1847 SMILES Strings for Envelope glycoprotein gp160

Compound Name
SMILES String
CC1=CN(C(=O)NC1=O)[C@H]2C[C@@H]([C@H](O2)CO)N=[N+]=[N-]
CCCCCCCCCCCCCCCCOCCCOP([O-])(=O)CO[C@H](C)Cn1cnc2c(N)ncnc12 |r|
C[C@H](Cn1cnc2c(N)ncnc12)OCP(O)(=O)OCCCO |r|
C[C@H](Cn1cnc2c(N)ncnc12)OCP(O)(=O)OCCCOCC(O)=O |r|
C[C@H](Cn1cnc2c(N)ncnc12)OCP(O)(=O)OCCCOCCCC(O)=O |r|
CC(=C)[C@@H]1CC[C@@]2(CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC=C(c6ccc(cc6)C(O)=O)C(C)(C)[C@@H]5CC[C@@]34C)[C@@H]12)C#Cc1ccccc1C(O)=O |r,t:18|
CC(=C)[C@@H]1CC[C@@]2(CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC=C(c6ccc(cc6)C(O)=O)C(C)(C)[C@@H]5CC[C@@]34C)[C@@H]12)C#Cc1ccsc1-c1nnn[nH]1 |r,t:18|
CC(=C)[C@@H]1CC[C@@]2(CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC=C(c6ccc(cc6)C(O)=O)C(C)(C)[C@@H]5CC[C@@]34C)[C@@H]12)c1nnco1 |r,t:18|
CN(C)Cc1nnc(o1)[C@]12CC[C@H]([C@@H]1[C@H]1CC[C@@H]3[C@@]4(C)CC=C(c5ccc(cc5)C(O)=O)C(C)(C)[C@@H]4CC[C@@]3(C)[C@]1(C)CC2)C(C)=C |r,t:23|
CC(=C)[C@@H]1CC[C@@]2(CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC=C(c6ccc(cc6)C(O)=O)C(C)(C)[C@@H]5CC[C@@]34C)[C@@H]12)c1nc[nH]n1 |r,t:18|
CC(=C)[C@@H]1CC[C@@]2(CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC=C(c6ccc(cc6)C(O)=O)C(C)(C)[C@@H]5CC[C@@]34C)[C@@H]12)c1ncn(CCN2CCS(=O)(=O)CC2)n1 |r,t:18|
CC(=C)[C@@H]1CC[C@@]2(CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC=C(c6ccc(cc6)C(O)=O)C(C)(C)[C@@H]5CC[C@@]34C)[C@@H]12)c1ncnn1C |r,t:18|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@H](CNCc1ccc(Cl)cc1)OC(=O)CC(C)(C)C(O)=O |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@H](CN(CCN(C)C)Cc1ccc(Cl)cc1)OC(=O)CC(C)(C)C(O)=O |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@@H](CNCc1ccc(Cl)cc1)OC(=O)CC(C)(C)C(O)=O |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@@H](CN(CCN(C)C)Cc1ccc(Cl)cc1)OC(=O)CC(C)(C)C(O)=O |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@@]1(CCNCc3ccc(Cl)cc3)CC(=O)C(C(C)C)=C21 |r,t:56|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@@]1(CCNCc3ccccc3)CC(=O)C(C(C)C)=C21 |r,t:55|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@@]1(CCNCc3cccc(Cl)c3)CC(=O)C(C(C)C)=C21 |r,t:56|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@@]1(CCNCc3cccc(Cl)c3F)CC(=O)C(C(C)C)=C21 |r,t:57|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@@]1(CCNC3(CC3)c3ccc(Cl)cc3)CC(=O)C(C(C)C)=C21 |r,t:59|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@@]1(CCN(CCN(C)C)Cc3ccc(Cl)cc3)CC(=O)C(C(C)C)=C21 |r,t:61|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@@]1(CCN(CCN(C)C)C3(CC3)c3ccc(Cl)cc3)CC(=O)C(C(C)C)=C21 |r,t:64|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@@]1(CCN(C)Cc3ccc(Cl)cc3)CC(=O)C(C(C)C)=C21 |r,t:57|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@@]1(CCN(Cc3ccc(Cl)cc3)C(C)=O)CC(=O)C(C(C)C)=C21 |r,t:59|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@@H](O)CNCc1ccc(Cl)cc1 |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@H](O)CNCc1ccc(Cl)cc1 |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@@H](CNCc1ccc(Cl)cc1)OC(C)=O |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@H](CNCc1ccc(Cl)cc1)OC(C)=O |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@@H](O)CN(CCN(C)C)Cc1ccc(Cl)cc1 |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@H](O)CN(CCN(C)C)Cc1ccc(Cl)cc1 |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@@H](CN(CCN(C)C)Cc1ccc(Cl)cc1)OC(C)=O |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@H](CN(CCN(C)C)Cc1ccc(Cl)cc1)OC(C)=O |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)CC(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@@H](O)CN(CCN(C)C)Cc1ccc(Cl)cc1 |r,t:45|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)CC(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@H](O)CN(CCN(C)C)Cc1ccc(Cl)cc1 |r,t:45|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@H](O)CNCc1ccccc1Cl |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@@H](O)CNCc1ccccc1Cl |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@@H](CNCc1ccc(F)cc1)OC(C)=O |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@H](CNCc1ccc(F)cc1)OC(C)=O |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@H](O)CN(C)Cc1ccc(Cl)cc1 |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@@H](O)CN(C)Cc1ccc(Cl)cc1 |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@H](O)CN(Cc1ccc(Cl)cc1)C(C)=O |r,t:44,@:21|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@@H](O)CN(Cc1ccc(Cl)cc1)C(C)=O |r,t:44,@:21|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@H](O)CN(Cc1ccccc1Cl)C(C)=O |r,t:44,@:21|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@@H](CN(CCN(C)C)Cc1ccccc1Cl)OC(C)=O |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@H](O)CNCc1cccc(Cl)c1 |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@@H](O)CNCc1cccc(Cl)c1 |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@@H](CNCc1cccc(Cl)c1)OC(C)=O |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@H](CNCc1cccc(Cl)c1)OC(C)=O |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@H](O)CN(CCN(C)C)Cc1cccc(Cl)c1 |r,t:44,@:21|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@@H](O)CN(CCN(C)C)Cc1cccc(Cl)c1 |r,t:44,@:21|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@@H](O)CN(Cc1cccc(Cl)c1)C(C)=O |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@H](O)CN(Cc1cccc(Cl)c1)C(C)=O |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@@H](O)CN(CC)Cc1ccccc1Cl |r,t:44,@:21|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@@H](O)CN(CCN(C)C)Cc1ccccc1Cl |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@H](O)CN(CCN(C)C)Cc1ccccc1Cl |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@H](CNCc1ccccc1)OC(C)=O |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@@H](CNCc1ccccc1)OC(C)=O |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@@H](O)CN(CCN(C)C)Cc1cccc(Cl)c1F |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@H](O)CN(CCN(C)C)Cc1cccc(Cl)c1F |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@@H](O)CNC(C)C |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@@H](O)CNC1CCCCC1 |r,t:44|
[H][C@@]1(CN(C(=O)O1)C1(CC1)c1ncc(Cl)cn1)[C@]12CC(=O)C(C(C)C)=C1[C@@]1([H])CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC2 |r,c:27|
[H][C@]1(CN(C(=O)O1)C1(CC1)c1ncc(Cl)cn1)[C@]12CC(=O)C(C(C)C)=C1[C@@]1([H])CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC2 |r,c:27|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)CC(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@H](O)CNCc1ccc(Cl)cc1 |r,t:45|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@@H](O)CN1CCc2ccccc2C1 |r,t:44,@:21|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@H](O)CN1CCc2ccccc2C1 |r,t:44,@:21|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CCC(C(C)C)=C21)C(O)CN1CCN(C)CC1 |r,t:43,@:21|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@@]1(CCNCc3ccc(Cl)cc3)CCC(C(C)C)=C21 |r,t:55,@:21|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CCC(C(C)C)=C21)[C@H](O)CNCC1CCCCC1 |r,t:43,@:21|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@H](O)CNC1CCCCC1 |r,t:44,@:21|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@H](O)CN(CCN(C)C)Cc1ccccc1 |r,t:44,@:21|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@@H](CN(CCN(C)C)Cc1ccc(F)cc1)OC(C)=O |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@H](CN(CCN(C)C)Cc1ccc(F)cc1)OC(C)=O |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)CC(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@@H](O)CNCc1ccc(Cl)cc1 |r,t:45|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)CC(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@H](O)CNCc1ccc(Cl)cc1 |r,t:45,@:22|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@H](O)CN(CCN(C)C)Cc1ccc(Cl)cc1Cl |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@@H](O)CN(CCN(C)C)Cc1ccccc1 |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@@H](O)CN(CCN(C)C)Cc1ccc(F)cc1 |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@@H](O)CNCc1ccc(F)cc1 |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@H](O)CN(CCN(C)C)Cc1ccc(F)cc1 |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@H](O)CNCc1ccc(F)cc1 |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@@H](O)CN(CCN(C)C)Cc1ccc(Cl)cc1Cl |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@]1(CC(=O)C(C(C)C)=C21)[C@@H](O)CN(CCN(C)C)C(=O)c1ccc(Cl)cc1 |r,t:44|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@@]1(CCNCc3ccccc3Cl)CC(=O)C(C(C)C)=C21 |r,t:56|
[H][C@]12CC[C@]3([H])[C@@]4(C)CC[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@]4([H])CC[C@@]3(C)[C@]1(C)CC[C@@]1(CCNC(=O)c3ccccc3)CC(=O)C(C(C)C)=C21 |r,t:56|
Cc1cc2nc(cn2c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O)-c1cccc(c1)-c1ccccc1 |r|
Cc1ccc(cc1)-c1cccc(c1)-c1cn2c(N3CCC(C)(C)CC3)c([C@H](OC(C)(C)C)C(O)=O)c(C)cc2n1 |r|
Cc1cc2nc(cn2c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O)-c1cccc(c1)-c1ccc(F)cc1 |r|
Cc1cc2nc(cn2c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O)-c1cccc(c1)-c1cccc(F)c1 |r|
Cc1cc2nc(cn2c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O)-c1cccc(c1)-c1ccc(F)cc1F |r|
Cc1ccc(c(F)c1)-c1cccc(c1)-c1cn2c(N3CCC(C)(C)CC3)c([C@H](OC(C)(C)C)C(O)=O)c(C)cc2n1 |r|
Cc1cc2nc(cn2c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O)-c1cccc(c1)-c1cccc(c1)C#N |r|
Cc1cc2nc(cn2c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O)-c1cccc(c1)-c1cnn(Cc2ccccc2)c1 |r|
Cc1cc2nc(cn2c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O)-c1cccc(c1)-c1cnn(C)c1 |r|
Cc1cc(-c2cccc(c2)-c2cn3c(N4CCC(C)(C)CC4)c([C@H](OC(C)(C)C)C(O)=O)c(C)cc3n2)n(C)n1 |r|
Cc1cc2nc(cn2c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O)-c1cccc(c1)-c1cc(nn1C)C(F)(F)F |r|
Cc1cc2nc(cn2c(c1[C@H](OC(C)(C)C)C(O)=O)-c1ccc2OCCc3ccnc1c23)-c1cccc(c1)-c1ccc(F)cc1 |r,wD:10.12,(5.32,1.7,;3.98,2.47,;2.65,1.7,;1.32,2.47,;-.15,1.99,;-1.05,3.24,;-.15,4.48,;1.32,4.01,;2.65,4.78,;3.98,4.01,;5.32,4.78,;5.32,6.32,;6.65,7.09,;7.98,7.86,;6.65,8.63,;7.98,6.32,;6.65,4.01,;7.98,4.78,;6.65,2.47,;2.65,6.32,;3.98,7.09,;3.98,8.63,;2.65,9.4,;2.65,10.94,;1.32,11.71,;-.02,10.94,;-.02,9.4,;-1.35,8.63,;-1.35,7.09,;-.02,6.32,;1.32,7.09,;1.32,8.63,;-2.59,3.24,;-3.36,1.91,;-4.9,1.91,;-5.67,3.24,;-4.9,4.57,;-3.36,4.57,;-5.67,5.91,;-4.9,7.24,;-5.67,8.57,;-7.21,8.57,;-7.98,9.91,;-7.98,7.24,;-7.21,5.91,)|
Cc1ccc(cc1)-c1c([C@H](OC(C)(C)C)C(O)=O)c(C)cc2nc(cn12)-c1cccc(c1)-c1ccc(F)cc1 |r|
Cc1cc2nc(cn2c(-c2cc(F)c3OCCCc3c2C)c1[C@H](OC(C)(C)C)C(O)=O)-c1cccc(c1)-c1ccc(F)cc1 |r,wD:22.26,(5.32,1.7,;3.98,2.47,;2.65,1.7,;1.32,2.47,;-.15,1.99,;-1.05,3.24,;-.15,4.48,;1.32,4.01,;2.65,4.78,;2.65,6.32,;3.98,7.09,;3.98,8.63,;5.32,9.4,;2.65,9.4,;2.65,10.94,;1.32,11.71,;-.02,10.94,;-.02,9.4,;1.32,8.63,;1.32,7.09,;-.02,6.32,;3.98,4.01,;5.32,4.78,;5.32,6.32,;6.65,7.09,;7.98,7.86,;6.65,8.63,;7.98,6.32,;6.65,4.01,;7.98,4.78,;6.65,2.47,;-2.59,3.24,;-3.36,1.91,;-4.9,1.91,;-5.67,3.24,;-4.9,4.57,;-3.36,4.57,;-5.67,5.91,;-4.9,7.24,;-5.67,8.57,;-7.21,8.57,;-7.98,9.91,;-7.98,7.24,;-7.21,5.91,)|
Cc1cc2nc(cn2c(-c2ccc(F)cc2)c1[C@H](OC(C)(C)C)C(O)=O)-c1cccc(c1)-c1ccc(F)cc1 |r|
Cc1cc2nc(cn2c(-c2ccc3OCCCc3c2)c1[C@H](OC(C)(C)C)C(O)=O)-c1cccc(c1)-c1ccc(F)cc1 |r|
Cc1cc2nc(cn2c(-c2ccc3OCCC(C)(C)c3c2)c1[C@H](OC(C)(C)C)C(O)=O)-c1cccc(c1)-c1ccc(F)cc1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cccc(Cl)c1)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)C1(C)CC1)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccc(C)cc1)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccc(Cl)cc1)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1Cl)c1ccc2OCOc2c1 |r|
COc1ccc(cc1)S(=O)(=O)NC(=O)N[C@@H](Cc1ccccc1)C(=O)N(C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1F)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Cc1ccccc1)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cc(Cl)cc(Cl)c1)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cc(Br)ccc1Br)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cc(C)ccc1C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1OC(F)(F)F)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cccc(Cl)c1Cl)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cc(F)ccc1C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C(F)(F)F)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccc(F)cc1F)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cccc(Br)c1)c1ccc2OCOc2c1 |r|
COc1cccc(c1)S(=O)(=O)NC(=O)N[C@@H](Cc1ccccc1)C(=O)N(C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccc(cc1)[NH+]=O)c1ccc2OCOc2c1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccc(F)cc1)c1ccc2OCOc2c1 |r|
COC(=O)c1ccccc1S(=O)(=O)NC(=O)N[C@@H](Cc1ccccc1)C(=O)N(C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)CCc1ccccc1)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)CCCc1ccccc1)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccc(F)c(F)c1)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccc(C)s1)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cccc(Cl)c1C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1Br)c1ccc2OCOc2c1 |r|
COc1ccc(OC)c(c1)S(=O)(=O)NC(=O)N[C@@H](Cc1ccccc1)C(=O)N(C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cccs1)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cc(Cl)sc1Cl)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1c(C)nn(C)c1Cl)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1F)c1ccc2OC(F)(F)Oc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)c1ccccc1F)c1ccc2OC(F)(F)Oc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1)c1ccc2OC(F)(F)Oc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OC(F)(F)Oc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1Cl)c1ccc2OC(F)(F)Oc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)c1ccccc1Cl)c1ccc2OC(F)(F)Oc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OC(F)(F)Oc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)c1ccccc1)c1ccc2OC(F)(F)Oc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)C1CC1)c1ccc2OCOc2c1 |r|
CC(C)S(=O)(=O)NC(=O)N[C@@H](Cc1ccccc1)C(=O)N(C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(C)(=O)=O)c1ccc2OCOc2c1 |r|
CC(C)CS(=O)(=O)NC(=O)N[C@@H](Cc1ccccc1)C(=O)N(C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)C(C)(C)C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)N(C)S(=O)(=O)c1ccccc1Br)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)N(C)S(=O)(=O)c1ccccc1-c1ccccc1)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1-c1cnn(C)c1)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1-c1ccoc1)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccc(Cl)cc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCOc2c1 |r|
CCOc1ccc(C[C@H](NC(=O)NS(=O)(=O)c2ccccc2C)C(=O)N(C)c2ccc3OCOc3c2)cc1 |r|
CN(C(=O)[C@H](Cc1ccccc1C)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1Cl)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1cccc(Cl)c1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCOc2c1 |r|
COc1ccc(C[C@H](NC(=O)NS(=O)(=O)c2ccccc2C)C(=O)N(C)c2ccc3OCOc3c2)cc1 |r|
CN(C(=O)[C@H](Cc1ccc(Br)cc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccc(OCC=C)cc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccc(Cl)c(Cl)c1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccc(F)c(F)c1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccc(cc1)C(F)(F)F)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1cccc(c1)C#N)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccc(cc1)C#N)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCOc2c1 |r|
COC(=O)c1cccc(C[C@H](NC(=O)NS(=O)(=O)c2ccccc2C)C(=O)N(C)c2ccc3OCOc3c2)c1 |r|
C[C@H]([C@H](NC(=O)NS(=O)(=O)c1ccccc1C)C(=O)N(C)c1ccc2OCOc2c1)c1ccccc1 |r|
CN(C(=O)[C@H](Cc1ccccc1C(N)=O)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccc(OCc2ccccc2)cc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccc(cc1)-c1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1F)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1cccc(c1)C(F)(F)F)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccc(C)cc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccc(NC(C)=O)cc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccc(Cl)cc1Cl)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)c(F)cc1F)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1Br)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1C#N)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCOc2c1 |r|
COc1cccc(C[C@H](NC(=O)NS(=O)(=O)c2ccccc2C)C(=O)N(C)c2ccc3OCOc3c2)c1 |r|
CN(C(=O)[C@@]1(C[C@H]1c1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1cccc(c1)C(N)=O)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1cccc(c1)S(=O)(=O)N1CCOCC1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccc(O)cc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1cccc2ccccc12)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@@H](NC(=O)NS(=O)(=O)c1ccccc1C)C1CCc2ccccc12)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1cccc(F)c1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1)c1ccccc1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1)c1ccc(Cl)cc1 |r|
COc1cccc(c1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1)c1cccc(C)c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1)c1ccc(F)cc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1)c1cccc(F)c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1)c1cccc2ccccc12 |r|
COc1ccccc1N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1 |r|
CCN(CC)CCN(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1 |r|
