2478 SMILES Strings for NACHT, LRR and PYD domains-containing protein 3

Compound Name
SMILES String
CC(C)NC(=O)c1c(O)c2ccccc2[nH]c1=O
CC1CC(=O)c2cnc(Nc3cccc(c3)C(F)(F)F)nc2C1
CCCCCC(=O)N1CCN(CCNC=C2C(=O)CC(CC2=O)c2ccco2)CC1 |(3.08,-11.51,;4.41,-10.74,;4.41,-9.2,;5.75,-8.43,;5.75,-6.89,;7.08,-6.12,;8.41,-6.89,;7.08,-4.58,;8.41,-3.81,;8.41,-2.27,;7.08,-1.5,;7.08,.04,;8.41,.81,;8.41,2.35,;9.75,3.12,;9.75,4.66,;8.41,5.43,;7.08,4.66,;8.41,6.97,;9.75,7.74,;11.08,6.97,;11.08,5.43,;12.42,4.66,;10.52,9.07,;9.89,10.48,;11.04,11.51,;12.37,10.74,;12.05,9.23,;5.75,-2.27,;5.75,-3.81,)|
Clc1cccc(NC(=O)c2cnn3cccnc23)c1
Cn1c2ccccc2c(O)c(C(=O)Nc2ncccn2)c1=O
Clc1ccc(NC(=O)Nc2ccc(cc2)C#N)cc1
Brc1cccc(NC(=O)c2cc3ccccc3o2)c1
CCN(CC)CCOc1ccc(cc1)/C(=C(\c2ccccc2)/Cl)/c3ccccc3
CCCCCCCCCn1c2CCCc2c(=N)c2CCCc12
Oc1c(ccc2oc(cc(=O)c12)-c1ccccc1Cl)[N+]([O-])=O
Cc1nc(C)c(CC=C)c(N=NCc2ccccc2O)n1 |w:10.9|
CC(=O)N(N=C1Sc2ccccc2C1=O)c1ccccc1C |w:4.3|
CCOC(=O)c1ccc2n(CC)c(COc3ccc(OC)cc3)nc2c1
CN(CCOc1ccccc1)c1ccc(cn1)S(=O)(=O)N1CCCCC1
COc1cc(CNCCc2ccccc2)ccc1OCc1ccc(Cl)nc1
COc1ccccc1CNC(=O)c1ccc(SC)cc1OC
Cc1onc(c1C(=O)N1CCN=C(C=C1)C(F)(F)F)-c1ccccc1Cl |c:12,14|
On1c(nc2cc(Cl)ccc2c1=O)-c1cccc(c1)C(F)(F)F
C(Oc1ccccc1)c1nnnn1-c1ccccc1
COc1ccc(CNC(=O)c2c(C)oc3c2C(=O)c2ccccc2C3=O)cc1
[#6](\[#7]=[#6]-1\[#7]-[#6]-[#6]-[#7]-1)-c1ccccc1-[#16]-c1cccc2ccccc12
CCOC(=O)N1C(=S)N(c2ccccc2Cl)C2(CCCCC2)C1=O
Cc1ccc(cc1)S(=O)(=O)N1CCN=C1SCc1ccccc1 |c:14|
Cc1cccc(NC(=O)N2CCN(Cc3ccc(Cl)cc3)CC2)c1
CCCCCCCCn1c2CCCc2c(=N)c2ccccc12
[O-][N+](=O)c1ccc[c-](C[NH+]=Nc2nc(NCc3ccccc3)nc(n2)N2CCOCC2)c1=O |w:10.10|
On1c(nc2ccc(Cl)cc2c1=O)-c1ccc(cc1)[N+]([O-])=O
On1c(nc2ccc(Br)cc2c1=O)-c1ccc(cc1)[N+]([O-])=O
CCN1\C(Oc2ccc(cc12)-c1ccccc1)=C\C=C\c1oc2ccc(cc2[n+]1CC)-c1ccccc1
CCCCCNC(=O)C(=O)C1C(=O)Nc2ccccc12
Cc1nc2ccc(Nc3nc4cc(ccc4o3)S(=O)(=O)N3CCOCC3)cc2s1
C[C@H]1C[C@H]2O[C@H]2C=CC=CC(=O)Cc2c(Cl)c(O)cc(O)c2C(=O)O1 |w:7.8,9.10|
COc1ccc(cc1)C2=CC(=O)c3ccccc3O2
Cc1cccc(c1)N1CCN(CC(O)COc2ccc(Cl)cc2)CC1
[O-][N+](=O)c1ccc(\[NH+]=N\c2ccc(=O)[c-](c2)C(=O)Nc2cccc(Cl)c2)c(Cl)c1
Oc1c(C=Nc2ccccn2)sc2ccccc12 |w:4.4|
Cc1ccc(cc1)C1=NOC(C)(C1)c1nnc(o1)-c1ccccc1 |t:8|
Brc1ccccc1C(=O)NCCCCc1ccccc1
CCCC1CCC(=CC1=O)c1ccc(OCC)cc1 |c:6|
COc1ccc(NC(=O)C#Cc2ccccc2)cc1
C1COC2C(C1)C(Nc1ccccc21)c1ccccc1
CCn1c2ccccc2nc2ccc(cc12)=[N+](CC)CC |(3.45,9.91,;4.73,9.17,;4.73,7.69,;3.45,6.95,;2.13,7.74,;.79,6.98,;.79,5.44,;2.13,4.68,;3.45,5.47,;4.73,4.73,;6.01,5.47,;7.34,4.68,;8.68,5.44,;8.68,6.98,;7.34,7.74,;6.01,6.95,;9.95,7.72,;9.95,9.2,;11.23,9.95,;11.24,6.99,;12.51,7.73,)|
CCSc1nsc(NC(=O)Nc2cccc(F)c2)n1
OC(=O)c1c(NC(=O)c2ccc(F)cc2)scc1-c1ccccc1
Oc1ccccc1C(=O)NNC(=S)NC(=O)c1ccc(F)cc1
COc1ccc(cc1)-c1nn(cc1C=O)-c1ccccc1
[O-][N+](=O)c1ccc(cc1)C(=O)NNC(=S)NC(=O)c1ccc(Br)cc1
Nc1ccc(Oc2cc(N)cc(Oc3ccccc3)c2)cc1
Brc1ccc(cc1)-n1cnc(c1)-c1ccccc1
Cc1ccc(NC(=O)c2nc(ncc2Cl)S(=O)(=O)Cc2ccccc2)cc1
Brc1cccc(c1)C(=O)NNC(=O)CN1CCCCC1
Cn1c2ccccc2c(O)c(C(=O)NNC(=O)c2ccccc2F)c1=O
Cc1cccc(c1)C(=O)NNC(=O)c1c(O)c2ccccc2n(C)c1=O
CN(CC(=O)N1CCc2ccccc2C1)c1ccccc1
Cc1cccc(c1)C(=O)ONC(=N)Cc1cccc2ccccc12
CCCOc1ccc(cc1)C(=O)NNC(=S)NC(=O)c1cccs1
CC(=O)Oc1c(I)cc(I)cc1C(=O)Nc1ccc(Cl)cc1
CCC1Nc2ncnc(N3CCN(CC3)c3ccccn3)c2N(Cc2ccc(Cl)cc2)C1=O
Oc1c(C(=O)NCCC2=CCCCC2)c(=O)nc2sccn12 |t:8|
Oc1c(C(=O)NCCCc2ccccc2)c(=O)nc2sccn12
CC1CC(C)CN(CCCNC(=O)c2c(O)nc3c(C)cccn3c2=O)C1
Fc1cccc2sc(nc12)N(CCCN1CCOCC1)C(=O)CCS(=O)(=O)c1ccccc1
Cc1csc2nc(=O)c(C(=O)NCCC3=CCCCC3)c(O)n12 |t:14|
COc1c(OC(C)=O)c(=O)n2c3ccccc3c3ccnc1c23
COc1cccc(NC(=O)c2ccccc2)c1
CC(N)C(=O)OC(C)(C)Cc1ccc(Cl)cc1
CC[N+](CC)=c1ccc2nc3ccc(N)cc3n(-c3ccccc3)c2c1 |(14.37,8.04,;13.04,7.27,;11.7,8.03,;11.7,9.57,;13.03,10.35,;10.37,7.26,;10.37,5.65,;8.98,4.86,;7.6,5.68,;6.26,4.91,;4.93,5.68,;3.55,4.86,;2.16,5.65,;2.16,7.26,;.83,8.03,;3.55,8.05,;4.93,7.22,;6.26,7.99,;6.26,9.53,;7.6,10.3,;7.6,11.84,;6.26,12.61,;4.93,11.84,;4.93,10.3,;7.6,7.22,;8.98,8.05,)|
CCC1Nc2ncnc(N3CCN(CC3)c3ccccn3)c2N(Cc2ccc(Br)cc2)C1=O
c1cc(ccc1NC(=O)Nc2ccc(c(c2)Cl)Cl)Cl
COC(=O)c1ccc(nc1)-c1cn(Cc2cc(Cl)ccc2OC)nn1
CCCOc1ccc(Cl)cc1Cn1cc(-c2ccc(C(=O)OC)cn2)nn1
COc1ccc(Cl)cc1Cn1cc(nn1)C(=O)N1CC(F)(F)C1
COc1ccc(Cl)cc1Cn1cc(nn1)-c1ccc(cc1)C(=O)N1CCC1
COc1ccc(Cl)cc1Cn1cc(-c2ccc(CO)cc2)nn1
CCCOc1ccc(Cl)cc1Cn1cc(nn1)S(=O)(=O)c1ccc(C)cc1
CCCOc1ccc(Cl)cc1Cn1cc(nn1)-c1ccccc1
O=C(Cc1c2CCCc2ccc1-c1ccnc(c1)C#N)NS(=O)(=O)c1ccn(n1)C1CC1
CC(C)c1cc(F)cc(-c2ccncc2)c1CC(=O)NS(=O)(=O)c1ccn(n1)C1CC1
COc4cc(c1cc(F)cc(C(C)C)c1CC(=O)NS(=O)(=O)c3cn(C2CC2)cn3)ccn4
COc1cc(ccn1)-c1cc(F)cc(C(C)C)c1CC(=O)NS(=O)(=O)c1ccn(n1)C1CC1
COc1cc(ccn1)-c1ccc2CCCc2c1CC(=O)NS(=O)(=O)c1cnn(n1)C1CC1
CC(C)c1cc(F)cc(-c2cccnc2)c1CC(=O)NS(=O)(=O)c1cn(cn1)C1CC1
CC(C)c1cc(F)cc(-c2ccnc(c2)C#N)c1CC(=O)NS(=O)(=O)c1cnn(n1)C1CC1
O=C(Cc1c2CCCc2ccc1-c1ccnc(c1)C#N)NS(=O)(=O)c1cnn(n1)C1CC1
CC(C)c1cc(F)cc(-c2ccnc(c2)C#N)c1CC(=O)NS(=O)(=O)c1cnn(c1)C1CC1
COc1cc(ccn1)-c1cc(F)cc(C(C)C)c1C(O)C(=O)NS(=O)(=O)c1cnn(c1)C1CC1
CC(C)c1cc(F)cc(-c2cccnc2)c1CC(=O)NS(=O)(=O)c1cnn(c1)C1CC1
CCC1(COC1)c1cc(nn1C(C)C)S(=O)(=O)NC(=O)Cc1c2CCCc2cc2CCCc12
COC1(COC1)c1cc(nn1C(C)C)S(=O)(=O)NC(=O)Cc1c2CCCc2ccc1-c1ccnc(c1)C#N
CCC1(COC1)c1cc(nn1C1CC1)S(=O)(=O)NC(=O)Cc1c2CCCc2cc2CCCc12
CC(N(C)C)c1cc(nn1C1CC1)S(=O)(=O)NC(=O)Cc1c2CCCc2cc2CCCc12
CC(C)c1cc(F)cc(C(C)C)c1CC(=O)NS(=O)(=O)c1cc(CN(C)C)n(n1)C1CC1
COc1cc(ccn1)-c1ccc2CCCc2c1CC(=O)NS(=O)(=O)c1ccn(n1)C1CC1
COc1cc(ccn1)-c1cc(F)cc(C(C)C)c1CC(=O)NS(=O)(=O)c1cnn(c1)C1CC1
O=C(Cc1c2CCCc2cc2CCCc12)NS(=O)(=O)c1cnn(c1)C1CC1
COc1cc(ccn1)-c1cc(F)cc(C(C)C)c1CC(=O)NS(=O)(=O)c1cnn(n1)C1CC1
COc1cc(ccn1)-c1cc(F)cc(C(C)C)c1CC(=O)NS(=O)(=O)c1ncn(n1)C1CC1
CC(C)c1cc(F)cc(-c2cccnc2)c1CC(=O)NS(=O)(=O)c1ncn(n1)C1CC1
COc1cc(ccn1)-c1ccc2CCCc2c1CC(=O)NS(=O)(=O)c1cnn(c1)C1CC1
CC(C)c1cc(F)cc(C(C)C)c1CC(=O)NS(=O)(=O)c1cnn(c1)C1CC1
CC(C)c1cc(F)cc(C(C)C)c1CC(=O)NS(=O)(=O)c1ncn(n1)C1CC1
CC(C)c1cc(F)cc(C(C)C)c1CC(=O)NS(=O)(=O)c1cnn(n1)C1CC1
CC(C)c1cc(F)cc(-c2cccnc2)c1CC(=O)NS(=O)(=O)c1cnn(n1)C1CC1
CC(C)c1cc(F)cc(C(C)C)c1CC(=O)NS(=O)(=O)c1cn(cn1)C1CC1
COC1(COC1)c1cc(nn1C(C)C)S(=O)(=O)NC(=O)Cc1c(cc(F)cc1C(C)C)C(C)C
O=C(Cc1c2CCCc2ccc1-c1ccnc(c1)C#N)NS(=O)(=O)c1cnn(c1)C1CC1
CC(C)c1cc(F)cc(-c2ccnc(c2)C#N)c1CC(=O)NS(=O)(=O)c1cn(cn1)C1CC1
Cc1oc(cc1C(C)(C)O)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
Cc1oc(cc1C(C)(C)O)[S@@](N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12 |r|
CC(C)(O)c1ncc(s1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
CC(C)(c1ncc(s1)[S@@](=NC(=O)Nc2c3c(cc4c2CCC4)CCC3)(=O)N)O
CC(C)(C)OC(=O)NS(=O)(=NC(=O)Nc1c2CCCc2cc2CCCc12)c1cnc(s1)C(C)(C)O
CNS(=O)(=NC(=O)Nc1c2CCCc2c(F)c2CCCc12)c1cc(cs1)C(C)(C)O
Cc1cc(sc1C(C)(C)O)S(N)(=O)=NC(=O)Nc1cc(C)nc(C)c1
CC(C)c1cc(F)cc(C(C)C)c1NC(=O)N=S(N)(=O)c1cc(c(C)o1)C(C)(C)O
CC(C)c1cc(F)cc(C(C)C)c1NC(=O)N=S(N)(=O)c1ccc(cc1)C(C)(C)O
Cc1sc(cc1C(C)(C)O)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
CC(C)(O)c1ccc(c(F)c1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
CC(C)(O)c1csc(c1)S(N)(=O)=NC(=O)Nc1c2CCCc2c(Cl)c2CCCc12
CC(C)c1cc(C#N)c(F)c(C(C)C)c1NC(=O)N=S(N)(=O)c1cnc(s1)C(C)(C)O
CC(C)n1ccc(n1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
CC(C)c1cc(OC(F)F)cc(C(C)C)c1NC(=O)N=S(N)(=O)c1sc(cc1F)C(C)(C)O
CCc1cc(OC(F)F)cc(C(C)C)c1NC(=O)N=S(N)(=O)c1cnc(s1)C(C)(C)O
Cc1cc(ccc1S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12)C(C)(C)O
CC(C)c1cc(OC(F)F)cc(C2CC2)c1NC(=O)N=S(N)(=O)c1cnc(s1)C(C)(C)O
CC(C)c1cc(F)cc(C(C)C)c1NC(=O)N=S(N)(=O)c1cnc(s1)C(C)(C)O
CC(C)c1cc(F)cc(C(C)C)c1NC(=O)N=S(N)(=O)c1cccc(c1)C(C)(C)O
CC(C)c1c(F)c(cc(C2CC2)c1NC(=O)N=S(N)(=O)c1cnc(s1)C(C)(C)O)C#N
CC(C)c1cc(OC(F)F)cc(C(C)C)c1NC(=O)N=S(N)(=O)c1sc(cc1C)C(C)(C)O
CC(C)c1cc(OC(F)F)cc(C(C)C)c1NC(=O)N=S(N)(=O)c1cnc(s1)C(C)(C)O
CC(C)(O)c1csc(c1)S(N)(=O)=NC(=O)Nc1c2CCCc2c(C#N)c2CCCc12
CC(C)(O)c1ncc(s1)S(N)(=O)=NC(=O)Nc1c2CCCc2c(OC(F)F)c2CCCc12
CN(C)Cc1ccc(cc1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
CC(C)c1cc(OC(F)F)cc(C2CC2)c1NC(=O)N=S(N)(=O)c1ccc(cc1C)C(C)(C)O
CC(C)(O)c1cc(F)c(s1)S(N)(=O)=NC(=O)Nc1c2CCCc2c(F)c2CCCc12
CC1CCc2c1cc1CCCc1c2NC(=O)N=S(N)(=O)c1cc(c(C)o1)C(C)(C)O
CC1CCc2cc3CCCc3c(NC(=O)N=S(N)(=O)c3cc(c(C)o3)C(C)(C)O)c12
CC(C)c1cc(C#N)c(F)c(C(C)C)c1NC(=O)N=S(N)(=O)c1cc(c(C)o1)C(C)(C)O
CC(C)(O)c1cccc(c1)S(N)(=O)=NC(=O)Nc1c2CCCc2c(F)c2CCCc12
CC(C)c1cc(cc(C(C)C)c1NC(=O)N=S(N)(=O)c1ncc(s1)C(C)(C)O)C#N
CC(C)c1cc(F)cc(C(C)C)c1NC(=O)N=S(N)(=O)c1ccc(CN(C)C)cc1
CC(C)c1cc(OC(F)F)cc(C2CC2)c1NC(=O)N=S(N)(=O)c1ccc(CN(C)C)cc1
CC(C)c1cc(OC(F)F)cc(C(C)C)c1NC(=O)N=S(N)(=O)c1ncc(s1)C(C)(C)O
CC(C)c1cc(F)cc(C(C)C)c1NC(=O)N=S(N)(=O)c1ncc(s1)C(C)(C)O
CC(C)c1cc(F)cc(C(C)C)c1NC(=O)N=S(N)(=O)c1cc(cs1)C(C)(C)O
CC(C)(O)c1ccc(c(F)c1)S(N)(=O)=NC(=O)Nc1c2CCCc2c(Cl)c2CCCc12
CC(C)c1cc(F)cc(C(C)C)c1NC(=O)N=S(N)(=O)c1ccc(cc1)S(C)(=O)=O
CC(C)(O)c1ncc(s1)S(N)(=O)=NC(=O)Nc1c2CCCc2c(C#N)c2CCCc12
CC(C)(O)c1ncc(s1)S(N)(=O)=NC(=O)Nc1c2CCCc2c(F)c2CCCc12
Cc1oc(cc1C(C)(C)O)S(N)(=O)=NC(=O)Nc1c2CCCc2c(F)c2CCCc12
CC(C)(O)c1cccc(c1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
CC(C)(O)c1ccc(c(F)c1)S(N)(=O)=NC(=O)Nc1c2CCCc2c(F)c2CCCc12
CN(C)Cc1ccc(c(F)c1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
CC(C)c1cc(F)cc(C(C)C)c1NC(=O)N=S(N)(=O)c1ccc(s1)C(C)(C)O
CC(C)(O)c1ccc(c(Cl)c1)S(N)(=O)=NC(=O)Nc1c2CCCc2c(F)c2CCCc12
CN(C)Cc1cccc(c1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
Cc1cc(ccc1C(C)(C)O)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
Cc1nc(sc1S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12)C(C)(C)O
CC(C)c1cc(OC(F)F)cc(C2CC2)c1NC(=O)N=S(N)(=O)c1ccc(cc1F)C(C)(C)O
CC(C)(O)c1ccc(F)c(c1)S(N)(=O)=NC(=O)Nc1c2CCCc2c(F)c2CCCc12
CC(C)(O)c1cc(F)cc(c1)S(N)(=O)=NC(=O)Nc1c2CCCc2c(F)c2CCCc12
CC(C)c1cc(OC(F)F)cc(C(C)C)c1NC(=O)N=S(N)(=O)c1cc(C)c(s1)C(C)(C)O
CC(C)(O)c1cc(ccc1F)S(N)(=O)=NC(=O)Nc1c2CCCc2c(F)c2CCCc12
Cc1nc(sc1S(N)(=O)=NC(=O)Nc1c2CCCc2c(F)c2CCCc12)C(C)(C)O
CC(C)(O)c1ccc(cc1F)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
CC(C)(O)c1csc(n1)S(N)(=O)=NC(=O)Nc1c2CCCc2c(F)c2CCCc12
CC(C)c1ccc(F)c(C(C)C)c1NC(=O)N=S(N)(=O)c1cnc(s1)C(C)(C)O
CC(C)c1cc(F)cc(C(C)C)c1NC(=O)N=S(N)(=O)c1cccc(c1)S(C)(=O)=O
CC(C)(O)c1cnc(s1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
CC(C)c1cc(cc(C(C)C)c1NC(=O)N=S(N)(=O)c1sc(cc1F)C(C)(C)O)C#N
CC(C)c1cc(cc(C(C)C)c1NC(=O)N=S(N)(=O)c1cc(cc(c1)C(C)(C)O)C(C)(C)O)C#N
CC(C)c1cc(cc(C(C)C)c1NC(=O)N=S(N)(=O)c1cc(cc(c1)C(C)(C)O)C#N)C#N
CC(C)c1cc(cc(C(C)C)c1NC(=O)N=S(N)(=O)c1ccc(c(CO)c1)C(C)(C)O)C#N
CC(C)(O)c1nc(CO)c(s1)S(N)(=O)=NC(=O)Nc1c2CCCc2c(C#N)c2CCCc12
CC(C)c1cc(cc(C(C)C)c1NC(=O)NS(=N)(=O)c1sc(nc1CO)C(C)(C)O)C#N
CC(C)c1cc(C#N)c(F)c(C(C)C)c1NC(=O)NS(=N)(=O)c1sc(nc1CO)C(C)(C)O
CC(C)c1cc(C#N)c(F)c(C(C)C)c1NC(=O)N=S(N)(=O)c1cnc(s1)C(C)(O)CO
CC(C)c1cc(cc(C(C)C)c1NC(=O)N=S(N)(=O)c1ccc(cc1)S(C)(=O)=O)C#N
CC(C)(O)c1csc(c1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
CC(C)(O)c1csc(c1)S(N)(=O)=NC(=O)Nc1c2CCCc2c(F)c2CCCc12
CC(C)(O)c1coc(c1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
CC(C)(O)c1csc(n1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
Cc1cc(NC(=O)N=S(N)(=O)c2ccc(s2)C(C)(C)O)cc(C)n1
CC(C)c1cc(cc(C(C)C)c1NC(=O)N=S(N)(=O)c1ccc(s1)C(C)(C)O)C#N
CC(C)c1cc(cc(C(C)C)c1NC(=O)N=S(N)(=O)c1sc(nc1CO)C(C)(C)O)C#N
CC(C)c1cc(C#N)c(F)c(C(C)C)c1NC(=O)N=S(N)(=O)c1sc(nc1CO)C(C)(C)O
CC(C)c1cc(F)cc(C(C)C)c1NC(=O)N=S(N)(=O)c1cc(Cl)c(Cl)s1
CC(C)c1cc(F)cc(C(C)C)c1NC(=O)N=S(N)(=O)c1cn(C)nc1C
CC(C)c1cc(F)cc(C(C)C)c1NC(=O)N=S(N)(=O)c1ccc2ccccc2c1
CC(C)c1cc(F)cc(C(C)C)c1NC(=O)N=S(N)(=O)c1ccc2OCCc2c1
CC(C)c1cc(F)cc(C(C)C)c1NC(=O)N=S(N)(=O)c1ccccc1-c1ccccc1
COCc1ccccc1S(N)(=O)=NC(=O)Nc1c(cc(F)cc1C(C)C)C(C)C
COc1cc(c(O)s1)S(N)(=O)=NC(=O)Nc1c(cc(F)cc1C(C)C)C(C)C
CC(C)c1cc(F)cc(C(C)C)c1NC(=O)N=S(N)(=O)c1cccnc1
CC(C)c1cc(F)cc(C(C)C)c1NC(=O)N=S(N)(=O)c1ccc2OCOc2c1
CC(C)c1cc(F)cc(C(C)C)c1NC(=O)N=S(N)(=O)c1cc(C)oc1C
CC(C)c1cc(F)cc(C(C)C)c1NC(=O)N=S(N)(=O)c1cnc2ccccc2c1
CC(C)c1cc(F)cc(C(C)C)c1NC(=O)N=S(N)(=O)c1cnc2CCCn12
CC(C)c1cc(F)cc(C(C)C)c1NC(=O)N=S(N)(=O)c1ccc(C)cn1
Cc1oc(cc1C(C)(C)O)S(N)(=O)=NC(=O)Nc1c2CCCc2nc2CCCc12
CC(C)c1cncc(C(C)C)c1NC(=O)N=S(N)(=O)c1cc(c(C)o1)C(C)(C)O
CC(C)(O)c1ncc(s1)S(N)(=O)=NC(=O)Nc1c2CCc2cc2CCCc12
CC(C)(O)c1ncc(s1)[S@@](N)(=O)=NC(=O)Nc1c2CCc2cc2CCCc12 |r|
CC(C)(O)c1ncc(s1)[S@](N)(=O)=NC(=O)Nc1c2CCc2cc2CCCc12 |r|
CC(C)(O)c1ncc(s1)S(N)(=O)=NC(=O)Nc1c2CCc2cc2CCc12
NS(=O)(=NC(=O)Nc1c2CCCc2c(F)c2CCCc12)c1ccc(O)cc1F
CC(C)(O)c1ncc(s1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2C(O)CCc12
COC1CN(Cc2ccc(cc2)S(N)(=O)=NC(=O)Nc2c3CCCc3cc3CCCc23)C1
COCCN(C)Cc1ccc(cc1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
NS(=O)(=NC(=O)Nc1c2CCCc2cc2CCCc12)c1ccc(CO)cc1
NS(=O)(=NC(=O)Nc1c2CCCc2cc2CCCc12)c1ccc(CN2CCOCC2)cc1
NS(=O)(=NC(=O)Nc1c2CCCc2cc2CCCc12)c1ccc(CN2CCC(F)(F)C2)cc1
NS(=O)(=NC(=O)Nc1c2CCCc2cc2CCCc12)c1ccc(CN2CCCC2)cc1
NS(=O)(=NC(=O)Nc1c2CCCc2cc2CCCc12)c1ccc(CN2CCC2)cc1
CN(CC=C)Cc1ccc(cc1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
