nnc2ccc(cc2c1N[C@@H](C)C1CCOCC1)-c1ccc(OCCCN(C)C)nc1 |r|
C[C@H](Nc1c(nnc2ccc(cc12)-c1ccc(OCCCN(C)C)nc1)C(N)=O)C1CCOCC1 |r|
CN(C)CCCOc1ccc(cn1)-c1ccc2ncc3n(C)c(=O)n(C4CCOCC4)c3c2c1
O=C(Cc1cccc(OCCCC2CCNCC2)c1)Nc1nc(cs1)-c1c[nH]c2ncccc12
CN1CCN(CCCOc2cccc(CC(=O)Nc3nc(cs3)-c3c[nH]c4ncccc34)c2)CC1
CS(=O)(=O)Nc1cccc(CC(=O)Nc2nc(cs2)-c2c[nH]c3ncccc23)c1
C[C@@H]1COCCN1c1cc(nc(n1)-c1cncc2[nH]ccc12)C1(CC1)S(C)(=O)=O |r|
C[C@@H]1COCCN1c1cc(nc(n1)-c1ccnc2[nH]ccc12)C1(CC1)[S@](C)(=N)=O |r|
CNc1nc2ccccc2n1-c1nc(cc(n1)C1(CC1)S(C)(=O)=O)N1CCOC[C@H]1C |r|
CNc1nc2ccccc2n1-c1nc(cc(n1)C1(CC1)[S@](C)(=N)=O)N1CCOC[C@H]1C |r|
C[C@@H]1C[C@H]1C(=O)N1CCN(C[C@H]1C)c1cnc(C#N)c(n1)-c1cnn(C)c1 |r|
Cc1cc2c(cccc2n1-c1nc2CCOCc2c(NCc2ccccc2)n1)C(N)=O
CN(C)C(=O)c1cc(CN2CCOc3c(F)cccc23)c2oc(cc(=O)c2c1)N1CCOCC1
C[C@@H](C1=Cc2cccc(c2C(=O)N1c3ccccc3)C#Cc4cnn(c4)C)NC(=O)c5c(nn6c5nccc6)N
CC(C)S(=O)(=O)c1ccc(cc1)-c1cnc(N)c(n1)-c1cc(no1)-c1ccc(cc1)[C@H](C)N |r|
CC(C)S(=O)(=O)c1ccc(cc1)-c1cnc(N)c(n1)-c1nnc(o1)-c1ccccc1
CNCc1ccc(-c2cc(on2)-c2nc(cnc2N)-c2ccc(cc2)S(=O)(=O)C(C)C)c(Cl)c1
CC(C)S(=O)(=O)c1ccc(cc1)-c1cnc(N)c(n1)-c1cc(no1)-c1ccc(cc1)[C@@H](C)N |r|
CC(C)S(=O)(=O)c1ccc(cc1)-c1cnc(N)c(n1)-c1cc(no1)-c1ccc(CNC2CCOCC2)cc1
CNCc1ccc(cc1)-c1cc(on1)-c1nc(cnc1N)-c1ccc(cc1)S(=O)(=O)C(C)C
CC(C)S(=O)(=O)c1ccc(cc1)-c1cnc(N)c(n1)-c1cc(no1)-c1ccc(CN)cc1
CC(C)S(=O)(=O)c1ccc(cc1)-c1cnc(N)c(n1)-c1nnc(s1)-c1ccccc1
CC(C)S(=O)(=O)c1ccc(cc1)-c1cnc(N)c(n1)-c1noc(n1)-c1ccccc1
CC(C)S(=O)(=O)c1ccc(cc1)-c1cnc(N)c(n1)-c1cc(on1)-c1ccccc1
CC(C)S(=O)(=O)c1ccc(cc1)-c1cnc(N)c(n1)C1CC(=NO1)c1ccccc1 |c:23|
CC(C)S(=O)(=O)c1ccc(cc1)-c1cnc(N)c(n1)-c1ncc(o1)-c1ccccc1
CNCc1ccc(cc1Cl)-c1cc(on1)-c1nc(cnc1N)-c1ccc(cc1)S(=O)(=O)C(C)C
CCNCc1ccc(cc1)-c1cc(on1)-c1nc(cnc1N)-c1ccc(cc1)S(=O)(=O)C(C)C
CC(C)S(=O)(=O)c1ccc(cc1)-c1cnc(N)c(n1)-c1cnc(o1)-c1ccccc1
CC(C)S(=O)(=O)c1ccc(cc1)-c1cnc(N)c(n1)-c1cn(nn1)-c1ccccc1
CC(C)S(=O)(=O)c1ccc(cc1)-c1cnc(N)c(n1)-c1nc(no1)-c1ccccc1
CC(C)S(=O)(=O)c1ccc(cc1)-c1cnc(N)c(n1)-c1cc(no1)-c1ccccc1
CN(C)c1ccc(cc1)C(=O)Nc1cccc(NC(=O)COc2ccc3c(c2)occc3=O)c1
C[C@H]1COCCN1c1nc(N2CCOC[C@H]2C)c2nc(sc2n1)-c1cc[nH]n1 |r|
COc1ccc(Nc2ncc3n(C)c(=O)n(-c4ccccc4)c3n2)c(C)c1
Cc1cc(ccc1Nc2ncc3c(n2)N(C(=O)N3C)C4CCC(CC4)O)OC
Cc1ccccc1Nc1ncc2n(C)c(=O)n([C@H]3CC[C@H](O)CC3)c2n1 |r,wU:20.21,wD:17.17,(63.68,-26.71,;63.69,-25.17,;65.03,-24.41,;65.04,-22.86,;63.69,-22.09,;62.36,-22.86,;62.37,-24.39,;61.03,-25.16,;59.7,-24.39,;58.37,-25.16,;57.03,-24.4,;57.03,-22.84,;55.88,-21.81,;54.38,-22.13,;56.51,-20.4,;55.74,-19.06,;58.04,-20.56,;59.06,-19.41,;60.57,-19.73,;61.59,-18.59,;61.12,-17.13,;62.15,-15.99,;59.62,-16.81,;58.58,-17.95,;58.37,-22.07,;59.71,-22.85,)|