CN(Cc1ccc(cc1)-c1noc(C)n1)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1c(F)cccc1F)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cc(F)ccc1F)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1c(Cl)cccc1Cl)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Cc1ccccc1Cl)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Cc1ccc(Cl)c(Cl)c1)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Cc1cccc(Cl)c1)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Cc1ccccc1C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Cc1ccc(cc1)C(F)(F)F)c1ccc2OCOc2c1 |r|
CC(C)C1CC1S(=O)(=O)NC(=O)N[C@@H](Cc1ccccc1)C(=O)N(C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)C1(Cc2ccccc2)CC1)c1ccc2OCOc2c1 |r|
COc1ccccc1S(=O)(=O)NC(=O)N[C@@H](Cc1ccccc1)C(=O)N(C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Cc1ccc(Cl)cc1)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Cc1ccc(F)cc1)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)C1CCCCC1)c1ccc2OCOc2c1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cccc(Br)c1)c1ccc(OC)cc1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1[N+]([O-])=O)c1ccc(OC)cc1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C(=O)OC)c1ccc(OC)cc1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cccc(Br)c1C)c1ccc(OC)cc1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cccc2ccccc12)c1ccc(OC)cc1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1F)c1ccc(OC)cc1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1c(F)cccc1F)c1ccc(OC)cc1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cccc(Cl)c1Cl)c1ccc(OC)cc1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cc(Br)ccc1C)c1ccc(OC)cc1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cccc(c1)-c1ccoc1)c1ccc(OC)cc1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cccc(-c2ccoc2)c1C)c1ccc(OC)cc1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cc(ccc1C)-c1ccoc1)c1ccc(OC)cc1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1-c1ccc(CO)cc1)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1-c1cccc(O)c1)c1ccc2OCOc2c1 |r|
COc1ccc(cn1)-c1ccccc1S(=O)(=O)NC(=O)N[C@@H](Cc1ccccc1)C(=O)N(C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1-c1cncnc1)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1-c1cccnc1)c1ccc2OCOc2c1 |r|
COc1ncccc1-c1ccccc1S(=O)(=O)NC(=O)N[C@@H](Cc1ccccc1)C(=O)N(C)c1ccc2OCOc2c1 |r|
COc1ncc(cn1)-c1ccccc1S(=O)(=O)NC(=O)N[C@@H](Cc1ccccc1)C(=O)N(C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1-c1ccc(cc1)C(N)=O)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1-c1ccsc1)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C(C)=C)c1ccc2OCOc2c1 |r|
CC(C)c1ccccc1S(=O)(=O)NC(=O)N[C@@H](Cc1ccccc1)C(=O)N(C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C=C)c1ccc2OCOc2c1 |r|
C\C=C/c1ccccc1S(=O)(=O)NC(=O)N[C@@H](Cc1ccccc1)C(=O)N(C)c1ccc2OCOc2c1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cccc(C=C)c1)c1ccc(OC)cc1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cccc(c1)C(C)=C)c1ccc(OC)cc1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cccc(\C=C/C)c1)c1ccc(OC)cc1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cccc(CC)c1)c1ccc(OC)cc1 |r|
CCCc1cccc(c1)S(=O)(=O)NC(=O)N[C@@H](Cc1ccccc1)C(=O)N(CC)c1ccc(OC)cc1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cccc(c1)C(C)C)c1ccc(OC)cc1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cc(CC)ccc1C)c1ccc(OC)cc1 |r|
CCCc1ccccc1S(=O)(=O)NC(=O)N[C@@H](Cc1ccccc1)C(=O)N(C)c1ccc2OCOc2c1 |r|
CCc1ccccc1S(=O)(=O)NC(=O)N[C@@H](Cc1ccccc1)C(=O)N(C)c1ccc2OCOc2c1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1N)c1ccc(OC)cc1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1-c1ccc(F)nc1)c1ccc2OCOc2c1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cccc(c1)-c1ccco1)c1ccc(OC)cc1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cccc(c1)-c1ccsc1Cl)c1ccc(OC)cc1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cccc(c1)-c1ccsc1)c1ccc(OC)cc1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cccc(c1)-c1ccnn1C)c1ccc(OC)cc1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cccc(c1)-c1csc2ccccc12)c1ccc(OC)cc1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cccc(c1)-c1cc2c(OC)cccc2[nH]1)c1ccc(OC)cc1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cccc(-c2ccco2)c1C)c1ccc(OC)cc1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cccc(-c2ccsc2Cl)c1C)c1ccc(OC)cc1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cccc(-c2ccsc2)c1C)c1ccc(OC)cc1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cccc(-c2ccnn2C)c1C)c1ccc(OC)cc1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cccc(-c2cnoc2)c1C)c1ccc(OC)cc1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cccc(-c2csc(c2)C(O)=O)c1C)c1ccc(OC)cc1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cccc(-c2csc3ccccc23)c1C)c1ccc(OC)cc1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cccc(-c2cc3c(OC)cccc3[nH]2)c1C)c1ccc(OC)cc1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1cccc(C)c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc(Cl)cc1 |r|
COc1ccccc1N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C |r|
COc1cccc(c1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1cccc(F)c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc(F)cc1 |r|
Cc1ccccc1S(=O)(=O)NC(=O)N[C@@H](Cc1ccccc1)C(=O)N1CCCc2ccccc12 |r|
COc1ccc2N(CCCc2c1)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C |r|
COc1ccc2N(CCOc2c1)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C |r|
Cc1ccccc1S(=O)(=O)NC(=O)N[C@@H](Cc1ccccc1)C(=O)N1CCCc2cc(O)ccc12 |r|
Cc1ccccc1S(=O)(=O)NC(=O)N[C@@H](Cc1ccccc1)C(=O)N1CCc2ccccc12 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc(C)c(C)c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1nc2ccccc2s1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2ccccc2c1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc(OC(F)(F)F)cc1 |r|
CN(C1CCCCC1)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C |r|
CN(Cc1ccccn1)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc(Cl)cc1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc(Cl)c(c1)C(F)(F)F |r|
CCCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc(Cl)c(Cl)c1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc(OC)cc1 |r|
CN(C)S(=O)(=O)c1ccc2N(CCc2c1)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C |r|
Cc1ccccc1S(=O)(=O)NC(=O)N[C@@H](Cc1ccccc1)C(=O)N1CCc2sccc2C1 |r|
[H][C@]12CN(C(=O)[C@H](Cc3ccccc3)NC(=O)NS(=O)(=O)c3ccccc3C)[C@]([H])(CO1)C2 |r,TLB:4:3:30.31:32|
Cc1ccccc1S(=O)(=O)NC(=O)N[C@@H](Cc1ccccc1)C(=O)N1CCC1 |r|
Cc1ccccc1S(=O)(=O)NC(=O)N[C@@H](Cc1ccccc1)C(=O)N1CCCC1c1cccnc1 |r|
Cc1ccccc1S(=O)(=O)NC(=O)N[C@@H](Cc1ccccc1)C(=O)N1CC(C)(C)C1 |r|
COC1CN(C1)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccn1)NC(=O)NS(=O)(=O)c1ccccc1C |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cn1cncn1)NC(=O)NS(=O)(=O)c1ccccc1C |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1cccnc1)NC(=O)NS(=O)(=O)c1ccccc1C |r|
COc1ccc(cc1)N(C)C(=O)[C@H](CC1CCCCC1)NC(=O)NS(=O)(=O)c1ccccc1C |r|
COc1ccc(cc1)N(C)C(=O)[C@H](CC1CCCC1)NC(=O)NS(=O)(=O)c1ccccc1C |r|
COc1ccc(cc1)N(C)C(=O)[C@@H](NC(=O)NS(=O)(=O)c1ccccc1C)[C@@H](C)c1ccccc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1cccs1)NC(=O)NS(=O)(=O)c1ccccc1C |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccncc1)NC(=O)NS(=O)(=O)c1ccccc1C |r|
COc1ccc(cc1)N(CC(F)(F)F)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1Br)c1ccc(OC)cc1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccc2n(CC)ccc2c1)c1ccc(OC)cc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)c1ccccc1F |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)c1ccccc1C |r|
COc1cc(cc(OC)c1OC)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C |r|
COc1ccc(N(C)C(=O)[C@H](Cc2ccccc2)NC(=O)NS(=O)(=O)c2ccccc2C)c(C)c1 |r|
COc1cc(C)c(cc1C)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C |r|
COc1ccc(cc1)N(Cc1ccccc1)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C |r|
COc1ccc(cc1)N(Cc1ccncc1)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C |r|
COc1ccc(cc1)N(CCc1ccccc1)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C |r|
COc1ccc(cc1)N(CC(C)C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccccc1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccccc1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccccc1C |r|
CC(C)N(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccccc1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2ncccc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2nc(C)ccc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2ncn(C)c2c1 |r|
CCn1c(C)nc2cc(ccc12)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2nccnc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCCc2c1 |r|
COc1ccc(cc1C)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc(OC)c(C)c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCCCc2c1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2ncccc2c1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCCCc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc(C)cc1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2nc(C)ccc2c1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1c(C)n(C)c2ccccc12 |r|
CCOc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc(NC(C)=O)c(O)c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2nc(C)oc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2sc(C)nc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2scnc2c1 |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc(O)c(NC=O)c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc(O)c(NC=O)c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1cccc(c1)C#N |r|
CN(C)C(=O)Nc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C |r|
COC(=O)Nc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1cccc(c1)C(N)=O |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2ncsc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2ncncc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc(cc1)C#N |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2cccnc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2cc[nH]c(=O)c2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc(F)c(c1)C(N)=O |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1cccc2[nH]cnc12 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc(F)c(c1)C(N)=O |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2cc[nH]c(=O)c2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2cccnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)c1ccccc1C)c1cc2ccccc2cn1 |r|
CNS(=O)(=O)c1cccc(c1)N(C)C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)c1ccccc1C |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccccc1F |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc(OC(F)(F)F)cc1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)c1ccccc1C)c1cccc2ncccc12 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)c1ccccc1C)c1cccc2cnccc12 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)c1ccccc1C)c1cccc(Cl)c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc(F)cc1F |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)c1ccccc1Cl)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)c1cc(F)ccc1F)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)c1ccccc1F)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)c1ccc(F)cc1F)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1Cl)c1ccc2CCCc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2CCCc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1)c1ccc2CCCc2c1 |r|
CN(C(=O)[C@H](CCc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCOc2c1 |r|
CN(C(=O)[C@@H](CCc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc2OCOc2c1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1cccc(C=C)c1)NC(=O)NS(=O)(=O)c1ccccc1C=C |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1cccc(OCCC=C)c1)NC(=O)NS(=O)(=O)c1ccccc1C=C |r|
CCN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1cccc(-c2ccnn2CC(C)C)c1C)c1ccc(OC)cc1 |r|
CCc1cccc(C[C@H](NC(=O)NS(=O)(=O)c2ccccc2CC)C(=O)N(C)c2ccc(OC)cc2)c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc(OCC=C)cc1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)c1ccccc1C)c1ccc(OCC(N)=O)cc1 |r|
C[C@H]1CCCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)nc3cc(nn23)-c2cccc(c2)-c2cc(ccc2O1)C(F)(F)F |r|
C[C@H]1CCCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)nc3cc(nn23)-c2cccc(c2)-c2cc(F)c(F)cc2O1 |r|
C[C@H]1CCCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)nc3cc(nn23)-c2cccc(c2)-c2c(F)cc(F)cc2O1 |r|
C[C@H]1C\C=C\COC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)nc3cc(nn23)-c2cccc(c2)-c2c(F)cc(C)cc2O1 |r,t:3|
C[C@H]1CCCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)nc3cc(nn23)-c2cccc(c2)-c2c(F)cc(C)cc2O1 |r|
CCc1ccc2O[C@@H](C)C\C=C\COC3(C)CCN(CC3)c3c([C@H](OC(C)(C)C)C(O)=O)c(C)nc4cc(nn34)-c3cccc(c3)-c2c1 |r,t:10|
CCc1ccc2O[C@@H](C)CCCCOC3(C)CCN(CC3)c3c([C@H](OC(C)(C)C)C(O)=O)c(C)nc4cc(nn34)-c3cccc(c3)-c2c1 |r|
COc1ccc2O[C@@H](C)CCCCCOC3(C)CCN(CC3)c3c([C@H](OC(C)(C)C)C(O)=O)c(C)nc4cc(nn34)-c3cccc(c3)-c2c1 |r|
CC1N=C2CC3=NN2C(N2CCC(C)(CC2)OC\C=C/[C@H](C)Oc2cc(F)ccc2-c2cccc3c2)=C1[C@H](OC(C)(C)C)C(O)=O |c:5,20,40,t:2|
C[C@H]1CCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)nc3cc(nn23)-c2cccc(c2)-c2ccc(F)cc2O1 |r|
C[C@@H]1Oc2ccc(C)c(F)c2-c2cccc(c2)-c2cc3nc(C)c([C@H](OC(C)(C)C)C(O)=O)c(N4CCC(C)(CC4)OC\C=C/1)n3n2 |c:46|
C[C@H]1CCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)nc3cc(nn23)-c2cccc(c2)-c2c(O1)ccc(C)c2F |r|
C[C@@H]1Oc2ccc(F)cc2-c2cccc(c2)-c2cc3nc(C)c([C@H](OC(C)(C)C)C(O)=O)c(N4CCC(C)(CC4)OC\C=C/1)n3n2 |c:45|
C[C@H]1CCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)nc3cc(nn23)-c2cccc(c2)-c2cc(F)ccc2O1 |r|
C[C@@H]1Oc2cc(C)ccc2-c2cccc(c2)-c2cc3nc(C)c([C@H](OC(C)(C)C)C(O)=O)c(N4CCC(C)(CC4)OC\C=C/1)n3n2 |c:45|
C[C@H]1CCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)nc3cc(nn23)-c2cccc(c2)-c2ccc(C)cc2O1 |r|
C[C@@H]1Oc2cc(C)cc(F)c2-c2cccc(c2)-c2cc3nc(C)c([C@H](OC(C)(C)C)C(O)=O)c(N4CCC(C)(CC4)OC\C=C/1)n3n2 |c:46|
C[C@H]1CCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)nc3cc(nn23)-c2cccc(c2)-c2c(F)cc(C)cc2O1 |r|
C[C@H]1CC\C=C/OC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)nc3cc(nn23)-c2cccc(c2)-c2cc(C)ccc2O1 |r,c:4|
CC1C\C=C\CCC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)nc3cc(nn23)-c2cccc(c2)-c2cc(C)ccc2O1 |r,w:2.2,t:3|
CC1CCCCCC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)nc3cc(nn23)-c2cccc(c2)-c2cc(C)ccc2O1 |r|
CC1C\C=C\CCC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)nc3cc(nn23)-c2cccc(c2)-c2cc(ccc2O1)[N+]#[C-] |r,w:2.2,t:3|
CC1CCCCCC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)nc3cc(nn23)-c2cccc(c2)-c2cc(ccc2O1)C(N)=O |r|
C[C@H]1CCCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)nc3cc(nn23)-c2cccc(c2)-c2cc(ccc2O1)C(=O)NCCC(C)(C)C |r|
C[C@H]1CCCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)nc3cc(nn23)-c2cc(ccc2F)-c2ccc(F)cc2O1 |r|
C[C@H]1CCCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)nc3cc(nn23)-c2cc(F)cc(c2)-c2ccc(F)cc2O1 |r|
C[C@H]1CCCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)nc3cc(nn23)-c2ccc(F)c(c2)-c2ccc(F)cc2O1 |r|
C[C@H]1COCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)cc3nc(cn23)-c2cccc(c2)-c2cc(F)c(F)cc2O1 |r|
C[C@H]1COCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)c(C)c3nc(cn23)-c2cccc(c2)-c2cc(F)c(F)cc2O1 |r|
C[C@H]1COCCOC2(C)CCN(CC2)c2c([C@@H](OC(C)(C)C)C(O)=O)c(C)c(C)c3nc(cn23)-c2cccc(c2)-c2cc(F)c(F)cc2O1 |r|
CCC(C)(C)O[C@H](C(O)=O)c1c(C)c(C)c2nc-3cn2c1N1CCC(C)(CC1)OCCOC[C@H](C)Oc1cc(F)c(F)cc1-c1cccc-3c1 |r|
C[C@H]1COCCOC2(C)CCN(CC2)c2c([C@H](O)C(O)=O)c(C)c(C)c3nc(cn23)-c2cccc(c2)-c2cc(F)c(F)cc2O1 |r|
C[C@H]1COCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)c(CO)c3nc(cn23)-c2cccc(c2)-c2cc(F)c(F)cc2O1 |r|
C[C@H]1COCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)cc3nc(c(Cl)n23)-c2cccc(c2)-c2cc(F)c(F)cc2O1 |r|
C[C@H]1COCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)c(C)c3nc(c(Cl)n23)-c2cccc(c2)-c2cc(F)c(F)cc2O1 |r|
C[C@H]1COCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)c(CO)c3nc(c(Cl)n23)-c2cccc(c2)-c2cc(F)c(F)cc2O1 |r|
C[C@H]1COCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)c(Cn3cccn3)c3nc(c(Cl)n23)-c2cccc(c2)-c2cc(F)c(F)cc2O1 |r|
COCc1c(C)c([C@H](OC(C)(C)C)C(O)=O)c2N3CCC(C)(CC3)OCCOC[C@H](C)Oc3cc(F)c(F)cc3-c3cccc(c3)-c3nc1n2c3Cl |r|
C[C@H]1COCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)c(Cn3ccnn3)c3nc(c(Cl)n23)-c2cccc(c2)-c2cc(F)c(F)cc2O1 |r|
C[C@H]1COCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)c(Cn3nccn3)c3nc(c(Cl)n23)-c2cccc(c2)-c2cc(F)c(F)cc2O1 |r|
C[C@H]1COCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)c(C(C)=C)c3nc(cn23)-c2cccc(c2)-c2cc(F)c(F)cc2O1 |r|
C[C@H]1COCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)c(C)c3nc(c(C)n23)-c2cccc(c2)-c2cc(F)c(F)cc2O1 |r|
CC(O)c1c(C)c([C@H](OC(C)(C)C)C(O)=O)c2N3CCC(C)(CC3)OCCOC[C@H](C)Oc3cc(F)c(F)cc3-c3cccc(c3)-c3cn2c1n3 |r|
C[C@H]1COCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)c(C#N)c3nc(cn23)-c2cccc(c2)-c2cc(F)c(F)cc2O1 |r|
C[C@H]1COCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)cc3nc(cn23)-c2cccc(c2)-c2c(F)cc(C)cc2O1 |r|
C[C@H]1COCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)c(C)c3nc(cn23)-c2cccc(c2)-c2c(F)cc(C)cc2O1 |r|
C[C@H]1COCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)c(C)c3nc(c(Cl)n23)-c2cccc(c2)-c2c(F)cc(C)cc2O1 |r|