CN(CC#C)Cc1ccc(cc1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
CN(CC1CC1)Cc1ccc(cc1)S(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
CN(CC(F)F)Cc1ccc(cc1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
COCc1ccc(cc1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
NCc1ccc(cc1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
NS(=O)(=NC(=O)Nc1c2CCCc2cc2CCCc12)c1ccc(CN2CCCC2=O)cc1
CN(C)S(=O)(=NC(=O)Nc1c2CCCc2cc2CCCc12)c1cc(cs1)C(C)(C)O
CNS(=O)(=NC(=O)Nc1c2CCCc2cc2CCCc12)c1cc(cs1)C(C)(C)O
CNS(=O)(=NC(=O)Nc1c2CCCc2cc2CCCc12)c1cnc(s1)C(C)(C)O
CN(C(=O)N=S(N)(=O)c1cnc(s1)C(C)(C)O)c1c2CCCc2cc2CCCc12
CNS(=O)(=NC(=O)N(C)c1c2CCCc2cc2CCCc12)c1cnc(s1)C(C)(C)O
CC(=O)NS(=O)(=NC(=O)Nc1c2CCCc2cc2CCCc12)c1cnc(s1)C(C)(C)O
COC(=O)CCC(=O)N(C)Cc1ccc(cc1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
CN(Cc1ccc(cc1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12)C(=O)CCC(O)=O
CC(C)c1ccc(C#N)c(C(C)C)c1NC(=O)N=S(N)(=O)c1ccc(s1)C(C)(C)O
CCc1ccc2cnn(C)c2c1NC(=O)N=S(N)(=O)c1ncc(s1)C(C)(C)O
CCc1ccc2cn(C)nc2c1NC(=O)N=S(N)(=O)c1ncc(s1)C(C)(C)O
CC(C)(O)c1cnc(s1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2OCCc12
CC(C)(O)c1cnc(s1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCOc12
CC(C)(O)c1cc(nn1-c1ccccc1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
CC(C)(O)c1ccc(cn1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
CN(Cc1ccc(cc1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12)C(=O)CCC#C
CC(C)(O)c1csc(n1)S(N)(=O)=NC(=O)Nc1c2CCc2cc2CCCc12
CC(C)(O)c1csc(n1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCOc12
Cc1nc(ccc1S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12)C(C)(C)O
Cc1sc(nc1C(C)(C)O)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
CC(N(C)C)c1ccc(cc1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
CN(C)C(C)(C)c1ccc(cc1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
CN(Cc1ccc(cc1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12)C(C)=O
CC(C)(O)c1cc(F)c(s1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
CN1CCc2cc(ccc2C1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
CN1CCc2ccc(cc2C1)S(=N)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
COc1cc(CN(C)C)ccc1S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
Cn1ncc2cc(ccc12)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
COC(C)(C)c1ccc(cc1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
CC(C)Cc1ccc(cn1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
CN(C)Cc1ccc(cn1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
CC(C)Cc1ccc(cc1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
CN(C)Cc1ccc(nc1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
CN(C)Cc1cc(F)c(s1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
CN(C)Cc1ccc(cc1F)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
CC(C)(O)c1cc(F)c(s1)S(N)(=O)=NC(=O)Nc1c2CCc2cc2CCCc12
CC(C)c1csc(c1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
CC1CCCN1c1ccc(cc1)S(=N)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
CC(C)c1nn(c(C(C)C)c1NC(=O)N=S(N)(=O)c1cc(cs1)C(C)(C)O)-c1ccccc1
CC(C)(O)c1ncc(s1)S(N)(=O)=NC(=O)Nc1cc2CCCc2c2CCCc12
CNCc1ccc(c(F)c1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
CC(C)c1ccc(cn1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
CC(C)(O)c1ncc(s1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCOc12
CCc1ccc2cn[nH]c2c1NC(=O)N=S(N)(=O)c1cnc(s1)C(C)(C)O
CC1CCc2c1cc1CCCc1c2NC(=O)N=S(N)(=O)c1cnc(s1)C(C)(C)O
CC1CCc2cc3CCCc3c(NC(=O)N=S(N)(=O)c3cnc(s3)C(C)(C)O)c12
CC(C)(O)c1ncc(s1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2C(=O)CCc12
CC(C)(O)c1ncc(s1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCC(=O)c12
COC(C)(C)c1ncc(s1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
CNCc1ccc(cc1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
CC(C)(O)c1cnc(s1)S(N)(=O)=NC(=O)Nc1c2CCCc2c(Br)c2CCCc12
CN(Cc1cccc(c1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12)C(C)=O
CC(C)(O)c1ncc(s1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCC(O)c12
CNS(=O)(=NC(=O)Nc1c2CCCc2cc2CCCc12)c1ccc(CN(C)C)cc1
CN1CCCC1c1ccc(cc1)S(=N)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
CC(=O)c1ncc(s1)S(N)(=O)=NC(=O)Nc1c2CCCc2cc2CCCc12
Cc1ccc(cc1C)-c1ccc(NC(=O)N=S(N)(=O)c2ncc(s2)C(C)(C)O)c2CCCc12
Cc1ccc(cc1C)-c1c2CCCc2c(NC(=O)N=[S@@](N)(=O)c2ncc(s2)C(C)(C)O)c2CCCc12 |r|
Cc1ccc(cc1C)-c1c2CCCc2c(NC(=O)N=[S@](N)(=O)c2ncc(s2)C(C)(C)O)c2CCCc12 |r|
CC(C)c1cc(F)cc(C(C)C)c1NC(=O)N=S(N)(=O)c1sc(C)nc1C
CC(C)c1cc(F)cc(C(C)C)c1NC(=O)N=S(N)(=O)c1cnc2n(C)ncc2c1
CC(C)c1cc(F)cc(C(C)C)c1NC(=O)N=S(N)(=O)c1cccc2c(cccc12)N(C)C
CN(C)S(=O)(=O)NC(=O)c1cnc(Nc2c3CCCc3cc3CCCc23)o1
O=C(NS(=O)(=O)N1CCOCC1)c1cnc(Nc2c3CCCc3cc3CCCc23)o1
O=C(NS(=O)(=O)N1CCCCC1)c1cnc(Nc2c3CCCc3cc3CCCc23)o1
O=C(NS(=O)(=O)N1CCCOCC1)c1cnc(Nc2c3CCCc3cc3CCCc23)o1
CC1COCCN1S(=O)(=O)NC(=O)c1cnc(Nc2c3CCCc3cc3CCCc23)o1
O=C(NS(=O)(=O)N1CCCC1)c1cnc(Nc2c3CCCc3cc3CCCc23)o1
CC(C)NS(=O)(=O)NC(=O)c1cnc(Nc2c3CCCc3cc3CCCc23)o1
O=C(NS(=O)(=O)NCc1ccccc1)c1cnc(Nc2c3CCCc3cc3CCCc23)o1
O=C(NS(=O)(=O)N1CCOCC11CCC1)c1cnc(Nc2c3CCCc3cc3CCCc23)o1
CC(C)C1COCCN1S(=O)(=O)NC(=O)c1cnc(Nc2c3CCCc3cc3CCCc23)o1
CCC1COCCN1S(=O)(=O)NC(=O)c1cnc(Nc2c3CCCc3cc3CCCc23)o1
COC1CN(C1Cl)S(=O)(=O)NC(=O)c1cnc(Nc2c3CCCc3cc3CCCc23)o1
CN(C)S(=O)(=O)NC(=O)c1coc(Nc2c3CCCc3cc3CCCc23)n1
CN(C)S(=O)(=O)NC(=O)c1cnc(Nc2c3CCCc3c(Cl)c3CCCc23)o1
CC(C)N(C)S(=O)(=O)NC(=O)c1cnc(Nc2c3CCCc3cc3CCCc23)o1
CCC1CN(CCO1)S(=O)(=O)NC(=O)c1cnc(Nc2c3CCCc3cc3CCCc23)o1
COC1CN(C1)S(=O)(=O)NC(=O)c1cnc(Nc2c3CCCc3cc3CCCc23)o1
Cn1cc(cn1)N(C1CCOCC1)S(=O)(=O)NC(=O)c1cnc(Nc2c3CCCc3cc3CCCc23)o1
CN(C)S(=O)(=O)NC(=O)c1cnc(Nc2cccc3CCCc23)o1
CC(C)N(C)S(=O)(=O)NC(=O)c1coc(Nc2c3CCCc3cc3CCCc23)n1
O=C(NS(=O)(=O)N1CCCC1)c1coc(Nc2c3CCCc3cc3CCCc23)n1
CCN(C(C)C)S(=O)(=O)NC(=O)c1cnc(Nc2c3CCCc3cc3CCCc23)o1
CN(C1CCOC1)S(=O)(=O)NC(=O)c1cnc(Nc2c3CCCc3cc3CCCc23)o1
CC1COCCN1S(=O)(=O)NC(=O)c1coc(Nc2c3CCCc3cc3CCCc23)n1
CN(C)S(=O)(=O)NC(=O)c1cnc(Nc2c3CCCc3c(F)c3CCCc23)o1
CN(C)S(=O)(=O)NC(=O)c1coc(Nc2c3CCCc3c(F)c3CCCc23)n1
CN(C)S(=O)(=O)NC(=O)c1coc(Nc2c3CCCc3c(Cl)c3CCCc23)n1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCC(O)C1)C(F)(F)F
Cc1ccc2CCCc2c1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCC(O)C1
Cc1ccc2CCCc2c1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCC1
Cc1ccc2CCCc2c1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCOCC1
CC1(O)CCN(C1)S(=O)(=O)NC(=O)c1coc(Nc2c3CCCc3c(F)c3CCCc23)n1
Clc1c2CCCc2c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCCC2)c2CCCc12
Fc1c2CCCc2c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCCC2)c2CCCc12
CO[C@@H]1CCN(C1)S(=O)(=O)NC(=O)c1coc(Nc2c3CCCc3c(Cl)c3CCCc23)n1 |r|
Clc1c2CCCc2c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCOCC2)c2CCCc12
COCC1CN(CCO1)S(=O)(=O)NC(=O)c1coc(Nc2c3CCCc3c(Cl)c3CCCc23)n1
COCCN(C(C)C)S(=O)(=O)NC(=O)c1coc(Nc2c3CCCc3c(Cl)c3CCCc23)n1
FC(F)(F)C1CCCN1S(=O)(=O)NC(=O)c1coc(Nc2c3CCCc3c(Cl)c3CCCc23)n1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCOCC1)C1CC1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCC(O)C1)C1CC1
CC(C)N(C)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
Cc1ccc(cc1Nc2nc(co2)C(=O)NS(=O)(=O)N3CCCOCC3)C(F)(F)F
CC1COCCN1S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CCC1CN(CCO1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CC(C)NS(=O)(=O)C1CCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CC1CCN(C1)S(=O)(=O)NC(=O)c1coc(Nc2c3CCCc3c(F)c3CCCc23)n1
CC1(C)CCN(C1)S(=O)(=O)NC(=O)c1coc(Nc2c3CCCc3c(F)c3CCCc23)n1
CN(C)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)F)n1
O=C(NS(=O)(=O)N1CCOCC1)c1csc(Nc2c3CCCc3cc3CCCc23)n1
CN(C)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(C)(F)F)n1
CC(C)n1nc2CCCc2c1Nc1nc(co1)C(=O)NS(=O)(=O)N(C)C
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCOCC1)C(C)(F)F
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCCC1)C(F)(F)F
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCOC2(COC2)C1)C(F)(F)F
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCC(CC1)S(C)(=O)=O)C(F)(F)F
CC1CCN(C1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCC(C)(C)C1)C(F)(F)F
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCC(F)(F)C1)C(F)(F)F
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCC(CS(C)(=O)=O)CC1)C(F)(F)F
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCC(F)(F)CC1)C(F)(F)F
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCC(CC1)C(F)(F)F)C(F)(F)F
CC(C)c1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N(C)C)C(F)(F)F
CC(C)c1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCOCC1)C(F)(F)F
CC(C)c1cc(Nc2nc(co2)C(=O)NS(=O)(=O)N(C)C)c(C)cc1Cl
CC(C)c1cc(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCOCC2)c(C)cc1Cl
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCNCC1)C(F)(F)F
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCN(CC1)S(C)(=O)=O)C(F)(F)F
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCOCC1)C(C)(F)F
CC(=O)N1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CC(=O)NC1CCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CN(C)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)S(F)(F)(F)(F)F)n1
CN(C)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C2CC2)n1
CN(C)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C2CCC2)n1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)NC1CCOCC1)C(F)(F)F
COC[C@@H]1CCCN1S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1 |r|
CC(C)n1cc(C)c(Nc2nc(co2)C(=O)NS(=O)(=O)N(C)C)n1
CC(C)c1ccc(C)c(Nc2nc(co2)C(=O)NS(=O)(=O)N(C)C)c1
CN(C)S(=O)(=O)NC(=O)c1coc(Nc2cc(cc(c2C)C(F)(F)F)C(F)(F)F)n1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCOCC1)C1CC1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCOCC1)C(F)F
CN(C)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C2(C)CC2)n1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCOCC1CO)C(F)(F)F
CC(C)NS(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CC(C)c1ccc(C)c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCCOCC2)c1
COCCN(C(C)C)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
COCC1CN(CCO1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCNC(=O)CC1)C(F)(F)F
CC(C)N(C(C)C)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
COC[C@H]1CCCN1S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1 |r|
C[C@H]1CCC[C@@H](C)N1S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1 |r|
CC(C)c1ccc(C)c(Nc2nc(cs2)C(=O)NS(=O)(=O)N(C)C)c1
CC(C)c1ccc(C)c(Nc2nc(cs2)C(=O)NS(=O)(=O)N2CCOCC2)c1
CC(C)c1ccc(C)c(Nc2nc(cs2)C(=O)NS(=O)(=O)N2CCCOCC2)c1
COC1CN(C1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CC1CCOCCN1S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CCc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCOCC1)C(F)(F)F
CCc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N(C)C)C(F)(F)F
COC(C)c1ccc(C)c(Nc2nc(co2)C(=O)NS(=O)(=O)N(C)C)c1
CN(C)S(=O)(=O)NC(=O)c1csc(Nc2cc(ccc2C)C(F)(F)F)n1
Cc1ccc(CC(F)(F)F)cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCOCC1
CCS(=O)(=O)N1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
Cc1ccc(cc1Nc1nc(cs1)C(=O)NS(=O)(=O)N1CCOCC1)C(F)(F)F
Cc1ccc(cc1Nc1nc(cs1)C(=O)NS(=O)(=O)N1CCCOCC1)C(F)(F)F
CN(C)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C2CC2)C(F)(F)F)n1
CN(C)S(=O)(=O)NC(=O)c1coc(Nc2cc(C)ccc2C)n1
CN(C)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(C)(C)C)n1
CC(C)c1ccc(C(C)C)c(Nc2nc(co2)C(=O)NS(=O)(=O)N(C)C)c1
CC(C)c1ccc(C(C)C)c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCCOCC2)c1
CC(C)c1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCOCC1)C(F)(F)F
Cc1ccc(C)c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCCOCC2)c1
CN(C)S(=O)(=O)NC(=O)c1coc(Nc2cc(ncc2C)C(F)(F)F)n1
Cc1cnc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCOCC1)C(F)(F)F
COC1COCCN(C1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CC(F)(F)C1)C(F)(F)F
CC1CCN1S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CN(C)C(=O)[C@@H]1CCCN1S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1 |r|
CN(C)C(=O)[C@H]1CCCN1S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1 |r|
CC(C)c1ccc(C)c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCOCC2C)c1
CCC1COCCN1S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(C)C)n1
CN(C)S(=O)(=O)NC(=O)c1csc(Nc2c3CCCc3ccc2C)n1
Cc1ccc2CCCc2c1Nc1nc(cs1)C(=O)NS(=O)(=O)N1CCOCC1
Cc1ccc2CCCc2c1Nc1nc(cs1)C(=O)NS(=O)(=O)N1CCCOCC1
CN(C)S(=O)(=O)NC(=O)c1coc(Nc2nc(ccc2C)C(F)(F)F)n1
Cc1ccc(nc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCOCC1)C(F)(F)F
CC(C)c1nn(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N(C)C)C(C)C
CC(C)c1nn(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCOCC1)C(C)C