Cn1c2cnc(Nc3ccccc3)nc2n([C@H]2CC[C@H](O)CC2)c1=O |r,wU:19.21,wD:16.17,(29.71,-38.04,;31.22,-37.72,;32.36,-38.76,;32.37,-40.31,;33.7,-41.07,;35.03,-40.3,;36.36,-41.07,;37.7,-40.3,;39.02,-41.08,;40.36,-40.32,;40.37,-38.77,;39.02,-38,;37.69,-38.77,;35.04,-38.76,;33.7,-37.98,;33.37,-36.47,;34.39,-35.32,;35.9,-35.64,;36.92,-34.51,;36.45,-33.04,;37.48,-31.91,;34.95,-32.72,;33.91,-33.87,;31.84,-36.31,;31.07,-34.98,)|
COc1ccc(C)c(Nc2ncc3n(C)c(=O)n([C@H]4CC[C@H](O)CC4)c3n2)c1 |r,wU:21.21,wD:18.17,(65.59,-35.67,;64.26,-36.43,;64.26,-37.97,;65.61,-38.75,;65.6,-40.29,;64.26,-41.06,;64.25,-42.6,;62.93,-40.28,;61.59,-41.05,;60.26,-40.28,;58.93,-41.04,;57.6,-40.28,;57.59,-38.73,;56.44,-37.69,;54.94,-38.01,;57.07,-36.28,;56.3,-34.94,;58.6,-36.44,;59.63,-35.29,;61.13,-35.61,;62.16,-34.48,;61.69,-33.01,;62.72,-31.87,;60.18,-32.69,;59.15,-33.83,;58.93,-37.95,;60.27,-38.73,;62.93,-38.74,)|
Cc1cc2nccn2cc1Nc1ncc2n(C)c(=O)n(C3CCOCC3)c2n1
COc1ccc(Nc2ncc3n(C)c(=O)n(C4CCCCC4)c3n2)c(C)c1
COc1ccc(Nc2ncc3n(C)c(=O)n([C@H]4CC[C@H](O)CC4)c3n2)cc1 |r,wU:19.19,wD:16.15,(17.81,-39.24,;16.48,-38.47,;15.15,-39.24,;15.15,-40.78,;13.81,-41.55,;12.48,-40.77,;11.14,-41.53,;9.81,-40.76,;8.49,-41.53,;7.15,-40.77,;7.15,-39.22,;6,-38.19,;4.5,-38.51,;6.63,-36.78,;5.86,-35.44,;8.16,-36.94,;9.18,-35.79,;10.68,-36.11,;11.71,-34.97,;11.24,-33.51,;12.27,-32.37,;9.73,-33.19,;8.7,-34.33,;8.48,-38.45,;9.82,-39.22,;12.48,-39.23,;13.81,-38.46,)|
Cc1c(Nc2ncc3n(C)c(=O)n([C@H]4CC[C@H](O)CC4)c3n2)ccc2nccn12 |r,wU:16.16,wD:13.12,(36.89,-53.69,;38.22,-54.46,;38.22,-55.99,;36.88,-56.76,;35.56,-55.99,;34.23,-56.76,;32.89,-56,;32.89,-54.45,;31.74,-53.41,;30.24,-53.73,;32.37,-52,;31.6,-50.67,;33.9,-52.16,;34.92,-51.01,;36.43,-51.33,;37.45,-50.2,;36.98,-48.73,;38.01,-47.6,;35.48,-48.41,;34.44,-49.56,;34.23,-53.67,;35.57,-54.45,;39.55,-56.77,;40.89,-56.01,;40.89,-54.46,;42.04,-53.42,;41.4,-52.01,;39.87,-52.18,;39.55,-53.69,)|
Cc1cc2ncnn2cc1Nc1ncc2n(C)c(=O)n(C3CCC(F)(F)CC3)c2n1
COc1ccc(Nc2ncc3n(C)c(=O)n(C4CCCC4)c3n2)c(C)c1
Cc1cc2nccn2cc1Nc1ncc2n(C)c(=O)n([C@H]3CC[C@H](O)CC3)c2n1 |r,wU:23.25,wD:20.21,(64.98,-58.36,;64.99,-56.83,;66.33,-56.06,;66.33,-54.51,;67.47,-53.48,;66.84,-52.07,;65.31,-52.23,;64.99,-53.74,;63.66,-54.51,;63.66,-56.05,;62.32,-56.81,;60.99,-56.04,;59.67,-56.81,;58.33,-56.05,;58.33,-54.5,;57.18,-53.47,;55.68,-53.79,;57.81,-52.06,;57.04,-50.72,;59.34,-52.22,;60.36,-51.07,;61.86,-51.39,;62.89,-50.25,;62.42,-48.79,;63.45,-47.65,;60.91,-48.47,;59.88,-49.61,;59.66,-53.73,;61,-54.5,)|
Cn1c2cnc(Nc3ccc4nccn4c3)nc2n([C@H]2CC[C@H](O)CC2)c1=O |r,wU:22.25,wD:19.21,(4.91,-54.43,;6.41,-54.11,;7.56,-55.15,;7.56,-56.7,;8.9,-57.46,;10.22,-56.69,;11.55,-57.46,;12.89,-56.69,;14.22,-57.47,;15.56,-56.71,;15.56,-55.16,;16.7,-54.12,;16.07,-52.71,;14.54,-52.88,;14.22,-54.39,;12.89,-55.16,;10.23,-55.15,;8.89,-54.37,;8.57,-52.86,;9.59,-51.71,;11.09,-52.03,;12.12,-50.9,;11.65,-49.44,;12.68,-48.3,;10.14,-49.11,;9.11,-50.26,;7.04,-52.7,;6.27,-51.37,)|