C[C@H]1COCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)cc3nc(cn23)-c2cccc(c2)-c2ccc(C)cc2O1 |r|
C[C@H]1COCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)c(C)c3nc(cn23)-c2cccc(c2)-c2ccc(C)cc2O1 |r|
C[C@H]1COCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)c(C)c3nc(c(Cl)n23)-c2cccc(c2)-c2ccc(C)cc2O1 |r|
C[C@H]1COCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)cc3nc(cn23)-c2cccc(c2)-c2cc(C)ccc2O1 |r|
C[C@H]1COCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)c(C)c3nc(cn23)-c2cccc(c2)-c2cc(C)ccc2O1 |r|
C[C@H]1COCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)c(C)c3nc(c(Cl)n23)-c2cccc(c2)-c2cc(C)ccc2O1 |r|
C[C@H]1COCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)c(C)c3nc(cn23)-c2cccc(c2)-c2cc(F)ccc2O1 |r|
C[C@H]1COCCOC2(C)CCN(CC2)c2c([C@H](OC(C)(C)C)C(O)=O)c(C)c(C)c3nc(c(Cl)n23)-c2cccc(c2)-c2cc(F)ccc2O1 |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccc(F)cc4)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4cccc(c4)C(F)(F)F)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1cccc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)c1 |r|
Cc1ccccc1CN1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1 |r|
Cc1ccc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)cc1 |r|
COc1cccc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)c1 |r|
Cc1nc(C)c(-c2ccc3CN(Cc4cccc(F)c4)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccc(cc4)C(F)(F)F)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccccc4F)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4cccc(c4)C(O)=O)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4cccc(c4)-c4ccccc4)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccccc4C(F)(F)F)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
CC(N1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1)c1ccccc1 |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccc(cc4)-c4ccccc4)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4cccc(c4C)C(F)(F)F)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1ccc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)cc1C(F)(F)F |r|
Cc1ccc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)cc1C |r|
Cc1ccc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)cc1F |r|
Cc1ccc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)c(C)c1 |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccc(F)cc4F)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4cccc(F)c4F)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccc(Cl)c(F)c4)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1cccc(Cl)c1CN1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1 |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccc(F)c(Cl)c4)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1cc(F)ccc1CN1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1 |r|
Cc1nc(C)c(-c2ccc3CN(Cc4cc(Cl)cc(Cl)c4)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccc(cc4)C(C)(C)C)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4cccc(Cl)c4)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1ccc(C)c(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)c1 |r|
Cc1nc(C)c(-c2ccc3CN(Cc4c(F)cccc4C(F)(F)F)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4cc(F)cc(F)c4)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4cccc(c4F)C(F)(F)F)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1cccc(C)c1CN1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1 |r|
Cc1nc(C)c(-c2ccc3CN(Cc4cc(F)c(F)c(F)c4)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccc(F)cc4Cl)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
CC(C)c1cccc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)c1 |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccc(F)c(F)c4)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4cc(F)ccc4F)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccc(Cl)cc4F)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4cccc(Cl)c4Cl)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccc(F)c(F)c4F)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4cc(Cl)ccc4F)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4cc(F)cc(Cl)c4)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4c(F)ccc(F)c4F)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4cc(F)ccc4Cl)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1cc(F)cc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)c1 |r|
Cc1ccc(F)cc1CN1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1 |r|
Cc1ccc(F)c(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)c1F |r|
Cc1nc(C)c(-c2ccc3CN(Cc4cc(F)c(F)cc4F)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4c(F)cccc4F)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1cccc(F)c1CN1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1 |r|
Cc1nc(C)c(-c2ccc3CN(Cc4cc(ccc4F)C(F)(F)F)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccc(Cl)cc4Cl)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1cccc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)c1F |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccccc4Cl)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccc(Cl)cc4)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1cc(C)c(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)c(C)c1 |r|
Cc1nc(C)c(-c2ccc3CN(Cc4c(F)cc(F)cc4F)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
CC(C)c1ccc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)cc1 |r|
CCc1ccc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)cc1 |r|
Cc1nc(C)c(-c2ccc3CN(Cc4cccc(c4)C#N)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccccc4C#N)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4cc(ccc4F)C#N)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccc(cc4)C#N)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1cc(ccc1CN1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1)C#N |r|
Cc1nc(C)c(-c2ccc3CN(Cc4cc(F)ccc4C(F)(F)F)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccc(F)c(c4)C(F)(F)F)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4cc(F)cc(c4)C(F)(F)F)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccc(F)cc4C(F)(F)F)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1cc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)ccc1F |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccc(F)c(C)c4C)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1ccc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)c(F)c1F |r|
Cc1ccc(F)c(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)c1 |r|
Cc1cc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)cc(C)c1F |r|
Cc1cc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)cc(F)c1F |r|
CC(C)c1ccccc1CN1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1 |r|
Cc1cc(C)c(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)cc1C |r|
Cc1cc(C)cc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)c1 |r|
Cc1cccc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)c1C |r|
Cc1nc(C)c(-c2ccc3CN(Cc4cccc(c4)C(C)(C)C)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4cccc(F)c4C)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
COc1cc(F)c(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)cc1F |r|
COc1cc(F)c(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)c(F)c1 |r|
Cc1nc(C)c(-c2ccc3CN(Cc4cc(Cl)cc(Cl)c4OCc4ccccc4)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
COc1cc(F)c(F)cc1CN1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1 |r|
COc1ccc(F)c(F)c1CN1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1 |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccccc4OCCO)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
COc1cc(F)cc(F)c1CN1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1 |r|
CCOc1cc(Cl)cc(Cl)c1CN1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1 |r|
COc1ccc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)c(Cl)c1Cl |r|
COc1ccc(F)c(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)c1F |r|
COc1cc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)c(F)cc1Cl |r|
COc1cc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)c(F)cc1F |r|
COc1c(F)cc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)cc1F |r|
Cc1nc(C)c(-c2ccc3CN(Cc4cc(F)cc(F)c4F)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
COc1ccc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)cc1F |r|
COc1c(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)cccc1C(F)(F)F |r|
COc1ccc(Cl)cc1CN1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1 |r|
COc1cc(Cl)cc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)c1 |r|
COc1cc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)ccc1F |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccc(OC(F)(F)F)cc4)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
CCOc1cccc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)c1 |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccc(OC(F)(F)F)c(Cl)c4)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccc(OC(F)F)cc4F)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccc(OC(F)(F)F)c(F)c4)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
COc1cc(ccc1CN1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1)C(F)(F)F |r|
Cc1nc(C)c(-c2ccc3CN(Cc4cccc(OC(F)(F)F)c4)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4cc(F)cc(OC(F)(F)F)c4)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
COc1cc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)cc(c1)C(F)(F)F |r|
Cc1nc(C)c(-c2ccc3CN(Cc4cc(Cl)cc(OC(F)(F)F)c4)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccccc4OC(F)F)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
COc1cccc(F)c1CN1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1 |r|
COc1ccc(F)c(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)c1 |r|
COc1cc(F)ccc1CN1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1 |r|
Cc1nc(C)c(-c2ccc3CN(Cc4cccc(OC(F)F)c4)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
COc1ccc(C)cc1CN1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1 |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccc(F)c(OC(F)(F)F)c4)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4cccc(OC(F)(F)C(F)F)c4)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
COc1cc(F)cc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)c1 |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccccc4OC(F)(F)F)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
COc1ccc(F)cc1CN1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1 |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccc(OC(F)(F)C(F)F)cc4)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
CCOc1cc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)c(F)cc1F |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccc(Cl)c(Cl)c4)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4c(Cl)cccc4Cl)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
COc1cccc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)c1Cl |r|
Cc1nc(C)c(-c2ccc3CN(Cc4cccc(Cl)c4F)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1cc(Cl)ccc1CN1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1 |r|
Cc1ccc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)cc1Cl |r|
Cc1ccc(Cl)cc1CN1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1 |r|
Cc1cc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)ccc1Cl |r|
Cc1nc(C)c(-c2ccc3CN(Cc4c(F)cc(Cl)cc4F)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4c(F)cccc4Cl)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
COc1ccc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)cc1Cl |r|
COc1cc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)ccc1Cl |r|
COc1ccc(cc1CN1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1)C(C)C |r|
COc1cc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)ccc1C |r|
COc1ccc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)cc1C |r|
COc1c(F)cccc1CN1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1 |r|
COc1ccc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)cc1C(C)C |r|
Cc1nc(C)c(-c2ccc3CN(Cc4c(O)cc(F)cc4F)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
COc1cccc(Cl)c1CN1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1 |r|
COc1ccc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)c(F)c1 |r|
COc1ccc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)c(C)c1C |r|
COc1cc(C)c(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)cc1C |r|
CCOc1ccc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)cc1 |r|
CC(C)Oc1ccc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)cc1 |r|
COc1ccc(cc1CN1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1)C(F)(F)F |r|
CC(C)Oc1ccccc1CN1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1 |r|
CC(C)COc1ccccc1CN1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1 |r|
CC(C)Oc1cccc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)c1 |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccc5OCCCc5c4)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccc5OCCOc5c4)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccc(OC(F)F)c(OC(F)F)c4)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4cccc5OCCOc45)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(Cc4c(F)cccc4Oc4ccccc4)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
CC(C)Oc1cc(C)c(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)c(C)c1 |r|
Cc1nc(C)c(-c2ccc3CN(Cc4ccc(cc4)C4(CC4)C#N)CCc3c2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
CCCCCCCCCOc1ccc(CN2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)cc1 |r|
Cc1cccc(Cl)c1CN1CCc2cc(ccc2C1)-c1cnc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1 |r|
Cc1ccccc1CN1CCc2cc(ccc2C1)-c1cnc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1 |r|
Cc1cccc(Cl)c1CN1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCCC(C)(C)C1 |r|
Cc1nc(C)c(-c2ccc3CN(CCc3c2)c2ncnc3c4ccccc4oc23)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(CCc3c2)c2nc3ccccc3c3ccccc23)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1ccc2c(c1)[nH]c1nc(nc(Cl)c21)N1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1 |r|
Cc1nc(C)c(-c2ccc3CN(CCc3c2)c2ccc3ccc4cccnc4c3n2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(CCc3c2)c2ncnc3c4ccccc4[nH]c23)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(CCc3c2)c2ncnc3sc4ccccc4c23)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(CCc3c2)c2ncnc3[nH]c4ccccc4c23)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(CCc3c2)c2ncnc3c4ccccc4sc23)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(CCc3c2)c2ncnc3c4cccnc4oc23)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(CCc3c2)c2ncnc3c4cc(F)ccc4oc23)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
CCOc1cccc2oc3c(ncnc3c12)N1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1 |r|
Cc1nc(C)c(-c2ccc3CN(CCc3c2)c2ncnc3c2oc2cccc(F)c32)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1ccc2[nH]c3c(ncnc3c2c1)N1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1 |r|
CCn1c2ccc(C)cc2c2ncnc(N3CCc4cc(ccc4C3)-c3c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c3N3CCC(C)(C)CC3)c12 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N1CCCc2ccccc12 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N(C)c1ccccc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccccc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccccc1Cl |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N(C)c1ccccc1Cl |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N1CCc2ccccc2C1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N1CC(C1)c1ccccc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N1CCc2ccccc12 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)n1c2ccccc2c2ccccc12 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N(C)c1ccccc1Cl)c1ccc2ncccc2c1 |r|
COc1ccccc1NS(=O)(=O)NC(=O)N[C@@H](Cc1ccccc1)C(=O)N(C)c1ccc2ncccc2c1 |r|
COc1ccccc1N(C)S(=O)(=O)NC(=O)N[C@@H](Cc1ccccc1)C(=O)N(C)c1ccc2ncccc2c1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N1CCCCC1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N(C)C |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccccc1Cl)c1ccc2ncccc2c1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccccc1C |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N(C)c1ccccc1C |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccccc1OC |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1cccc(Cl)c1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1cccc(OC)c1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1cccnc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccc(Cl)cc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N(C)c1ccccc1OC |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1cccc(C)c1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N(C)c1cccc(C)c1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccc(C)cc1 |r|
COc1ccc(NS(=O)(=O)NC(=O)N[C@@H](Cc2ccccc2)C(=O)N(C)c2ccc(OC)cc2)cc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N(C)c1ccc(OC)cc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ncccn1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N(C)CC(=O)N(C)C |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N1CCc2cccnc12 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1nccc2ccccc12 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)NCCc1ccccc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N(C)c1cccc(OC)c1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N(C)c1ccc(Cl)cc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccc2[nH]cnc2c1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N(C)c1cccc(Cl)c1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)NCc1ccccc1F |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)NCc1ccccn1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N(C)C(c1ccccc1)c1ccccc1 |r|