COCC1CN(CCCO1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CC1COCCN(C1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CN1CCN(CCC1=O)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CN(C)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C2(CC2)C#N)n1
CN1C(=O)CCC11CCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CC(CC#N)c1ccc(C)c(Nc2nc(co2)C(=O)NS(=O)(=O)N(C)C)c1
Cc1ccc2CCCc2c1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCOCC1
CC(C)c1ccc(C)c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCOCC2(C)C)c1
CN(C)S(=O)(=O)N1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CCCS(=O)(=O)N1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
COC(=O)N1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CCC(=O)N1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCN(CC1)S(=O)(=O)C1CC1)C(F)(F)F
Cc1ncc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCOCC1)C(F)(F)F
CC(C)c1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N(C)C)C(F)F
CC(C)c1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCOCC1)C(F)F
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCOCC1)C1(CC1)C#N
CN(CC#N)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCC(CC1)C#N)C(F)(F)F
CN(C)C(=O)CN(C)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CC(C)(C)c1ccc(c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCCOCC2)c1)C(C)(C)C
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCOCC1)C(C)(C)C
Cc1ccc(C)c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCCOCC2)c1C
Cc1cccc(C)c1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCOCC1
CC(C)c1cn(nc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCOCC1)C(C)C
CC(C)c1cn(nc1Nc1nc(co1)C(=O)NS(=O)(=O)N(C)C)C(C)C
CC(C)c1ccc2CCCc2c1Nc1nc(co1)C(=O)NS(=O)(=O)N(C)C
CC(C)c1ccc2CCCc2c1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCOCC1
COCC1CN(CCO1)S(=O)(=O)NC(=O)c1coc(Nc2c3CCCc3ccc2C(C)C)n1
COC1COCCN(C1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C(C)C)C(F)(F)F)n1
CCS(=O)(=O)C1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C(C)C)C(F)(F)F)n1
CC(C)c1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCN(C)CC1)C(F)(F)F
CC(C)c1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCC1CO)C(F)(F)F
CC(C)c1ccc(nc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCOCC1)C(F)(F)F
CCCCS(=O)(=O)N1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCOCC(C1)C#N)C(F)(F)F
CC(C)CS(=O)(=O)N1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CCN(C)S(=O)(=O)N1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCN(CC1)S(=O)(=O)CCC(F)(F)F)C(F)(F)F
CN(Cc1ccccn1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CN(C)CCN(C)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(C)(C)C)n1
CN(Cc1cccnc1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CC(C)c1ccc(cc1Nc1ncc(o1)C(=O)NS(=O)(=O)N1CCCOCC1)C(F)(F)F
COc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCOCC1)C(F)(F)F
CC(C)N(C)S(=O)(=O)NC(=O)c1coc(Nc2nn(cc2C(C)C)C(C)C)n1
CC(C)c1cn(nc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCC1)C(C)C
Cc1ccc(Br)cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCOCC1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCC(CC1)C#N)C(F)(F)F
Cc1cc(C#N)c(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCOCC1)C(F)(F)F
CN(C)C(=O)C1COCCN(C1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCCCC1)C(F)(F)F
CCC(=O)N(C)C1COCCN(C1)S(=O)(=O)NC(=O)c1coc(Nc2ccccc2)n1
CC(C)n1cc(C)c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCCOCC2)n1
COC1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCC(=O)CC1)C(F)(F)F
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCC(CC#N)CC1)C(F)(F)F
COCC1COCCN(C1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
Cc1cn(CC(F)(F)F)nc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCOCC1
Cc1cn(nc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCOCC1)C1CCCC1
CCCN1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CCCN1CCCN(CC1=O)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCC(O)CC1)C(F)(F)F
CN(C)C(=O)C1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
COC1CCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
COC1CCCN(C1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CCCS(=O)(=O)N1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cn(nc2C(C)C)C(C)C)n1
CCCCS(=O)(=O)N1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cn(nc2C(C)C)C(C)C)n1
CN(CCNC(C)=O)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CN(Cc1ccccc1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
COCCN(CCOC)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CN(C1CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCCC11CC1)C(F)(F)F
CC(C)c1ccc(C)c(Nc2nc(co2)C(=O)NS(=O)(=O)N(C)Cc2ccccn2)c1
CCC(CC)n1cc(C)c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCCOCC2)n1
CC(C)n1cc(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCCOCC2)c(n1)C(F)(F)F
CC(C)c1nn(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCN(CC1)S(=O)(=O)CC(C)(C)C)C(C)C
CC1CCCCN1S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CN(C)C1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CC1CCCN1S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CC(C)c1ccc(OC(F)(F)F)c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCCOCC2)c1
CC(C)c1ccc(c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCCOCC2)c1)C(F)(F)F
CCCCS(=O)(=O)N1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2nn(cc2C(C)C)C(C)C)n1
CC(n1cc(C)c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCCOCC2)n1)C(F)(F)F
COCC(C)(C)n1cc(C)c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCCOCC2)n1
CCCCS(=O)(=O)N1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2nn(cc2C)C(C)C)n1
CCCCC(=O)N1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCN(CC1)c1ncccn1)C(F)(F)F
CC(C)c1cn(nc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCOCCC1C)C(C)C
COC1COCCN(C1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(C)(F)F)n1
CC(C)c1ccnc(n1)N1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCCC1C(F)F)C(F)(F)F
Cc1cn(nc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCOCC1)C1CCC1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCOCC(F)(F)C1)C(F)(F)F
CC(C)c1nn(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCC(CC1)C#N)C(C)C
CC(C)n1cc(C)c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCCC(CC2)C#N)n1
CC(C)n1cc(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCCOCC2)c(n1)C(C)(C)C
CC(C)n1cc(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCCOCC2)c(n1)C1CC1
CC(C)n1cc(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCCOCC2)c(n1)C1CCC1
CCCCS(=O)(=O)N1CCN(CC(F)C1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCN(CC(F)C1)S(=O)(=O)CCCF)C(F)(F)F
COC1CCN(C1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CCC(C)n1cc(C)c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCCOCC2)n1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1C[C@H]2COC[C@@H]2C1)C(F)(F)F |r|
CC(C)c1cc(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCCOCC2)n(n1)C(C)C
CCCCS(=O)(=O)N1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(C)ccc2C)n1
CCCCS(=O)(=O)N1CCN(CC(C1)OC)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
COC1CN(CCN(C1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1)S(=O)(=O)CCCF
CN(CC1CCCCC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CC(C)N(Cc1ccccc1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CN(CC1CCCC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
COc1ccnc(n1)N1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Cc2cc(ccc2C)C(F)(F)F)n1
Cc1ccnc(n1)N1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CC(C)n1cc(C)c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCOCC(F)(F)C2)n1
Cc1cc(F)c(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCOCC1)C(F)(F)F
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCN(CC1)c1ccncn1)C(F)(F)F
CCCC(=O)N1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCN(CC1)C(=O)C1CCOC1)C(F)(F)F
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCc2nncn2CC1)C(F)(F)F
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCN(CC1)S(=O)(=O)C1CCOC1)C(F)(F)F
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCC(C1)C#N)C(F)(F)F
CCCS(=O)(=O)N1CCN(CC(F)C1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CCCC(=O)N1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C(C)C)C(F)F)n1
CCCS(=O)(=O)N1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C(C)C)C(F)F)n1
CCCCS(=O)(=O)N1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C(C)C)C(F)F)n1
CC(C)c1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCN(CC1)S(=O)(=O)C1CCOC1)C(F)F
CC(C)c1nn(C(C)C)c(C)c1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCOCC1
CCCS(=O)(=O)N1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(C)ccc2C)n1
Cc1ccc(C)c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCCN(CC2)S(=O)(=O)C2CC2)c1
CC1CN(CCCO1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CC1COCCCN1S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CN(C1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1)C(C)=O
CCCC1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCC(F)(F)CC1)C(F)(F)F
COCCCN(C)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CN(Cc1cnccn1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CN(Cc1cnn(C)c1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCS(=O)(=O)CC1)C(F)(F)F
CCC1(CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1)C#N
CCS(=O)(=O)N1CCCN(C(C)C1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CCS(=O)(=O)N1CCCN(CC1C)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
Cc1nn(C(F)F)c(C)c1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCOCC1
COC1COCCN(C1)S(=O)(=O)NC(=O)c1coc(Nc2cc(c(F)cc2C)C(F)(F)F)n1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCN(CC1)c1cnccn1)C(F)(F)F
CCN(C)C(=O)C1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CCCCS(=O)(=O)N1CCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CCCCC1(CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1)C#N
COCCC1(CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1)C#N
CCCS(=O)(=O)N1CCN(CC(C1)OC)S(=O)(=O)NC(=O)c1coc(Nc2cc(C)ccc2C)n1
CCS(=O)(=O)N1CCN(CC(C1)OC)S(=O)(=O)NC(=O)c1coc(Nc2cc(C)ccc2C)n1
C\C=C\C(C)C(=O)C1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCn2nccc2C1)C(F)(F)F
CCC(=O)N(C)C1CCCN(C1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CCCS(=O)(=O)N1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(CC)ccc2C)n1
CCCS(=O)(=O)N1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(C)ccc2CC)n1
CCCS(=O)(=O)N1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(CC)ccc2CC)n1
CN(C)C(=O)C1(C)CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CN(C)C(=O)C1(CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1)C#N
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCC(CC1)(C#N)C(=O)N1CCCC1)C(F)(F)F
CC1CCN(CCO1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CN(C)C(=O)C1CCN(CCO1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCOC(CC1)C#N)C(F)(F)F
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCN(CC1)c1ncccn1)C(F)(F)F
CN(C)S(=O)(=O)N1CCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CC(C)S(=O)(=O)N1CCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
COCCN(Cc1ccccc1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CCCS(=O)(=O)N1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2ccccc2C)n1
CCCS(=O)(=O)N1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)F)n1
CCCS(=O)(=O)N1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cccc3ocnc23)n1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCOC(CO)CC1)C(F)(F)F
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCC(CC1)n1cccn1)C(F)(F)F
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCN(CC1)c1ccccc1)C(F)(F)F
Cc1ccc(C)c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCCN(CC2)c2ncccn2)c1
CN(C)S(=O)(=O)C1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
COCN1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CN(CCn1cccn1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CN(CCS(C)(=O)=O)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCn2nccc12)C(F)(F)F
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCC(CC1)c1ccccc1)C(F)(F)F
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCC(C1)c1ccccc1)C(F)(F)F
Cc1noc(n1)C1(C)CCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
Cc1nnc(o1)C1(C)CCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CN(CCc1ccccn1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CCCS(=O)(=O)N1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(C)cc(C)c2C)n1
CCCS(=O)(=O)N1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(C)c(C)cc2C)n1
CCCS(=O)(=O)N1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(Cl)ccc2C)n1
CCCS(=O)(=O)N1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(Br)ccc2C)n1