Cn1c2cnc(Nc3ccc4ncnn4c3)nc2n([C@H]2CC[C@H](O)CC2)c1=O |r,wU:22.25,wD:19.21,(3.6,-8.19,;5.1,-7.87,;6.25,-8.9,;6.25,-10.46,;7.59,-11.22,;8.91,-10.45,;10.24,-11.22,;11.58,-10.45,;12.91,-11.23,;14.25,-10.47,;14.25,-8.92,;15.39,-7.88,;14.76,-6.47,;13.23,-6.64,;12.91,-8.15,;11.58,-8.92,;8.92,-8.91,;7.58,-8.13,;7.26,-6.62,;8.28,-5.47,;9.78,-5.79,;10.81,-4.66,;10.34,-3.19,;11.37,-2.05,;8.83,-2.87,;7.8,-4.02,;5.73,-6.46,;4.96,-5.12,)|
COc1ccc(Nc2ncc3[nH]c(=O)n([C@H]4CC[C@H](O)CC4)c3n2)c(C)c1 |r,wU:18.18,wD:15.14,(42.18,-22.41,;40.84,-21.64,;39.51,-22.42,;38.17,-21.65,;36.84,-22.42,;36.84,-23.97,;35.5,-24.73,;34.17,-23.97,;32.85,-24.73,;31.52,-23.97,;31.51,-22.42,;30.37,-21.39,;30.99,-19.99,;30.22,-18.65,;32.52,-20.15,;33.54,-19.01,;35.04,-19.33,;36.06,-18.19,;35.59,-16.73,;36.62,-15.59,;34.09,-16.41,;33.06,-17.55,;32.84,-21.65,;34.18,-22.43,;38.17,-24.74,;38.17,-26.28,;39.51,-23.97,)|
CCC(CC)CNc1c(cnc2ccc(cc12)C#N)C(N)=O
COc1cc2ncnc(-n3nc(nc3N)-c3ccccn3)c2cc1OC
C[C@@H](Nc1c(cnc2ccc(cc12)C#N)C(N)=O)c1ccc(Cl)cc1 |r|
C[C@@H](Nc1c(cnc2ccc(cc12)-c1cccnc1)C(N)=O)c1ccc(Cl)cc1 |r|
COCc1ccc(cn1)-c1ccc2ncc(C(N)=O)c(N[C@@H](C)C3CCOCC3)c2c1 |r|
COCc1ccc(cn1)-c1cc2c(N[C@@H](C)c3ccn(C)n3)c(cnc2cc1F)C(N)=O |r|
O=c1cc(oc(c1)-c1cccc2Cc3ccccc3Sc12)N1CCOCC1
COc1ncc(cc1NS(C)(=O)=O)-c1cc2COCc2c(NC(=O)CN2CCOCC2)c1
C[C@@H]1COCCN1c1cc(-c2ccnn2C)c2ccnc(-c3ccn[nH]3)c2n1 |r|
Cc1nc(NC(=O)NCCc2cn(CC(F)F)cn2)sc1C#Cc1cccnc1
COc1cc(cnc1OC)C#Cc1sc(NC(=O)NCCOCC2CC2)nc1C
Cc1nc(NC(=O)NCCOCC2CC2)sc1C#Cc1ccc2cncn2c1
C[C@@H](CNC(=O)Nc1nc(C)c(s1)C#Cc1cncc(C)c1)OCC1CC1 |r|
C[C@@H](CNC(=O)Nc1nc(C)c(s1)C#Cc1cnc(C)c(C)c1)OCC1CC1 |r|
C[C@H]1CN(CC(=O)Nc2ccc3Sc4c(Cc3c2)cccc4-c2cc(=O)cc(o2)N2CCOCC2)C[C@@H](C)O1
COc1ccc2Sc3c(Cc2c1)cccc3-c1cc(=O)cc(o1)N1CCOCC1
C[C@H](CN1C[C@H](C)O[C@H](C)C1)Oc1ccc2Sc3c(Cc2c1)cccc3-c1cc(=O)cc(o1)N1CCOCC1 |r|
C[C@H](CN1CCOCC1)Oc2ccc3c(c2)Cc4cccc(c4S3)C5=CC(=O)C=C(O5)N6CCOCC6
COC[C@@H](C)Oc1ccc2Sc3c(Cc2c1)cccc3-c1cc(=O)cc(o1)N1CCOCC1 |r|
O=c1cc(oc(c1)-c1cccc2Cc3cc(OC4COC4)ccc3Sc12)N1CCOCC1
Nc1ccc(cn1)-c1nc(N2CCOCC2)c2ncn(CCCCCCC(=O)NO)c2n1
OCc1cccc(c1)-c1nc(N2CCOCC2)c2ncn(CCCCCCC(=O)NO)c2n1
Nc1ncc(cn1)-c1nc(N2CCOCC2)c2ncn(CCCCCCC(=O)NO)c2n1
COc1ncc(cn1)-c1nc(N2CCOCC2)c2ncn(CCCCCCC(=O)NO)c2n1
Nc1ncc(cn1)-c1nc(N2CCOCC2)c2ccn(CCCCCCC(=O)NO)c2n1
COc1ccc(cn1)-c1nc(N2CCOCC2)c2sc(CN(C)c3ncc(cn3)C(=O)NO)cc2n1
O=c1cc(cc([nH]1)N1CCCCC[C@@H]1Cc1ccccc1)N1CCOCC1 |r|
[H][C@]12C[C@@]1([H])[C@H](Cc1ccccc1)N(C2)c1cc(cc(=O)[nH]1)N1CCOCC1 |r|
[H][C@@]12C[C@]1([H])[C@H](Cc1ccccc1)N(C2)c1cc(cc(=O)[nH]1)N1CCO[C@H](C)C1 |r|
C[C@@H]1CCN([C@H]1Cc1ccccc1)c1nc(cc(=O)[nH]1)N1CCOCC1 |r|