CCc1ccc(CN(C)S(=O)(=O)NC(=O)N[C@@H](Cc2ccccc2)C(=O)N(C)c2ccc(OC)cc2)cc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N1CCN(C)CC1c1ccccc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)NCc1nccs1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N1Cc2ccncc2C1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)NCc1cnc2ccccc2c1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1cc(F)cc(F)c1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)NCc1cccc(c1)-n1cccn1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1cc(F)ccc1F |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1cc(Cl)ccc1F |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccc(F)cc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccc(F)c(F)c1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccc(NC(=O)N(C)C)cc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N1CCCCC1c1ccccc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)NCc1ccc2nc(C)[nH]c2c1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)NCc1cncn1C |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)NCc1ccccc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)NCc1cccc(F)c1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)NC(C)c1cccc(C)n1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)NCc1cc(C)on1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)NC(C)c1cnn(C)c1C |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1cccc(c1)C(N)=O |r|
COC(=O)Nc1ccc(NS(=O)(=O)NC(=O)N[C@@H](Cc2ccccc2)C(=O)N(C)c2ccc(OC)cc2)cc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)NCc1nccn1C |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)NC(C)c1csc(C)n1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)NC(C)c1cccnc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)NCc1n[nH]c2ccccc12 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)NC(C)c1ncnn1C |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N(C)Cc1n[nH]c(=O)[nH]1 |r|
CCOc1ccc(cc1)N(CC)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N1CCc2cc(C)ccc12 |r|
CCOc1ccc(cc1)N(CC)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N1CCc2cccnc12 |r|
CCOc1ccc(cc1)N(CC)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N1CCc2c1cccc2Cl |r|
CCOc1ccc(cc1)N(CC)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N1CCc2ccccc12 |r|
CCOc1ccc(cc1)N(CC)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N1CCc2cc(OC)cc(C)c12 |r|
CCOc1ccc(cc1)N(CC)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)n1ccc2ccccc12 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N1CCc2c1cccc2Cl |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N1CCc2cc(C)ccc12 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N1CCc2cc(Cl)cc(Cl)c12 |r|
CCOc1ccc(cc1)N(CC)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N1CCc2cc(Cl)cc(Cl)c12 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1cccc2ccccc12 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccc2ccccc2c1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccccc1C#N |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccccc1F |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1cccc2ncccc12 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1cccc(c1)C#N |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1cccc(F)c1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccc2CCCc2c1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccc(Cl)c(Cl)c1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccc(C)c(C)c1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1cc(C)cc(C)c1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccc(cc1)C#N |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccc(Br)cc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccc(NC(C)=O)cc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccc(Oc2ccccc2)cc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccc(cc1)C(C)=O |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccc(cc1)C(C)(C)C |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccc(cc1)C(C)C |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccccc1C(N)=O |r|
CCN(c1ccccc1)S(=O)(=O)NC(=O)N[C@@H](Cc1ccccc1)C(=O)N(C)c1ccc(OC)cc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccc2ncsc2c1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N(C(C)C)c1ccccc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccccc1OC(F)(F)F |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1cccc(c1)-c1cnco1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccc(cc1)C(F)(F)F |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccc(cc1)-c1ccccc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1cccc(Cl)c1Cl |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccccc1-c1ccccc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccc(OCc2ccccc2)cc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccccc1Oc1ccccc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccc(OC(F)(F)F)cc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1cccc(OC(F)(F)F)c1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1cccc(Oc2ccccc2)c1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1cccc(c1)-c1ccccc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccc(cc1)-c1cnco1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccc(Cc2ccncc2)cc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccc(OC(C)C)cc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1cccc(c1)C(C)(C)C |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccccc1NC(C)=O |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccc(cc1)S(=O)(=O)N1CCCC1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccc(cc1)S(=O)(=O)N1CCOCC1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccc(cc1)-n1cccc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1cccc(NS(C)(=O)=O)c1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1cccc(c1)S(=O)(=O)N1CCOCC1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccc2CS(=O)(=O)Cc2c1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1cc(Cl)cc(Cl)c1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccc(Cl)cc1Cl |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)NCC(=O)N1CCCC1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)NCC(=O)N(C)C |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N1CCc2cc(OC)cc(C)c12 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)NCC(=O)N1CCN(CC1)c1ccccc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)NCC(=O)N1CCOCC1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)Nc1ccccc1C(F)(F)F |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)n1ccc2cccnc12 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)n1ccc2c(F)c(F)c(F)c(F)c12 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N1Cc2ccccc2S1(=O)=O |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)n1ccc2cnccc12 |r|
CCOc1ccc(NS(=O)(=O)NC(=O)N[C@@H](Cc2ccccc2)C(=O)N(C)c2ccc(OC)cc2)cc1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)n1ccc2ccncc12 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)n1c(C)cc2ccncc12 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)n1nc(-c2ccccc2)c2ccccc12 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)n1c(C)cc2ccc(OC)cc12 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)n1c(C)cc2cc(F)c(O)cc12 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)n1ncc2c(Cl)nc(Cl)cc12 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2ccccc12)c1ccc2scnc2c1 |r|
CCN(c1ccccc1)S(=O)(=O)NC(=O)N[C@@H](Cc1cc(F)cc(F)c1)C(=O)N(C)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)Nc1ccc(C)cc1)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)Nc1ccc(cc1)C(C)(C)C)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cc(F)ccc12)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccc(F)c12)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)n1ccc2nccnc12)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N(C)c1ccccn1)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)Nc1ccccn1)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)Nc1ccccc1)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)Nc1cccc(Cl)c1)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N(C)c1ccccc1F)c1ccc2scnc2c1 |r|
COc1ccc(cn1)N(C)S(=O)(=O)NC(=O)N[C@@H](Cc1cc(F)cc(F)c1)C(=O)N(C)c1ccc2scnc2c1 |r|
COc1cccc(c1)N(C)S(=O)(=O)NC(=O)N[C@@H](Cc1cc(F)cc(F)c1)C(=O)N(C)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N(C)c1cccnc1)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCCC1c1ccccn1)c1ccc2scnc2c1 |r|
CCN(c1cccnc1)S(=O)(=O)NC(=O)N[C@@H](Cc1cc(F)cc(F)c1)C(=O)N(C)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCCC1c1ccccc1)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)n1ncc2c(Cl)cccc12)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)n1ncc2cc(F)ccc12)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCCc2ccccc12)c1ccc2scnc2c1 |r|
C[C@@H]1Cc2cccnc2N1S(=O)(=O)NC(=O)N[C@@H](Cc1cc(F)cc(F)c1)C(=O)N(C)c1ccc2scnc2c1 |r|
C[C@H]1Cc2cccnc2N1S(=O)(=O)NC(=O)N[C@@H](Cc1cc(F)cc(F)c1)C(=O)N(C)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)n1ccc2cccnc12)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cc(Br)cnc12)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2nccnc12)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCCc2cccnc12)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1ccc2sc(C)nc2c1 |r|
C[C@@H]1CCc2ccccc2N1S(=O)(=O)NC(=O)N[C@@H](Cc1cc(F)cc(F)c1)C(=O)N(C)c1ccc2scnc2c1 |r|
C[C@H]1CCc2ccccc2N1S(=O)(=O)NC(=O)N[C@@H](Cc1cc(F)cc(F)c1)C(=O)N(C)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCCc2ccc(C)nc12)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1ccc2OCCOc2c1 |r|
CC1CN(c2ncccc12)S(=O)(=O)NC(=O)N[C@@H](Cc1cc(F)cc(F)c1)C(=O)N(C)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1ccc(C)nc1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1ccc(Cl)cc1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1ccc(=O)n(C)c1 |r|
CCc1ccc(cc1)N(C)C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12 |r|
CCc1ccc(cn1)N(C)C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCOc2cccnc12)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1ccc(C)cn1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1ccc2sc(=O)[nH]c2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1ccc2n(C)cnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1ccc(OC(F)(F)F)cc1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1ccc2n(C)ncc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1ccc(cc1)N1CCOCC1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2c1nccc2Cl |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1ccc(nc1)C(F)(F)F |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1ccc(cc1)C1CC1 |r|
COc1ccc(cn1)N(C)C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1ccc(nc1)C(F)F |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1ccc(cc1)C(N)=O |r|
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1ccc(Cl)c(C)c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1ccc(OC(F)F)nc1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2c1nccc2Cl)c1ccc2scnc2c1 |r|
COc1ccc2CCN(c2n1)S(=O)(=O)NC(=O)N[C@@H](Cc1cc(F)cc(F)c1)C(=O)N(C)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2ccncc12)c1ccc2scnc2c1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2ccncc12 |r|
CN(C)S(=O)(=O)NC(=O)N[C@@H](Cc1cc(F)cc(F)c1)C(=O)N(C)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2ccnnc12)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1cnc(C)nc1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1cnc(C)c(Cl)c1 |r|
CCCc1ccc(cc1)N(C)C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1cnc2scnc2c1 |r|
CC(C)Oc1ccc(cn1)N(C)C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1cc(C)cc(F)c1 |r|
CCc1ccc(cn1)N(C)C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N(C)C |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cncnc12)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)n1ccc2cncnc12)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cncnc12)c1ccc(C)c(F)c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1ccc(C#N)c(C)c1 |r|
CCN(CC)S(=O)(=O)NC(=O)N[C@@H](Cc1cc(F)cc(F)c1)C(=O)N(C)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCCC1)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCOCC1)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCCCC1)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1ccc(Cl)c(C)c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1ccc(F)c(C)c1 |r|
CC(C)c1ccc(cn1)N(C)C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12 |r|
COc1cncc(c1)N(C)C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(N)(=O)=O)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1ccc(C)c(Cl)c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1cccnc1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1ccc2sc(=O)n(C)c2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1cnc(C)c(C)c1 |r|
COc1ccc(cc1F)N(C)C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCC(F)(F)CC1 |r|
COc1ccc(cc1F)N(C)C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCCCC1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCC[C@H]1C(=O)N(C)C |r|
CN(C)C(=O)[C@@H]1CCCN1S(=O)(=O)NC(=O)N[C@@H](Cc1cc(F)cc(F)c1)C(=O)N(C)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CC[C@H](O)C1)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1ccc(Cl)c(c1)C#N |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CC[C@@H](O)C1)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)N1CCN(C)S1(=O)=O)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1ccc(CC(F)F)cc1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)N(C)S(=O)(=O)N1CCc2cccnc12)c1ccc2scnc2c1 |r|
CN(C)C(=O)[C@H]1CCCN1S(=O)(=O)NC(=O)N[C@@H](Cc1cc(F)cc(F)c1)C(=O)N(C)c1ccc2scnc2c1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCC[C@@H]1C(=O)N(C)C |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCN(C)CC1)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)Nc1cccnc1)c1ccc2scnc2c1 |r|
CCNS(=O)(=O)NC(=O)N[C@@H](Cc1cc(F)cc(F)c1)C(=O)N(C)c1ccc2scnc2c1 |r|
CN(CCO)S(=O)(=O)NC(=O)N[C@@H](Cc1cc(F)cc(F)c1)C(=O)N(C)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)NCc1ccccc1)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)NCC1CC1)c1ccc2scnc2c1 |r|
COC1CN(C1)S(=O)(=O)NC(=O)N[C@@H](Cc1cc(F)cc(F)c1)C(=O)N(C)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CC(C)(O)C1)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CC(F)(F)C1)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1ccc2sc(C)nc2c1F |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCC[C@H]1CO)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)NC1CCC1)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCC(Cc2ccccc2)CC1)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)NCc1ccccn1)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)NCc1cccnc1)c1ccc2scnc2c1 |r|
CC(C)NS(=O)(=O)NC(=O)N[C@@H](Cc1cc(F)cc(F)c1)C(=O)N(C)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)NCCNC(C)=O)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)NCCO)c1ccc2scnc2c1 |r|
CN(Cc1ccccc1)S(=O)(=O)NC(=O)N[C@@H](Cc1cc(F)cc(F)c1)C(=O)N(C)c1ccc2scnc2c1 |r|
CC(C)CN(C)S(=O)(=O)NC(=O)N[C@@H](Cc1cc(F)cc(F)c1)C(=O)N(C)c1ccc2scnc2c1 |r|
CCCN(C)S(=O)(=O)NC(=O)N[C@@H](Cc1cc(F)cc(F)c1)C(=O)N(C)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)NC1CC1)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)NCC(C)(C)C)c1ccc2scnc2c1 |r|
CC(C)CNS(=O)(=O)NC(=O)N[C@@H](Cc1cc(F)cc(F)c1)C(=O)N(C)c1ccc2scnc2c1 |r|
CC(C)CCNS(=O)(=O)NC(=O)N[C@@H](Cc1cc(F)cc(F)c1)C(=O)N(C)c1ccc2scnc2c1 |r|
CCCNS(=O)(=O)NC(=O)N[C@@H](Cc1cc(F)cc(F)c1)C(=O)N(C)c1ccc2scnc2c1 |r|
CC(C)N(C)S(=O)(=O)NC(=O)N[C@@H](Cc1cc(F)cc(F)c1)C(=O)N(C)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCN(CC1)C(C)=O)c1ccc2scnc2c1 |r|
COCCN(C)S(=O)(=O)NC(=O)N[C@@H](Cc1cc(F)cc(F)c1)C(=O)N(C)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)NCc1cnc(C)cn1)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCNC(=O)C1)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCC(C1)c1ccccc1)c1ccc2scnc2c1 |r|
COCCNS(=O)(=O)NC(=O)N[C@@H](Cc1cc(F)cc(F)c1)C(=O)N(C)c1ccc2scnc2c1 |r|
CCN(C)S(=O)(=O)NC(=O)N[C@@H](Cc1cc(F)cc(F)c1)C(=O)N(C)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCC(O)CC1)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCC(CC1)c1ccccc1)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2ccccc2C1)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)NCCc1ccccc1)c1ccc2scnc2c1 |r|
CN(C)C(=O)C1Cc2cccnc2N1S(=O)(=O)NC(=O)N[C@@H](Cc1cc(F)cc(F)c1)C(=O)N(C)c1ccc2scnc2c1 |r|
CN(C)C(=O)C1Cc2cccnc2N1S(=O)(=O)NC(=O)N[C@H](Cc1cc(F)cc(F)c1)C(=O)N(C)c1ccc2scnc2c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1ccc2scnc2c1F |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1ccc2cncnc2c1 |r|
COc1ccc(cc1)N(C)C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12 |r|
COc1ccc(cc1)N(C1CC1)C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCCC1=O)c1ccc2scnc2c1 |r|
Fc1cc(F)cc(C[C@H](NC(=O)NS(=O)(=O)N2CCc3cccnc23)C(=O)N(CCOCc2ccccc2)c2ccc3scnc3c2)c1 |r|
CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)NS(=O)(=O)N1CCc2cccnc12)c1ccc(OC(F)F)cc1 |r|
CCN(CC)S(=O)(=O)NC(=O)N[C@@H](Cc1cc(F)cc(F)c1)C(=O)N(C)c1ccc(OC(F)F)cc1 |r|