CN(C)S(=O)(=O)N1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(C)ccc2C)n1
COC1COCCN(C1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(C)C)n1
COCC1CCN(CCO1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(C)C)n1
COCC(C)CN(C)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
Cc1cc(C)n(n1)C1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
Cc1cnn(c1)C1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
COCC1CCN(CCO1)S(=O)(=O)NC(=O)c1coc(Nc2cc(C)ccc2C)n1
Cc1ccc(C)c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCCC(CC2)C#N)c1
CCOCC1CCN(CCO1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CCCS(=O)(=O)C1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2nn(cc2C)C(C)C)n1
COC[C@@H]1CCCN1S(=O)(=O)NC(=O)c1coc(Nc2cc(C)ccc2C)n1 |r|
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCOCC(C1)n1cccn1)C(F)(F)F
CCOCC1CCN(CCO1)S(=O)(=O)NC(=O)c1coc(Nc2cc(C)ccc2C)n1
COCC1CCN(C1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CC(C)c1ccc(C)cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCOCC1
COCC1CCN(CCO1)S(=O)(=O)NC(=O)c1coc(Nc2cc(C)ccc2C(C)C)n1
COC1COCCN(C1)S(=O)(=O)NC(=O)c1coc(Nc2cc(C)ccc2C(C)C)n1
CCCS(=O)(=O)C1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(C)ccc2C(C)C)n1
C[C@H]1CN(CCCC1c1ncccn1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1 |r|
C[C@@H]1CN(CCCN1c1ncccn1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1 |r|
CCOC[C@@H]1CCCN1S(=O)(=O)NC(=O)c1coc(Nc2cc(C)ccc2C)n1 |r|
CCCS(=O)(=O)C1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2nc(ccc2C(C)C)C(F)(F)F)n1
CCCS(=O)(=O)C1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C(C)C)C(F)(F)F)n1
CC(C)S(=O)(=O)C1CCCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CCOC1COCCN(C1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CCOC1COCCN(C1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(C)C)n1
COC[C@@H]1CCCN1S(=O)(=O)NC(=O)c1coc(Nc2cc(C)ccc2C(C)C)n1 |r|
CCCOCC1CCN(CCO1)S(=O)(=O)NC(=O)c1coc(Nc2cc(C)ccc2C)n1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCOC(COC(F)F)CC1)C(F)(F)F
CCOCC1CCN(CCO1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(C)C)n1
CC(C)c1ccc(C)c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCOC(COC(F)F)CC2)c1
COCC1CCN(CCO1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)F)n1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCOC(COC(F)F)CC1)C(F)F
COc1ccc(C(C)C)c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCCOCC2)c1
Cc1cc(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCCOCC2)c(C)cc1Cl
COC1COCCN(C1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)F)n1
CCOCC1CCN(CCO1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)F)n1
CCOCC1CCN(CCO1)S(=O)(=O)NC(=O)c1coc(Nc2nn(cc2C)C(C)C)n1
CC(C)c1cc(F)c(C)cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCOCC1
CCOCC1CCN(CCO1)S(=O)(=O)NC(=O)c1coc(Nc2cc(C)c(F)cc2C(C)C)n1
CC(C)c1cc(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCCOCC2)c(C)cc1F
CCOCC1CCN(CCO1)S(=O)(=O)NC(=O)c1coc(Nc2cc(C(C)C)c(F)cc2C)n1
CN(C)C(=O)CCN(C)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
Cc1cc(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCCOCC2)c(C)cc1F
CCOCC1CCN(CCO1)S(=O)(=O)NC(=O)c1coc(Nc2cc(C)c(F)cc2C)n1
CC(C)c1ccc(C)c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCOC(CN(C)C)CC2)c1
Cc1ccc(C)c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCOC(COCC3CCC3)CC2)c1
COC1COCCN(C1)S(=O)(=O)NC(=O)c1coc(Nc2cc(C(C)C)c(F)cc2C)n1
CCOCC1CCN(CCO1)S(=O)(=O)NC(=O)c1coc(Nc2nn(cc2C(C)C)C(C)C)n1
COCCOCC1CCN(CCO1)S(=O)(=O)NC(=O)c1coc(Nc2cc(C)ccc2C)n1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCOCC1c1ccccc1)C(F)(F)F
COC[C@@H]1CCN(CCO1)S(=O)(=O)NC(=O)c1coc(Nc2cc(C)c(F)cc2C)n1 |r|
CC(C)c1cc(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCOC(CO)CC2)c(C)cc1F
Cc1ccc(C)c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCOC(CC#N)CC2)c1
CC(C)c1cc(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCOCC(O)C2)c(C)cc1F
CC(C)c1cc(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCOCC(C)(O)C2)c(C)cc1F
CCOCC1CCN(CCO1)S(=O)(=O)NC(=O)c1coc(Nc2cc(OC)c(F)cc2C)n1
Cc1cc(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCOC(COCC(C)(C)O)CC2)c(C)cc1F
COC[C@H]1CCN(CCO1)S(=O)(=O)NC(=O)c1coc(Nc2cc(C)c(F)cc2C)n1 |r|
Cc1cc(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCOC(CC2)C(C)(C)O)c(C)cc1F
CC(C)OCC1CCN(CCO1)S(=O)(=O)NC(=O)c1coc(Nc2cc(C)c(F)cc2C)n1
CC(C)S(=O)(=O)CC1CCN(CCO1)S(=O)(=O)NC(=O)c1coc(Nc2cc(C)c(F)cc2C)n1
COCCOC[C@@H]1CCN(CCO1)S(=O)(=O)NC(=O)c1coc(Nc2cc(C)c(F)cc2C)n1 |r|
CCOC[C@H]1OCCN(C[C@@H]1OC)S(=O)(=O)NC(=O)c1coc(Nc2cc(C)c(F)cc2C)n1 |r|
CCOC[C@@H]1OCCN(C[C@H]1OC)S(=O)(=O)NC(=O)c1coc(Nc2cc(C)c(F)cc2C)n1 |r|
OC1CCN(C1)S(=O)(=O)NC(=O)c1coc(Nc2c3CCCc3c(Cl)c3CCCc23)n1
Clc1c2CCCc2c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCS(=O)(=O)CC2)c2CCCc12
CS(=O)(=O)C1CCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2c3CCCc3c(Cl)c3CCCc23)n1
C[C@H]1CCCN1S(=O)(=O)NC(=O)c1coc(Nc2c3CCCc3c(Cl)c3CCCc23)n1 |r|
C[C@@H]1CCCN1S(=O)(=O)NC(=O)c1coc(Nc2c3CCCc3c(Cl)c3CCCc23)n1 |r|
Clc1c2CCCc2c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCCn3nccc23)c2CCCc12
CS(=O)(=O)C1CCN(C1)S(=O)(=O)NC(=O)c1coc(Nc2c3CCCc3c(Cl)c3CCCc23)n1
FC1(F)CCN(C1)S(=O)(=O)NC(=O)c1coc(Nc2c3CCCc3c(Cl)c3CCCc23)n1
Clc1c2CCCc2c(Nc2nc(co2)C(=O)NS(=O)(=O)N2C3CCC2CC3)c2CCCc12
Clc1c2CCCc2c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CC3CCC(C2)O3)c2CCCc12
OC1CCN(C1)S(=O)(=O)NC(=O)c1coc(Nc2c3CCCc3c(F)c3CCCc23)n1
Fc1c2CCCc2c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCOCC2)c2CCCc12
CC(=O)N1CCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2c3CCCc3c(Cl)c3CCCc23)n1
CS(=O)(=O)N1CCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2c3CCCc3c(Cl)c3CCCc23)n1
Clc1c2CCCc2c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CC3CC2CO3)c2CCCc12
Clc1c2CCCc2c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCOC3(COC3)C2)c2CCCc12
CS(=O)(=O)C1CCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2c3CCCc3c(F)c3CCCc23)n1
Fc1c2CCCc2c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CC3CCC(C2)O3)c2CCCc12
Fc1c2CCCc2c(Nc2nc(co2)C(=O)NS(=O)(=O)N2C[C@@H]3COC[C@@H]3C2)c2CCCc12 |r|
Clc1c2CCCc2c(Nc2nc(co2)C(=O)NS(=O)(=O)N2C[C@@H]3COC[C@@H]3C2)c2CCCc12 |r|
CC(=O)NC1CCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2c3CCCc3c(F)c3CCCc23)n1
CN(C)C(=O)C1CCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2c3CCCc3c(F)c3CCCc23)n1
CN1CCN(CC1=O)S(=O)(=O)NC(=O)c1coc(Nc2c3CCCc3c(F)c3CCCc23)n1
Clc1c2CCCc2c(Nc2nc(co2)C(=O)NS(=O)(=O)N2CCC(=O)C2)c2CCCc12
CN(C)S(=O)(=O)C1CCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2c3CCCc3c(F)c3CCCc23)n1
CCOC(=O)c1c2CN(Cc2nn1C)S(=O)(=O)NC(=O)c1coc(Nc2c3CCCc3c(F)c3CCCc23)n1
CN(C)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
CN(C)S(=O)(=O)NC(=O)c1coc(Nc2c3CCCc3ccc2C)n1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCOCC1)C(F)(F)F
COC(=O)CC1COCCN1S(=O)(=O)NC(=O)c1coc(Nc2c3CCCc3c(Cl)c3CCCc23)n1
COC(=O)C1COCCN1S(=O)(=O)NC(=O)c1coc(Nc2c3CCCc3c(Cl)c3CCCc23)n1
CN(C)C1CCN(C1)S(=O)(=O)NC(=O)c1coc(Nc2c3CCCc3c(F)c3CCCc23)n1
CN(C)S(=O)(=O)C1CCN(CC1)S(=O)(=O)NC(=O)c1coc(Nc2cc(ccc2C)C(F)(F)F)n1
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CCCC1)C(F)(F)F
Cc1ccc(cc1Nc1nc(co1)C(=O)NS(=O)(=O)N1CC2CCC(C1)O2)C(F)(F)F
Clc1ccccc1-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
O=c1[nH]c(nc2nn(cc12)-c1ccccc1)N1CCCC1
Cc1ccccc1-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
CN(C)c1nc2nn(cc2c(=O)[nH]1)-c1ccccc1Cl
Cc1ccccc1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
Cc1ccc(cc1-n1cc2c(n1)nc([nH]c2=O)N1CCCC1)C(F)(F)F
COc1ccccc1CN(C)c1nc2nn(cc2c(=O)[nH]1)-c1ccccc1C
FC(F)(F)c1ccccc1-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
FC(F)(F)Oc1ccccc1-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
Fc1cccc(F)c1-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
Cc1cccc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
Cc1ccccc1-n1cc2c(n1)nc([nH]c2=O)N1CCC(F)(F)C1
COc1nc(nc2nn(cc12)-c1ccccc1C)N1CCCC1
Cc1ccccc1-n1cc2c(n1)nc(N1CCCC1)n(C)c2=O
Cc1ccccc1-n1cc2c(n1)nc([nH]c2=O)N1CCCCC1
Cc1ccccc1-n1cc2c(n1)nc([nH]c2=O)N1CCC1
CC1COCCN1c1nc2nn(cc2c(=O)[nH]1)-c1ccccc1C
CCCN(C)c1nc2nn(cc2c(=O)[nH]1)-c1ccccc1C
CCCNc1nc2nn(cc2c(=O)[nH]1)-c1ccccc1C
CN(C)c1nc2nn(cc2c(=O)[nH]1)-c1ccccc1C
Cc1ccccc1-n1cc2c(n1)nc([nH]c2=O)N1CCC(O)C1
Cc1ccccc1-n1cc2c(n1)nc([nH]c2=O)N1CCCCCC1
CC(C)N(C)c1nc2nn(cc2c(=O)[nH]1)-c1ccccc1C
Cc1ccccc1-n1cc2c(n1)nc(Nc1ccccc1)[nH]c2=O
FC(F)(F)c1ccccc1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
Cc1ccccc1-n1cc2c(n1)nc([nH]c2=O)N1CCC(C1)C#N
Cc1ccccc1-n1cc2c(n1)nc([nH]c2=O)N1CCC(C1)c1ccccc1
CCOC1CCN(C1)c1nc2nn(cc2c(=O)[nH]1)-c1ccccc1C
Clc1cccc(Cl)c1-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
CC(C)c1ccccc1-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
Fc1ccc(c(Cl)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
COC1CN(C1)c1nc2nn(cc2c(=O)[nH]1)-c1ccccc1C
Cc1ccccc1-n1cc2c(n1)nc([nH]c2=O)N1CC(F)(F)C1
CC(C)CNc1nc2nn(cc2c(=O)[nH]1)-c1ccccc1C
CNc1nc2nn(cc2c(=O)[nH]1)-c1ccccc1C
Cc1ccccc1-n1cc2c(n1)nc([nH]c2=O)N1CCC(C)(O)C1
Cc1ccccc1-n1cc2c(n1)nc([nH]c2=O)N1CCC1Cc1ccccc1
Cc1ccccc1-n1cc2c(n1)nc([nH]c2=O)N1CCC1(C)C
Cc1ccc(cc1)-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
COC[C@H]1CCCN1c1nc2nn(cc2c(=O)[nH]1)-c1ccccc1C |r|
COC[C@@H]1CCCN1c1nc2nn(cc2c(=O)[nH]1)-c1ccccc1C |r|
Cc1cccc(c1)-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
Cc1ccc(c(C)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
Cc1ccc(C)c(c1)-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
Cc1cccc(c1C)-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
CCOC1CCN(C1)c1nc2nn(cc2c(=O)[nH]1)-c1c(C)cccc1C
FC(F)(F)c1ccc(cc1)-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
COC1CN(C1)c1nc2nn(cc2c(=O)[nH]1)-c1c(C)cccc1C
Cc1cccc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CC(C1)OCC(F)(F)F
Cc1ccc(cc1C)-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
Cc1cccc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CC(C1)C(F)(F)F
COC1CCN(C1)c1nc2nn(cc2c(=O)[nH]1)-c1c(C)cccc1C
Cc1n(nc2nc([nH]c(=O)c12)N1CCCC1)-c1ccc(C)cc1C
COC1CCN(C1)c1nc2nn(cc2c(=O)[nH]1)-c1ccc(C)cc1C
CCOC1CCN(C1)c1nc2nn(cc2c(=O)[nH]1)-c1ccc(C)cc1C
Cc1ccc(c(C)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
COC1CN(C1)c1nc2nn(cc2c(=O)[nH]1)-c1ccc(C)cc1C
COCCNc1nc2nn(cc2c(=O)[nH]1)-c1ccc(C)cc1C
CCCCNc1nc2nn(cc2c(=O)[nH]1)-c1ccccc1C
Cc1cc(Br)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
Cc1cc(C)c(c(C)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
Cc1cc(C)cc(c1)-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
CNc1nc2nn(cc2c(=O)[nH]1)-c1ccc(C)cc1C
CN(C(C)=O)c1nc2nn(cc2c(=O)[nH]1)-c1ccc(C)cc1C
Cc1cc(ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCCC1)C1=CCCCC1 |t:26|
O=c1[nH]c(nc2nn(cc12)-c1cccc2ccccc12)N1CCCC1
Cc1cc(Br)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
COC1CCN(C1)c1nc2nn(cc2c(=O)[nH]1)-c1ccc(Br)cc1C
Cc1cc(ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCCC1)C#N
COCC1CN(CCO1)c1nc2nn(cc2c(=O)[nH]1)-c1ccc(Br)cc1C
CC(=O)N1CCN(CC1)c1nc2nn(cc2c(=O)[nH]1)-c1ccc(Br)cc1C
Cc1cc(Br)ccc1-n1cc2c(n1)nc(NCc1ccccc1)[nH]c2=O
Cc1cc(Br)ccc1-n1cc2c(n1)nc([nH]c2=O)N1Cc2ccccc2C1
Cc1cc(Br)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CC(F)(F)C1
Cc1cc(Br)cnc1-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
Cc1cc(Br)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCNC(=O)C1
Cc1cc(Br)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCS(=O)(=O)CC1
CNc1nc2nn(cc2c(=O)n1C)-c1ccc(C)cc1C
CC(=C)c1ccc(c(C)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
Cc1cc(ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCCC1)C1CC1
CC(C)c1ccc(c(C)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
CN1CCN(CC1)c1nc2nn(cc2c(=O)[nH]1)-c1ccc(C)cc1C
Cc1ccc(c(C)c1)-n1cc2c(n1)nc([nH]c2=O)N1CC(F)(F)C(F)(F)C1
FC(F)(F)c1ccc(c(Cl)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
Cc1ccc(c(Cl)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
Cc1cc(Br)ccc1-n1cc2c(n1)nc(N1CCOCC1)n(C)c2=O
Cc1cc(Br)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCC(C1)C#N
Cc1cc(Br)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCN(CC1)S(C)(=O)=O
Cc1cc(C)c(c(C)c1)-n1cc2c(n1)nc([nH]c2=O)N1CC(F)(F)C1
COC1CCN(C1)c1nc2nn(cc2c(=O)[nH]1)-c1c(C)cc(C)cc1C
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
Cc1cc(Cl)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
Cc1cc(C)c(c(C)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
Fc1cc(Cl)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
Cc1cc(ncc1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1)C(F)(F)F
Cc1cc(ncc1-n1cc2c(n1)nc([nH]c2=O)N1CC(F)(F)C1)C(F)(F)F
Cc1cc(C)c(c(C)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCCOCC1