CN(C)C\C=C\C(=O)Nc1ccc(O[C@@H]2CCC[C@H](C2)Nc2ncc(Cl)c(n2)-c2c[nH]c3ccccc23)cc1 |r|
OCc1cccc(c1)-c1ccc2ncc3nnc(C4CCOCC4)n3c2c1
CN(C)CCCOc1ccc(cn1)-c1ccc2ncc3nnc(C4CCOCC4)n3c2c1
FC(F)c1cccc(c1)-c1ccc2ncc3nnc(C4CCOCC4)n3c2c1
FC(F)c1ccc(cc1)-c1ccc2ncc3nnc(C4CCOCC4)n3c2c1
Clc1cccc(c1)-c1ccc2ncc3nnc(C4CCOCC4)n3c2c1
FC(F)(F)Oc1cccc(c1)-c1ccc2ncc3nnc(C4CCOCC4)n3c2c1
NS(=O)(=O)c1cccc(c1)-c1ccc2ncc3nnc(C4CCOCC4)n3c2c1
CS(=O)(=O)c1ccc(F)c(c1)-c1ccc2ncc3nnc(C4CCOCC4)n3c2c1
CS(=O)(=O)c1cccc(c1)-c1ccc2ncc3nnc(C4CCOCC4)n3c2c1
Cc1cncc(c1)-c1ccc2ncc3nnc(C4CCOCC4)n3c2c1
FC(F)c1cncc(c1)-c1ccc2ncc3nnc(C4CCOCC4)n3c2c1
NS(=O)(=O)c1cncc(c1)-c1ccc2ncc3nnc(C4CCOCC4)n3c2c1
CS(=O)(=O)c1cncc(c1)-c1ccc2ncc3nnc(C4CCOCC4)n3c2c1
FC(F)(F)c1cncc(c1)-c1ccc2ncc3nnc(C4CCOCC4)n3c2c1
Cc1cc(cnc1F)-c1ccc2ncc3nnc(C4CCOCC4)n3c2c1
Cc1nc2ccc(cc2n2c(nnc12)C1CCOCC1)-c1cncc(c1)C(F)F
FC(F)c1cncc(c1)-c1ccc2ncc3nnc(C4CCOCC4)n3c2c1F
FC(F)c1cncc(c1)-c1cc(F)c2ncc3nnc(C4CCOCC4)n3c2c1
FC(F)c1cncc(c1)-c1ccc2ncc3[nH]nc(C4CCOCC4)c3c2c1
Cn1nc(C2CCOCC2)c2c1cnc1ccc(cc21)-c1cncc(c1)C(F)F
Cn1nc2cnc3ccc(cc3c2c1C1CCOCC1)-c1cncc(c1)C(F)F
Cc1nc(C2CCOCC2)n2c1cnc1ccc(cc21)-c1cncc(c1)C(F)F
[H][C@@]12COC[C@]1([H])[C@H]2c1nnc2cnc3ccc(cc3n12)-c1cncc(c1)C(F)F |r|
FC(F)c1cncc(c1)-c1ccc2ncc3nnc(C4=CCOCC4)n3c2c1 |t:20|
FC(F)c1cncc(c1)-c1ccc2ncc3nnc(C4=CCCOCC4)n3c2c1 |t:20|
[H][C@@]12CCC[C@]1([H])[C@H]2c1nnc2cnc3ccc(cc3n12)-c1cncc(c1)C(F)F |r|
FC(F)c1cncc(c1)-c1ccc2ncc3nnc(C4=CCCCC4)n3c2c1 |t:20|
FC(F)c1cncc(c1)-c1ccc2ncc3nnc(C4=CCCCCC4)n3c2c1 |t:20|
CO[C@H]1CC[C@H](CC1)c1nnc2cnc3ccc(cc3n12)-c1cncc(c1)C(F)F |r,wU:5.8,2.1,(26.22,-45.52,;25.75,-46.98,;26.79,-48.11,;28.29,-47.78,;29.33,-48.92,;28.86,-50.39,;27.36,-50.72,;26.32,-49.58,;29.9,-51.52,;31.42,-51.35,;32.06,-52.74,;30.93,-53.78,;30.94,-55.33,;29.61,-56.11,;28.27,-55.34,;26.93,-56.12,;25.6,-55.34,;25.6,-53.8,;26.93,-53.03,;28.27,-53.79,;29.6,-53.02,;24.27,-53.03,;22.94,-53.8,;21.61,-53.04,;21.61,-51.49,;22.94,-50.72,;24.27,-51.49,;22.94,-49.19,;24.26,-48.42,;21.61,-48.42,)|
CO[C@H]1CC[C@@H](CC1)c1nnc2cnc3ccc(cc3n12)-c1cncc(c1)C(F)F |r,wU:5.8,wD:2.1,(43.27,-45.09,;42.81,-46.55,;43.84,-47.68,;43.38,-49.15,;44.41,-50.29,;45.91,-49.96,;46.38,-48.49,;45.35,-47.35,;46.95,-51.09,;48.48,-50.92,;49.11,-52.31,;47.98,-53.34,;48,-54.9,;46.66,-55.68,;45.32,-54.91,;43.99,-55.69,;42.65,-54.91,;42.66,-53.37,;43.99,-52.6,;45.32,-53.36,;46.65,-52.59,;41.32,-52.6,;40,-53.37,;38.67,-52.61,;38.66,-51.06,;39.99,-50.29,;41.33,-51.06,;39.99,-48.76,;41.32,-47.99,;38.66,-47.99,)|
c1cc(oc1)c2nc3c4cc(ccc4nc(n3n2)N)Cl
Cc1cc2c(c(c1)[C@H](C)Nc3ccccc3)OC(=CC2=O)N4CCOCC4
CN1C(=O)CN(C2CCOCC2)c2nc(Nc3cn4ncnc4cc3C)ncc12
CN1C(=O)C2(CCOCC2)c2nc(Nc3cc4cccnc4cc3C)ncc12
CN1C(=O)CN(C2CCOCC2)c2nc(Nc3cc4nccnc4cc3C)ncc12