CN(C)S(=O)(=O)NC(=O)N[C@@H](Cc1cc(F)cc(F)c1)C(=O)N(C)c1ccc(OC(F)F)cc1 |r|
CN1CCN(CCOc2ccc(cc2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)CC1 |r|
Cc1nc(C)c(-c2ccc(OCCC3CCCCC3)cc2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc(OCCN3CCOCC3)cc2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc(OCC3(CC3)c3ccc(F)cc3)cc2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc(OCCN3CCSCC3)cc2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc(OC3CCCC3c3ccc(F)cc3)cc2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1c(Cl)cccc1NS(=O)(=O)c1ccc2NC(C3CC=CC3c2c1)c1ccc(cc1)C(O)=O |c:21|
OC(=O)CCCN1C(=S)S\C(=C/c2ccc(o2)-c2nc3ccccc3s2)C1=O
CCC(Sc1nc2ccsc2c(=O)n1Cc1ccc(cc1)C(O)=O)C(=O)Nc1ccc(C)c(Cl)c1
COc1cc(CN=Nc2ccc(Cl)c(c2)C(O)=O)ccc1OC(=O)c1ccccc1F |w:7.7|
COc1cc(CN=Nc2ccc(Cl)c(c2)C(O)=O)ccc1OC(=O)c1ccc(F)cc1 |w:7.7|
OC(=O)c1cc(ccc1Cl)N=NCc1ccc(cc1)-c1ccccc1 |w:10.10|
COc1ccc(cc1)C(=O)Oc1ccc(CN=Nc2ccc(Cl)c(c2)C(O)=O)cc1OC |w:17.18|
Cc1ccc(c(C)c1)-n1c(O)c(C=Nc2ccccc2-c2n[nH]c(=S)[nH]c2=O)c2ccccc2c1=O |w:13.14,(4.41,6.16,;5.75,5.39,;5.75,3.85,;7.08,3.08,;8.41,3.85,;8.41,5.39,;9.75,6.16,;7.08,6.16,;9.75,3.08,;9.75,1.54,;8.41,.77,;11.08,.77,;11.08,-.77,;9.75,-1.54,;9.75,-3.08,;11.08,-3.85,;11.08,-5.39,;9.75,-6.16,;8.41,-5.39,;8.41,-3.85,;7.08,-3.08,;7.08,-1.54,;5.75,-.77,;4.41,-1.54,;3.08,-.77,;4.41,-3.08,;5.75,-3.85,;5.75,-5.39,;12.42,1.54,;13.79,.72,;15.19,1.51,;15.19,3.11,;13.79,3.9,;12.42,3.08,;11.08,3.85,;11.08,5.39,)|
COc1ccccc1NS(=O)(=O)c1cccc(c1)-n1c(O)c(C=Nc2ccccc2C(O)=O)c2ccccc2c1=O |w:23.25|
Fc1ccc(cc1)N1C(=S)NC(=O)C(=Cc2ccco2)C1=O |w:14.15|
CC1(C)CC(=O)C2=C(C1)c1c(NC2c2cc(cc(c2O)[N+]([O-])=O)[N+]([O-])=O)ccc2ccccc12 |c:6|
Oc1c(\C=c2/sc3nc4ccccc4n3c2=O)cc(cc1[N+]([O-])=O)[N+]([O-])=O
COc1ccc(OC)c(c1)N1C(=S)NC(=O)C(=Cc2ccco2)C1=O |w:17.18|
Cc1ccc(cc1Cl)-n1cccc1\C=C1\C(=N)N2C(SN=C2S(C)(=O)=O)=NC1=O |c:22,28|
CS(=O)(=O)C1=NSC2=NC(=O)\C(=C/c3cccn3-c3ccc(Cl)cc3)C(=N)N12 |t:4,7|
Cc1cc(C)cc(c1)-n1cccc1\C=C1/C(=O)N=C2SN=C(N2C1=N)S(C)(=O)=O |c:22,t:19|
CC(C)S(=O)(=O)C1=NSC2=NC(=O)\C(=C/c3ccc(o3)-c3ccccc3)C(=N)N12 |t:6,9|
CC(C)S(=O)(=O)C1=NSC2=NC(=O)\C(=C/c3ccc(o3)-c3cccc(c3)C(O)=O)C(=N)N12 |t:6,9|
Cc1ccc(cc1)S(=O)(=O)Oc1ccc(\C=C2/C(=O)N=C3SN=C(N3C2=N)S(C)(=O)=O)cc1 |c:23,t:20|
CS(=O)(=O)C1=NSC2=NC(=O)\C(=C/c3ccc(OS(=O)(=O)c4ccccc4)cc3)C(=N)N12 |t:4,7|
CCS(=O)(=O)C1=NSC2=NC(=O)\C(=C/c3ccc(OS(=O)(=O)c4ccccc4)cc3)C(=N)N12 |t:5,8|
CCC=c1[nH]n(-c2ccccc2)c(=O)c1=Cc1ccc(OCc2ccc(cc2)C(O)=O)cc1 |w:2.1,15.17|
OC(=O)c1ccccc1N[NH+]=C1C(=O)[N-]c2ccc(cc12)[N+]([O-])=O |w:10.10|
CC(C)NC(=O)c1sc(=S)n2c1[nH]c(=O)c1ccc(cc21)C(=O)NCCc1ccc(Cl)cc1
[O-][N+](=O)c1c[c-](\C=C(/C#N)c2[nH+]c3ccccc3s2)ccc1=O
Oc1c(cc([N+]([O-])=O)c2oc(c(Br)c12)-c1ccccc1)[N+]([O-])=O
Oc1ccccc1C(=O)NNC=C1C(=O)NC(=S)N(C2CCCCC2)C1=O |w:11.11|
COc1cc(\C=N\NS(=O)(=O)c2ccc3ccccc3c2)ccc1OCc1ccc(cc1)C(O)=O
CSc1nnc(-c2ccccc2N=Cc2c(C)[nH]n(-c3ccc4ccccc4c3)c2=O)c(=O)[nH]1 |w:12.12|
CCOC(=O)C1=C(C)N=c2sc(=Cc3ccc(OCC(O)=O)cc3)c(=O)n2C1c1ccc(OC(C)C)cc1 |c:5,t:8|
COC(=O)c1sc(cc1NC(=O)c1ccccc1C(O)=O)-c1ccc(cc1)C(C)(C)C
CCC(C)(C)C1CCc2c(C1)sc(NC(=O)c1ccccc1C(O)=O)c2C#N
Fc1ccc(cc1)N1C(=S)NC(=O)C(=Cc2ccoc2)C1=O |w:14.15|
CCOC(=O)c1sc(nc1C)N1C(C(C(=O)c2ccc(C)o2)C(=O)C1=O)c1cccc(c1)[N+]([O-])=O
COc1cc(\C=C2/SC(=O)N(C2=O)c2ccccc2Cl)cc(c1O)[N+]([O-])=O
CCOc1cc(\C=C2/SC(=O)N(CC(=O)Nc3ccccc3F)C2=O)cc(c1O)[N+]([O-])=O
c1c(c(c(c(c1Cl)Cl)Cc2c(c(cc(c2Cl)Cl)Cl)O)O)Cl
CC(C)(C)c1cc(cc(c1O)C(C)(C)C)-c1cs\c(=[NH+]/c2ccccc2)n1Cc1ccc(cc1)C(O)=O
Cc1n(Cc2ccccc2)c(=O)cc2[n-]n(-c3nc4ccccc4s3)c(=O)c12
OC(=O)c1ccccc1C(=O)N(Cc1cccc(Oc2ccc(Cl)cc2)c1)[C@H]1CCCc2ccccc12
OC(=O)c1cccc(NC(=O)C(=C\c2ccc(OCc3ccc(Cl)cc3)cc2)\C#N)c1
O=c1[nH]c2cc3OCCOc3cc2cc1C(N1CCSCC1)c1nnnn1C1CCCC1
CCOC(=O)c1c(C)[nH]sc1=S
CCOC(=O)CSc1nc(N)c(C#N)c(-c2ccc(OC)cc2)c1C#N
CCOc1cccc(c1)-c1nn2c(nnc2s1)-c1ccco1
Cc1nc(SCC(=O)Nc2ccc3OCCOc3c2)c2oc3ccccc3c2n1
Oc1ccccc1-c1n[nH]c2C(=O)N(CC3CCCO3)C(c12)c1cccc(Cl)c1
Cc1cc(=O)oc2cc(NC(=O)C3COc4ccccc4O3)ccc12
COc1cc(ccc1OCc1c(C)noc1C)C(=O)Oc1ccccc1
CCOc1ccc(OCC)c(NC(=O)c2[nH]c(C)c(C(C)=O)c2C)c1
Fc1ccc(NC(=O)c2ccc3c(c2)nc2CCCCCn2c3=O)c(Cl)c1
COc1ccc(NC(=O)c2oc3ccccc3c2NC(=O)C2CC2)cc1
CCSc1nnc(NC(=O)c2cc3CCCCc3s2)s1
COC(=O)Cc1c(C)c2c(O)cc(C)cc2oc1=O
Cc1ccc(o1)-c1c2CCCCc2[nH]c(=S)c1C#N
Cc1cc(NC(=O)CSc2nc(nc3sc(C)c(C)c23)C2CC2)no1
COc1cc2[nH]c(=S)n(NC(=O)c3ccccc3)c(=O)c2cc1OC
c1nc2ccccc2n1-c1ccc(cc1)-c1ccnc(n1)-c1ccccc1
Cc1cc2ccccc2n1CCNC(=O)C1CCCCC1
COc1ccc(OC)c(c1)S(=O)(=O)Nc1ccc(cc1)C(C)=O
CCn1c(=S)[nH]c2nc3CCCCc3cc2c1=O
Cc1cccc(NC(=O)C2CCCN(C2)S(=O)(=O)c2cccc3nsnc23)c1
CC(C)c1ccc(cc1)-c1c(C#N)c(N)nc(SCC(=O)N2CCCCC2)c1C#N
Cc1nc(SCC(=O)NCCc2ccccc2)c2oc3ccccc3c2n1
O=C(Nc1nnc(SCc2ccccc2)s1)c1cc2CCCCc2s1
COc1ccc(cc1)C(=O)Nc1ccccc1C(=O)N(Cc1ccco1)C(C(C)C)C(N)=O
Cc1n(nc2c1c(C)n[nH]c2=S)-c1ccc(C)cc1
COC(=O)Nc1nc(c(s1)C(=O)c1ccccc1)-c1ccccc1
COCc1cc(C)n(CC(=O)Nc2ccc(Cl)cc2Cl)c(=O)c1C#N
Clc1ccc(cc1)-c1c2CCCc2nc2sc3c([nH]cnc3=O)c12
Cc1c(Cl)c(nn1C)-c1n[nH]c(=S)n1-c1ccc(F)cc1
CCCc1nc(SCC(=O)Nc2nnc(CC)s2)c2c(C)c(C)sc2n1
Cc1ccc(NC(=S)Nc2nc(CC(=O)Nc3ccccc3)cs2)cc1
S=c1[nH]cnc2c3ccccc3[nH]c12
C1CN(CCO1)c1ccc(cc1)-c1ccc2ccccc2n1
COc1ccc(cc1)C(=O)\C=C1\Sc2cc3OCOc3cc2N1C
COc1cc(CN(C2CCCCC2C)S(=O)(=O)c2ccc(cc2)S(=O)(=O)NC2CC2)cc(OC)c1OC
Cc1ccc2[nH]c3c(nc[nH]c3=S)c2c1
CCc1ccccc1NC(=O)COc1ccc2oc(cc(=O)c2c1)-c1ccc(OC)cc1
Cc1ccc(cc1)-n1c(=S)[nH]c2c3ccccc3oc2c1=O
O=c1n(-c2ccccc2)c(=S)[nH]c2c3ccccc3oc12
COc1ccc(cc1)-n1c(=S)[nH]c2c3ccccc3oc2c1=O
Cc1cccc(Nc2nc3c(nnn3c3ccccc23)S(=O)(=O)c2ccccc2)c1C
COc1ccc2[nH]c3c(nc[nH]c3=S)c2c1
COc1ccc(NC(=O)c2c(NC(=O)CNCC(C)C)sc3CCCc23)c(OC)c1
CCn1c(=S)[nH]c2-c3ccccc3CC(C)(C)c2c1=O
NS(=O)(=O)c1ccc(CCNC(=O)CCCCCn2c(=S)[nH]c3ccc(Br)cc3c2=O)cc1
CC1CCN(CCCn2c(=S)[nH]c3c4ccccc4sc3c2=O)CC1
COc1ccccc1NS(=O)(=O)c1cccc(NC(=O)c2[nH]c(C)c(C(C)=O)c2C)c1
CCC(=O)c1ccc(OCC(=O)c2ccc3OCC(=O)Nc3c2)cc1
S=c1[nH]c2ccccc2c2ccccc12
S=c1[nH]c2ccccc2n2cccc12
O=C(Nc1ccc2OCOc2c1)C1CCN(CC1)c1ccc(cc1)S(=O)(=O)N1CCOCC1
COc1ccc(cc1OC)-c1c(C)nn2c(cc(C)nc12)N1CCC(CC1)C(=O)N1CCCCC1
Cc1ccc2nc(cn2c1)-c1cc(no1)-c1ccccc1
COc1ccc(cc1)-c1c(C#N)c(N)nc(Sc2ccc(Cl)cc2)c1C#N
Nn1c(=S)[nH]c2sc3CCCCc3c2c1=O
NS(=O)(=O)c1ccc(CCNC(=O)c2ccc(cc2)-c2ccccc2)cc1
COc1ccc(C(=O)Nc2nnc(Cc3ccccc3)s2)c(OC)c1
CC1(C)Cc2ccccc2-c2[nH]c(=S)[nH]c(=O)c12
CCOC(=O)c1c(C)n(CC=C)c2c1cc(O)c1ccccc21
CCC1(C)Cc2ccccc2-c2nc(SC)[nH]c(=O)c12
S=c1[nH]c(Cc2ccccc2)nc2ccccc12
CCOc1ccc2cc(C(=O)NCc3ccccc3)c(=N)oc2c1
COCCNC(=O)c1cnc2ccc(cc2c1O)S(=O)(=O)Nc1ccc(F)cc1F
COc1ccccc1Cn1c(=S)[nH]c2ccc(F)cc2c1=O
COc1ccc(Br)cc1-c1nc2n(Cc3ccccc3)c(=O)[nH]c(=O)c2n1C
CSc1ccc(cc1)C(=O)NC1CCSc2ccccc12
Fc1ccccc1C(=O)Nc1nnc(s1)-c1ccccc1F
COC(=O)c1cc(-c2ccc(Br)cc2)c2c(n1)n(C)c(=O)[nH]c2=O
S=c1[nH]cnc2n(ncc12)-c1ccccc1
CCN(CC)c1ccc(cc1)-c1sc(Nc2ccc(CC)cc2)n[n+]1-c1ccccc1
Clc1ccccc1CNC(=O)CCCn1c(=S)[nH]c2cc3OCOc3cc2c1=O
Fc1ccccc1C1C(C(=O)c2ccc3OCCOc3c2)C(=O)C(=O)N1Cc1ccncc1
Brc1cccc(c1)C1C(C(=O)c2ccc3OCCOc3c2)C(=O)C(=O)N1CCCn1ccnc1
COc1ccc2cc([nH]c2c1)C(=O)N1CCc2ccccc2C1
COc1ccc(C(=O)NC(=S)Nc2ccc3[nH]c(=O)[nH]c3c2)c(OC)c1
COc1cccc(NC(=O)Cn2c3ccc(OC)cc3c3nc4SCCn4c(=O)c23)c1
CSc1ccc(cc1)S(=O)(=O)Nc1ccccc1C(=O)N1CCOCC1
CC(=O)c1cccc(NC(=O)c2cccc(c2)N2C(=O)c3ccccc3C2=O)c1
COC(=O)c1ccc(NC(=O)c2ccc(NC(=O)c3ccco3)cc2)cc1
CCCc1cc(=O)oc2cc(OCC(=O)Nc3ccc(cc3)S(N)(=O)=O)ccc12
Clc1cccc(NC(=O)Cn2cnc3c4cc5CCCCc5nc4oc3c2=O)c1
CCSc1nnc(NC(=O)C(Cc2ccccc2)n2cccc2)s1
Cc1sc2ncnc(N3CCC(CC3)C(=O)Nc3ccc(cc3)C#N)c2c1C
[O-][N+](=O)c1ccc(cc1)N1CCN(CC1)C(=O)c1cc(ccc1N1CCOCC1)[N+]([O-])=O
CCN(c1ccc(cc1)C(=O)CN1C(=O)NC2(CCOc3ccccc23)C1=O)S(C)(=O)=O
CN(CC(=O)Nc1ccc(C)cc1)C(=O)COc1ncnc2ccc(Br)cc12
COc1ccc(NC(=O)COC(=O)c2ccc3OCOc3c2)c(OC)c1
O=C(Oc1ccccc1)Oc1ccc2c(c1)oc(=O)c1ccccc21
CCCCc1nc2sc3c(SCC(=O)NCc4ccco4)ncnc3c2c2CCCc12
CCOC(=O)c1sc(S)nc1C
COc1ccc(C(=O)NCCN(C)C)c2nc3ccccc3cc12
COc1cc(OC)cc(c1)-c1c(Sc2ccccc2)c2cc(ccc2n1C)-c1ccc(OC)c(OC)c1
COc1ccc(cc1)-c1c(Sc2ccccc2)c2cc(ccc2n1C)-c1ccc2OCOc2c1
COC(=O)C1=C(C)N(Cc2ccccc2C(F)(F)F)C(NCc2ccc(OC)cc2)=NC1c1cccc(c1)C(F)(F)F |c:4,31|
Cc1nc(C)c(-c2ccc3CN(CCc3c2)c2nc3ncc(cc3s2)C(F)(F)F)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(CCc3c2)c2nc3cccnc3s2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(CCc3c2)c2nc3c(Cl)cncc3s2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(CCc3c2)c2nc3ccc(Cl)cc3s2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(CCc3c2)c2nc3cc(Cl)c(Cl)cc3s2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1ccc2sc(nc2c1)N1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1 |r|
Cc1nc(C)c(-c2ccc3CN(CCc3c2)c2nc3c(Cl)cccc3s2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(CCc3c2)c2nc3ccc(F)cc3s2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1ccc2nc(sc2c1)N1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1 |r|
Cc1nc(C)c(-c2ccc3CN(CCc3c2)c2nc3ncccc3s2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(CCc3c2)c2nc3cnccc3s2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
COc1ccc2nc(sc2c1)N1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1 |r|
Cc1nc(C)c(-c2ccc3CN(CCc3c2)c2nc3ccccc3s2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(CCc3c2)c2ncnc3sccc23)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1csc2c(ncnc12)N1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1 |r|
Cc1nc(C)c(-c2ccc3CN(CCc3c2)c2ncnc3n(C)ncc23)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(CCc3c2)c2nc3ccccc3n2C)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(CCc3c2)c2noc3ccccc23)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(N2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)c2cnn(C)c2n1 |r|
Cc1nc(C)c(-c2ccc3CN(CCc3c2)c2ncnc3[nH]ccc23)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(CCc3c2)c2nc(O)c3[nH]cnc3n2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(CCc3c2)c2ncnc3cc[nH]c23)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
CNc1nc(nc2nc[nH]c12)N1CCc2cc(ccc2C1)-c1c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c1N1CCC(C)(C)CC1 |r|
Cc1nc(C)c(-c2ccc3CN(CCc3c2)c2nccc3[nH]cnc23)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
Cc1nc(C)c(-c2ccc3CN(CCc3c2)c2ncc3cc[nH]c3n2)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
COc1nc(N2CCc3cc(ccc3C2)-c2c(C)nc(C)c([C@H](OC(C)(C)C)C(O)=O)c2N2CCC(C)(C)CC2)c2cc[nH]c2n1 |r|
Cc1nc(C)c(-c2ccc3CN(CCc3c2)c2ncnc3cc(sc23)C(C)(C)C)c(N2CCC(C)(C)CC2)c1[C@H](OC(C)(C)C)C(O)=O |r|
COc1ccc(c(F)c1)[C@@]1(CC(C)(C)C)NC(=N)N([C@H](COC(=O)N(C)C)c2ccc(Cl)c(c2)-c2ncccc2C)C1=O |r|
CN(C)C(=O)OC[C@@H](N1C(=N)N[C@@](C2CC2)(C1=O)c1cc(F)cc(F)c1)c1ccc(Cl)c(c1)-c1ncc(s1)-c1ccccc1 |r|
CN(C)C(=O)OC[C@@H](N1C(=N)N[C@@](C2CC2)(C1=O)c1cc(F)cc(F)c1)c1ccc(Cl)c(c1)-c1ncc(s1)N1CCOCC1 |r|
CN(C)C(=O)OC[C@@H](N1C(=N)N[C@@](C2CC2)(C1=O)c1cc(F)cc(F)c1)c1ccc(Cl)c(c1)-c1ncc(o1)-c1ccccc1 |r|
CN(C)C(=O)OC[C@@H](N1C(=N)N[C@@](C2CC2)(C1=O)c1cc(F)cc(F)c1)c1ccc(Cl)c(c1)-c1nccs1 |r|
CN(C)C(=O)OC[C@@H](N1C(=N)N[C@@](C2CC2)(C1=O)c1cc(F)cc(F)c1)c1ccc(Cl)c(c1)-c1nc(cs1)-c1ccccc1 |r|
CC(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC(C)C)c2cccc(c2)-c2ocnc2C)C1=O)c1ccccc1 |r|
COc1ccc(c(F)c1)[C@@]1(CC(C)(C)C)NC(=N)N([C@H](COC(=O)N(C)C)c2ccc(Cl)c(c2)-c2ccccn2)C1=O |r|
COc1ccc(c(F)c1)[C@@]1(CC(C)(C)C)NC(=N)N([C@H](COC(=O)N(C)C)c2ccc(Cl)c(c2)-c2nccn2C)C1=O |r|
COc1ccc(c(F)c1)[C@@]1(CC(C)(C)C)NC(=N)N([C@H](COC(=O)N(C)C)c2ccc(Cl)c(c2)-c2ncccc2F)C1=O |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2CC2)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1F)-c1cnn(c1)C(F)F |r|
Cc1cccnc1-c1cc(ccc1Cl)[C@@H](COC(=O)NC1CC1)N1C(=N)N[C@@](CC(C)(C)C)(C1=O)c1ccc(cc1F)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2CC2)c2ccc(Cl)c(c2)-c2ncccc2Cl)C1=O)c1ccc(cc1F)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2CC2)c2ccc(Cl)c(c2)-c2ncccn2)C1=O)c1ccc(cc1F)-c1cnn(c1)C(F)F |r|
COc1ccnc(n1)-c1cc(ccc1Cl)[C@@H](COC(=O)NC1CC1)N1C(=N)N[C@@](CC(C)(C)C)(C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2CC2)c2ccc(Cl)c(c2)-c2ncc[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2CC2)c2ccc(Cl)c(c2)-c2nccc(=O)[nH]2)[C@H]1O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
Cn1ncnc1-c1cc(ccc1Cl)[C@@H](COC(=O)NC1CC1)N1C(=N)N[C@@](CC(C)(C)C)(C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2CC2)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ccccn2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2CC2)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1F)-c1cnccn1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2CC2)c2ccc(Cl)c(c2)-c2nc(Cl)c[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2CC2)c2ccc(Cl)c(c2)-c2nc(Cl)c(Cl)[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2CC2)c2ccc(Cl)c(c2)-c2cc[nH]n2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnccn1 |r|
CC(C)(C)C[C@@]1(NC(=N)C([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnccn1 |r|
CC(C)(C)C[C@@]1(NC(=N)C([C@H](COC(=O)NC2CC2)c2ccc(Cl)c(c2)-c2ncn[nH]2)[C@H]1O)c1ccc(cc1)-c1cnccn1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(N)=O)c2ccc(Cl)c(c2)-c2c[nH]cn2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2CC2)c2ccc(Cl)c(c2)-c2c[nH]cn2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(C)CC2)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(C)CC2)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F)C(F)(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(C)CC2)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnccn1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2CC2)c2ccc(Cl)c(c2)-c2ncn(n2)C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2CC2)c2ccc(Cl)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2CC2)c2ccc(Cl)c(c2)-c2cn(cn2)C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2CC2)c2ccc(Cl)c(c2)-c2cncn2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2CC2)c2ccc(Cl)c(c2)-c2ncnn2C2CC2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2CC2)c2ccc(Cl)c(c2)-c2nncs2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
Cc1nnc([nH]1)-c1cc(ccc1Cl)[C@@H](COC(=O)NC1CC1)N1C(=N)N[C@@](CC(C)(C)C)(C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
Cn1cc(nn1)-c1cc(ccc1Cl)[C@@H](COC(=O)NC1CC1)N1C(=N)N[C@@](CC(C)(C)C)(C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](CO)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(C)CC2)c2ccc(Cl)c(c2)-c2ncnn2C2CC2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2CC2)c2ccc(Cl)c(c2)-c2nnc(s2)C2CC2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC(C)(C)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](CO)c2ccc(Cl)c(c2)-c2ncnn2C2CC2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(C)CC2)c2ccc(Cl)c(c2)-c2ccccn2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2CC2)c2ccc(Cl)c(c2)-c2ncns2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N2CC(F)(F)C2)c2ccc(Cl)c(c2)-c2ccccn2)C1=O)c1ccc(cc1)-c1cnn(c1)C1CC1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(C)CC2)c2ccc(Cl)c(c2)-c2nncs2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(C)CC2)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C1CC1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(C)CC2)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1ccccn1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncnn2C2CC2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C1CC1)C(F)(F)F |r|
CC(C)(C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(C)CC2)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C1CC1)C(F)(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(C)CC2)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(CC(F)(F)F)c1 |r|
CC(C)(NC(=O)OC[C@@H](N1C(=N)N[C@@](CC(C)(C)C(F)(F)F)(C1=O)c1ccc(cc1)-c1cnn(c1)C1CC1)c1ccc(Cl)c(c1)-c1ncn[nH]1)C(F)F |r|
CC(C)(CF)NC(=O)OC[C@@H](N1C(=N)N[C@@](CC(C)(C)C(F)(F)F)(C1=O)c1ccc(cc1)-c1cnn(c1)C1CC1)c1ccc(Cl)c(c1)-c1ncn[nH]1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C1CC1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1ccccn1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N2CC(F)(F)C2)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC(C)(C)C)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC(C)(C)C(F)F)c2ccc(Cl)c(c2)-c2ncn(n2)C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(C)CC2)c2ccc(Cl)c(c2)-c2ncn(n2)C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)C#N)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2nnn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N2CC(C)(C)C2)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N2CC(C)(F)C2)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N2CC(F)(F)C2)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C1CC1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC(C)(C)C(F)F)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC(C)(C)C(F)F)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C1CC1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N(CC(F)F)C2CC2)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CN(C)C(=O)OC[C@@H](N1C(=N)N[C@@](CC(C)(C)C)(C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F)c1ccc(Cl)c(c1)-c1ncn[nH]1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N2CC3(COC3)C2)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N2CC(C2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N2CC(C2)S(C)(=O)=O)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N2CC(C)(C2)C#N)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N2CCC2)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N2CC3(CC3)C2)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC1CCN1C(=O)OC[C@@H](N1C(=N)N[C@@](CC(C)(C)C)(C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F)c1ccc(Cl)c(c1)-c1ncn[nH]1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC(C)(C)C(F)F)c2ccc(Cl)c(c2)-c2nccn2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC(C)(C)C(F)F)c2ccc(Cl)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC(C)(C)C(F)F)c2ccc(Cl)c(c2)-c2nncn2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N2CC3(CCO3)C2)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)F)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2COC2)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N(CC(F)(F)F)C2CC2)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