Cc1cc(C)c(c(C)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCN(CC1)C(=O)OC(C)(C)C
Cc1cc(C)c(c(C)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCNCC1
Cc1cc(C)c(c(C)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCN(CC1)S(=O)(=O)C1CC1
OCc1cc(Br)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
Cc1cc(C)c(c(C)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCC(O)CC1
COC1CCN(CC1)c1nc2nn(cc2c(=O)[nH]1)-c1c(C)cc(C)cc1C
Cc1cc(C)c(c(C)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCCC(O)C1
COC1CCCN(C1)c1nc2nn(cc2c(=O)[nH]1)-c1c(C)cc(C)cc1C
CC1CCN(C1)c1nc2nn(cc2c(=O)[nH]1)-c1c(C)cc(C)cc1C
CNC(=O)C1CCN(C1)c1nc2nn(cc2c(=O)[nH]1)-c1c(C)cc(C)cc1C
CC(=O)NC1CCN(C1)c1nc2nn(cc2c(=O)[nH]1)-c1c(C)cc(C)cc1C
Cc1cc(C)c(c(C)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCC(C1)S(C)(=O)=O
CN(C)C1CCN(C1)c1nc2nn(cc2c(=O)[nH]1)-c1c(C)cc(C)cc1C
Cc1cc(C)c(c(C)c1)-n1cc2c(n1)nc([nH]c2=O)N1CC2C(C1)C2(F)F
Cc1cc(C)c(c(C)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCC(CO)CC1
Cc1cc(C)c(c(C)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCCC(CO)C1
Cc1cc(C)c(c(C)c1)-n1cc2c(n1)nc([nH]c2=O)N1CC2COCC2C1
Cc1cc(C)c(c(C)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCC2(COC2)CC1
Cc1cc(ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCCC1)C#C
CCc1ccc(c(C)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
Cc1nc(ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1)C(F)(F)F
Cc1cc(cnc1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1)C(F)(F)F
Cc1cc(cnc1-n1cc2c(n1)nc([nH]c2=O)N1CC(F)(F)C1)C(F)(F)F
Cc1cc(cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1)C1CC1
Clc1ccc(c(Cl)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
FC(F)(F)c1ccc(c(Cl)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
FC(F)(F)c1ccc(c(Cl)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCCOCC1
CC(O)c1cc(Br)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
CC(=O)c1cc(Br)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
CC(C)(C)OC(=O)N1CCCN(CC1)c1nc2nn(cc2c(=O)[nH]1)-c1ccc(cc1Cl)C(F)(F)F
FC(F)(F)c1ccc(c(Cl)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCCNCC1
CC(=O)N1CCCN(CC1)c1nc2nn(cc2c(=O)[nH]1)-c1ccc(cc1Cl)C(F)(F)F
CS(=O)(=O)N1CCCN(CC1)c1nc2nn(cc2c(=O)[nH]1)-c1ccc(cc1Cl)C(F)(F)F
CC(C)Oc1nc(nc2nn(cc12)-c1ccc(Br)cc1C)N1CCOCC1
COc1nc(nc2nn(cc12)-c1ccc(Br)cc1C)N1CCN(CC1)S(C)(=O)=O
Cc1cc(Br)ccc1-n1cc2c(n1)nc(N1CCN(CC1)S(C)(=O)=O)n(C)c2=O
Cc1cc(Br)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCN(CC1)S(=O)(=O)C1CC1
Cc1cc(Br)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCN(CC1)C(=O)C1CC1
COCC(=O)N1CCN(CC1)c1nc2nn(cc2c(=O)[nH]1)-c1ccc(Br)cc1C
Cc1cc(Br)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCCOCC1
COCc1cc(Cl)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
COCc1cc(Cl)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCCOCC1
Cc1cc(Br)cc(Cl)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
Cc1cc(C)c(c(Cl)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
Cc1cc(Br)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCN(CC1)c1ncccn1
OC(C1CC1)c1cc(Br)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
Cc1n(nc2nc([nH]c(=O)c12)N1CCCC1)-c1ccc(cc1)C(F)(F)F
Cc1cc(Br)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCN(C2CC2)C(=O)C1
Cc1cc(Br)ccc1-n1cc2c(OCCO)nc(nc2n1)N1CCOCC1
COCCOc1nc(nc2nn(cc12)-c1ccc(Br)cc1C)N1CCOCC1
Cc1cc(Br)ccc1-n1cc2c(OCC3CC3)nc(nc2n1)N1CCOCC1
Cc1cc(Br)ccc1-n1cc2c(OCC#N)nc(nc2n1)N1CCOCC1
FC(F)(F)c1cnc(c(Cl)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
Cc1cc(Cl)cc(CO)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
Cc1cc(Br)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CC2CC1CO2
Cc1cc(Cl)cc(C=O)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
COCc1cc(Cl)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CC(F)(F)C1
Cc1cc(Cl)cc(C(O)C2CC2)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
Cc1cc(Br)ccc1-n1cc2c(n1)nc(N1CCOCC1)n(CCO)c2=O
Cc1cc(Cl)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
Cc1cc(Cl)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCCOCC1
Cc1cc(Cl)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
Cc1cc(Cl)cc(C(=O)C2CC2)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
Cc1cc(Cl)cc(C#N)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
Cc1cc(Br)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CC2CC(C1)O2
Cc1n(nc2nc([nH]c(=O)c12)N1CCCC1)-c1ccc(cc1Cl)C(F)(F)F
COc1ccc(c(C)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
Cc1cc(Br)ccc1-n1cc2c(n1)nc(N1CCOCC1)n(CC#N)c2=O
Cc1cc(Br)ccc1-n1cc2c(n1)nc(N1CCN(CC1)S(C)(=O)=O)n(CC#N)c2=O
Cc1cc(Br)cc(c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1)C(F)(F)F
Cc1cc(cc(c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1)C(F)(F)F)C1CC1
FC(F)(F)c1cc(Cl)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
FC(F)(F)c1cc(ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1)C1CC1
OCC1CCCN1c1nc2nn(cc2c(=O)[nH]1)-c1ccc(cc1Cl)C(F)(F)F
CC(C)(C)OC(=O)N1CC2CN(CC2C1)c1nc2nn(cc2c(=O)[nH]1)-c1ccc(cc1Cl)C(F)(F)F
OCCC1CN(C1)c1nc2nn(cc2c(=O)[nH]1)-c1ccc(cc1Cl)C(F)(F)F
FC1CN(C1)c1nc2nn(cc2c(=O)[nH]1)-c1ccc(cc1Cl)C(F)(F)F
OC1CN(C1)c1nc2nn(cc2c(=O)[nH]1)-c1ccc(cc1Cl)C(F)(F)F
OC1CC2(C1)CN(C2)c1nc2nn(cc2c(=O)[nH]1)-c1ccc(cc1Cl)C(F)(F)F
FC(F)(F)c1ccc(c(Cl)c1)-n1cc2c(n1)nc(NC1CCOCC1)[nH]c2=O
CNc1nc2nn(cc2c(=O)[nH]1)-c1c(C)cc(Br)cc1C
FC(F)(F)c1ccc(c(Cl)c1)-n1cc2c(n1)nc([nH]c2=O)N1CC2CNCC2C1
CC(=O)N1CC2CN(CC2C1)c1nc2nn(cc2c(=O)[nH]1)-c1ccc(cc1Cl)C(F)(F)F
CC(C)c1cc(Cl)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
Fc1cc(cc(Cl)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1)C(F)(F)F
FC(F)(F)c1cc(Cl)c(c(OCC2CC2)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
Cc1cc(Br)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CC2(COC2)C1
COC[C@@H]1CCN(CCO1)c1nc2nn(cc2c(=O)[nH]1)-c1ccc(Br)cc1C |r|
COC[C@H]1CCN(CCO1)c1nc2nn(cc2c(=O)[nH]1)-c1ccc(Br)cc1C |r|
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCC(C1)C(C)(C)O
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1C[C@@H]2C[C@H]1CO2 |r|
Brc1ccc(c(c1)C1CC1)-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1C[C@H]2C[C@@H]1CO2 |r|
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CC(F)C1
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CC2(CC(O)C2)C1
Cc1cc(OC(F)(F)F)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
FC(F)(F)c1cnc(c(Br)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
Cc1cc(ncc1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1)C1CC1
COC1(C)CN(C1)c1nc2nn(cc2c(=O)[nH]1)-c1c(C)cc(Br)cc1C
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CC2(COC2)C1
COc1cc(Cl)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
FC(F)(F)Oc1cc(Br)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
Cc1cc(cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1C[C@@H]2C[C@H]1CO2)C1CC1 |r|
FC(F)(F)Oc1cc(ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1)C1CC1
Cc1cc(cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1C[C@H]2C[C@@H]1CO2)C1CC1 |r|
O=c1[nH]c(nc2nn(cc12)-c1ccc(cc1C1CC1)C1CC1)N1CCOCC1
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CC2CC(C1)O2
COC1(C)CN(C1)c1nc2nn(cc2c(=O)n1C)-c1c(C)cc(Br)cc1C
C[C@@H]1COCCN1c1nc2nn(cc2c(=O)[nH]1)-c1c(C)cc(Br)cc1C |r|
C[C@H]1CN(CCO1)c1nc2nn(cc2c(=O)[nH]1)-c1c(C)cc(Br)cc1C |r|
C[C@@H]1CN(CCO1)c1nc2nn(cc2c(=O)[nH]1)-c1c(C)cc(Br)cc1C |r|
COC1COCCN(C1)c1nc2nn(cc2c(=O)[nH]1)-c1c(C)cc(Br)cc1C
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CC2CC1C2 |(2.88,2.83,;3.65,1.5,;5.2,1.5,;5.96,.13,;7.5,.13,;5.22,-1.2,;3.65,-1.2,;2.88,-2.53,;2.88,.16,;1.34,.16,;.42,1.42,;-1.04,.96,;-1.04,-.62,;.44,-1.11,;-2.39,-1.46,;-3.74,-.66,;-3.76,.86,;-2.44,1.68,;-2.44,3.22,;-5.07,-1.43,;-5.25,-2.98,;-6.75,-3.22,;-7.5,-1.93,;-6.48,-.82,;-6.08,-2.31,)|
FC(F)(F)c1cc(Cl)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CC2CC1CN2S(C)(=O)=O
COCC(=O)N1CC2CC1CN2c1nc2nn(cc2c(=O)[nH]1)-c1c(C)cc(Br)cc1C
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1C2CC1CN(C2)S(C)(=O)=O
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CC2CC(C1)N2S(C)(=O)=O
C[C@H]1COCCN1c1nc2nn(cc2c(=O)[nH]1)-c1c(C)cc(Br)cc1C |r|
C[C@H]1CN(C[C@@H](C)O1)c1nc2nn(cc2c(=O)[nH]1)-c1c(C)cc(Br)cc1C |r|
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOC2(CC2)C1
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc(NCC1CC1)[nH]c2=O
CNc1nc2nn(cc2c(=O)[nH]1)-c1c(C)cc(cc1C)C1CC1
Cc1cc(cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CC2CC(C1)O2)C1CC1
Cc1cccc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
COCC(=O)N1CC2CC1CN2c1nc2nn(cc2c(=O)[nH]1)-c1c(C)cc(cc1C)C1CC1
CC(C)c1cc(cnc1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1)C(F)(F)F
Cc1cc(cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1)C(F)(F)F
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1C2CCC1CC(F)(F)C2
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CC2CCC(C1)C2(F)F
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCC2CC12
FC(F)(F)c1cc(Br)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
Cc1cc(ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1)C1CC1
FC(F)c1cc(Br)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
FC(F)c1cc(ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1)C1CC1
CN1CCCC(C1)Nc1nc2nn(cc2c(=O)[nH]1)-c1c(C)cc(Br)cc1C
CN1CCN(CC1)c1nc2nn(cc2c(=O)[nH]1)-c1c(C)cc(Br)cc1C
CNc1nc2nn(cc2c(=O)n1C)-c1c(C)cc(Br)cc1C
CCC1COCCN1c1nc2nn(cc2c(=O)[nH]1)-c1c(C)cc(Br)cc1C
Cc1cc(cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1C[C@H]2C[C@@H]1CO2)C(F)(F)F |r|
Cc1cc(cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1C[C@@H]2C[C@H]1CO2)C(F)(F)F |r|
CC(C)CNc1nc2nn(cc2c(=O)[nH]1)-c1c(C)cc(Br)cc1C
COc1cc(C)c(c(C)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
Cc1cc(Br)cc(F)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
Cc1cc(cc(F)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1)C1CC1
Oc1cc(cc(Cl)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1)C(F)(F)F
C[C@@H]1COCCN1c1nc2nn(cc2c(=O)[nH]1)-c1ccc(Br)cc1C(F)(F)F |r|
FC(F)(F)c1cc(Br)ccc1-n1cc2c(n1)nc([nH]c2=O)N1C[C@H]2C[C@@H]1CO2 |r|
FC(F)(F)c1cc(Br)ccc1-n1cc2c(n1)nc([nH]c2=O)N1C[C@@H]2C[C@H]1CO2 |r|
C[C@@H]1COCCN1c1nc2nn(cc2c(=O)[nH]1)-c1ccc(cc1C(F)(F)F)C1CC1 |r|
FC(F)(F)c1cc(ccc1-n1cc2c(n1)nc([nH]c2=O)N1C[C@H]2C[C@@H]1CO2)C1CC1 |r|
FC(F)(F)c1cc(ccc1-n1cc2c(n1)nc([nH]c2=O)N1C[C@@H]2C[C@H]1CO2)C1CC1 |r|
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOC2(COC2)C1
Cc1cc(c(C)cc1Cl)-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc(NCC(F)(F)F)[nH]c2=O
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc(NCCF)[nH]c2=O
COCc1cc(Br)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
Cc1cc(cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1)C1CCC1
Nc1cc(cc(Cl)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1)C(F)(F)F
Fc1cc(Br)cc(c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1)C(F)(F)F
Fc1cc(cc(c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1)C(F)(F)F)C1CC1
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc(NC1COC1)[nH]c2=O
C[C@@H]1COCCN1c1nc2nn(cc2c(=O)[nH]1)-c1c(C)cc(cc1C)C1CC1 |r|
Cc1cc(cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1)C1(CC1)C(F)(F)F
Cc1cc(cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CC2CC(C1)O2)C(F)(F)F
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CC2CCC(C1)O2
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CC2COC(C2)C1
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
Cc1cc(cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCCC1)C(F)(F)F
Cc1c(Cl)ccc(c1C)-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCC(F)(F)C1
C[C@@H]1CCCN1c1nc2nn(cc2c(=O)[nH]1)-c1c(C)cc(Br)cc1C |r|
C[C@H]1CCCN1c1nc2nn(cc2c(=O)[nH]1)-c1c(C)cc(Br)cc1C |r|
Cc1cc(cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCCC1)C1CC1
Cc1cc(cc(Cl)c1-n1cc2c(n1)nc([nH]c2=O)N1C[C@H]2C[C@@H]1CO2)C1CC1 |r|
Cc1cc(cc(Cl)c1-n1cc2c(n1)nc([nH]c2=O)N1C[C@@H]2C[C@H]1CO2)C1CC1 |r|
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOC2CC12
C[C@@H]1CN(CCN1c1nc2nn(cc2c(=O)[nH]1)-c1c(C)cc(cc1C)C1CC1)C(C)=O |r|
CC(C)N(C)c1nc2nn(cc2c(=O)[nH]1)-c1c(C)cc(Br)cc1C
CCc1cc(C)c(c(C)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
Cc1cc(cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1)C(=C)C(F)(F)F
CC(c1cc(C)c(c(C)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1)C(F)(F)F
Cc1cc(cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CC2CCC(C1)O2)C(F)(F)F
Cc1cc(Br)cc(Cl)c1-n1cc2c(n1)nc([nH]c2=O)N1CC2CC(C1)O2
Cc1cc(cc(Cl)c1-n1cc2c(n1)nc([nH]c2=O)N1CC2CC(C1)O2)C1CC1
Cc1cc(OC(F)F)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
Cc1cc(cc(F)c1-n1cc2c(n1)nc([nH]c2=O)N1C[C@H]2C[C@@H]1CO2)C1CC1 |r|