CN1C(=O)CN(C2CCOCC2)c2nc(Nc3cc4cccnc4cc3C)ncc12
Cc1cc2ncnn2cc1Nc1ncc2NC(=O)CN(C3CCOCC3)c2n1
CCN1C(=O)CN(C2CCOCC2)c2nc(Nc3cn4ncnc4cc3C)ncc12
CC(C)N1C(=O)CN(C2CCOCC2)c2nc(Nc3cn4ncnc4cc3C)ncc12
Cc1cc2ncnn2cc1Nc1ncc2N(C3CC3)C(=O)CN(C3CCOCC3)c2n1
CN1C(=O)C2(CCC(CC2)OCC(F)F)c2nc(Nc3cn4ncnc4cc3C)ncc12
CC(C)N1C(=O)C2(CCOCC2)c2nc(Nc3cn4ncnc4cc3C)ncc12
CCN1C(=O)C2(CCOCC2)c2nc(Nc3cn4ncnc4cc3C)ncc12
CN1C(=O)C2(CCC2)c2nc(Nc3cn4ncnc4cc3C)ncc12
CN1C(=O)C(C)(C)c2nc(Nc3cn4ncnc4cc3C)ncc12
[2H]C([2H])([2H])N1C(=O)C2(CCOCC2)c2nc(Nc3cn4ncnc4cc3C)ncc12
CN1C(=O)C2(CCC(C)(C)CC2)c2nc(Nc3cn4ncnc4cc3C)ncc12
CN1C(=O)C2(CCC3(CC3)CC2)c2nc(Nc3cn4ncnc4cc3C)ncc12
Cc1cc2ncnn2cc1Nc1ncc2n(C)c(=O)n(N3CC4CCC(C3)O4)c2n1
Cc1cc2ncnn2cc1Nc1ncc2n(C)c(=O)n(N3CCOCC3)c2n1
C[C@H](CNc1cc(ncn1)-c1cnc(C)nc1)c1cccc2c(ccnc12)-c1noc(=O)[nH]1 |r|
C[C@@H](CNc1cc(ncn1)-c1cnc(C)nc1)c1cccc2c(ccnc12)C1=NCCN1 |r,t:31|
COc1ccc(Nc2cc(c(F)cc2Cl)-c2ncnc3cc(ccc23)N2CCOCC2)nn1
COc1ccc(nn1)C1(CC1)c1cc(c(F)cc1Cl)-c1ncnc2cc(ccc12)N1CCOCC1
CN(C)CCCOc1ncc(cc1NS(=O)(=O)C(F)(F)F)-c1ccc2ncc3N(C)C(=O)C4(CCC4)c3c2c1
C[C@@H]1CN(CCO1)c1cc(O[C@@H]2CC[C@@H](CC2)Nc2ncccn2)c2nccnc2c1 |r,wU:11.11,14.18,1.0,(6.01,-5,;4.68,-4.23,;4.68,-2.69,;3.35,-1.92,;2.01,-2.69,;2.01,-4.23,;3.35,-5,;3.35,-.38,;2.01,.38,;1.99,1.91,;.66,2.68,;-.67,1.91,;-2.01,2.68,;-3.34,1.91,;-3.34,.37,;-2.01,-.4,;-.67,.37,;-4.67,-.4,;-4.67,-1.94,;-3.34,-2.71,;-3.34,-4.24,;-4.68,-5.01,;-6,-4.25,;-6.01,-2.71,;3.33,2.7,;3.33,4.24,;4.66,5.01,;5.99,4.24,;5.99,2.7,;4.67,1.93,;4.67,.4,)|
Fc1cnc(N[C@H]2CC[C@H](CC2)Oc2cc(cc3nccnc23)N2CCOCC2)[nH]c1=O |r,wU:9.12,6.5,(-4.67,-5.78,;-4.67,-4.24,;-5.99,-3.48,;-6,-1.94,;-4.66,-1.17,;-4.66,.37,;-3.33,1.14,;-3.33,2.68,;-2,3.45,;-.66,2.68,;-.66,1.14,;-2,.37,;.67,3.45,;2,2.68,;2.02,1.15,;3.36,.39,;4.68,1.17,;4.68,2.7,;6,3.47,;6,5.01,;4.67,5.78,;3.34,5.01,;3.34,3.47,;3.36,-1.15,;4.69,-1.92,;4.69,-3.46,;3.36,-4.23,;2.02,-3.46,;2.02,-1.92,;-3.33,-1.94,;-3.33,-3.47,;-2,-4.24,)|
CN1CCC(CC1)n1c2nc(Nc3cn4ncnc4cc3C)ncc2n(C)c1=O
Cc1cc2ncccc2cc1Nc1ncc2n(C)c(=O)n([C@H]3CCN(CCO)C3)c2n1 |r|
COCCN1CC[C@@H](C1)n1c2nc(Nc3cc4cccnc4cc3C)ncc2n(C)c1=O |r|
Cc1cc2ncccc2cc1Nc1ncc2n(C)c(=O)n([C@H]3CCN(C3)C3COC3)c2n1 |r|
CN1C[C@@H](F)[C@@H](C1)n1c2nc(Nc3cc4cccnc4cc3C)ncc2n(C)c1=O |r|
CN1C[C@H](F)[C@@H](C1)n1c2nc(Nc3cc4cccnc4cc3C)ncc2n(C)c1=O |r|
Cc1cc2ncccc2cc1Nc1ncc2n(C)c(=O)n([C@@H]3CNC[C@@H]3F)c2n1 |r|
O=c1cc(oc2c(csc12)-c1ccc2OCCOc2c1)N1CCOCC1
CC(C)n1nc2ncnc(N)c2c1C1C=c2cc(O)ccc2=N1 |c:24,t:16|
C[C@H](c1ccccc1)n1nnc2cnc3ccc(cc3c12)-c1ccc(OCCCN(C)C)nc1 |r|
Oc1cc(cc2n(Cc3ccccc3)c3ccccc3c(=O)c12)N1CCOCC1
C[C@@H]1COCCN1c1nc(nc2c1CN(C(=O)c1ccc3OCOc3c1)C2(C)C)-c1cccc2[nH]ccc12 |r|
C[C@@H]1COCCN1c1nc(nc2c1CN(C(=O)c1cccc(c1)S(C)(=O)=O)C2(C)C)-c1cccc2[nH]ccc12 |r|