Cn1cnc(n1)-c1cc(ccc1Cl)[C@@H](COC(=O)NC(C)(C)C(F)F)N1C(=N)N[C@@](C[C@@]2(C)CC2(F)F)(C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
Cn1cnc(n1)-c1cc(ccc1Cl)[C@@H](COC(=O)NC(C)(C)C(F)F)N1C(=N)N[C@@](C[C@]2(C)CC2(F)F)(C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
Cn1cnc(n1)-c1cc(ccc1Cl)[C@@H](COC(=O)NC(C)(C)C(F)F)N1C(=N)N[C@@](CC2(C)CC2)(C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N2CC(C2)C(F)F)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N2CC(F)(F)C2)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C1COC1 |r|
CC(C)(F)C[C@@]1(NC(=N)N([C@H](COC(=O)N2CC(F)(F)C2)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC(C)(CO)CO)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N2CC(F)(F)C2)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1ncccn1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1ncccn1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC(C)(C)C)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C1COC1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)Nc2ccccc2)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)Nc2ccccn2)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1F)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N2CC(F)(F)C2)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1F)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1F)-c1ncccn1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC(C)(C)C)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1F)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC(C)(C)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncn[nH]2)C1=O)c1ccc(cc1F)-c1ccccn1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)C2=NC=NC2C(F)F)C1=O)c1ccc(cc1)-c1ncccn1 |r,c:34,t:32|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1)-c1cnc(nc1)C#N |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1)-c1cnsc1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1)-c1ccn2ccnc2c1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1)-c1cnc2ccccn12 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1)-c1cnc(nc1)C(F)(F)F |r|
CC(C)(C)C[C@@H]1N(C(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(F)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@H]1N(C(=N)N([C@H](COC(=O)NC(C)(C)C(F)F)c2ccc(F)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@H]1N(C(=N)N([C@H](COC(=O)NC(C)(C)C(F)F)c2ccc(Cl)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1)-c1ncccn1 |r|
CC(C)(F)C[C@@H]1N(C(=N)N([C@H](COC(=O)NC(C)(C)C(F)F)c2ccc(Cl)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(Br)cc1 |r|
CC(C)(F)C[C@@]1(NC(=N)N([C@H](COC(=O)NC(C)(C)C(F)F)c2ccc(Cl)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1)-c1ncccn1 |r|
Cn1ncnc1-c1cc(ccc1Cl)[C@@H](COC(=O)NC(C)(C)C(F)F)N1C(=N)N[C@@](CC(C)(C)F)(C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(F)C[C@@]1(NC(=N)N([C@H](COC(=O)NC(C)(C)C(F)F)c2ccc(Cl)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
Cn1ncnc1-c1cc(ccc1Cl)[C@@H](COC(=O)NC(C)(C)C(F)F)N1C(=N)N[C@@](CC(C)(C)C(F)(F)F)(C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(F)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C1CC1 |r|
CC(C)(F)C[C@@]1(NC(=N)N([C@H](COC(=O)NC(C)(C)C(F)F)c2ccc(Cl)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1F)-c1ncccn1 |r|
CC(C)(F)C[C@@]1(NC(=N)N([C@H](COC(=O)NC(C)(C)C(F)F)c2ccc(Cl)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1F)-c1cnn(c1)C1CC1 |r|
CC(C)(F)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C1CC1)C(F)(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(-c2cnn(c2)C2CC2)c(F)c1F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1)-c1cn(nn1)C1CC1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1)-n1cc(F)cn1 |r|
CC1(C[C@@]2(NC(=N)N([C@H](COC(=O)NC3(CC3)C(F)(F)F)c3ccc(Cl)c(c3)-c3ncnn3C(F)F)C2=O)c2ccc(cc2)-c2cnn(c2)C2CC2)CC1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(C#N)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(C(N)=O)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1F)-c1ncn(n1)C1CC1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1F)-c1cnn(n1)C1CC1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(-c2cnn(n2)C2CC2)c(F)c1 |r|
CC(C)(Cl)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1)-c1cnn(n1)C1CC1 |r|
C[C@H](NC(=O)OC[C@@H](N1C(=N)N[C@@](CC(C)(C)C)(C1=O)c1ccc(cc1)-c1cnn(n1)C1CC1)c1ccc(Cl)c(c1)-c1ncnn1C(F)F)C(F)(F)F |r|
C[C@H](NC(=O)OC[C@@H](N1C(=N)N[C@@](CC(C)(C)C)(C1=O)c1ccc(-c2cn(nn2)C23CC(C2)C3)c(F)c1)c1ccc(Cl)c(c1)-c1ncnn1C(F)F)C(F)(F)F |r|
CC(C)(C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1)-c1cnn(n1)C1CC1)C1CC1 |r|
C[C@H](NC(=O)OC[C@@H](N1C(=N)N[C@@](CC(C)(C)C2CC2)(C1=O)c1ccc(cc1)-c1cnn(n1)C1CC1)c1ccc(Cl)c(c1)-c1ncnn1C(F)F)C(F)(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1F)-c1cnn(CC(F)F)n1 |r|
CC(C)(C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1)-c1cnn(n1)C1CC1)C(F)(F)F |r|
C[C@H](NC(=O)OC[C@@H](N1C(=N)N[C@@](CC(C)(C)C(F)(F)F)(C1=O)c1ccc(cc1)-c1cnn(n1)C1CC1)c1ccc(Cl)c(c1)-c1ncnn1C(F)F)C(F)(F)F |r|
CC(C)(C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1)-c1cnn(n1)C1CC1)C(F)F |r|
CC(C)(C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)F)c2ccc(Cl)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1)-c1cnn(n1)C1CC1)C(F)(F)F |r|
CC(C)(C[C@@]1(NC(=N)N([C@H](COC(=O)NCC(F)(F)F)c2ccc(Cl)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1)-c1cnn(n1)C1CC1)C(F)(F)F |r|
CC(C)(C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(C)CC2)c2ccc(Cl)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1)-c1cnn(n1)C1CC1)C(F)(F)F |r|
CC(C)(C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-c2ncnn2C2CC2)C1=O)c1ccc(cc1)-c1cnn(n1)C1CC1)C(F)(F)F |r|
CC(C)(C[C@@]1(NC(=N)N([C@H](CNC(=O)CC(F)(F)F)c2ccc(Cl)c(c2)-c2ncnn2C(F)F)C1=O)c1ccc(cc1)-c1cnn(n1)C1CC1)C(F)(F)F |r|
C[C@H](C(=O)NC[C@@H](N1C(=N)N[C@@](CC(C)(C)C(F)(F)F)(C1=O)c1ccc(cc1)-c1cnn(n1)C1CC1)c1ccc(Cl)c(c1)-c1ncnn1C(F)F)C(F)(F)F |r|
C[C@@H](C(=O)NC[C@@H](N1C(=N)N[C@@](CC(C)(C)C(F)(F)F)(C1=O)c1ccc(cc1)-c1cnn(n1)C1CC1)c1ccc(Cl)c(c1)-c1ncnn1C(F)F)C(F)(F)F |r|
C[C@H](NC(=O)OC[C@@H](N1C(=N)N[C@@](CC(C)(C)C)(C1=O)c1ccc(cc1)-c1cnn(n1)C(F)F)c1ccc(Cl)c(c1)-c1ncnn1C(F)F)C(F)(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(C)CC2)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)Nc2ccccc2)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)Nc2ccccn2)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC(C)(C)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC(C)(C)C)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N2CC(F)(F)C2)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC(C)(C)C(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](CO)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1ncccn1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC(C)(C)C(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1ncccn1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC(C)(C)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1ncccn1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1ccccn1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC(C)(C)C)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1ccccn1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2cc(F)c(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2cc(F)c(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1ccccn1 |r|
CC(C)(F)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1F)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1F)-c1ccccn1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1F)-c1ncccn1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC(C)(C)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1F)-c1ncccn1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1F)-c1cncs1 |r|
Cc1ncsc1-c1ccc(c(F)c1)[C@@]1(CC(C)(C)C)NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnccn1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1F)-c1cnccn1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC(F)F)CC2)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N[C@@H]2C[C@H]2C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N[C@H]2C[C@@H]2C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N[C@@H]2CC2C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N[C@H]2C[C@@H]2C(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N[C@@H]2C[C@H]2C(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
Cn1nccc1-c1ccc(cc1)[C@@]1(CC(C)(C)C)NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O |r|
Cn1ccc(n1)-c1ccc(cc1)[C@@]1(CC(C)(C)C)NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C1CC1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1F)-c1cnn(c1)C1CC1 |r|
Cn1ccc(n1)-c1ccc(c(F)c1)[C@@]1(CC(C)(C)C)NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1ccc(F)cn1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1ncc(F)cn1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1ccsn1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cncs1 |r|
CC(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1F)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1F)-c1ccc(nc1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)C#N |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1ccc(cc1)C#N |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1ccc(OC(F)F)cc1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1ccc2OC(F)(F)Oc2c1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)N1CCn2c(C1)nnc2C(F)(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC(C)(C)C(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc2ncc(Br)cc2c1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1F)-c1ncns1 |r|
CC(C)(F)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnccn1 |r|
CC(C)(F)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1ncccn1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2CC2(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N[C@@H]2CC2(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1ccnn1C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)C([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1ccn(n1)C1CC1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1F)-c1ccn(n1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)C([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1F)-c1ccn(n1)C1CC1 |r|
CC(C)(C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1ccn(n1)C(F)F)C#N |r|
Cc1cc(on1)-c1ccc(cc1)[C@@]1(CC(C)(C)C)NC(=N)C([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1F)-c1cnn(c1)S(C)(=O)=O |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N[C@@H]2C[C@@H]2F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N[C@H]2C[C@H]2F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)C2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1F)-c1nncn1C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N[C@@H]2C[C@H]2F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N[C@H]2C[C@@H]2F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NCC(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NCC(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N[C@@H]2CC2(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(-c2cnn(c2)C(F)F)c(F)c1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N[C@H]2CC2(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(-c2cnn(c2)C(F)F)c(F)c1 |r|
Cn1ccc(n1)-c1ccc(cc1F)[C@@]1(CC(C)(C)C)NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(-c2cnn(c2)S(C)(=O)=O)c(F)c1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(-c2cnn(c2)S(=O)(=O)C2CC2)c(F)c1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)S(C)(=O)=O |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2CC2(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(-c2cnn(c2)S(C)(=O)=O)c(F)c1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N[C@@H]2CC22CC2)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N[C@H]2CC22CC2)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2CC2(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C1CC1 |r|
Cn1ccc(n1)-c1ccc(cc1F)[C@@]1(CC(C)(C)C)NC(=N)N([C@H](COC(=O)NC2CC2(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O |r|
CC(C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F)CS(C)(=O)=O |r|
Cn1ccc(n1)-c1ccc(cc1)[C@@]1(CC(C)(C)C)NC(=N)N([C@H](COC(=O)N[C@H]2CC2(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O |r|
Cn1ccc(n1)-c1ccc(cc1)[C@@]1(CC(C)(C)C)NC(=N)N([C@H](COC(=O)NCC(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O |r|
C[C@@H](CC#N)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
C[C@H](CC#N)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2CC2(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(-c2cnn(c2)C2CC2)c(F)c1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NCC(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C1CC1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NCC(C)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(-c2cnn(c2)C(F)F)c(F)c1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NCC(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(-c2cnn(c2)S(C)(=O)=O)c(F)c1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NCC(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(-c2cnn(c2)S(=O)(=O)C2CC2)c(F)c1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(-c2cnn(c2)S(C)(=O)=O)c(F)c1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(-c2cnn(c2)C2CC2)c(F)c1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NCC(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(-c2cnn(c2)C2CC2)c(F)c1 |r|
CC(C)(C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)S(C)(=O)=O)C(F)(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(n1)C1CC1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1F)-c1cnn(n1)C1CC1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(-c2cnn(n2)C2CC2)c(F)c1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(c(F)c1)-n1nccn1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc2c(nccc2c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-n1nccn1 |r|
Cn1c2ccc(cc2ccc1=O)[C@@]1(CC(C)(C)C)NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O |r|
C[C@@H](NC(=O)OC[C@@H](N1C(=N)N[C@@](CC(C)(C)C)(C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F)c1ccc(Cl)c(c1)-n1ncnc1C(F)F)C(F)(F)F |r|
C[C@H](NC(=O)OC[C@@H](N1C(=N)N[C@@](CC(C)(C)C)(C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F)c1ccc(Cl)c(c1)-n1ncnc1C(F)F)C(F)(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(-c2cnn(n2)C2CC2)c(F)c1F |r|
COc1ccc(c(F)c1F)[C@@]1(CC(C)(C)C)NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc2nc(ccc2c1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-n1ccnn1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(-c2cn(nn2)C2CC2)c(F)c1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc2nc(ccc2c1)C1CC1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc2nc(ccc2c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-n1cncn1 |r|
C[C@@H](NC(=O)OC[C@@H](N1C(=N)N[C@@](CC(C)(C)C)(C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F)c1ccc(Cl)c(c1)-n1ncnc1C(F)F)C(F)F |r|
C[C@H](NC(=O)OC[C@@H](N1C(=N)N[C@@](CC(C)(C)C)(C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F)c1ccc(Cl)c(c1)-n1ncnc1C(F)F)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(c(F)c1)-n1cnnn1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1nnn(n1)C1CC1 |r|
Cn1nnc(n1)-c1ccc(cc1)[C@@]1(CC(C)(C)C)NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O |r|
Cn1nnnc1-c1ccc(cc1)[C@@]1(CC(C)(C)C)NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O |r|
C[C@H](NC(=O)OC[C@@H](N1C(=N)N[C@@](CC(C)(C)C)(C1=O)c1ccc(cc1)-c1cnn(n1)C1CC1)c1ccc(Cl)c(c1)-n1ncnc1C(F)F)C(F)(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-n1cnnc1 |r|
CC(C)(C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F)C1CC1 |r|
CC(C)(C)C[C@@]1(NC(=N)N(C(COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc2nc(ccc2c1)C#Cc1ccccc1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(c(F)c1)-c1cccc(c1)S(C)(=O)=O |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(C#Cc2cnn(c2)C(F)F)c(F)c1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(c(F)c1)-c1ccc(cc1)S(C)(=O)=O |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cn(nn1)C1CC1 |r|
C[C@H](NC(=O)OC[C@@H](N1C(=N)N[C@@](CC(C)(C)C)(C1=O)c1ccc(cc1)-c1cn(nn1)C1CC1)c1ccc(Cl)c(c1)-n1ncnc1C(F)F)C(F)(F)F |r|
C[C@H](NC(=O)OC[C@@H](N1C(=N)N[C@@](CC(C)(C)C)(C1=O)c1ccc(cc1)-c1cnn(c1)C1CC1)c1ccc(Cl)c(c1)-n1ncnc1C(F)F)C(F)(F)F |r|
C[C@H](NC(=O)OC[C@@H](N1C(=N)N[C@@](CC(C)(C)C)(C1=O)c1ccc(-c2cnn(c2)C2CC2)c(F)c1)c1ccc(Cl)c(c1)-n1ncnc1C(F)F)C(F)(F)F |r|
C[C@H](NC(=O)OC[C@@H](N1C(=N)N[C@@](CC(C)(C)C)(C1=O)c1ccc(cc1F)-c1cnn(c1)C1CC1)c1ccc(Cl)c(c1)-n1ncnc1C(F)F)C(F)(F)F |r|
CC(C)(CC#N)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C1CC1 |r|
C[C@H](NC(=O)OC[C@@H](N1C(=N)N[C@@](CC(C)(C)C)(C1=O)c1ccc(cc1)-c1cn(nn1)C1(CC1)C(F)(F)F)c1ccc(Cl)c(c1)-n1ncnc1C(F)F)C(F)(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cn(nn1)C1(CC1)C(F)(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COc2ccc(F)cc2F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