Cc1cc(cc(F)c1-n1cc2c(n1)nc([nH]c2=O)N1C[C@@H]2C[C@H]1CO2)C1CC1 |r|
CC(C)c1cc(C)c(c(C)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
CCOc1cc(Br)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
CC(C)Oc1cc(Br)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
COc1cc(Br)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
Brc1ccc(c(OC2CCC2)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
CC(C)(C)c1ccc(c(Br)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
COc1ccc(c(Br)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCCO1
OC(C1CC1)c1cc(Br)ccc1-n1cc2c(n1)nc([nH]c2=O)N1C[C@H]2C[C@@H]1CO2 |r|
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc(N1CC3CC(C1)O3)n(C)c2=O
Cn1c(nc2nn(cc2c1=O)-c1ccc(Br)cc1C(F)(F)F)N1CC2CC(C1)O2
Cc1cc(cc(C)c1-n1cc2c(n1)nc(N1CC3CC(C1)O3)n(C)c2=O)C1CC1
Cn1c(nc2nn(cc2c1=O)-c1ccc(cc1C(F)(F)F)C1CC1)N1CC2CC(C1)O2
COC(C1CC1)c1cc(Br)ccc1-n1cc2c(n1)nc([nH]c2=O)N1C[C@H]2C[C@@H]1CO2 |r|
COC(C1CC1)c1cc(ccc1-n1cc2c(n1)nc([nH]c2=O)N1C[C@H]2C[C@@H]1CO2)C1CC1 |r|
CO[C@@H]1CCN(C1)c1nc2nn(cc2c(=O)[nH]1)-c1c(C)cc(Br)cc1C |r|
CO[C@@H]1CCN(C1)c1nc2nn(cc2c(=O)[nH]1)-c1c(C)cc(cc1C)C1CC1 |r|
CO[C@H]1CCN(C1)c1nc2nn(cc2c(=O)[nH]1)-c1c(C)cc(Br)cc1C |r|
CO[C@H]1CCN(C1)c1nc2nn(cc2c(=O)[nH]1)-c1c(C)cc(cc1C)C1CC1 |r|
Clc1ccc(c(CC2CC2)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
O=c1[nH]c(nc2nn(cc12)-c1ccc(cc1CC1CC1)C1CC1)N1CCOCC1
CC(C)Cc1ccccc1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCC(C1)C#N
Cc1cc(cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCC(C1)C#N)C1CC1
FC(F)Oc1ccc(c(c1)C(F)(F)F)-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1
Cc1cc(cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCCOCC1)C1CC1
Cc1cc(cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1)N1CCC1
Cc1cc(cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCC1)C1CC1
Cc1cc(cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1)C(F)F
Cc1cc(cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1C[C@H]2C[C@@H]1CO2)C(F)F |r|
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCCCO1
Cc1cc(cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCCCO1)C1CC1
CONc1nc2nn(cc2c(=O)[nH]1)-c1c(C)cc(Br)cc1C
COCCN(C)c1nc2nn(cc2c(=O)[nH]1)-c1c(C)cc(Br)cc1C
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCCCCO1
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCCO1
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCc2cccnc12
Cc1ccc(c(c1)-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1)C(F)(F)F
CC(C)n1nc(C)c(c1C)-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
Cc1nn(C2CCC2)c(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
COc1cc(C)c(c(C)c1)-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
CC(C)n1nc(c(c1C)-n1cc2c(n1)nc([nH]c2=O)N1CCCC1)C(F)(F)F
CCC(C)n1nc(C)c(c1C)-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
CONc1nc2nn(cc2c(=O)[nH]1)-c1c(C)cc(cc1C)C1CC1
Cc1cc(cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCCO1)C1CC1
Cc1nn(C2CCCC2)c(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCCC1
Cc1cc(cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCCO1)C(C)(F)F
Cc1cc(OC(F)F)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCCO1
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1=O
Cc1cc(OC(F)F)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1=O
FC(F)(F)c1cc(Br)ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCOCCO1
FC(F)(F)c1cc(ccc1-n1cc2c(n1)nc([nH]c2=O)N1CCOCCO1)C1CC1
Cc1cc(cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCCO1)C(F)(F)F
Cc1cc(CC(F)F)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCCO1
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc(NCCOCCO)[nH]c2=O
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N(CCO)CCO
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOC=C1 |c:26|
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOCC1O
Cc1cc(Br)cc(C)c1-n1cc2c(n1)nc([nH]c2=O)N1CCOC(O)C1
[#6]-[#8]-c1cc(ccn1)-c1c(-[#6])cc2-[#6]-[#6]-[#6]-c2c1-[#7]-[#6](=O)-[#7]S(=O)(=O)c1ccn(n1)-[#6]-1-[#6]\[#6](-[#6]-1)=[#6](/F)F
CC(C)(O)c1cc(co1)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
Cc1ccccc1-n1cc2c(=O)[nH]c(-c3ccn(C)n3)nc2n1
COc1cc(C)c(-n2cc3c(=O)[nH]c(-c4ccn(C)n4)nc3n2)c(C)c1
COc1cc(C)c(-n2cc3c(=O)[nH]c(-c4cnn(C)c4)nc3n2)c(C)c1
Cc1cc(C2CC2)cc(C)c1-n1cc2c(=O)[nH]c(-c3ccn(C)n3)nc2n1
Cc1cc(C2CC2)cc(C)c1-n1cc2c(=O)[nH]c(-c3ccnn3C)nc2n1
Cc1cn(C)nc1-c1nc2nn(-c3c(C)cc(C4CC4)cc3C)cc2c(=O)[nH]1
Cc1cc(Br)cc(C)c1-n1cc2c(=O)[nH]c(-c3ncoc3C)nc2n1
Cc1cc(C(F)(F)C(F)(F)F)cc(C)c1-n1cc2c(=O)[nH]c(-c3ccn(C)n3)nc2n1
Cc1cc(OC(F)F)cc(C)c1-n1cc2c(=O)[nH]c(-c3ccn(C)n3)nc2n1
Cc1cc(Br)cc(C)c1-n1cc2c(=O)[nH]c(-c3ccn(C)n3)nc2n1
Cc1cc(Br)cc(C)c1-n1cc2c(=O)[nH]c(-c3cnn(C)c3)nc2n1
Cc1cc(Br)cc(C)c1-n1cc2c(=O)[nH]c(-c3ccncn3)nc2n1
Cc1cc(C2CC2)cc(C)c1-n1cc2c(=O)[nH]c(-c3cc[nH]n3)nc2n1
Cc1nnc(-c2nc3nn(-c4c(C)cc(Br)cc4C)cc3c(=O)[nH]2)o1
Cc1cc(Br)cc(C)c1-n1cc2c(=O)[nH]c(-c3ccnnc3)nc2n1
COCCn1ccc(-c2nc3nn(-c4c(C)cc(Br)cc4C)cc3c(=O)[nH]2)n1
COCCn1nccc1-c1nc2nn(-c3c(C)cc(Br)cc3C)cc2c(=O)[nH]1
Cc1cc(C2CC2)cc(C)c1-n1cc2c(=O)[nH]c(-c3ccn(C(F)F)n3)nc2n1
Cc1cc(C2CC2)cc(C)c1-n1cc2c(=O)[nH]c(-c3ccn(C4COC4)n3)nc2n1
COCCn1ccc(-c2nc3nn(-c4c(C)cc(C5CC5)cc4C)cc3c(=O)[nH]2)n1
Cc1cc(Br)cc(C)c1-n1cc2c(=O)[nH]c(-c3cn(C)nn3)nc2n1
Cc1cc(Br)cc(C)c1-n1cc2c(=O)[nH]c(-c3cnccn3)nc2n1
Cc1cc(Br)cc(C)c1-n1cc2c(=O)[nH]c(-c3cccnn3)nc2n1
Cc1ncc(-c2nc3nn(-c4c(C)cc(Br)cc4C)cc3c(=O)[nH]2)o1
Cc1cc(-c2nc3nn(-c4c(C)cc(Br)cc4C)cc3c(=O)[nH]2)no1
Cc1cc(C2CC2)cc(C)c1-n1cc2c(=O)[nH]c(-c3cn(C)nn3)nc2n1
Cc1cc(OC(F)F)cc(C)c1-n1cc2c(=O)[nH]c(-c3cccnn3)nc2n1
Cc1cc(C2CC2)cc(C)c1-n1cc2c(=O)[nH]c(-c3ccnnc3)nc2n1
Cc1cc(C(F)(F)F)cc(C)c1-n1cc2c(=O)[nH]c(-c3ccn(C)n3)nc2n1
CCn1ccc(-c2nc3nn(-c4c(C)cc(Br)cc4C)cc3c(=O)[nH]2)n1
Cc1cc(Br)cc(C)c1-n1cc2c(=O)[nH]c(-c3cc(C(F)(F)F)ncn3)nc2n1
Cc1cc(Br)cc(C)c1-n1cc2c(=O)[nH]c(-c3ccnc(C(F)(F)F)n3)nc2n1
Cc1cc(C(F)(F)F)cc(C)c1-n1cc2c(=O)[nH]c(-c3ccncc3F)nc2n1
COc1nccc(-c2nc3nn(-c4c(C)cc(Br)cc4C)cc3c(=O)[nH]2)n1
Cc1cc(Br)cc(C)c1-n1cc2c(=O)[nH]c(-c3ccncc3F)nc2n1
Cc1cc(C2CC2)cc(C)c1-n1cc2c(=O)[nH]c(-c3ccncc3F)nc2n1
Cc1cc(Br)cc(C)c1-n1cc2c(=O)[nH]c(-c3nn(C)cc3F)nc2n1
Cc1cc(C2CC2)cc(C)c1-n1cc2c(=O)[nH]c(-c3nn(C)cc3F)nc2n1
Cc1cc(C2CC2)cc(C)c1-n1cc2c(=O)[nH]c(-c3cn(C)cn3)nc2n1
COCc1cc(C2CC2)cc(C)c1-n1cc2c(=O)[nH]c(-c3ccn(C)n3)nc2n1
Cc1cc(C(C)(F)F)cc(C)c1-n1cc2c(=O)[nH]c(-c3cn(C)cn3)nc2n1
Cc1cc(C(C)(F)F)cc(C)c1-n1cc2c(=O)[nH]c(-c3ccncn3)nc2n1
Cc1cc(C2CC2)cc(C)c1-n1cc2c(=O)[nH]c(-c3ccncn3)nc2n1
Cc1cccc(C)c1-n1cc2c(=O)[nH]c(-c3ccn(C)n3)nc2n1
Cc1cc(C2(F)CC2)cc(C)c1-n1cc2c(=O)[nH]c(-c3ccn(C)n3)nc2n1
Cc1cc(C2CC2)cc(C)c1-n1cc2c(=O)[nH]c(-c3cnn(C)c3)nc2n1
Cc1cc(I)cc(C)c1-n1cc2c(=O)[nH]c(-c3ccn(C)n3)nc2n1
Cc1cc(C2CC2)cc(CO)c1-n1cc2c(=O)[nH]c(-c3ccn(C)n3)nc2n1
Cc1csc(-c2nc3nn(-c4c(C)cc(C5CC5)cc4C)cc3c(=O)[nH]2)n1
Cc1cc(C2CC2)cc(C)c1-n1cc2c(=O)[nH]c(-c3cscn3)nc2n1
Cc1cc(C2CC2)cc(C)c1-n1cc2c(=O)[nH]c(-c3cnn4c3OCCC4)nc2n1
Cc1cc(C2CC2)cc(C)c1-n1cc2c(=O)[nH]c(-c3cc4n(n3)CCOC4)nc2n1
Cc1cc(C2CC2)cc(C)c1-n1cc2c(=O)[nH]c(-c3cc4n(n3)CCCO4)nc2n1
Cn1ccc(-c2nc3nn(-c4cc5c(cc4Cl)OCCC5)cc3c(=O)[nH]2)n1
Cc1cc(C2CC2)cc(C)c1-n1cc2c(=O)[nH]c(-c3cc4n(n3)CCC4)nc2n1
Cc1cc(C(C)(F)F)cc(C)c1-n1cc2c(=O)[nH]c(-c3cscn3)nc2n1
Cn1ccc(-c2nc3nn(-c4cc5c(cc4Cl)CCC5)cc3c(=O)[nH]2)n1
Cc1cc(C(C)(F)F)cc(C)c1-n1cc2c(=O)[nH]c(-c3nc[nH]n3)nc2n1
Cc1cc(C(F)(F)C(F)(F)F)cc(C)c1-n1cc2c(=O)[nH]c(-c3ncn(C)n3)nc2n1
CC1(CCN2CC(S(=O)(=O)NC(=O)Nc3c4c(cc5c3CCC5)CCC4)C2)N=N1
CS(=O)(=O)N1CCC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)CC1
CC(=O)N1CCC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)CC1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CN2CCC1CC2
CCN1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
CCN1CCC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)CC1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CCN(C(=O)C2CC2)CC1
CC(=O)N1CCC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)CC1
CCN1CCCC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
CCC(=O)N1CCC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)CC1
CC(C)C(=O)N1CCC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)CC1
COCC(=O)N1CCC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)CC1
COC(=O)N1CCC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)CC1
N#CCN1CCC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)CC1
CC(C)n1cc(S(=O)(=O)NC(=O)Nc2c(-c3ccnc(C#N)c3)ccc3c2CCC3)ncc1=O
Cn1cc(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)c(=O)n(C)c1=O
CCCCCCn1cc(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)c(=O)[nH]c1=O
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CN(C2CCC2)C1
CCCN1CCC(S(=O)(=O)CC(=O)Nc2c3c(cc4c2CCC4)CCC3)CC1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CCN(C2COC2)CC1
CN(C)C(=O)CN1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CCN(CCF)CC1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CCN(C2CC2)CC1
CCN1CC(N2CCC(S(=O)(=O)NC(=O)Nc3c4c(cc5c3CCC5)CCC4)CC2)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CCN(C(=O)C2CCC2)CC1
CCNC(=O)N1CCC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)CC1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CCCN(C(=O)NC2CCC2)C1
CNC(=O)N1CCC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)CC1
CS(=O)(=O)N1CCC(S(=O)(=O)CC(=O)Nc2c3c(cc4c2CCC4)CCC3)CC1
CCNC(=O)N1CCC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
CC(C)N1CCCC(S(=O)(=O)CC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
CCC(=O)N1CCCC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
CC(C)NC(=O)N1CCCC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CCCN(CCF)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CNc2ccccc2C1
CC(C)N1CCCC(S(=O)(=O)CC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
CCN1CCC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
CC(=O)N1CCC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
O=C(CS(=O)(=O)C1CCN(C2CC2)C1)Nc1c2c(cc3c1CCC3)CCC2
CN(C)C(=O)N1CCC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
CC(C)N1CCC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CNC1
O=C(CS(=O)(=O)C1CCN(C2CC2)C1)Nc1c2c(cc3c1CCC3)CCC2
CCN1CCC(N2CCC(S(=O)(=O)NC(=O)Nc3c4c(cc5c3CCC5)CCC4)C2)CC1
CC(C)N1[C@@H]2CC[C@H]1C[C@@H](S(=O)(=O)NC(=O)Nc1c3c(cc4c1CCC4)CCC3)C2
CC(C)N1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
CC(C)N1CCC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)CC1
CCN1CCC(N2CCC(S(=O)(=O)NC(=O)Nc3c4c(cc5c3CCC5)CCC4)CC2)CC1
O=C(CS(=O)(=O)C1CCN(C2CC2)C1)Nc1c2c(cc3c1CCC3)CCC2
CCN1CC2(CC(S(=O)(=O)NC(=O)Nc3c4c(cc5c3CCC5)CCC4)C2)C1
CC(C)N1CC(N2CCC(S(=O)(=O)CC(=O)Nc3c4c(cc5c3CCC5)CCC4)C2)C1
CCN1[C@@H]2CC[C@H]1C[C@@H](S(=O)(=O)NC(=O)Nc1c3c(cc4c1CCC4)CCC3)C2
CCN1CC(S(=O)(=O)CC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CCN(C(=O)C(F)(F)F)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CCNC1
CC(=O)N1CCCC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CCCN(CC2CC2)C1
N#CCN1CCCC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
C#CCN1CCCC(S(=O)(=O)CC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
CN1CCCC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
CN(C)C(=O)N1CCC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)CC1
CC(C)N1CC(N2CCC(S(=O)(=O)NC(=O)Nc3c4c(cc5c3CCC5)CCC4)CC2)C1
CC(C)N1CC2(CC(S(=O)(=O)NC(=O)Nc3c4c(cc5c3CCC5)CCC4)C2)C1
CN1CC2(CC(S(=O)(=O)NC(=O)Nc3c4c(cc5c3CCC5)CCC4)C2)C1
CCC(CC)N1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
CCN1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)Cc2ccccc21
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CCN(CC(F)(F)F)CC1
CC(C)N1CCC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1=O
CC(C)N1[C@@H]2CC[C@H]1C[C@H](S(=O)(=O)NC(=O)Nc1c3c(cc4c1CCC4)CCC3)C2
CCN1[C@@H]2CC[C@H]1C[C@H](S(=O)(=O)NC(=O)Nc1c3c(cc4c1CCC4)CCC3)C2
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CN(C(=O)OCc2ccccc2)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CN(Cc2ccccc2)C1
CCN1CCC(N2CC(S(=O)(=O)NC(=O)Nc3c4c(cc5c3CCC5)CCC4)C2)CC1
CC(=O)N1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CN(C2CCOCC2)C1
CCCN1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
CC(C)(C)OC(=O)N1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
COC(=O)CN1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
CC(=O)N1CC(N2CCC(S(=O)(=O)NC(=O)Nc3c4c(cc5c3CCC5)CCC4)CC2)C1
CN1CC(N2CCC(S(=O)(=O)NC(=O)Nc3c4c(cc5c3CCC5)CCC4)CC2)C1
CCC(CC)N1CCC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
CCC(C)N1CCC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
CCCCN1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
CC(C)(O)CN1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CN(C2CC2)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CN(C(CF)CF)C1
N#CCN1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
COCCN1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CN(CC2CCCCC2)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CN(Cc2cccnc2)C1