CC(C)NC(=O)N(C)c1cnc2ccc(cc2n1)-c1ccc(OCCCN2CCCCC2)nc1
Cn1c2cnc3ccc(cc3c2n(-c2ccc(cc2)C(C)(C)C#N)c1=O)-c1cnc2ccccc2c1
Cn1c(=O)n(C2CCCC2)c2cc(Nc3ccccc3)ncc21
Cc1ccc(Nc2cc3c(cn2)n(C)c(=O)n3C2CCCC2)cc1
Cc1cccc(Nc2cc3c(cn2)n(C)c(=O)n3C2CCCC2)c1
Cc1ccccc1Nc1cc2c(cn1)n(C)c(=O)n2C1CCCC1
COc1ccc(Nc2cc3c(cn2)n(C)c(=O)n3C2CCCC2)cc1
COc1cccc(Nc2cc3c(cn2)n(C)c(=O)n3C2CCCC2)c1
COc1ccccc1Nc1cc2c(cn1)n(C)c(=O)n2C1CCCC1
Cn1c(=O)n(C2CCCC2)c2cc(Nc3ccc(Cl)cc3)ncc21
Cn1c(=O)n(C2CCCC2)c2cc(Nc3cccc(Cl)c3)ncc21
Cn1c(=O)n(C2CCCC2)c2cc(Nc3ccccc3Cl)ncc21
Cn1c(=O)n(C2CCCC2)c2cc(Nc3ccc([N+](=O)[O-])cc3)ncc21
Cn1c(=O)n(C2CCCC2)c2cc(Nc3cccc([N+](=O)[O-])c3)ncc21
Cn1c(=O)n(C2CCCC2)c2cc(Nc3ccccc3[N+](=O)[O-])ncc21
Cn1c(=O)n(C2CCCC2)c2cc(Nc3ccc(N)cc3)ncc21
Cn1c(=O)n(C2CCCC2)c2cc(Nc3cccc(N)c3)ncc21
Cn1c(=O)n(C2CCCC2)c2cc(Nc3ccccc3N)ncc21
CC(=O)Nc1ccc(Nc2cc3c(cn2)n(C)c(=O)n3C2CCCC2)cc1
CC(=O)Nc1cccc(Nc2cc3c(cn2)n(C)c(=O)n3C2CCCC2)c1
CC(=O)Nc1ccccc1Nc1cc2c(cn1)n(C)c(=O)n2C1CCCC1
Cn1c(=O)n(C2CCCC2)c2cc(Nc3ccc(C#N)cc3)ncc21
Cn1c(=O)n(C2CCCC2)c2cc(Nc3cccc(C#N)c3)ncc21
Cn1c(=O)n(C2CCCC2)c2cc(Nc3ccccc3C#N)ncc21
Cn1c(=O)n(C2CCCC2)c2cc(Nc3ccc(C(F)(F)F)cc3)ncc21
Cn1c(=O)n(C2CCCC2)c2cc(Nc3cccc(C(F)(F)F)c3)ncc21
Cn1c(=O)n(C2CCCC2)c2cc(Nc3ccccc3C(F)(F)F)ncc21
CC(=O)c1ccc(Nc2cc3c(cn2)n(C)c(=O)n3C2CCCC2)cc1
CC(=O)c1cccc(Nc2cc3c(cn2)n(C)c(=O)n3C2CCCC2)c1
Cn1c(=O)n(C2CCCC2)c2cc(Nc3ccc(S(C)(=O)=O)cc3)ncc21
Cn1c(=O)n(C2CCCC2)c2cc(Nc3cccc(S(C)(=O)=O)c3)ncc21
Cn1c(=O)n(C2CCCC2)c2cc(Nc3ccccc3S(C)(=O)=O)ncc21
Cn1c(=O)n(C2CCCC2)c2cc(Nc3ccc(OCc4ccccc4)cc3)ncc21
Cn1c(=O)n(C2CCCC2)c2cc(Nc3cccc(OCc4ccccc4)c3)ncc21
Cn1c(=O)n(C2CCCC2)c2cc(Nc3ccccc3OCc3ccccc3)ncc21
Cn1c(=O)n(C2CCCC2)c2cc(Nc3ccc(O)cc3)ncc21
Cn1c(=O)n(C2CCCC2)c2cc(Nc3cccc(O)c3)ncc21
Cn1c(=O)n(C2CCCC2)c2cc(Nc3ccccc3O)ncc21
Cn1c(=O)n(C2CCCC2)c2cc(Nc3ccc(C(C)(C)C#N)cc3)ncc21
Cc1ccc(Nc2cc3c(cn2)n(C)c(=O)n3C2CCCC2)c(C)c1
Cc1cccc(Nc2cc3c(cn2)n(C)c(=O)n3C2CCCC2)c1C
Cc1ccc(Nc2cc3c(cn2)n(C)c(=O)n3C2CCCC2)cc1C
Cc1c(Cl)cccc1Nc1cc2c(cn1)n(C)c(=O)n2C1CCCC1
Cc1cc(Cl)ccc1Nc1cc2c(cn1)n(C)c(=O)n2C1CCCC1
Cc1ccc(Cl)cc1Nc1cc2c(cn1)n(C)c(=O)n2C1CCCC1
Cc1cc(S(C)(=O)=O)ccc1Nc1cc2c(cn1)n(C)c(=O)n2C1CCCC1
Cc1ccc(S(C)(=O)=O)cc1Nc1cc2c(cn1)n(C)c(=O)n2C1CCCC1
Cc1cc(C#N)ccc1Nc1cc2c(cn1)n(C)c(=O)n2C1CCCC1
Cc1cc(Nc2cc3c(cn2)n(C)c(=O)n3C2CCCC2)ccc1C#N
COc1ccc(Nc2cc3c(cn2)n(C)c(=O)n3C2CCCC2)c(C)c1
COc1ccc(C)c(Nc2cc3c(cn2)n(C)c(=O)n3C2CCCC2)c1
Cc1cc(OCc2ccccc2)ccc1Nc1cc2c(cn1)n(C)c(=O)n2C1CCCC1
Cc1cc(O)ccc1Nc1cc2c(cn1)n(C)c(=O)n2C1CCCC1
Cc1cc(F)ccc1Nc1cc2c(cn1)n(C)c(=O)n2C1CCCC1
Cc1cc(OC(F)(F)F)ccc1Nc1cc2c(cn1)n(C)c(=O)n2C1CCCC1
Cc1cc(OC(F)F)ccc1Nc1cc2c(cn1)n(C)c(=O)n2C1CCCC1
CCOc1ccc(Nc2cc3c(cn2)n(C)c(=O)n3C2CCCC2)c(C)c1
Cc1cc(OCCN(C)C)ccc1Nc1cc2c(cn1)n(C)c(=O)n2C1CCCC1