C[C@H](NC(=O)OC[C@@H](N1C(=N)N[C@@](CC(C)(C)C)(C1=O)c1ccn2nccc2c1)c1ccc(Cl)c(c1)-n1ncnc1C(F)F)C(F)(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(-c2cnn(c2)C2CC2)c(Cl)c1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1Cl)-c1cnn(c1)C1CC1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cn(nc1F)C1CC1 |r|
CC(C)n1ncc(n1)-c1ccc(cc1)[C@@]1(CC(C)(C)C)NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cn[nH]n1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)C(F)(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2CC2)c2ccc(Cl)c(c2)-n2cncn2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2cncn2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(C)CC2)c2ccc(Cl)c(c2)-n2cncn2)C1=O)c1ccc(-c2cnn(c2)C(F)F)c(F)c1F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(C)CC2)c2cccc(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
Cc1ncn(n1)-c1cc(ccc1Cl)[C@@H](COC(=O)NC1(C)CC1)N1C(=N)N[C@@](CC(C)(C)C)(C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(C)CC2)c2ccc(Cl)c(c2)-n2cnc(n2)C2CC2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2cncn2)C1=O)c1ccc(cc1)-c1cnn(c1)C1CC1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2cncn2)C1=O)c1ccc(cc1)-c1ccccn1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N2CC(F)(F)C2)c2ccc(Cl)c(c2)-n2cncn2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC(C)(C)C)c2ccc(Cl)c(c2)-n2cncn2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC(C)(C)C(F)(F)F)c2ccc(Cl)c(c2)-n2cncn2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2CC2)c2ccc(Cl)c(c2)-n2cncn2)C1=O)c1ccc(cc1)-c1cnn(c1)C1CC1 |r|
CN(C1CC1)C(=O)OC[C@@H](N1C(=N)N[C@@](CC(C)(C)C)(C1=O)c1ccc(cc1)-c1cnn(c1)C1CC1)c1ccc(Cl)c(c1)-n1cncn1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](CO)c2ccc(Cl)c(c2)-n2cncn2)C1=O)c1ccc(cc1)-c1ncccn1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](CO)c2ccc(Cl)c(c2)-n2cncn2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
Cc1ncnn1-c1cc(ccc1Cl)[C@@H](COC(=O)NC1(C)CC1)N1C(=N)N[C@@](CC(C)(C)C)(C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC23CC(C2)(C3)C(F)(F)F)c2ccc(Cl)c(c2)-n2cncn2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N(CC(F)F)C2CC2)c2ccc(Cl)c(c2)-n2cncn2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2cncn2)C1=O)c1ccc(cc1)-c1cccc(=O)[nH]1 |r|
CC(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2cncn2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC(C)(C)C(F)F)c2ccc(Cl)c(c2)-n2cncn2)C1=O)c1ccc(cc1)C#CC(C)(C)S(C)(=O)=O |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2cncn2)C1=O)c1ccc(cc1)-c1ccns1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(C)CC2)c2ccc(OC(F)(F)F)c(c2)-n2cncn2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(C)CC2)c2ccc(Cl)c(c2)-n2ncnc2C2CC2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
Cc1ncnn1-c1cc(ccc1Cl)[C@@H](COC(=O)NC1(CC1)C(F)F)N1C(=N)N[C@@](CC(C)(C)C)(C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2cncn2)C1=O)c1ccc(cc1)-c1ncon1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(cc2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(F)c(c2)N2C=NCN2C(F)F)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r,c:33|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2cccc(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1ccsn1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2cccn2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(C)CC2)c2ccc(Cl)c(c2)-n2cc(cn2)-c2ccccn2)C1=O)c1cc(F)cc(F)c1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(C)CC2)c2ccc(Cl)c(c2)-n2cccn2)C1=O)c1cc(F)cc(F)c1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(C)CC2)c2ccc(Cl)c(c2)-n2cccn2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CCC1(CC1)NC(=O)OC[C@@H](N1C(=N)N[C@@](CC(C)(C)C)(C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F)c1ccc(Cl)c(c1)-n1cccn1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(C)CC2)c2ccc(Cl)c(c2)-n2ccnn2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)N2CC(F)(F)C2)c2ccc(Cl)c(c2)-n2cccn2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(C)CC2)c2ccc(Cl)c(c2)-n2cccn2)C1=O)c1cc(F)cc(F)c1)C(F)(F)F |r|
CC(C)(C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(C)CC2)c2ccc(Cl)c(c2)-n2cccn2)C1=O)c1ccc(Cl)cc1)C(F)(F)F |r|
CC(C)(C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(C)CC2)c2ccc(Cl)c(c2)-n2cccn2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F)C(F)(F)F |r|
CC(C)(C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(C)CC2)c2ccc(Cl)c(c2)-n2cccn2)C1=O)c1ccc(cc1)-c1cnn(c1)C1CC1)C(F)(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(C)CC2)c2ccc(Cl)c(c2)-n2cc(cn2)C2CC2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(C)CC2)c2ccc(Cl)c(c2)-n2cc(cn2)C#N)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(C)CC2)c2ccc(Cl)c(c2)-n2cnnn2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
FC(F)n1cc(cn1)-c1ccc(cc1)[C@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2cccn2)C1=O)C#CC1CC1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2nccn2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(C)CC2)c2cc(c(Cl)cn2)-n2cncn2)C1=O)c1ccc(cc1)-c1cnn(c1)C(F)F |r|
CC(C)(C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(n1)C1CC1)C(F)(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](CNC(=O)C2CC2)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(n1)C1CC1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](CNC(=O)C2(C)CC2)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(n1)C1CC1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](CNC(=O)CC(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(n1)C1CC1 |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](CNC(=O)CC2CC2)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(n1)C1CC1 |r|
C[C@H](C(=O)NC[C@@H](N1C(=N)N[C@@](CC(C)(C)C)(C1=O)c1ccc(cc1)-c1cnn(n1)C1CC1)c1ccc(Cl)c(c1)-n1ncnc1C(F)F)C(F)(F)F |r|
C[C@@H](C(=O)NC[C@@H](N1C(=N)N[C@@](CC(C)(C)C)(C1=O)c1ccc(cc1)-c1cnn(n1)C1CC1)c1ccc(Cl)c(c1)-n1ncnc1C(F)F)C(F)(F)F |r|
CC(C)(C)C[C@@]1(NC(=N)N([C@H](CNS(=O)(=O)C2CC2)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(n1)C1CC1 |r|
CC(C)C(=O)NC[C@@H](N1C(=N)N[C@@](CC(C)(C)C(F)(F)F)(C1=O)c1ccc(cc1)-c1cnn(n1)C1CC1)c1ccc(Cl)c(c1)-n1ncnc1C(F)F |r|
C[C@H](C(=O)NC[C@@H](N1C(=N)N[C@@](CC(C)(C)C(F)(F)F)(C1=O)c1ccc(cc1)-c1cnn(n1)C1CC1)c1ccc(Cl)c(c1)-n1ncnc1C(F)F)C(F)(F)F |r|
C[C@@H](C(=O)NC[C@@H](N1C(=N)N[C@@](CC(C)(C)C(F)(F)F)(C1=O)c1ccc(cc1)-c1cnn(n1)C1CC1)c1ccc(Cl)c(c1)-n1ncnc1C(F)F)C(F)(F)F |r|
CC(C)(C[C@@]1(NC(=N)N([C@H](CNC(=O)CC(F)(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(n1)C1CC1)C(F)(F)F |r|
CC(C)(C[C@@]1(NC(=N)N([C@H](COC(=O)NC2(CC2)C(F)F)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(n1)C1CC1)C(F)(F)F |r|
CC(C)(C[C@@]1(NC(=N)N([C@H](CNC(=O)OC2CC2)c2ccc(Cl)c(c2)-n2ncnc2C(F)F)C1=O)c1ccc(cc1)-c1cnn(n1)C1CC1)C(F)(F)F |r|
COC(=O)NC[C@@H](N1C(=N)N[C@@](CC(C)(C)C(F)(F)F)(C1=O)c1ccc(cc1)-c1cnn(n1)C1CC1)c1ccc(Cl)c(c1)-n1ncnc1C(F)F |r|
CCOP(=O)(CCOCc1ccc2c(NC(c3ccccc3)(c3ccccc3)c3ccccc3)ncnn12)OCC
CCOP(=O)(CO[C@H](C)Cc1ccc2c(NC(c3ccccc3)(c3ccccc3)c3ccc(OC)cc3)ncnn12)OCC |r|
CCOP(=O)(COCCc1ccc2c(NC(c3ccccc3)(c3ccccc3)c3ccc(OC)cc3)ncnn12)OCC
CSc1nc(N)nn2c(C[C@@H](C)OCc3ccccc3)nnc12 |r|
CCOP(=O)(CO[C@H](C)Cc1cnc2c(N)ncnn12)OCC |r|
CSc1nc(N)nn2c(C[C@@H](C)OCc3ccccc3)ncc12 |r|
CN(c1ccccc1)c1ncnc2c(I)cnn12
CCOP(=O)(COC(C)Cc1ccc2c(NC(c3ccccc3)(c3ccccc3)c3ccc(OC)cc3)nc(F)nn12)OCC |w:7.7|
COc1ccc(cc1)C(Nc1nc(NC(c2ccccc2)(c2ccccc2)c2ccc(OC)cc2)c2ccc(I)n2n1)(c1ccccc1)c1ccccc1
CCOP(=O)(COC(CF)Cc1cnn2c(N)ncnc12)OCC |w:7.7|
CC(C)OC(=O)OCOP(=O)(CO[C@H](C)Cc1ccc2c(N)ncnn12)OCOC(=O)OC(C)C |r|
CC(C)OC(=O)OCOP(=O)(CO[C@H](C)Cc1cnc2c(N)ncnn12)OCOC(=O)OC(C)C |r|
CC(C)OC(=O)OCOP(=O)(CO[C@H](C)Cc1cnn2c(N)ncnc12)OCOC(=O)OC(C)C |r|
CC(C)OC(=O)OCOP(=O)(CO[C@@H](C)Cc1cnn2c(N)ncnc12)OCOC(=O)OC(C)C |r|
C[C@H](Cc1cnn2c(N)ncnc12)OCP(O)(O)=O |r|
C[C@@H](Cc1cnn2c(N)ncnc12)OCP(O)(O)=O |r|
Oc1c2C(=O)N3CN(Cc4ccc(F)cc4C3)n2cc(C(=O)NCc2c(F)cc(F)cc2F)c1=O
Oc1c2C(=O)N3CN(Cc4cc(F)ccc4C3)n2cc(C(=O)NCc2c(F)cc(F)cc2F)c1=O
C[C@H]1C=CCN2CN1C(=O)c1c(O)c(=O)c(cn21)C(=O)NCc1c(F)cc(F)cc1F |r,c:2|
Oc1c2C(=O)N3CCCCN(C3Cc3ccccc3)n2cc(C(=O)NCc2c(F)cc(F)cc2F)c1=O |TLB:12:11:19.2.3:7.6.8.9|
C[C@@H]1C\C=C/[C@H](C)N2CN1n1cc(C(=O)NCc3c(F)cc(F)cc3F)c(=O)c(O)c1C2=O |r,c:3|
C[C@H]1CCC[C@@H](C)N2CN1C(=O)c1c(O)c(=O)c(cn21)C(=O)NCc1c(F)cc(F)cc1F |r|
C[C@@H]1C\C=C/CN2CN1n1cc(C(=O)NCc3ccc(F)cc3F)c(=O)c(O)c1C2=O |r,c:3|
C[C@@H]1CCCCN2CN1n1cc(C(=O)NCc3ccc(F)cc3F)c(=O)c(O)c1C2=O |r|
C[C@@H]1C\C=C/CN2CN1n1cc(C(=O)NCc3c(F)cc(F)cc3F)c(=O)c(OCc3ccccc3)c1C2=O |r,c:3|
C[C@@H]1CCCCN2CN1n1cc(C(=O)NCc3c(F)cc(F)cc3F)c(=O)c(O)c1C2=O |r|
C[C@@H]1C\C=C/[C@H](C)N2CN1n1cc(C(=O)NCc3c(F)cc(F)cc3F)c(=O)c(OCc3ccccc3)c1C2=O |r,c:3|
C[C@H]1C\C=C/[C@H](C)N2CN1n1cc(C(=O)NCc3c(F)cc(F)cc3F)c(=O)c(O)c1C2=O |r,c:3|
C[C@@H]1CCC[C@@H](C)N2CN1C(=O)c1c(O)c(=O)c(cn21)C(=O)NCc1c(F)cc(F)cc1F |r|
C[C@H]1CCC[C@H](C)N2CN1C(=O)c1c(O)c(=O)c(cn21)C(=O)NCc1c(F)cc(F)cc1F |r|
C[C@H]1C=C[C@@H](C)N2CN1C(=O)c1c(O)c(=O)c(cn21)C(=O)NCc1c(F)cc(F)cc1F |r,c:2|
C[C@H]1C=C[C@H](C)N2CN1C(=O)c1c(O)c(=O)c(cn21)C(=O)NCc1c(F)cc(F)cc1F |r,c:2|
C[C@H]1CC[C@H](C)N2CN1C(=O)c1c(O)c(=O)c(cn21)C(=O)NCc1c(F)cc(F)cc1F |r|
C[C@H]1C=C[C@@H](C)N2CN1C(=O)c1c(O)c(=O)c(cn21)C(=O)NCc1ccc(F)cc1F |r,c:2|
C[C@H]1C=C[C@H](C)N2CN1C(=O)c1c(O)c(=O)c(cn21)C(=O)NCc1ccc(F)cc1F |r,c:2|
C[C@H]1CC[C@H](C)N2CN1C(=O)c1c(O)c(=O)c(cn21)C(=O)NCc1ccc(F)cc1F |r|
CO[C@H]1[C@H](C)N2CN([C@H](C)[C@H]1OC)n1cc(C(=O)NCc3c(F)cc(F)cc3F)c(=O)c(O)c1C2=O
CO[C@@H]1C[C@@H](C)N2CN([C@H]1C)C(=O)c1c(O)c(=O)c(cn21)C(=O)NCc1c(F)cc(F)cc1F |r|
C[C@@H]1C[C@H](F)[C@H](C)N2CN1n1cc(C(=O)NCc3c(F)cc(F)cc3F)c(=O)c(O)c1C2=O |r|
C[C@@H]1CC(F)(F)[C@H](C)N2CN1n1cc(C(=O)NCc3c(F)cc(F)cc3F)c(=O)c(O)c1C2=O |r|
C[C@H]1C=C(F)[C@@H](C)N2CN1C(=O)c1c(O)c(=O)c(cn21)C(=O)NCc1c(F)cc(F)cc1F |r,t:2|
C[C@H]1CC[C@@H](C)N2CN1C(=O)c1c(O)c(=O)c(cn21)C(=O)NCc1ccc(F)cc1F |r|
C[C@@H]1C[C@H](O)[C@H](O)CN2CN1n1cc(C(=O)NCc3ccc(F)cc3F)c(=O)c(O)c1C2=O |r|
CO[C@H]1C[C@@H](C)N2CN(C[C@H]1OC)C(=O)c1c(O)c(=O)c(cn21)C(=O)NCc1ccc(F)cc1F |r|
C[C@H]1CCCCN2CN1n1cc(C(=O)NCc3ccc(F)cc3F)c(=O)c(O)c1C2=O |r|
C[C@H]1C\C=C/CN2CN1n1cc(C(=O)NCc3ccc(F)cc3F)c(=O)c(O)c1C2=O |r,c:3|
C[C@H]1C=C[C@@H](CF)N2CN1C(=O)c1c(O)c(=O)c(cn21)C(=O)NCc1ccc(F)cc1F |r,c:2|
C[C@H]1CC[C@@H](CF)N2CN1C(=O)c1c(O)c(=O)c(cn21)C(=O)NCc1ccc(F)cc1F |r|
CO[C@@H]1C=C[C@H](C)N2CN1n1cc(C(=O)NCc3c(F)cc(F)cc3F)c(=O)c(O)c1C2=O |r,c:3|
C[C@H]1C=CC(C)(C)N2CN1C(=O)c1c(O)c(=O)c(cn21)C(=O)NCc1c(F)cc(F)cc1F |r,c:2|
C[C@@H]1C=C[C@H](CF)[N@@]2CN1n1cc(C(=O)NCc3ccc(F)cc3F)c(=O)c(O)c1C2=O |r,c:2,THB:27:29:8:1.2.3.4,11:10:8:1.2.3.4,31:30:8:1.2.3.4|
C[C@@H]1C=C[C@H](CF)[N@]2CN1n1cc(C(=O)NCc3ccc(F)cc3F)c(=O)c(O)c1C2=O |r,c:2,THB:27:29:8:1.2.3.4,11:10:8:1.2.3.4,31:30:8:1.2.3.4|
C[C@@H]1C=C[C@H](CF)N2CN1n1cc(C(=O)NCc3c(F)cc(F)cc3F)c(=O)c(O)c1C2=O |r,c:2|
C[C@@H]1C=C[C@H](CF)N2CN1n1cc(C(=O)NCc3c(F)cc(F)cc3F)c(=O)c(OCc3ccccc3)c1C2=O |r,c:2|
C[C@@H]1C[C@H](F)[C@H](C)N2CN1n1cc(C(=O)NCc3ccc(F)cc3F)c(=O)c(O)c1C2=O |r|
C[C@@H]1C[C@@H](F)[C@H](C)N2CN1n1cc(C(=O)NCc3ccc(F)cc3F)c(=O)c(O)c1C2=O |r|
C[C@@H]1CC(F)(F)[C@H](C)N2CN1n1cc(C(=O)NCc3ccc(F)cc3F)c(=O)c(O)c1C2=O |r|
C[C@@H]1C=C(F)[C@H](C)N2CN1n1cc(C(=O)NCc3c(F)cc(F)cc3F)c(=O)c(O)c1C2=O |r,t:2|
C[C@@H]1C[C@@H](C(F)F)[C@H](C)N2CN1n1cc(C(=O)NCc3c(F)cc(F)cc3F)c(=O)c(O)c1C2=O |r|
C[C@@H]1C[C@@H](CF)[C@H](C)N2CN1n1cc(C(=O)NCc3c(F)cc(F)cc3F)c(=O)c(O)c1C2=O |r|
C[C@H]1C[C@H](F)[C@H](C)N2CN1n1cc(C(=O)NCc3ccc(F)cc3F)c(=O)c(O)c1C2=O |r|
C[C@H]1CC(F)(F)[C@H](C)N2CN1n1cc(C(=O)NCc3ccc(F)cc3F)c(=O)c(O)c1C2=O |r|
C[C@@H]1N2CN([C@H](C)c3nc[nH]c13)n1cc(C(=O)NCc3ccc(F)cc3F)c(=O)c(O)c1C2=O |r|
CO[C@@H]1[C@H](C)N2CN([C@H](C)[C@@H]1OC)n1cc(C(=O)NCc3c(F)cc(F)cc3F)c(=O)c(O)c1C2=O |r|
C[C@H]1C=C(C)[C@@H](C)N2CN1C(=O)c1c(O)c(=O)c(cn21)C(=O)NCc1ccc(F)cc1F |r,t:2|
C[C@@H]1C=C[C@@H](C)N2CN1C(=O)c1c(O)c(=O)c(cn21)C(=O)NCc1c(F)cc(F)cc1F |r,c:2|
C[C@@H]1CC[C@@H](C)N2CN1C(=O)c1c(O)c(=O)c(cn21)C(=O)NCc1c(F)cc(F)cc1F |r|
C[C@@H]1CC[C@@H](C)N2CN1C(=O)c1c(O)c(=O)c(cn21)C(=O)NCc1ccc(F)cc1F |r|
C[C@@H]1C=C[C@@H](C)N2CN1C(=O)c1c(O)c(=O)c(cn21)C(=O)NCc1ccc(F)cc1F |r,c:2|
C[C@@H]1C=CCN2CN1n1cc(C(=O)NCc3c(F)cc(F)cc3F)c(=O)c(O)c1C2=O |r,c:2|
CC[C@@H]1C=C[C@H](C)N2CN1n1cc(C(=O)NCc3c(F)cc(F)cc3F)c(=O)c(O)c1C2=O |r,c:3|
CC[C@@H]1CC[C@H](C)N2CN1n1cc(C(=O)NCc3c(F)cc(F)cc3F)c(=O)c(O)c1C2=O |r|
CC(C)[C@@H]1C=C[C@H](C)N2CN1n1cc(C(=O)NCc3c(F)cc(F)cc3F)c(=O)c(O)c1C2=O |r,c:4|
CC(C)[C@@H]1CC[C@H](C)N2CN1n1cc(C(=O)NCc3c(F)cc(F)cc3F)c(=O)c(O)c1C2=O
C[C@H]1C=C[C@@H](CF)N2CN1C(=O)c1c(O)c(=O)c(cn21)C(=O)NCc1c(F)cc(F)cc1F |r,c:2|
C[C@H]1CC[C@@H](CF)N2CN1C(=O)c1c(O)c(=O)c(cn21)C(=O)NCc1c(F)cc(F)cc1F |r|
C[C@H]1CC[C@@H](C(F)F)N2CN1C(=O)c1c(O)c(=O)c(cn21)C(=O)NCc1c(F)cc(F)cc1F |r|
COC[C@@H]1C=C[C@H](C)N2CN1n1cc(C(=O)NCc3c(F)cc(F)cc3F)c(=O)c(OCc3ccccc3)c1C2=O |r,c:4|
C[C@H]1C=C[C@H](CF)N2CN1C(=O)c1c(O)c(=O)c(cn21)C(=O)NCc1c(F)cc(F)cc1F |r,c:2|
COC[C@@H]1C=C[C@H](C)N2CN1n1cc(C(=O)NCc3ccc(F)cc3F)c(=O)c(O)c1C2=O |r,c:4|
COC[C@@H]1CC[C@H](C)N2CN1n1cc(C(=O)NCc3ccc(F)cc3F)c(=O)c(O)c1C2=O |r|
C[C@H]1C=C[C@]2(CCOC2)N2CN1C(=O)c1c(O)c(=O)c(cn21)C(=O)NCc1c(F)cc(F)cc1F |r,c:2|
C[C@H]1CCC2(CCOC2)N2CN1C(=O)c1c(O)c(=O)c(cn21)C(=O)NCc1c(F)cc(F)cc1F |r|
C[C@H]1[C@@H]2C[C@@H]2[C@H](C)N2CN1C(=O)c1c(O)c(=O)c(cn21)C(=O)NCc1c(F)cc(F)cc1F |r|
C[C@H]1[C@@H]2C[C@@H]2[C@@H](C)N2CN1C(=O)c1c(O)c(=O)c(cn21)C(=O)NCc1c(F)cc(F)cc1F |r|
C[C@@H]1C=CC(C)(C)N2CN1n1cc(C(=O)NCc3ccc(F)cc3F)c(=O)c(O)c1C2=O |r,c:2|
C[C@H]1C=CC(C)(C)N2CN1n1cc(C(=O)NCc3ccc(F)cc3F)c(=O)c(O)c1C2=O |r,c:2|
C[C@H]1C=CC(C)(C)N2CN1n1cc(C(=O)NCc3ccc(F)cc3F)c(=O)c(OCc3ccccc3)c1C2=O |r,c:2|
C[C@@H]1CCC(C)(C)N2CN1n1cc(C(=O)NCc3ccc(F)cc3F)c(=O)c(O)c1C2=O |r|
C[C@H]1CCC(C)(C)N2CN1n1cc(C(=O)NCc3ccc(F)cc3F)c(=O)c(O)c1C2=O |r|
C[C@H]1CC[C@@H](CF)N2CN1n1cc(C(=O)NCc3ccc(F)cc3F)c(=O)c(O)c1C2=O |r|
C[C@H]1C=C[C@@H](CF)N2CN1n1cc(C(=O)NCc3ccc(F)cc3F)c(=O)c(O)c1C2=O |r,c:2|
C[C@@H]1CC[C@H](CF)N2CN1n1cc(C(=O)NCc3ccc(F)cc3F)c(=O)c(O)c1C2=O |r|
C[C@@H]1C[C@H](F)[C@H](CF)N2CN1n1cc(C(=O)NCc3c(F)cc(F)cc3F)c(=O)c(O)c1C2=O |r|
CC1N2[C@@H](C)C=C[C@@H](C)N1n1cc(C(=O)NCc3c(F)cc(F)cc3F)c(=O)c(O)c1C2=O |r,c:5,TLB:0:1:10.30.31:5.3.7.6|
CCC1N2[C@@H](C)C=C[C@@H](C)N1n1cc(C(=O)NCc3c(F)cc(F)cc3F)c(=O)c(O)c1C2=O |r,c:6,TLB:33:32:2:7.8.6.4,5:4:32.31.11:2,THB:12:11:2:7.8.6.4,9:8:32.31.11:2,29:31:2:7.8.6.4|
C[C@H]1C=CC2(CCC2)N2CN1C(=O)c1c(O)c(=O)c(cn21)C(=O)NCc1c(F)cc(F)cc1F |r,c:2|
CC[C@H]1C=C[C@H](C)N2CN1n1cc(C(=O)NCc3c(F)cc(F)cc3F)c(=O)c(O)c1C2=O |r,c:3|
Oc1c2C(=O)N3CN(CCCC3)n2cc(C(=O)NCc2c(F)cc(F)cc2F)c1=O
COc1cnc(OC)c2[nH]cc(C(=O)C(=O)N3CCN(CC3)C(=O)c3ccccc3)c12
COc1cnc(-n2cnc(C)n2)c2[nH]cc(C(=O)C(=O)N3CCN(CC3)C(=O)c3ccccc3)c12
CC(C)C1=C(O)C(=O)\C(=C/N[C@H]2[C@H](O)O[C@H](CO)[C@@H](O)[C@@H]2O)c2c(O)c(c(C)cc12)-c1c(C)cc2C(C(C)C)=C(O)C(=O)\C(=C/N[C@H]3[C@H](O)O[C@H](CO)[C@@H](O)[C@@H]3O)c2c1O |r,wU:47.50,55.59,50.53,12.12,20.21,15.15,wD:11.10,46.48,53.56,18.18,c:3,t:41,(10.32,-5.58,;9,-6.36,;7.66,-5.6,;9.01,-7.9,;10.34,-8.65,;11.67,-7.87,;10.36,-10.19,;11.7,-10.95,;9.03,-10.97,;9.04,-12.51,;10.38,-13.27,;10.39,-14.81,;9.05,-15.58,;7.72,-14.81,;9.06,-17.11,;10.39,-17.88,;10.4,-19.42,;11.73,-20.19,;11.73,-17.1,;13.06,-17.87,;11.72,-15.56,;13.05,-14.78,;7.7,-10.21,;6.38,-10.99,;6.39,-12.53,;5.04,-10.23,;5.03,-8.69,;3.69,-7.93,;6.35,-7.91,;7.7,-8.67,;3.71,-11,;3.72,-12.55,;5.06,-13.32,;2.39,-13.32,;1.05,-12.56,;-.3,-13.34,;-.28,-14.88,;-1.61,-15.65,;1.06,-15.64,;-1.62,-12.57,;-2.96,-13.33,;-1.62,-11.02,;-2.95,-10.25,;-.29,-10.25,;-.3,-8.71,;-1.63,-7.94,;-1.64,-6.4,;-.3,-5.63,;1.04,-6.39,;-.3,-4.09,;-1.63,-3.32,;-1.63,-1.78,;-.3,-1.01,;-2.97,-4.09,;-4.31,-3.32,;-2.96,-5.64,;-4.31,-6.41,;1.05,-11.01,;2.38,-10.24,;2.37,-8.7,)|
CC(C)C1=C(O)C(=O)C(=C/NC(C)C(=O)NC(C)C([O-])=O)c2c(O)c(c(C)cc12)-c1c(C)cc2C(C(C)C)=C(O)C(=O)C(=C/NC(C)C(=O)NC(C)C([O-])=O)c2c1O |c:3,t:39|
CC(C)C1=C(O)C(=O)C(=C/NC(C)S([O-])(=O)=O)c2c(O)c(c(C)cc12)-c1c(C)cc2C(C(C)C)=C(O)C(=O)C(=C/NC(C)S([O-])(=O)=O)c2c1O |c:3,t:35|
CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)CCNC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](NC(C)=O)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)CC)C(N)=O |r|
Cc1ccc(cc1)-c1ccc2CCCC(=Cc2c1)C(=O)Nc1ccc(C[N+](C)(C)C2CCOCC2)cc1 |c:15|
C[C@@H]1CN(CCN1C(=O)C(=O)c2c[nH]c3c2c(ccn3)OC)C(=O)c4ccccc4
C[C@@H]1CN(CCN1C(=O)C(=O)c1c[nH]c2nccc(OCCOCCOCCOCCOCCOCCn3cc(COCCOCCOCCOCCNc4ccc(cc4[N+]([O-])=O)[N+]([O-])=O)nn3)c12)C(=O)c1ccccc1 |r|
COc1ccc(-c2ccco2)c2[nH]cc(C(=O)C(=O)N3CCN(CC3)C(=O)c3ccccc3)c12
COc1ccc(-c2ccc(CNC(=O)COCCOCCOCCOCCn3cc(COCCOCCOCCOCCNc4ccc(cc4[N+]([O-])=O)[N+]([O-])=O)nn3)o2)c2[nH]cc(C(=O)C(=O)N3CCN(CC3)C(=O)c3ccccc3)c12
OC(=O)C(Cc1c([nH]c2ccccc12)-c1cc(cc(c1)C(O)=O)C(O)=O)NC(=O)CCC(CCC(=O)NC(Cc1c([nH]c2ccccc12)-c1cc(cc(c1)C(O)=O)C(O)=O)C(O)=O)(CCC(=O)NC(Cc1c([nH]c2ccccc12)-c1cc(cc(c1)C(O)=O)C(O)=O)C(O)=O)[N+]([O-])=O
OC(=O)C(Cc1c([nH]c2ccccc12)-c1cc(cc(c1)C(O)=O)C(O)=O)NC(=O)CCOCC(COCCC(=O)NC(Cc1c([nH]c2ccccc12)-c1cc(cc(c1)C(O)=O)C(O)=O)C(O)=O)(COCCC(=O)NC(Cc1c([nH]c2ccccc12)-c1cc(cc(c1)C(O)=O)C(O)=O)C(O)=O)COCCC(=O)NC(Cc1c([nH]c2ccccc12)-c1cc(cc(c1)C(O)=O)C(O)=O)C(O)=O
COc1cccc(CN2CCc3ccc(cc23)-c2ccc3ccn(Cc4cccc(c4)C(O)=O)c3c2)c1
COC(=O)c1cccc(Cn2ccc3ccc(cc23)-c2ccc3cnn(Cc4cccc(c4)C(O)=O)c3c2)c1
COC(=O)c1cc(Cn2ccc3ccc(cc23)-c2ccc3ccn(Cc4cccc(c4)C(O)=O)c3c2)cc(c1)C(=O)OC
OC(=O)c1cc(F)cc(Cn2ccc3ccc(cc23)-c2ccc3ccn(Cc4cccc(c4)C(=O)OC(F)(F)F)c3c2)c1