CN(C)C(=O)CN1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CN(CCCl)C1
CC(C)(C)N1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CN(CC2CC2)C1
[N-]=[N+]=NCCN1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CN(CC(F)(F)F)C1
CC(C)CN1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CN(C2CCCCC2)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CN(C2CCCC2)C1
CC(=N)N1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
CCN1CCC(S(=O)(=O)NC(=O)Nc2c(-c3ccnc(OC)c3)cc(F)cc2C(C)C)CC1
CN(C)CCN1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CN(Cc2ccncc2)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CN(Cc2ccccn2)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CN(Cc2cccnc2Br)C1
CC(C)(C)OC(=O)N1CC(N2CC(S(=O)(=O)NC(=O)Nc3c4c(cc5c3CCC5)CCC4)C2)C1
CSCCN1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CN(CCF)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CN(C2CSC2)C1
CN1CC(N2CC(S(=O)(=O)NC(=O)Nc3c4c(cc5c3CCC5)CCC4)C2)C1
CC(C(F)F)N1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
CC(C)(C)OC(=O)/N=C(/NC(=O)OC(C)(C)C)N1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
N=C(N)N1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CN(C2CNC2)C1
CC(C)(C)CN1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CN(C2COC2)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CN(C2CS(=O)C2)C1
CC1CC(N2CC(S(=O)(=O)NC(=O)Nc3c4c(cc5c3CCC5)CCC4)C2)C1
CC1(C)CC(N2CC(S(=O)(=O)NC(=O)Nc3c4c(cc5c3CCC5)CCC4)C2)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CN(C2CS(=O)(=O)C2)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CN(C2CCOC2)C1
CCC(C)N1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
Cn1ccnc1CN1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
CC1(C)CCC1N1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CN(Cc2cncnc2)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CN(CC2CCC2)C1
CN(C(=O)OC(C)(C)C)/C(=N\C(=O)OC(C)(C)C)N4CC(S(=O)(=O)NC(=O)Nc3c1CCCc1cc2CCCc23)C4
C/C(CN1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1)=N/O
CNC(=N)N1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
CC(CO)N1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
CC(C(F)F)N1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
C=CCN1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
C#CCN1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CN(CCCO)C1
CC(C)(C)CN1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
C[Si](C)(C)CN1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
CC(O)CN1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CN(CCCCO)C1
CC1(CCN2CC(S(=O)(=O)NC(=O)Nc3c4c(cc5c3CCC5)CCC4)C2)N=N1
Cn1cc(CN2CC(S(=O)(=O)NC(=O)Nc3c4c(cc5c3CCC5)CCC4)C2)ccc1=O
Cn1ccc(CN2CC(S(=O)(=O)NC(=O)Nc3c4c(cc5c3CCC5)CCC4)C2)cc1=O
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CN(CCC2CCOC2)C1
CCC(C)N1CC(S(=O)(=O)NC(=O)Nc2c(C(C)C)cc(F)cc2C(C)C)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CN(CC2CCOC2)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CN(CC2CCCO2)C1
CN1CC(N2[C@@H]3CC[C@H]2C[C@@H](S(=O)(=O)NC(=O)Nc2c4c(cc5c2CCC5)CCC4)C3)C1
CCN1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)CC1=O
CC(C)N1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)CC1C(=O)N(C)C
COC1CN(C)CC1S(=O)(=O)NC(=O)Nc1c2c(cc3c1CCC3)CCC2
CCN1CC(OC)C(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
CC(C)(C)[Si](C)(C)OCCN1CC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)C1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)C1CN(CCO)C1
COc1cc(-c2ccc3c(c2NC(=O)NS(=O)(=O)c2ccc(=O)n(C(C)C)c2)CCC3)ccn1
CC(C)n1cc(S(=O)(=O)NC(=O)Nc2c(-c3ccnc(C#N)c3)ccc3c2CCC3)ccc1=O
CC(C)n1cc(S(=O)(=O)NC(=O)Nc2c(-c3ccnc(C#N)c3)ccc3c2CCC3)ncc1=O
COc1cc(ccn1)-c1ccc2CCCc2c1NC(=O)NS(=O)(=O)c1cn(C(C)C)c(=O)cn1
CC(C)c1cc(F)cc(-c2ccnc(C#N)c2)c1NC(=O)NS(=O)(=O)C1CN(C(C)C)C1
COc1cc(-c2cc(F)cc(C(C)C)c2NC(=O)NS(=O)(=O)C2CN(C(C)C)C2)ccn1
COc1cc(-c2ccc3c(c2NC(=O)NS(=O)(=O)C2CN(C(C)C)C2)CCC3)ccn1
CC(C)N1CC(S(=O)(=O)NC(=O)Nc2c(-c3ccncc3)cc(F)c3c2CCC3)C1
CC(C)c1cc(F)cc(-c2ccnc(C#N)c2)c1NC(=O)NS(=O)(=O)C1CN(C2CCC2)C1
COc1cc(-c2cc(F)cc(C(C)C)c2NC(=O)NS(=O)(=O)C2CN(C3CCC3)C2)ccn1
COc1cc(-c2ccc3c(c2NC(=O)NS(=O)(=O)C2CN(C4CCC4)C2)CCC3)ccn1
O=C(Nc1c(-c2ccncc2)cc(F)c2c1CCC2)NS(=O)(=O)C1CN(C2CCC2)C1
CCN1CC(S(=O)(=O)NC(=O)Nc2c(-c3ccnc(C#N)c3)cc(F)cc2C(C)C)C1
CCN1CC(S(=O)(=O)NC(=O)Nc2c(-c3ccnc(OC)c3)cc(F)cc2C(C)C)C1
CCN1CC(S(=O)(=O)NC(=O)Nc2c(-c3ccnc(OC)c3)ccc3c2CCC3)C1
CCN1CC(S(=O)(=O)NC(=O)Nc2c(-c3ccncc3)cc(F)c3c2CCC3)C1
CC(C)c1cc(F)cc(-c2ccnc(C#N)c2)c1NC(=O)NS(=O)(=O)C1CN(Cc2cccnc2)C1
COc1cc(-c2ccc3c(c2NC(=O)NS(=O)(=O)C2CN(Cc4cccnc4)C2)CCC3)ccn1
O=C(Nc1c(-c2ccncc2)cc(F)c2c1CCC2)NS(=O)(=O)C1CN(Cc2cccnc2)C1
CC(C)c1cc(F)cc(-c2ccnc(C#N)c2)c1NC(=O)NS(=O)(=O)c1ccc(=O)n(C(C)C)c1
COc1cc(-c2cc(F)cc(C(C)C)c2NC(=O)NS(=O)(=O)c2ccc(=O)n(C(C)C)c2)ccn1
CC(C)n1cc(S(=O)(=O)NC(=O)Nc2c(-c3ccncc3)cc(F)c3c2CCC3)ccc1=O
CC(C)c1cc(F)cc(-c2cccnc2)c1NC(=O)NS(=O)(=O)C1CN(C(C)C)C1
CC(C)c1cc(F)cc(-c2cccnc2)c1NC(=O)NS(=O)(=O)C1CCN(C(C)C)CC1
COc1cc(-c2cc(F)cc(C(C)C)c2NC(=O)NS(=O)(=O)C2CN(Cc3cccnc3)C2)ccn1
COc1cc(-c2ccc3c(c2NC(=O)NS(=O)(=O)c2cnc(=O)n(C(C)C)c2)CCC3)ccn1
COc1cc(-c2ccc3c(c2NC(=O)NS(=O)(=O)c2ccn(C(C)C)c(=O)c2)CCC3)ccn1
CC(C)n1ccc(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)cc1=O
CC(C)n1cc(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)ncc1=O
CC(C)n1cccc(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)c1=O
C[C@@H](O)Cn1cc(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)ccc1=O
CN(C)CCn1cc(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)ccc1=O
CC(C)n1cc(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)ccc1=O
CCN1CCC(S(=O)(=O)NC(=O)Nc2c(-c3ccnc(OC)c3)cc(F)c3c2CCC3)CC1
CCC(C)N1CC(S(=O)(=O)NC(=O)Nc2c(C(C)C)cc(Cl)cc2C(C)C)C1
CCN1CCC(S(=O)(=O)NC(=O)Nc2c(-c3ccnc(OC)c3)ccc3c2CCC3)CC1
CCN1CCC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CC=C3)CC1
CCN1CCC(S(=O)(=O)NC(=O)Nc2c(-c3ccnc(C#N)c3)ccc3c2CCC3)CC1
CCN1CCC(S(=O)(=O)NC(=O)Nc2c(-c3ccnc(OC)c3)cc(F)cc2C(C)C)CC1
CCN1CCC(S(=O)(=O)NC(=O)Nc2c(-c3ccncc3)ccc3c2CCC3)CC1
[2H]C([2H])([2H])C([2H])([2H])N1CCC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)CC1
CCN1CCCC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)CC1
CN1CCCC(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)CC1
COc1ccc(cc1C(=O)NCCc2ccc(cc2)S(=O)(=O)NC(=O)NC3CCCCC3)Cl
CC(C)c1cc(Cl)cc(C(C)C)c1NC(=O)NS(=O)(=O)c1cccc(c1)C(C)O
CC(C)c1cc(Cl)cc(C(C)C)c1NC(=O)NS(=O)(=O)c1cccc(c1)C(C)(C)O
CC(C)(c1cc(oc1)S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)O
[H][C@@]12O[C@]1(C)CC\C=C(C)\CC[C@@]1([H])C(=C)C(=O)C[C@]21[H] |r,c:8|
[O-][N+](=O)\C=C\c1ccc2OCOc2c1
[H][C@]12O[C@@]11[C@@](C)(CC[C@]3([H])[C@@]4(C)C=CC(=O)C(C)(C)[C@]4([H])C=C[C@@]13C)[C@@H](OC2=O)c1ccoc1 |r,c:13,23|
CC(C)(O)c1coc(c1)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2[C@H](O)CCc12 |r|
CC(C)(O)c1coc(c1)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2[C@@H](O)CCc12 |r|
CC(C)(O)c1coc(c1)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2C(O)CCc12
CC(C)(O)c1coc(c1)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCC(O)c12
CC(C)(O)c1coc(c1)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CC(O)Cc12
CC(=O)OC[C@H]1OCC(=O)C=C1 |r,c:10|
[H][C@@]12CO[C@@]([H])(O1)C(=O)C(F)=C2 |r,c:11|
OC[C@H]1OCC(=O)C[C@@H]1O |r|
CCCCCCCC(=O)OC[C@H]1OCC(=O)C=C1 |r,c:16|
CC(=O)OC[C@H]1OCC(=O)C(F)=C1 |r,c:11|
[H][C@@]12CO[C@@]([H])(O1)C(OC(C)=O)=C(F)C2C(C)=O |r,t:12|
[H][C@]12CO[C@]([H])(O1)C(=O)C=C2 |r,c:10|
C1C(=O)[C@H]([C@@H]([C@H](O1)CO)O)O
OC[C@H]1OCC(=O)C=C1 |r,c:7|
CCCC(=O)OC[C@H]1OCC(=O)C=C1 |r,c:12|
[2H]C1([2H])CCc3c1cc2CCCc2c3NC(=O)NS(=O)(=O)c4cc(C(C)(C)O)co4
[2H]C([2H])([2H])C(O)(c4coc(S(=O)(=O)NC(=O)Nc3c1CCCc1cc2CCCc23)c4)C([2H])([2H])[2H]
[2H]C1([2H])CCc3c1cc2c(CCC2([2H])[2H])c3NC(=O)NS(=O)(=O)c4cc(C(C)(C)O)co4
[2H]C4([2H])CCc3cc1CCC([2H])([2H])c1c(NC(=O)NS(=O)(=O)c2cc(C(C)(C)O)co2)c34
COc1ccc(C\C(=N/O)c2nc3ccc(Cl)cc3o2)cc1
COc1ccc(C\C(=N/O)c2nc3ccc(OC)cc3o2)cc1
Cc1ccc2nc(oc2c1)C(\Cc1ccccc1)=N\O
COc1ccccc1C(=O)O\N=C(/C)c1nc2ccccc2o1
c1cc(ccc1C=CC(=O)c2ccc(cc2O)O)O
O\N=C(/Cc1ccccc1)c1nc2ccc(Cl)cc2o1
COc1ccc(Cl)cc1C(=O)NCCc1ccc(cc1)S(=O)(=O)N1CCCC1
CNS(=O)(=O)c1ccc(CCNC(=O)c2ccc(OC)c(Cl)c2)cc1
CNS(=O)(=O)c1ccc(CCNC(=O)c2cc(Cl)ccc2O)cc1
CNS(=O)(=O)c1ccc(CCNC(=O)c2cccc(Cl)c2OC)cc1
CNS(=O)(=O)c1ccc(CCNC(=O)c2ccccc2)cc1
CNS(=O)(=O)c1ccc(CCNC(=O)c2cccc(Cl)c2)cc1
CNS(=O)(=O)c1ccc(CCNC(=O)c2cc(Cl)ccc2OC)cc1
CCCCN(CCCC)S(=O)(=O)c1ccc(CCNC(=O)c2cc(Cl)ccc2OC)cc1
CNS(=O)(=O)c1ccc(CCCCNC(=O)c2cc(Cl)ccc2OC)cc1
CNS(=O)(=O)c1ccc(CCCNC(=O)c2cc(Cl)ccc2OC)cc1
COc1ccc(Cl)cc1C(=O)NCCc1ccc(cc1)S(=O)(=O)N1CCCCC1
COc1ccc(Cl)cc1C(=O)NCCc1ccc(cc1)S(=O)(=O)NCCc1ccccc1
COc1ccc(Cl)cc1C(=O)NCCc1ccc(cc1)S(=O)(=O)NCc1ccc(Cl)cc1
COc1ccc(Cl)cc1C(=O)NCCc1ccc(cc1)S(=O)(=O)NCc1ccc(O)cc1
COc1ccc(CNS(=O)(=O)c2ccc(CCNC(=O)c3cc(Cl)ccc3OC)cc2)cc1
CCCCNS(=O)(=O)c1ccc(CCNC(=O)c2cc(Cl)ccc2OC)cc1
CCCN(CCC)S(=O)(=O)c1ccc(CCNC(=O)c2cc(Cl)ccc2OC)cc1
CCCNS(=O)(=O)c1ccc(CCNC(=O)c2cc(Cl)ccc2OC)cc1
CNS(=O)(=O)c1ccc(CCNC(=O)c2c(Cl)cccc2OC)cc1
CNS(=O)(=O)c1ccc(CCNC(=O)c2ccc(Cl)cc2OC)cc1
COc1ccc(Cl)cc1C(=O)NCCc1ccc(cc1)S(=O)(=O)N1CCC1
COc1ccc(Cl)cc1C(=O)NCCc1ccc(cc1)S(=O)(=O)Nc1ccccc1
COc1ccc(Cl)cc1C(=O)NCCc1ccc(cc1)S(=O)(=O)N1CCNCC1
CNS(=O)(=O)c1ccc(CCNC(=O)c2cc(Cl)cc(OC)c2)cc1
CNS(=O)(=O)c1ccc(CCNC(=O)c2ccccc2OC)cc1
COc1ccc(Cl)cc1C(=O)NCCc1ccc(cc1)S(=O)(=O)N1CCOCC1
COc1ccc(Cl)cc1C(=O)NCCc1ccc(cc1)S(=O)(=O)NCc1ccc(cc1)C(F)(F)F
COc1ccc(Cl)cc1C(=O)NCCc1ccc(cc1)S(=O)(=O)NCc1ccccc1
CCN(CC)S(=O)(=O)c1ccc(CCNC(=O)c2cc(Cl)ccc2OC)cc1
Nc1nc2cc(ccc2c2[nH]c(CN3C[C@@H](CC3=O)c3ccccc3)nc12)-n1cccn1 |r|
CCN(Cc1nc2c(N)nc3cc(ccc3c2[nH]1)-c1ccccc1)C(C)=O
Nc1nc2cc(ccc2c2[nH]c(CN3CCCC3=O)nc12)-c1cccs1
CCN(Cc1nc2c(N)nc3cc(ccc3c2[nH]1)C1=CCCC1)C(C)=O |t:21|
CCN(Cc1nc2c(N)nc3cc(ccc3c2n1CC)-c1ccn[nH]1)C(=O)CC
CCN(Cc1nc2c(N)nc3cc(ccc3c2n1C)-c1cc[nH]n1)C(=O)OC(C)(C)C
CCN(C)Cc1nc2c(N)nc3cc(ccc3c2[nH]1)-c1cc[nH]n1
Cc1ccc(cc1)-c1ccc2c3[nH]c(CN4CCCC4=O)nc3c(N)nc2c1
Cc1cccc(c1)-c1ccc2c3[nH]c(CN4CCCC4=O)nc3c(N)nc2c1
Nc1nc2cc(ccc2c2[nH]c(CN3CCCC3=O)nc12)-c1ccccc1
CCn1c(CN2CCCC2=O)nc2c(N)nc3cc(ccc3c12)-c1cccs1
Nc1nc2cc(ccc2c2[nH]c(CN3CCCC3=O)nc12)-c1ccccc1F
COc1ccc2C(=O)N(C(=O)c2c1)c1ccccc1
Cc1cccc(c1C)Nc2ccccc2C(=O)O
CCn1c(nc2cc(C)ccc12)-c1ccccc1
CC1Cc2o\c(=N\C3CCCCC3)sc2C(=O)C1
CS(=O)(=O)CCC#N
COc1ccc(Cl)cc1C(=O)NCCc1ccc(cc1)S(=O)(=O)NO
NS(=O)(=O)c1ccc(CCNC(=O)C(=C)Cc2ccccc2Cl)cc1
CC(=O)C1=C(N[B-]([O+]=C1N)(c1ccccc1)c1ccccc1)C(Cl)(Cl)Cl |c:7,t:3|
[O-][N+](=O)c1ccc(cc1)-c1nc2ccccc2c(=O)[nH]1
c1cc(ccc1C2=CC(=O)c3c(cc(cc3O2)O)O)O
OC(=O)c1ccc(\C=C2/SC(=S)N(Cc3cccc(c3)C(F)(F)F)C2=S)cc1
Cc1ccc(cc1)S(=O)(=O)/C=C/C#N
CCC1=C(C)CN(C(=O)NCCc2ccc(cc2)S(=O)(=O)NC(=O)Nc2c3CCCc3cc3CCCc23)C1=O |c:2|
COc1ccc(Cl)cc1C(=O)NCCc1ccc(cc1)S(N)(=O)=O
CCCOc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)C=C
CCCOc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)c1cscn1
COc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)C=C
CCC(=O)N(CCc1ccc(cc1)S(=O)(=O)NCC#C)Cc1cc(Cl)ccc1OC
CCCCCC(=O)N(CCc1ccc(cc1)S(=O)(=O)NCC#C)Cc1cc(Cl)ccc1OC
COc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)CC=C
CCCOc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)Cc1ccccc1
CCCOc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)Cc1ccc(OC)cc1
CCCOc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)Cc1ccccn1
CCCOc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)Cc1c[nH]c2ccccc12
CCCOc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)Cc1ccsc1
CCCOc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)c1ccoc1
CCCOc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)c1cnsn1
CCCOc1ccc(Br)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)Cc1ccsc1
CCCOc1ccc(F)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)Cc1ccsc1
CCCCOc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)Cc1ccsc1
COc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)Cc1ccccc1
CCCOc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)CCc1ccccc1
CCCOc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)c1ccsc1
COc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)Cc1ccsc1
CCCOc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)Cc1ccncc1
CCCOc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)c1nc[nH]n1
CCCOc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)c1cnccn1
CCC(C)Oc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)Cc1ccsc1
CCCOc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)Cc1c[nH]cn1
CCCCCOc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)Cc1ccsc1
CCCN(CCc1ccc(cc1)S(=O)(=O)NCC#C)Cc1cc(Cl)ccc1OC
Cc1ccc(cc1)S(=O)(NC(=O)Nc1c2CCCc2cc2CCCc12)=NC#N
Cc1ccc(cc1)S(=O)(=O)N\C(Nc1c2CCCc2cc2CCCc12)=N/C#N
OP(=O)(NC(=O)Nc1c2CCCc2cc2CCCc12)c1ccccc1