Cc1cc(N2CCOCC2)ccc1Nc1cc2c(cn1)n(C)c(=O)n2C1CCCC1
Cc1cc(N2CCN(C)CC2)ccc1Nc1cc2c(cn1)n(C)c(=O)n2C1CCCC1
COc1ccc(Nc2cc3c(cn2)n(C)c(=O)n3C2CCCC2)c(C(F)(F)F)c1
COc1ccc(Nc2cc3c(cn2)n(C)c(=O)n3C2CCCC2)c(C#N)c1
COc1ccc(Nc2cc3c(cn2)n(C)c(=O)n3C2CCCC2)c(Cl)c1
COc1ccc(Nc2cc3c(cn2)n(C)c(=O)n3C2CCCC2)c(OC)c1
COc1ccc(N(C)c2cc3c(cn2)n(C)c(=O)n3C2CCCC2)c(C)c1
COCCn1c(=O)n(C2CCCC2)c2cc(Nc3ccc(OC)cc3C)ncc21
COc1ccc(Nc2cc3c(cn2)n(CCOCc2ccccc2)c(=O)n3C2CCCC2)c(C)c1
COc1ccc(Nc2cc3c(cn2)n(CCO)c(=O)n3C2CCCC2)c(C)c1
COc1ccc(Nc2cc3c(cn2)n(C(C)C)c(=O)n3C2CCCC2)c(C)c1
COc1ccc(Nc2cc3c(cn2)n(C2CCCC2)c(=O)n3C2CCCC2)c(C)c1
COc1ccc(Nc2cc3c(cn2)n(Cc2ccccc2)c(=O)n3C2CCCC2)c(C)c1
COCCn1c(=O)n(C)c2cnc(Nc3ccc(OC)cc3C)cc21
COc1ccc(Nc2cc3c(cn2)n(C)c(=O)n3C2COC2)c(C)c1
COc1ccc(Nc2cc3c(cn2)n(C)c(=O)n3C2CCOC2)c(C)c1
COc1ccc(Nc2cc3c(cn2)n(C)c(=O)n3C2CCOCC2)c(C)c1
COc1ccc(Nc2cc3c(cn2)n(C)c(=O)n3CC2CCOCC2)c(C)c1
COc1ccc(Nc2cc3c(cn2)n(C)c(=O)n3CCC2CCOCC2)c(C)c1
COc1ccc(Nc2cc3c(cn2)n(C)c(=O)n3C2CCC(OC)CC2)c(C)c1
COc1ccc(Nc2cc3c(cn2)n(C)c(=O)n3C2CCC(OCc3ccccc3)CC2)c(C)c1
COc1ccc(Nc2cc3c(cn2)n(C)c(=O)n3C2CCC(O)CC2)c(C)c1
COc1ccc(Nc2cc3c(cn2)n(C)c(=O)n3-c2ccccc2)c(C)c1
COc1ccc(-n2c(=O)n(C)c3cnc(Nc4ccc(OC)cc4C)cc32)cc1
COc1ccc(Nc2cc3c(cn2)n(C)c(=O)n3-c2ccc(OCc3ccccc3)cc2)c(C)c1
COc1ccc(Nc2cc3c(cn2)n(C)c(=O)n3-c2ccc(O)cc2)c(C)c1
COc1ccc(Nc2cc3c(cn2)n(C)c(=O)n3-c2ccc(C(C)(C)C#N)cc2)c(C)c1
COc1ccc(Nc2cc3c(cn2)n(C)c(=O)n3C2CCN(C(=O)OC(C)(C)C)CC2)c(C)c1
COc1ccc(Nc2cc3c(cn2)n(C)c(=O)n3C2CCNCC2)c(C)c1
COc1ccc(Nc2cc3c(cn2)n(C)c(=O)n3CC2CCN(C(=O)OC(C)(C)C)CC2)c(C)c1
COc1ccc(Nc2cc3c(cn2)n(C)c(=O)n3CC2CCNCC2)c(C)c1
COc1ccc(Nc2cc3c(cn2)n(C)c(=O)n3C2CCC(NC(=O)OC(C)(C)C)CC2)c(C)c1
COc1ccc(Nc2cc3c(cn2)n(C)c(=O)n3C2CCC(N)CC2)c(C)c1
COc1ccc(Nc2cc3c(cn2)n(C)c(=O)n3C2CCN(C)CC2)c(C)c1
COc1ccc(Nc2cc3c(cn2)n(C)c(=O)n3CC2CCN(C)CC2)c(C)c1
COc1ccc(N(C(=O)OCc2ccccc2)c2cc3c(cn2)n(C)c(=O)n3C2CCOCC2)c(C)c1
CNCc1ccc(cc1)-c1cc(on1)-c1nc(cnc1N)-c1ccc(cc1)S(=O)(=O)C(C)C
C[C@@H]1COCCN1c1cc(nc(n1)-c1cc[nH]c2nccc12)C1(CC1)[S@](C)(=N)=O |r|
C[C@@H]1COCCN1c1nc(-c2ccnc3[nH]ccc23)nc2c1ccn2S(C)(=O)=O
COc1ccc2c(c1)CCN2c1ncc2c(n1)n(C1CCOCC1)c(=O)n2C
Cn1c(=O)n(C2CCOCC2)c2nc(N3CCc4cc(C#N)ccc43)ncc21
CC(=O)c1ccc2c(c1)CCN2c1ncc2c(n1)n(C1CCOCC1)c(=O)n2C
COC(=O)c1ccc2c(c1)CCN2c1ncc2c(n1)n(C1CCOCC1)c(=O)n2C
Cc1cc(-c2nc[nH]n2)ccc1Nc1ncc2c(n1)n(C1CCOCC1)c(=O)n2C
Cc1nc(-c2cn[nH]c2)ccc1Nc1ncc2c(n1)n(C1CCOCC1)c(=O)n2C
Cc1cc(-c2ncn(C)n2)ccc1Nc1ncc2c(n1)n(C1CCOCC1)c(=O)n2C
Cc1nc(-c2ccnn2C)ccc1Nc1ncc2c(n1)n(C1CCOCC1)c(=O)n2C
COc1cncc(-c2ccc(Nc3ncc4c(n3)n(C3CCOCC3)c(=O)n4C)c(C)n2)c1
COc1ccc(-c2ccc(Nc3ncc4c(n3)n(C3CCOCC3)c(=O)n4C)c(C)n2)cn1
COc1ccc(-c2cc(C)c(Nc3ncc4c(n3)n(C3CCOCC3)c(=O)n4C)cn2)cn1
COc1ccc(-c2cc(C)c(Nc3ncc4c(n3)n(C3CCOCC3)c(=O)n4C)cn2)cc1OC