CC(C)(C)OC(=O)Nc1cccc(Cn2ccc3ccc(cc23)-c2ccc3ccn(Cc4cccc(c4)C(O)=O)c3c2)c1
Cn1ncc2ccc(cc12)-c1ccc2ccn(Cc3cc(F)cc(c3)C(O)=O)c2c1
CC(C)(C)OC(=O)N1CCc2ccc(cc12)-c1ccc2ccn(Cc3cccc(c3)C(O)=O)c2c1
Cn1ccc2cc(F)c(cc12)-c1ccc2ccn(Cc3cc(F)cc(c3)C(O)=O)c2c1
COC(=O)c1cc(F)cc(Cn2ccc3ccc(cc23)-c2ccc3ccn(Cc4cccc(c4)C(O)=O)c3c2)c1
OC(=O)c1cccc(Cn2ccc3ccc(cc23)-c2ccc3ccn(Cc4cccc(OC(F)(F)F)c4)c3c2)c1
COc1cccc(Cn2ccc3cc(F)c(cc23)-c2ccc3ccn(Cc4cccc(c4)C(O)=O)c3c2)c1
COc1cc(Cn2ccc3ccc(cc23)-c2ccc3ccn(Cc4cccc(c4)C(O)=O)c3c2)cc(c1)C(O)=O
CC(=O)Nc1cccc(Cn2ccc3ccc(cc23)-c2ccc3ccn(Cc4cccc(c4)C(O)=O)c3c2)c1
CC(C)(C)OC(=O)N1CCC(Cn2ccc3ccc(cc23)-c2ccc3ccn(Cc4cccc(c4)C(O)=O)c3c2)CC1
Cc1ccc(cc1)S(=O)(=O)n1ccc2ccc(cc12)-c1ccc2ccn(Cc3cccc(c3)C(O)=O)c2c1
Cn1cc2ccc(cc2n1)-c1ccc2ccn(Cc3cc(F)cc(c3)C(O)=O)c2c1
Cn1ccc2ccc(cc12)-c1ccc2CCN(Cc3cccc(c3)C(O)=O)c2c1
COc1cccc(Cn2ccc3ccc(cc23)-c2ccc3cn(Cc4cccc(c4)C(O)=O)nc3c2)c1
COc1cccc(CNc2cccc(c2)-c2ccc3ccn(Cc4cccc(c4)C(O)=O)c3c2)c1
COC(=O)c1cccc(Cn2ncc3ccc(cc23)-c2ccc3ccn(Cc4cccc(c4)C(O)=O)c3c2)c1
Cn1ccc2ccc(cc12)-c1ccc2ccn(Cc3cc(F)cc(c3)C(O)=O)c2c1
OC(=O)c1cccc(Cn2ccc3ccc(cc23)-c2ccc3ccn(Cc4cccc(c4)[N+]([O-])=O)c3c2)c1
Nc1ccc(Cn2ccc3ccc(cc23)-c2ccc3ccn(Cc4cccc(c4)C(O)=O)c3c2)cc1
Cn1ncc2ccc(cc12)-c1ccc2cnn(Cc3ccc(F)c(c3)C(O)=O)c2c1
COc1cccc(CN(C)c2cccc(c2)-c2ccc3ccn(Cc4cccc(c4)C(O)=O)c3c2)c1
COc1cccc(CN(C(=O)OC(C)(C)C)c2cccc(c2)-c2ccc3ccn(Cc4cccc(c4)C(O)=O)c3c2)c1
COC(=O)c1cccc(Cn2ccc3cc(F)c(cc23)-c2ccc3ccn(Cc4cccc(c4)C(O)=O)c3c2)c1
CC(C)(C)OC(=O)c1cccc(Cn2ccc3ccc(cc23)-c2ccc3ccn(Cc4cccc(c4)C(O)=O)c3c2)c1
CC(C)(C)OC(=O)n1ccc2ccc(cc12)-c1ccc2ccn(Cc3cccc(c3)C(O)=O)c2c1
CN(C(=O)OC(C)(C)C)c1cccc(c1)-c1ccc2ccn(Cc3cccc(c3)C(O)=O)c2c1
Cn1ccc2ccc(cc12)-c1ccc2cnn(Cc3cc(F)cc(c3)C(O)=O)c2c1
COc1cccc(Cn2ccc3ccc(cc23)-c2ccc3c(C)cn(Cc4cccc(c4)C(O)=O)c3c2)c1
Cc1cn(C(=O)OC(C)(C)C)c2cc(ccc12)-c1ccc2ccn(Cc3cccc(c3)C(O)=O)c2c1
COC(=O)c1ccc(Cn2ccc3ccc(cc23)-c2ccc3ccn(Cc4cccc(c4)C(O)=O)c3c2)c(OC)c1
CC[C@H](C)[C@H](NC(C)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)CC)C(=O)NC1CCSCc2cccc(CSCCC(NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](C)NC1=O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC(C)C)C(N)=O)c2 |r|
CC[C@H](C)[C@H](NC(C)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)CC)C(=O)NC1CCSCc2cccc(CSCCC(NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](C)NC1=O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC(C)C)C(N)=O)c2 |r|
CC[C@H](C)[C@H](NC(C)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@H]1CSCc2cccc(CSC[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](C)NC(=O)[C@H](C)NC1=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC(C)C)C(N)=O)c2 |r|
CC[C@H](C)[C@H](NC(C)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@H]1CSCc2cccc(CSC[C@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CCCCN)NC1=O)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC(C)C)C(N)=O)c2 |r|
CC[C@H](C)[C@H](NC(C)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@H]1CSCc2cccc(CSC[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(O)=O)NC1=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC(C)C)C(N)=O)c2 |r|
CC[C@H](C)[C@H](NC(C)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@H]1CSCc2cccc(CSC[C@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC1=O)[C@@H](C)CC)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC(C)C)C(N)=O)c2 |r|
CC[C@H](C)[C@H](NC(C)=O)C(=O)N[C@H]1CSCc2cccc(CSC[C@H](NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](C)NC1=O)[C@@H](C)CC)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC(C)C)C(N)=O)c2 |r|
CC[C@H](C)[C@H](NC(C)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC(C)C)C(N)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CO)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)C(CO)NC(=O)[C@@H](NC(=O)[C@H](Cc1ccc(O)cc1)NC(C)=O)[C@@H](C)O)[C@@H](C)CC)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](Cc1ccccc1)C(N)=O
CC[C@H](C)[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CCSC)NC(=O)[C@@H](N)CCC(O)=O)[C@@H](C)O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCCN)C(O)=O |r|
CC[C@H](C)[C@H](NC(C)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@H]1CSCc2cccc(CSC[C@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(N)=O)NC1=O)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC(C)C)C(N)=O)c2 |r|
CC[C@H](C)[C@H](NC(C)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@H]1CSCc2cccc(CSC[C@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](C)NC1=O)C(=O)N[C@@H](CC(C)C)C(N)=O)c2 |r|
CC[C@H](C)[C@H](NC(C)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@H]1CSCc2cccc(CSC[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](C)NC1=O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC(C)C)C(N)=O)c2 |r|
CC[C@H](C)[C@H](NC(C)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)CC)C(=O)NC1CCSCc2cccc(CSCCC(NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](C)NC1=O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC(C)C)C(N)=O)c2 |r|
CS(=O)(=O)N1CCC[C@@H](C1)C(=O)Nc1ccc(Cl)cc1 |r|
COC(=O)N1CCC[C@@H](C1)C(=O)Nc2ccc(c(c2)F)Cl
CCOC(=O)N1CCC[C@@H](C1)C(=O)Nc2ccc(c(c2)F)Cl
CS(=O)(=O)N1CCC[C@@H](C1)C(=O)Nc2ccc(c(c2)F)Cl
CC1(C)CC(CC(C)(C)N1)NC(=O)C(=O)Nc1ccc(cn1)C(F)(F)F
CC1(C)CC(CC(C)(C)N1)NC(=O)C(=O)Nc1ccc(F)nc1
Brc1ccc(NC(=O)C(=O)NC2CCNC3(CCCCC3)C2)cn1
Fc1ccc(NC(=O)C(=O)NC2CCNC3(CCCCC3)C2)cn1
CC1(CC(CC(N1)(C)C)NC(=O)C(=O)Nc2ccc(cc2)Cl)C
CC1(C)CC(CC(C)(C)N1)NC(=O)C(=O)Nc1cnc(F)c(F)c1
CC1(C)CC(CC(C)(C)N1)NC(=O)C(=O)Nc1ccc(Cl)nc1
CC1(C)CC(CC(C)(C)N1)NC(=O)C(=O)Nc1cccnc1Cl
CC1(C)CC(CC(C)(C)N1)NC(=O)C(=O)Nc1ccnc(Br)c1
CC1(C)CC(CC(C)(C)N1)NC(=O)C(=O)Nc1ccncc1
Cc1cccc(NC(=O)C(=O)NC2CC(C)(C)NC(C)(C)C2)n1
CC1(C)CC(CC(C)(C)N1)NC(=O)C(=O)Nc1ccc(I)cn1
CC1(C)CC(CC(C)(C)N1)NC(=O)C(=O)Nc1ccc(F)cn1
CC1(C)CC(CC(C)(C)N1)NC(=O)C(=O)Nc1ccnc(Cl)c1
CC1(C)CC(CC(C)(C)N1)NC(=O)C(=O)Nc1ccc(Cl)cn1
CC1(C)CC(CC(C)(C)N1)NC(=O)C(=O)Nc1cccnc1
c1cc2c(cc1Cl)[C@@](OC(=O)N2)(C#CC3CC3)C(F)(F)F
COc1ccc(NC(=O)C(=O)NC2CC(C)(C)NC(C)(C)C2)cn1
CC1(C)CC(CC(C)(C)N1)NC(=O)C(=O)Nc1ccnc(F)c1
CC1(C)CC(CC(C)(C)N1)NC(=O)C(=O)Nc1ccc(Br)cn1
CC1(C)CC(CC(C)(C)N1)NC(=O)C(=O)Nc1ccc(Br)nc1
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CC1(C)CC(CC(C)(C)N1)NC(=O)c1ccc([nH]1)-c1ccc(Cl)c(F)c1
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[#7]\[#6](-[#7])=[#7]\[#7]=[#6]-[#6]-1=[#6](Cl)-c2ccccc2-[#6]-[#6]-[#6]-1 |w:5.5,c:6|
COC(=O)C(=O)N1CCC[C@@H]1C(=O)N[C@H](Cc1ccccc1)C(=O)OCc1ccccc1
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OCCN1CCCC(CNC(=O)C(=O)Nc2ccc(Cl)c(F)c2)C1
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Fc1cc(NC(=O)C(=O)NC2CCNC3(CCC3)C2)ccc1Cl
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Fc1cc(NC(=O)C(=O)NC2CCN(C2)C2CCCCC2)ccc1Cl
Fc1cc(NC(=O)C(=O)NCC2CCN(C2)C2CC2)ccc1Cl
Fc1cc(NC(=O)C(=O)N[C@@H]2CCN(Cc3ccccc3)C2)ccc1Cl |r|
Fc1cc(NC(=O)C(=O)N[C@H]2CCN(Cc3ccccc3)C2)ccc1Cl |r|
CCN1CCCC1CNC(=O)C(=O)Nc1ccc(Cl)c(F)c1
CCN1CCCC1CNC(=O)C(=O)Nc1ccc(Cl)cc1
CC(NC(=O)C(=O)Nc1ccc(Cl)c(F)c1)c1ccc2OCC(=O)Nc2c1
Fc1cc(NC(=O)C(=O)NCC2NCCc3ccccc23)ccc1Cl
c1cc(c(cc1NC(=O)C(=O)NC[C@@]23CCC[C@@H]2CNC3)F)Cl
Cn1ccnc1C(O)(CCNC(=O)C(=O)Nc1ccc(Cl)c(F)c1)C(F)(F)F
Fc1cc(NC(=O)C(=O)Nc2cccc3[nH]ncc23)ccc1Cl
Fc1cc(NC(=O)C(=O)NC2CCc3[nH]ncc3C2)ccc1Cl
Fc1cc(NC(=O)C(=O)Nc2cnn3CCCNc23)ccc1Cl
Fc1cc(NC(=O)C(=O)NCc2[nH]nc3CCCCCc23)ccc1Cl
CCc1n[nH]c(NC(=O)C(=O)Nc2ccc(Cl)c(F)c2)c1CC
CCn1ncnc1C(C)NC(=O)C(=O)Nc1ccc(Cl)c(F)c1
Cc1n[nH]c(C)c1CNC(=O)C(=O)Nc1ccc(Cl)c(F)c1
CN(C)C1(CNC(=O)C(=O)Nc2ccc(Cl)c(F)c2)CCN(C)CC1
CC(C)(CNC(=O)C(=O)Nc1ccc(Cl)c(F)c1)N1CCOCC1
CC1CN(CCNC(=O)C(=O)Nc2ccc(Cl)c(F)c2)CC(C)O1
CC(CNC(=O)C(=O)Nc1ccc(Cl)c(F)c1)N1CCCCC1C
CC(C)N1CCCCC1CCNC(=O)C(=O)Nc1ccc(Cl)c(F)c1
CN1CCCC(C1)ONC(=O)C(=O)Nc1ccc(Cl)c(F)c1
CN1CCCC(CNC(=O)C(=O)Nc2ccc(Cl)c(F)c2)C1
CN1CCCC(C1)NC(=O)C(=O)Nc1ccc(Cl)c(F)c1
CCCN1CCCC(C1)NC(=O)C(=O)Nc1ccc(Cl)c(F)c1
CC1(C)CC(CC(C)(C)[N+]1(C)[O-])NC(=O)C(=O)Nc1ccc(Cl)c(F)c1 |(20.21,-44.3,;18.73,-44.71,;19.49,-46.04,;17.41,-45.48,;16.08,-44.71,;16.06,-43.17,;17.4,-42.4,;16.62,-41.06,;18.16,-41.06,;18.74,-43.17,;19.49,-41.83,;20.27,-43.17,;14.75,-45.49,;13.41,-44.72,;13.4,-43.18,;12.08,-45.5,;12.09,-47.04,;10.74,-44.73,;9.41,-45.51,;8.08,-44.74,;6.75,-45.52,;6.75,-47.06,;5.41,-47.83,;8.08,-47.83,;8.08,-49.37,;9.42,-47.06,)|
CC1(C)CC(CC(C)(C)O1)NC(=O)C(=O)Nc1ccc(Cl)c(F)c1
CC1(C)C2CCC1(C)C(C2)NC(=O)C(=O)Nc1ccc(Cl)c(F)c1 |THB:10:8:1:4.5|
CC1(C)CC(CC(C)(C)C1)NC(=O)C(=O)Nc1ccc(Cl)c(F)c1
CCN1CCC(CNC(=O)C(=O)Nc2ccc(Cl)c(F)c2)CC1
CN1CCC(CNC(=O)C(=O)Nc2ccc(Cl)c(F)c2)CC1
Fc1cc(NC(=O)C(=O)NCC2CCNCC2)ccc1Cl
Fc1cc(NC(=O)C(=O)NC2CCN(CC2)C(=O)c2ccccc2)ccc1Cl
CC(C)(C)OC(=O)N1CCC(CC1)NC(=O)C(=O)Nc1ccc(Cl)c(F)c1
CC(C)N1CCC(CC1)NC(=O)C(=O)Nc1ccc(Cl)c(F)c1
CCCN1CCC(CC1)NC(=O)C(=O)Nc1ccc(Cl)c(F)c1
CN1CCC(CC1)NC(=O)C(=O)Nc1ccc(Cl)c(F)c1
CC1(CC(CC(N1C)(C)C)NC(=O)C(=O)Nc2ccc(c(c2)F)Cl)C
CC1(C)CC(CC(C)(C)N1)NCC(=O)Nc1ccc(Cl)c(F)c1
CN(C1CC(C)(C)NC(C)(C)C1)C(=O)C(=O)Nc1ccc(Cl)c(F)c1
CN(C(=O)C(=O)NC1CC(C)(C)NC(C)(C)C1)c1ccc(Cl)cc1
CC1(C)CC(CC(C)(C)N1)NC(=O)CCC(=O)Nc1ccc(Br)cc1
CC1(C)CC(CC(C)(C)N1)NC(=O)CC(=O)Nc1ccc(Br)cc1
CC1(C)CC(CNC(=O)C(=O)Nc2ccc(Cl)c(F)c2)CC(C)(C)N1
CC1(C)CC(CC(C)(C)N1)NC(=O)C(=O)Nc1ccc(Cl)c(F)c1
CN1CCCN(CC1)C(=O)COc1ccc(Cl)cc1
CN1CCC(CC1)NC(=O)Nc1ccc(Cl)cc1Cl
Clc1ccc(NC(=O)CSc2[nH]c(=O)nc3CCCCc23)cc1
Clc1ccc(OCC(=O)Nc2ccc3[nH]c(=O)[nH]c3c2)cc1
Nc1ccc(cc1)C(=O)CC(=O)Nc1ccc(Cl)cc1
C[C@@H](Sc1nc(N)cc(=O)[nH]1)C(=O)Nc1ccc(Cl)cc1 |r|
Clc1ccc(cc1Cl)C(=O)Nc1ccc2C(=O)NC(=O)c2c1
Clc1c(sc2cc(Cl)ccc12)C(=O)Nc1ccnc(=O)[nH]1
Clc1ccc(NC(=O)Nc2ncnc3nc[nH]c23)cc1
Clc1ccc(NC(=O)c2cc3CCCCc3[nH]c2=O)cc1
Cc1cc(SCC(=O)Nc2ccc(Cl)cc2)[nH]c(=O)n1
Clc1ccc(OCC(=O)Nc2cc(=O)[nH]c(=O)[nH]2)cc1
CC1(C)CC(CC(C)(C)N1)NC(=O)C(=O)Nc1ccc(cc1)-n1cc(CCCCCO)nn1
CC1(C)CC(CC(C)(C)N1)NC(=O)C(=O)Nc1ccc(cc1)-n1cc(nn1)-c1ccccc1
CC1(C)CC(CC(C)(C)N1)NC(=O)C(=O)Nc1ccc(cc1)-n1cc(CCc2ccccc2)nn1
CC1(C)CC(CC(C)(C)N1)NC(=O)C(=O)Nc1ccc2ccccc2c1
CC1(C)CC(CC(C)(C)N1)NC(=O)C(=O)Nc1c[nH]c2ncccc12
CC(C)c1cccc(NC(=O)C(=O)NC2CC(C)(C)NC(C)(C)C2)c1
CC(C)c1ccccc1NC(=O)C(=O)NC1CC(C)(C)NC(C)(C)C1
CC1(C)CC(CC(C)(C)N1)NC(=O)C(=O)Nc1ccc(cc1)N=[N+]=[N-]
CC(C)COc1cc(Cl)ccc1NC(=O)C(=O)NC1CC(C)(C)NC(C)(C)C1
CC1(C)CC(CC(C)(C)N1)NC(=O)C(=O)Nc1cccc(OCc2ccccc2)c1
CC1(C)CC(CC(C)(C)N1)NC(=O)C(=O)Nc1ccc(Cl)c(OCc2ccccc2)c1
CC(C)Oc1cc(NC(=O)C(=O)NC2CC(C)(C)NC(C)(C)C2)ccc1Cl
COc1cc(NC(=O)C(=O)NC2CC(C)(C)NC(C)(C)C2)ccc1Cl
Fc1cc(NC(=O)C(=O)NCc2ccccc2CN2CCOCC2)ccc1Cl
CC(NC(=O)C(=O)Nc1ccc(Cl)c(F)c1)C(N1CCOCC1)c1ccccc1Cl
CN1CCN(CC1)C(CNC(=O)C(=O)Nc1ccc(Cl)c(F)c1)c1ccccc1Cl
CN1CCN(CC1)C(CNC(=O)C(=O)Nc1ccc(Cl)c(F)c1)c1cccs1
Fc1cc(NC(=O)C(=O)NCC(N2CCCC2)c2ccc(Cl)cc2)ccc1Cl
Fc1cc(NC(=O)C(=O)NCC(N2CCCC2)c2ccco2)ccc1Cl
CN(C)C(CNC(=O)C(=O)Nc1ccc(Cl)c(F)c1)N1CCCC1
CN(C)C(CNC(=O)C(=O)Nc1ccc(Cl)c(F)c1)c1ccco1
CCN(CC)C(CNC(=O)C(=O)Nc1ccc(Cl)c(F)c1)CC(C)C
CC(NC(=O)C(=O)Nc1ccc(Cl)c(F)c1)c1ccc(cc1)S(N)(=O)=O
CNS(=O)(=O)Cc1ccc(CNC(=O)C(=O)Nc2ccc(Cl)c(F)c2)cc1
Nc1ncc(CNC(=O)C(=O)Nc2ccc(Cl)c(F)c2)cn1
CNC(=O)c1ccc(CNC(=O)C(=O)Nc2ccc(Cl)c(F)c2)cc1
CC1(C)Cc2c(C#N)c(NC(=O)C(=O)Nc3ccc(Cl)c(F)c3)sc2C(C)(C)N1
CC1(C)CC(CC(C)(C)N1)NC(=O)C(=O)Nc1ccc(Cl)cc1OCc1ccccc1
CCOc1cc(Cl)ccc1NC(=O)C(=O)NC1CC(C)(C)NC(C)(C)C1
COc1cc(Cl)ccc1NC(=O)C(=O)NC1CC(C)(C)NC(C)(C)C1
CC1(C)CC(CC(C)(C)N1)NC(=O)C(=O)Nc1ccc(Cl)cc1C(F)(F)F
Cc1cc(Cl)ccc1NC(=O)C(=O)NC1CC(C)(C)NC(C)(C)C1
CC1(C)CC(CC(C)(C)N1)NC(=O)C(=O)Nc1ccc(Cl)cc1Cl
NC(=O)C1CCN(CCC(=O)Nc2ccc(Br)cc2)CC1
CC(C)c1ccc(C)cc1OCC(=O)NNC(=O)Nc1ccc(Cl)cc1
C[C@H]1CCCN(CCC(=O)Nc2ccc(Cl)cc2)C1 |r|
CCOC(=O)[C@H]1CCCN(CCC(=O)Nc2ccc(Br)cc2)C1 |r|
C[C@H]1CN(CCC(=O)Nc2ccc(Br)cc2)C[C@@H](C)O1 |r|
Cc1cc(NC(=O)C(=O)c2c[nH]c3ccccc23)ccc1Br
Brc1ccc(NC(=O)CN2CCCCCC2)cc1
CCNC(=S)N1CCN(CC(=O)Nc2ccc(Br)cc2)CC1
CC(C)C1CCN(CCC(=O)Nc2ccc(Br)cc2)CC1
Clc1ccc(NC(=O)C(=O)NC[C@@H]2COC3(CCCC3)O2)cc1 |r|
COc1cccc(CNC(=O)C(=O)Nc2ccc(Cl)cc2)c1
CC(CC(=O)Nc1ccc(Br)cc1)Nc1cccc(CO)c1
CC1CCCN(CCC(=O)Nc2ccc(Br)cc2)C1
Brc1ccc(NC(=O)C(=O)NCC2OCCc3ccccc23)cc1
Brc1ccc(NC(=O)C(=O)Nc2cccc3ccccc23)cc1
CCN1CCCC1CNC(=O)C(=O)Nc1c(C)c(C)sc1C(=O)OC
Brc1ccc(NC(=O)CSCc2cc(=O)[nH][nH]2)cc1
COc1cccc(NC(=O)C(=O)Nc2ccc(Cl)cc2)c1
Brc1ccc(NC(=O)C(=O)NCc2ccc3OCOc3c2)cc1
COc1cccc(N[C@@H](C)C(=O)Nc2ccc(Br)cc2)c1 |r|
CN(CC(=O)Nc1ccc(Br)cc1)Cc1cn(C)nc1C
Brc1ccc(NC(=O)C(=O)NCC2COc3ccccc3O2)cc1
Brc1ccc(NC(=O)c2cc(CN3CCCC3)on2)cc1
CC1(C)CC(CC(C)(C)N1)NC(=O)C(=O)NCCc1ccc(Cl)cc1
Brc1ccc(NC(=O)C(=O)NCc2ccco2)cc1
CC1(C)CC(CC(C)(C)N1)=NNC(=O)c1[nH]nc2CCCCc12 |(-.58,-3.08,;-.26,-4.59,;.77,-3.45,;-1.76,-4.91,;-2.24,-6.39,;-1.2,-7.53,;.29,-7.19,;1.83,-7.19,;.77,-8.66,;.77,-5.73,;-3.74,-6.72,;-4.22,-8.19,;-5.71,-8.51,;-6.75,-7.37,;-6.19,-9.98,;-5.29,-11.23,;-6.19,-12.47,;-7.65,-12,;-8.98,-12.76,;-10.33,-11.99,;-10.33,-10.45,;-8.98,-9.68,;-7.65,-10.45,)|
CC1Sc2cc(ccc2NC1=O)C(=O)NC1CC(C)(C)NC(C)(C)C1
CC1(C)CC(CC(C)(C)N1)NC(=O)C(=O)Nc1ccc2cc[nH]c2c1
CC1(C)CC(=O)c2cc(C(=O)Nc3ccc(Cl)cc3)c(=O)[nH]c2C1
C[C@H](Sc1nc(N)cc(N)n1)C(=O)Nc1ccc(Cl)cc1 |r|
Clc1ccc(NC(=O)COC(=O)c2n[nH]c3ccccc23)nc1
CC1(C)NC(=O)N(C[C@H](O)COc2ccc(Cl)cc2)C1=O |r|
Clc1ccc(NC(=O)NCCc2cnc[nH]2)cc1Cl
Clc1ccc(NC(=O)C(=O)c2c[nH]c3ccccc23)cc1
CN(C)c1ccc(C)c(NC(=O)COc2ccc(Cl)cc2)c1
Cc1cc(OCC(=O)NCc2nnc[nH]2)ccc1Cl
CC1(C)OC(=O)N(CCC(=O)Nc2ccc(Cl)cc2)[C@@]1(C)O |r|
Oc1ccc2cc(C(=O)Nc3ccc(Cl)cc3)c(=N)oc2c1
Clc1ccc(NC(=O)c2cc(n[nH]2)-n2cnnc2)cc1
Cc1cccc(-c2cc([nH]n2)C(=O)Nc2ccc(Cl)cc2)c1O
CC(C)C[C@@H]1NC(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CO)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]2CSSC[C@H](NC(=O)[C@H](C)NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](CC4=CC=CC=C4)NC(=O)[C@H](CC4=CN=CN4)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(N)=O)NC(=O)CCSSC[C@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)CNC(=O)[C@H](CC(C)C)NC1=O)C(=O)N[C@@H](C)C(=O)N1CCC[C@@H]1C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC1=CC=C(C=C1)C1=CC=CC=C1)C(=O)N3)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N2)C(=O)N[C@@H](C(C)C)C(N)=O |r,c:62,64,74,157,159,164,166,t:60,72,155,162|
CC(C)C[C@@H]1NC(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CO)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]2CSSC[C@H](NC(=O)[C@H](C)NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](CC4=CC=CC=C4)NC(=O)[C@H](CC4=CN=CN4)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(N)=O)NC(=O)CCSSC[C@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)CNC(=O)[C@H](CC(C)C)NC1=O)C(=O)N[C@@H](C)C(=O)N1CCC[C@@H]1C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC1=CC=C(OCCC4CCCCC4)C=C1)C(=O)N3)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N2)C(=O)N[C@@H](C(C)C)C(N)=O |r,c:62,64,74,169,t:60,72,155,157|
CC(C)C[C@@H]1NC(=O)[C@H](CO)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]2CSSC[C@H](NC(=O)[C@H](C)NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](CC4=CC=CC=C4)NC(=O)[C@H](CC4=CN=CN4)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(N)=O)NC(=O)CCSSC[C@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)CNC1=O)C(=O)N[C@@H](C)C(=O)N1CCC[C@@H]1C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC1=CC=C(OCCCCO)C=C1)C(=O)N3)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N2)C(=O)N[C@@H](C(C)C)C(N)=O |r,c:50,52,62,165,t:48,60,155,157|
[H][C@]1(CSSC[C@@H]2NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@]3([H])CSSC[C@]([H])(NC(=O)[C@H](CC4=CC=CC=C4)NC(=O)[C@@H](NC(=O)[C@H]4CCCN4C(=O)[C@H](C)NC(=O)[C@]([H])(CSSCCC(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC4=CN=CN4)C(=O)N[C@@H](CC4=CC=CC=C4)C(=O)N3)NC(=O)[C@H](CCCNC(N)=N)NC(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CO)NC(=O)[C@H](CCCCN)NC2=O)[C@@H](C)O)C(=O)N[C@@H](C)C(=O)N1)C(=O)N[C@@H](C(C)C)C(N)=O |r,c:53,55,108,119,121,t:51,106,117|
CC(C)C[C@@H]1NC(=O)[C@H](CO)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]2CSSC[C@H](NC(=O)[C@H](C)NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](CC4=CC=CC=C4)NC(=O)[C@H](CC4=CN=CN4)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(N)=O)NC(=O)CCSSC[C@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)CNC1=O)C(=O)N[C@@H](C)C(=O)N1CCC[C@@H]1C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC1=CC=C(OCCC4CCCC4)C=C1)C(=O)N3)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N2)C(=O)N[C@@H](C(C)C)C(N)=O |r,c:50,52,62,168,t:48,60,155,157|
CC(C)C[C@@H]1NC(=O)[C@H](CO)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]2CSSC[C@H](NC(=O)[C@H](C)NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](CC4=CC=CC=C4)NC(=O)[C@H](CC4=CN=CN4)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(N)=O)NC(=O)CCSSC[C@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)CNC1=O)C(=O)N[C@@H](C)C(=O)N1CCC[C@@H]1C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC1=CC=C(OCC4CCCCC4)C=C1)C(=O)N3)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N2)C(=O)N[C@@H](C(C)C)C(N)=O |r,c:50,52,62,168,t:48,60,155,157|
CC(C)C[C@@H]1NC(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CO)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]2CSSC[C@H](NC(=O)[C@H](C)NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](CC4=CC=CC=C4)NC(=O)[C@H](CC4=CN=CN4)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(N)=O)NC(=O)CCSSC[C@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)CNC(=O)[C@H](CC(C)C)NC1=O)C(=O)N[C@@H](C)C(=O)N1CCC[C@@H]1C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC1=CC=C(OCCC4=CC=CC=C4)C=C1)C(=O)N3)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N2)C(=O)N[C@@H](C(C)C)C(N)=O |r,c:62,64,74,164,166,169,t:60,72,155,157,162|
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