Cc1cc(-c2cccnc2)ncc1Nc1ncc2c(n1)n(C1CCOCC1)c(=O)n2C
Cc1cc(-c2cn[nH]c2)ncc1Nc1ncc2c(n1)n(C1CCOCC1)c(=O)n2C
Cc1cc(-c2ccoc2)ncc1Nc1ncc2c(n1)n(C1CCOCC1)c(=O)n2C
Cc1cc(-c2ccco2)ncc1Nc1ncc2c(n1)n(C1CCOCC1)c(=O)n2C
Cc1cc(-c2ccsc2)ncc1Nc1ncc2c(n1)n(C1CCOCC1)c(=O)n2C
Cc1cc(-c2cccs2)ncc1Nc1ncc2c(n1)n(C1CCOCC1)c(=O)n2C
Cc1cc(-c2ccc(C=O)o2)ncc1Nc1ncc2c(n1)n(C1CCOCC1)c(=O)n2C
Cc1cc(-c2cnn(C)c2)ncc1Nc1ncc2c(n1)n(C1CCOCC1)c(=O)n2C
Cc1cc(-c2ccnn2C)ncc1Nc1ncc2c(n1)n(C1CCOCC1)c(=O)n2C
Cc1cc(-c2cn(C)nc2C)ncc1Nc1ncc2c(n1)n(C1CCOCC1)c(=O)n2C
Cc1cc(-c2cn(C)nc2C(F)(F)F)ncc1Nc1ncc2c(n1)n(C1CCOCC1)c(=O)n2C
Cc1cc(-c2cnn(C(F)F)c2)ncc1Nc1ncc2c(n1)n(C1CCOCC1)c(=O)n2C
Cc1ccc(-c2cnn(C)c2)cc1Nc1ncc2c(n1)n(C1CCOCC1)c(=O)n2C
Cc1ncc(-c2cnn(C)c2)cc1Nc1ncc2c(n1)n(C1CCOCC1)c(=O)n2C
Cc1cnc(-c2cnn(C)c2)cc1Nc1ncc2c(n1)n(C1CCOCC1)c(=O)n2C
Cn1cc(-c2ccc3c(c2)CCN3c2ncc3c(n2)n(C2CCOCC2)c(=O)n3C)cn1
Cc1cc(-c2cnn(C)c2)ncc1Nc1ncc2c(n1)n([C@H]1CCOC1)c(=O)n2C
Cc1cc(-c2cnn(C)c2)ncc1Nc1ncc2c(n1)n(C1CCCCC1C)c(=O)n2C
Cc1cc(-c2cnn(C)c2)ncc1Nc1ncc2c(n1)n([C@@]13C[C@@H]4C[C@@](C)(C[C@@](C)(C4)C1)C3)c(=O)n2C
Cc1cc(-c2cnn(C)c2)ncc1Nc1ncc2c(n1)n(C1CCNCC1)c(=O)n2C
CC(=O)N1CCC(n2c(=O)n(C)c3cnc(Nc4cnc(-c5cnn(C)c5)cc4C)nc32)CC1
Cc1cc(-c2cnn(C)c2)ncc1Nc1ncc2c(n1)n(C1CCN(S(C)(=O)=O)CC1)c(=O)n2C
Cc1cc(-c2cnn(C)c2)ncc1Nc1ncc2c(n1)n(C1CCN(C(=O)C3CC3)CC1)c(=O)n2C
Cc1cc(-c2cnn(C)c2)ncc1Nc1ncc2c(n1)n(C1CCN(S(=O)(=O)C3CC3)CC1)c(=O)n2C
Cc1cc(-c2cnn(C)c2)ncc1Nc1ncc2c(n1)n(C1CCN(S(=O)(=O)C(F)(F)F)CC1)c(=O)n2C
Cc1cc(-c2cnn(C)c2)ncc1Nc1ncc2c(n1)n(C1CCN(C(=O)C3CC3(F)F)CC1)c(=O)n2C
COc1ccc(Nc2ncc3c(n2)N(C2CCOCC2)Cc2nccn2-3)c(C)c1
Cc1cc2cccnc2cc1Nc1ncc2c(n1)N(C1CCOCC1)Cc1nccn1-2
Cc1cc2ncnn2cc1Nc1ncc2c(n1)N(C1CCOCC1)Cc1nccn1-2
c1cn2c(n1)CN(C1CCOCC1)c1nc(Nc3ccc4nccnc4c3)ncc1-2
Cc1cnc(-c2cnn(C)c2)cc1Nc1ncc2c(n1)N(C1CCOCC1)Cc1nccn1-2
c1cnc2cc(Nc3ncc4c(n3)N(C3CCOCC3)Cc3nncn3-4)ccc2n1
COc1ccc(Nc2ncc3c(n2)N(C2CCOCC2)Cc2nnc(C)n2-3)c(C)c1
Cc1cc2ncnn2cc1Nc1ncc2c(n1)N(C1CCOCC1)Cc1nncn1-2
Cc1nnc2n1-c1cnc(Nc3ccc4nccnc4c3)nc1N(C1CCOCC1)C2
Cc1cc2cccnc2cc1Nc1ncc2c(n1)N(C1CCOCC1)Cc1nncn1-2
Cc1cc2cccnc2cc1Nc1ncc2c(n1)N(C1CCOCC1)Cc1nnc(C)n1-2
Cc1cc2ncnn2cc1Nc1ncc2c(n1)N(C1CCOCC1)Cc1nnc(C)n1-2
Cc1cnc(-c2cnn(C)c2)cc1Nc1ncc2c(n1)N(C1CCOCC1)Cc1nnc(C)n1-2
Cc1cnc(-c2cnn(C)c2)cc1Nc1ncc2c(n1)N(C1CCOCC1)Cc1nncn1-2
Cn1c(=O)n(C(C)(C)C#N)c2c3cc(-c4cnc5ccccc5c4)ccc3ncc21
Cc1ccc(C(=O)Nc2cccc(C(F)(F)F)c2)cc1Nc1nc(-c2cccnc2)nc2c1cnn2C
COc1cccc2cc(-c3nc([C@H]4CC[C@H](C(=O)O)CC4)n4ncnc(N)c34)[nH]c12
Nc1nccn2c1c(-c1cc3cccc(Cl)c3[nH]1)nc2[C@H]1CC[C@H](C(=O)O)CC1
COc1ncc(cc1NS(=O)(=O)c1ccc(F)cc1F)-c1ccc2nccc(-c3ccnnc3)c2c1
Oc1cccc(c1)-c1nc(N2CCOCC2)c2oc3ncccc3c2n1
CCOc1cc(ccc1Nc2ncc3c(n2)N(c4ccccc4C(=O)N3C)C)N5CCC(CC5)O
CC1=CN2C(=O)C=C(N=C2C(=C1)[C@@H](C)Nc3ccccc3C(=O)O)N4CCOCC4