Cc1ccc(cc1)S(=O)(=O)NC(=O)C(=O)Nc1c2CCCc2cc2CCCc12
Cc1ccc(cc1)S(=O)(=O)NS(=O)(=O)Nc1c2CCCc2cc2CCCc12
Cc1ccc(cc1)S(=O)(=O)NC(=O)Cc1c2CCCc2cc2CCCc12
Cc1ccc(cc1)S(=O)(=O)NC(=O)C(O)c1c2CCCc2cc2CCCc12
Cc1ccc(cc1)S(=O)(=O)NC(=O)C(=O)c1c2CCCc2cc2CCCc12
Cc1ccc(cc1)S(=O)(=O)Nc1c(Nc2c3CCCc3cc3CCCc23)c(=O)c1=O
O=C(Nc1c2CCCc2cc2CCCc12)NC1(COC1)c1ccccc1
FC(F)(F)C(NC(=O)Nc1c2CCCc2cc2CCCc12)c1ccccc1
O=C(NC(C#N)c1ccccc1)Nc1c2CCCc2cc2CCCc12
Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
O=C(Nc1c2CCCc2cc2CCCc12)NS(=O)(=O)c1ccccc1
O=C(Nc1c2CCCc2cc2CCCc12)NS(=O)(=NC#N)c1ccccc1
CN=S(=O)(NC(=O)Nc1c2CCCc2cc2CCCc12)c1ccc(C)cc1
Cc1ccc(cc1)S(=O)(NC(=O)Nc1c2CCCc2cc2CCCc12)=NCC(F)(F)F
CON=S(=O)(NC(=O)Nc1c2CCCc2cc2CCCc12)c1ccc(C)cc1
Cc1ccc(cc1)S(=O)(NC(=O)Nc1c2CCCc2cc2CCCc12)=Nc1ccc(F)cc1
Cc1ccc(cc1)S(=O)(NC(=O)Nc1c2CCCc2cc2CCCc12)=Nc1ccn[nH]1
Cc1ccc(cc1)S(=O)(NC(=O)Nc1c2CCCc2cc2CCCc12)=NC(N)=O
CCOC(=O)N=S(=O)(NC(=O)Nc1c2CCCc2cc2CCCc12)c1ccc(C)cc1
CC(=O)N=S(=O)(NC(=O)Nc1c2CCCc2cc2CCCc12)c1ccc(C)cc1
Cc1ccc(cc1F)S(=O)(NC(=O)Nc1c2CCCc2cc2CCCc12)=NC#N
O=C(Nc1c2CCCc2cc2CCCc12)NS(=O)(=NC#N)c1ccc(cc1)C#N
O=C(Nc1c2CCCc2cc2CCCc12)NS(=O)(=NC#N)c1cccc(c1)C#N
O=C(Nc1c2CCCc2cc2CCCc12)NS(=O)(=NC#N)c1ccncc1
O=C(Nc1c2CCCc2cc2CCCc12)NS(=O)(=NC#N)c1cccnc1
O=C(Nc1c2CCCc2cc2CCCc12)NS(=O)(=NC#N)c1ccccn1
C\C(=N/NS(=O)(=O)c1ccc(C)cc1)c1nc2ccccc2o1
COc1ccc(cc1)S(=O)(=O)N\N=C(/C)c1nc2ccccc2o1
OC(=O)c1ccc(\C=C2/SC(=S)N(C2=O)c2cccc(c2)C(F)(F)F)cc1
CN1CCN(CC1)C(=O)c1ccc(\C=C2/SC(=S)N(C2=O)c2cccc(c2)C(F)(F)F)cc1
FC(F)(F)c1cccc(c1)N1C(=S)S\C(=C/c2ccc(cc2)C(=O)N2CCOCC2)C1=O
OC1CCN(CC1)C(=O)c1ccc(\C=C2/SC(=S)N(C2=O)c2cccc(c2)C(F)(F)F)cc1
CN1CCN(CC1)C(=O)c1ccc(\C=C2/SC(=S)N(C2=O)c2cccc(OC(F)(F)F)c2)cc1
FC(F)(F)Oc1cccc(c1)N1C(=S)S\C(=C/c2ccc(cc2)C(=O)N2CCOCC2)C1=O
CN1CCN(CC1)C(=O)c1ccc(\C=C2/SC(=S)N(C2=O)c2cccc(c2)[N+]([O-])=O)cc1
FC(F)(F)c1cccc(c1)N1C(=S)S\C(=C/c2ccc(cc2)C(=O)Nc2ccccc2)C1=O
OC(=O)c1ccc(\C=C2/SC(=S)N(Cc3cccc(c3)C(F)(F)F)C2=O)cc1
OC(=O)c1ccc(\C=C2/SC(=S)N(CCc3cccc(c3)C(F)(F)F)C2=O)cc1
OC(=O)c1ccc(\C=C2/SC(=S)N(CCCc3cccc(c3)C(F)(F)F)C2=O)cc1
FC(F)(F)c1cccc(CN2C(=S)S\C(=C/c3ccc(cc3)-c3nnn[nH]3)C2=O)c1
FC(F)(F)c1cccc(CCN2C(=S)S\C(=C/c3ccc(cc3)-c3nnn[nH]3)C2=O)c1
FC(F)(F)c1cccc(CCCN2C(=S)S\C(=C/c3ccc(cc3)-c3nnn[nH]3)C2=O)c1
CN1CCN(CC1)C(=O)c1ccc(\C=C2/SC(=S)N(Cc3cccc(c3)C(F)(F)F)C2=O)cc1
OC(=O)c1ccc(\C=C2/SC(=O)N(Cc3cccc(c3)C(F)(F)F)C2=O)cc1
FC(F)(F)c1cccc(CN2C(=O)S\C(=C/c3ccc(cc3)-c3nnn[nH]3)C2=O)c1
OC(=O)c1ccc(\C=C2/SC(=S)N(Cc3cccc(OC(F)(F)F)c3)C2=O)cc1
OC(=O)c1ccc(\C=C2/SC(=S)N(Cc3cccc(F)c3)C2=O)cc1
OC(=O)c1ccc(\C=C2/SC(=S)N(Cc3cccnc3)C2=O)cc1
OC(=O)c1ccc(\C=C2/SC(=S)N(Cc3ccc(cc3)-c3ccccc3)C2=O)cc1
[H][C@@]12C\C(=N\OC(=O)CCCCCCCCCCC)C(C)=C(CCc3ccoc3)[C@@]1(C)CCCC2(C)C |r,t:20|
[H][C@@]12C\C(=N\OC(=O)c3ccc(cc3)C(=O)O\N=C3\C[C@@]4([H])C(C)(C)CCC[C@]4(C)C(CCc4ccoc4)=C3C)C(C)=C(CCc3ccoc3)[C@@]1(C)CCCC2(C)C |r,c:40,t:45|
O=C(Nc1c2CCCc2cc2CCCc12)NS(=O)(=O)\C=C\c1nccs1
CC(C)(O)c1coc(\C=C\S(=O)(=O)NC(=O)Nc2c3CCCc3cc3CCCc23)c1
O=C(Nc1c2CCCc2cc2CCCc12)NS(=O)(=O)\C=C\c1cccs1
O=C(Nc1c2CCCc2cc2CCCc12)NS(=O)(=O)\C=C\c1ccsc1
O=C(Nc1c2CCCc2cc2CCCc12)NS(=O)(=O)\C=C\c1ccncc1
O=C(Nc1c2CCCc2cc2CCCc12)NS(=O)(=O)\C=C\c1ccccn1
Cc1csc(\C=C\S(=O)(=O)NC(=O)Nc2c3CCCc3cc3CCCc23)n1
Cc1cnc(\C=C\S(=O)(=O)NC(=O)Nc2c3CCCc3cc3CCCc23)s1
O=C(Nc1c2CCCc2cc2CCCc12)NS(=O)(=O)\C=C\c1cncs1
O=C(Nc1c2CCCc2cc2CCCc12)NS(=O)(=O)\C=C\c1cscn1
CC(C)(O)c1csc(\C=C\S(=O)(=O)NC(=O)Nc2c3CCCc3cc3CCCc23)n1
OCc1csc(\C=C\S(=O)(=O)NC(=O)Nc2c3CCCc3cc3CCCc23)n1
CCSCc1csc(\C=C\S(=O)(=O)NC(=O)Nc2c3CCCc3cc3CCCc23)n1
CC[S+]([O-])Cc1csc(\C=C\S(=O)(=O)NC(=O)Nc2c3CCCc3cc3CCCc23)n1
CCS(=O)(=O)Cc1csc(\C=C\S(=O)(=O)NC(=O)Nc2c3CCCc3cc3CCCc23)n1
CN(C)C(=O)c1csc(\C=C\S(=O)(=O)NC(=O)Nc2c3CCCc3cc3CCCc23)n1
O=C(Nc1c2CCCc2cc2CCCc12)NS(=O)(=O)\C=C\c1nc2ccccc2s1
Cc1c2CCCc2c(NC(=O)NS(=O)(=O)\C=C\c2nccs2)c2CCCc12
O=C(Nc1c2CCOc2cc2CCOc12)NS(=O)(=O)\C=C\c1nccs1
CC(C)c1cccc(C(C)C)c1NC(=O)NS(=O)(=O)\C=C\c1nccs1
COc1cccc(OC)c1NC(=O)NS(=O)(=O)\C=C\c1nccs1
Fc1cccc(c1NC(=O)NS(=O)(=O)\C=C\c1nccs1)C(F)(F)F
FC(F)(F)c1ccc(c(NC(=O)NS(=O)(=O)\C=C\c2nccs2)c1)C(F)(F)F
FC(F)(F)c1ccccc1NC(=O)NS(=O)(=O)\C=C\c1nccs1
Cc1cc(C)c(C)c(NC(=O)NS(=O)(=O)\C=C\c2nccs2)c1C
CC(C)(O)c1coc(c1)S(=O)(=O)[N-]C(=O)Nc1c2CCCc2cc2CCCc12
CC(C)(O)c1coc(c1)S(=O)(=O)NC(=O)Nc1cccc2CCCc12
CC(C)(O)c1coc(c1)S(=O)(=O)[N-]C(=O)Nc1ccccc1
O=C(Nc1c2CCCc2cc2CCCc12)[N-]S(=O)(=O)c1ccco1
O=C(Nc1c2CCCc2cc2CCCc12)[N-]S(=O)(=O)c1ccccc1
CS(=O)(=O)[N-]C(=O)Nc1c2CCCc2cc2CCCc12
OC(=O)CC(=O)Nc1c2CCCc2cc2CCCc12
COC(=O)CC(=O)Nc1c2CCCc2cc2CCCc12
O=C(CS(=O)(=O)Nc1ccccc1)Nc1c2CCCc2cc2CCCc12
O=C(CNS(=O)(=O)c1ccccc1)Nc1c2CCCc2cc2CCCc12
OC(=O)CNC(=O)Nc1c2CCCc2cc2CCCc12
COC(=O)CNC(=O)Nc1c2CCCc2cc2CCCc12
CCOC(=O)CNC(=O)Nc1c2CCCc2cc2CCCc12
CC(C)OC(=O)CNC(=O)Nc1c2CCCc2cc2CCCc12
CC(C)(C)OC(=O)CNC(=O)Nc1c2CCCc2cc2CCCc12
CNC(=O)CNC(=O)Nc1c2CCCc2cc2CCCc12
CN(C)C(=O)CNC(=O)Nc1c2CCCc2cc2CCCc12
Cc1nc(CNC(=O)Nc2c3CCCc3cc3CCCc23)no1
Cc1nnc(CNC(=O)Nc2c3CCCc3cc3CCCc23)o1
CCOC(=O)CNC(=O)Nc1c2CCCc2cc2CCCCc12
CCOC(=O)CNC(=O)Nc1cc2CCCc2c2CCCCc12
CCOC(=O)CNC(=O)Nc1c2CCCc2c(Cl)c2CCCc12
CCOC(=O)CNC(=O)Nc1c2CCCc2nc2CCCc12
COC(=O)CNC(=O)Nc1c(cccc1C(C)C)C(C)C
CCOC(=O)CNC(=O)Nc1c(C)cccc1C
CCOC(=O)CNC(=O)NC12CC3CC(CC(C3)C1)C2 |TLB:17:12:19:16.18.15,17:16:19:12.11.13,THB:15:14:11:16.18.17,15:16:11:14.19.13|
CCOC(=O)CNC(=O)NC(c1ccccc1)c1ccccc1
COC(=O)C(C)(C)NC(=O)Nc1c2CCCc2cc2CCCc12
COC(=O)C(Cc1ccccc1)NC(=O)Nc1c2CCCc2cc2CCCc12
COC(=O)[C@H](Cc1ccccc1)NC(=O)Nc1c2CCCc2cc2CCCc12 |r|
COC(=O)[C@@H](Cc1ccccc1)NC(=O)Nc1c2CCCc2cc2CCCc12 |r|
COC(=O)C(CCc1ccccc1)NC(=O)Nc1c2CCCc2cc2CCCc12
COC(=O)C(Cc1ccccc1O)NC(=O)Nc1c2CCCc2cc2CCCc12
COC(=O)C(Cc1cccc(O)c1)NC(=O)Nc1c2CCCc2cc2CCCc12
COC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)Nc1c2CCCc2cc2CCCc12 |r|
COC(=O)[C@@H](Cc1cccc(c1)C#N)NC(=O)Nc1c2CCCc2cc2CCCc12 |r|
COC(=O)[C@@H](Cc1ccc(cc1)C#N)NC(=O)Nc1c2CCCc2cc2CCCc12 |r|
COC(=O)[C@@H](Cc1ccccn1)NC(=O)Nc1c2CCCc2cc2CCCc12 |r|
COC(=O)[C@@H](Cc1cccnc1)NC(=O)Nc1c2CCCc2cc2CCCc12 |r|
COC(=O)[C@@H](Cc1ccncc1)NC(=O)Nc1c2CCCc2cc2CCCc12 |r|
CCOC(=O)C(Cc1ccncn1)NC(=O)Nc1c2CCCc2cc2CCCc12
COC(=O)[C@@H](Cc1cncnc1)NC(=O)Nc1c2CCCc2cc2CCCc12 |r|
COC(=O)[C@@H](Cc1cccnn1)NC(=O)Nc1c2CCCc2cc2CCCc12 |r|
CCOC(=O)C(Cc1ccnnc1)NC(=O)Nc1c2CCCc2cc2CCCc12
CCOC(=O)[C@@H](Cc1ncccn1)NC(=O)Nc1c2CCCc2cc2CCCc12 |r|
CCOC(=O)[C@@H](Cc1cnccn1)NC(=O)Nc1c2CCCc2cc2CCCc12 |r|
COc1c(ccc(c1)/C=C/C(=O)CC(=O)/C=C/c2cc(c(cc2)O)OC)O
COc1cc(\C=C\C(=O)c2ccccc2)c(OC)c2ccoc12
[H][C@@]12CCC(C)=C3CC[C@@](C)(O)[C@]3([H])[C@@]1([H])OC(=O)[C@H]2CN(C)CCCOc1no[n+]([O-])c1S(=O)(=O)c1ccccc1 |r,t:5|
[H][C@@]12CCC(C)=C3CC[C@@](C)(O)[C@]3([H])[C@@]1([H])OC(=O)[C@H]2CN(C)CCOc1no[n+]([O-])c1S(=O)(=O)c1ccccc1 |r,t:5|
[H][C@]12O[C@@]1(C)CC\C=C(C)\CC[C@@]1([H])[C@H](CN(C)CCCOc3no[n+]([O-])c3S(=O)(=O)c3ccccc3)C(=O)O[C@]21[H] |r,c:8|
[H][C@]12O[C@@]1(C)CC\C=C(C)\CC[C@@]1([H])[C@H](CN(C)CCOc3no[n+]([O-])c3S(=O)(=O)c3ccccc3)C(=O)O[C@]21[H] |r,c:8|
[H][C@@]12CCC(C)=C3CC[C@@](C)(O)[C@]3([H])[C@@]1([H])OC(=O)C2=C |r,t:5|
[O-][n+]1onc(c1S(=O)(=O)c1ccccc1)S(=O)(=O)c1ccccc1
[H][C@]12O[C@@]1(C)CC\C=C(C)\CC[C@@]1([H])C(=C)C(=O)O[C@]21[H] |r,c:8|
CS(=O)(=O)N1CCCc2ccc(cc12)N(S(=O)(=O)c1ccccc1[N+]([O-])=O)S(=O)(=O)c1ccccc1[N+]([O-])=O
CC(=O)c1ccc(cc1)S(=O)(=O)N(c1ccc2CCCN(c2c1)S(C)(=O)=O)S(=O)(=O)c1ccc(cc1)C(C)=O
CS(=O)(=O)N1CCCc2ccc(cc12)N(S(=O)(=O)c1ccc(cc1)-c1ccccc1)S(=O)(=O)c1ccc(cc1)-c1ccccc1
CC(C)(C)c1ccc(cc1)S(=O)(=O)N(c1ccc2CCCN(c2c1)S(C)(=O)=O)S(=O)(=O)c1ccc(cc1)C(C)(C)C
CCCCS(=O)(=O)N(c1ccc2CCCN(c2c1)S(C)(=O)=O)S(=O)(=O)CCCC
CS(=O)(=O)N1CCCc2ccc(cc12)N(S(=O)(=O)CCN1C(=O)c2ccccc2C1=O)S(=O)(=O)CCN1C(=O)c2ccccc2C1=O
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(NS(C)(=O)=O)cc12
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(NS(=O)(=O)CC)cc12
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(NS(=O)(=O)C3CC3)cc12
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(NS(=O)(=O)C=C)cc12
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(NS(=O)(=O)C3CCCCC3)cc12
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(NS(=O)(=O)c3ccccc3)cc12
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(NS(=O)(=O)c3cccnc3)cc12
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(NS(=O)(=O)c3ccc(C)cc3)cc12
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(NS(=O)(=O)c3ccc(F)cc3)cc12
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(NS(=O)(=O)c3ccc(cc3)C(F)(F)F)cc12
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(NS(=O)(=O)c3ccc(OC)cc3)cc12
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(cc12)S(N)(=O)=O
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(cc12)S(=O)(=O)NC
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(cc12)S(=O)(=O)NC(C)C
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(cc12)S(=O)(=O)NOC
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(cc12)S(=O)(=O)NCCN(C)C
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(cc12)S(=O)(=O)N(C)C
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(cc12)S(=O)(=O)N(CCC)CCC
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(NC(C)=O)cc12
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(NC(=O)C=C)cc12
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(NC(=O)C(C)C)cc12
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(NC(=O)CCCC)cc12
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(NC(=O)C(C)(C)C)cc12
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(NC(=O)c3ccccc3)cc12
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(NC(=O)c3ccc(OC)cc3)cc12
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(NC(=O)NC(C)C)cc12
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(NC(=O)NCCC)cc12
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(NC(=O)NC3CCCC3)cc12
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(NC(=O)NC3CCCCC3)cc12
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(NC(=O)Nc3ccc(C)cc3)cc12
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(NC(=O)Nc3ccc(OC)cc3)cc12
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(NC(=O)Nc3ccc(cc3)C#N)cc12
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(NC(=O)Nc3ccc(Cl)cc3)cc12
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(NS(=O)(=O)NC)cc12
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(NS(=O)(=O)N(C)C)cc12
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(NS(=O)(=O)NC(C)C)cc12
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(N)cc12
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccccc12
Cc1cc(cc(c1OC(C)(C)C(=O)O)C)/C=C/C(=O)c2ccc(cc2)SC
COc1c(C)cc(\C=C\C(=O)c2ccc(SC)cc2)cc1C
COc1c(C)cc(\C=C\C(=O)c2ccc(N)cc2)cc1C
COc1c(C)cc(\C=C\C(=O)c2ccc(cc2)N(C)C)cc1C
COc1c(C)cc(\C=C\C(=O)c2ccc(NC(=O)NC(C)C)cc2)cc1C
CCCNC(=O)Nc1ccc(cc1)C(=O)\C=C\c1cc(C)c(OC)c(C)c1
COc1c(C)cc(\C=C\C(=O)c2ccc(NC(=O)Nc3ccc(F)cc3)cc2)cc1C
COc1c(C)cc(\C=C\C(=O)c2ccc(NC(=O)Nc3ccc(C)cc3)cc2)cc1C
CSc1ccc(cc1)C(=O)\C=C\c1cc(C)c(OCC(O)=O)c(C)c1
CSc1ccc(cc1)C(=O)\C=C\c1cc(C)c(OCCO)c(C)c1
CCC(Oc1c(C)cc(\C=C\C(=O)c2ccc(SC)cc2)cc1C)C(O)=O
CSc1ccc(cc1)C(=O)\C=C\c1cc(C)c(OCC(=C)C(O)=O)c(C)c1
CSc1ccc(cc1)C(=O)\C=C\c1cc(C)c(OCCCCC(O)=O)c(C)c1
CCCNC(=O)Oc1c(C)cc(\C=C\C(=O)c2ccc(SC)cc2)cc1C
CSc1ccc(cc1)C(=O)\C=C\c1cc(C)c(OCCCN2CCOCC2)c(C)c1
CSc1ccc(cc1)C(=O)\C=C\c1ccc2OCCc2c1
CSc1ccc(cc1)C(=O)\C=C\c1cc(C)c(O)c(C)c1
CSc1ccc(cc1)C(=O)\C=C\c1ccc(cc1)C(O)=O
CSc1ccc(cc1)C(=O)\C=C\c1ccc(O)cc1
CSc1ccc(cc1)C(=O)\C=C\c1ccc(O)c(C)c1
COc1cc(\C=C\C(=O)c2ccc(SC)cc2)ccc1O
CSc1ccc(cc1)C(=O)\C=C\c1ccc(O)c(F)c1
CSc1ccc(cc1)C(=O)\C=C\c1ccc(O)cc1F
CSc1ccc(cc1)C(=O)\C=C\c1ccc(O)c(Cl)c1
CSc1ccc(cc1)C(=O)\C=C\c1cc(C)c(O)cc1C
CSc1ccc(cc1)C(=O)\C=C\c1c(C)cc(O)cc1C
COc1cc(\C=C\C(=O)c2ccc(SC)cc2)cc(OC)c1O
CCc1cc(\C=C\C(=O)c2ccc(SC)cc2)cc(CC)c1O
CSc1ccc(cc1)C(=O)\C=C\c1ccc(O)c(O)c1
Cc1cc(\C=C\C(=O)c2ccc(F)cc2)cc(C)c1O
Cc1cc(\C=C\C(=O)c2ccc(Cl)cc2)cc(C)c1O
Cc1cc(\C=C\C(=O)c2ccc(I)cc2)cc(C)c1O
C[S+]([O-])c1ccc(cc1)C(=O)\C=C\c1cc(C)c(O)c(C)c1
Cc1cc(\C=C\C(=O)c2ccc(cc2)S(C)(=O)=O)cc(C)c1O
Cc1cc(\C=C\C(=O)c2ccc(cc2)-c2ccccc2)cc(C)c1O
Cc1cc(\C=C\C(=O)c2ccc(cc2)-c2cccs2)cc(C)c1O
Cc1ccc(s1)-c1ccc(cc1)C(=O)\C=C\c1cc(C)c(O)c(C)c1
Cc1cc(\C=C\C(=O)c2ccc(NS(=O)(=O)c3ccc(F)cc3)cc2)cc(C)c1O
CC(C)NS(=O)(=O)Nc1ccc(cc1)C(=O)\C=C\c1cc(C)c(O)c(C)c1
Cc1cc(\C=C\C(=O)c2ccc(NC(=O)C=C)cc2)cc(C)c1O
CCN(CC)C(=S)SSC(=S)N(CC)CC
COc1cc(OC)cc(\C=C\c2ccc(OCc3ccc(cc3)C(F)(F)F)cc2)c1
COc1cc(OC)c(\C=C\[N+]([O-])=O)c(\C=C\c2ccc(O)cc2)c1
COc1cc(OC)c(-c2cnn[nH]2)c(\C=C\c2ccc(OCC(=O)NCc3ccccc3)cc2)c1
COc1cc(OC)c(\C=C\[N+]([O-])=O)c(\C=C\c2ccc(OCC(=O)NCc3ccc(Br)cc3)cc2)c1
COc1cc(OC)c(\C=C\[N+]([O-])=O)c(\C=C\c2ccc(OCC(=O)NCc3ccncc3)cc2)c1
CCCCNC(=O)COc1ccc(\C=C\c2cc(OC)cc(OC)c2\C=C\[N+]([O-])=O)cc1
COc1cc(OC)c(\C=C\[N+]([O-])=O)c(\C=C\c2ccc(N)cc2)c1
COc1cc(OC)c(\C=C\[N+]([O-])=O)c(\C=C\c2ccc(NC(=O)CCCl)cc2)c1
COc1cc(OC)c(\C=C\[N+]([O-])=O)c(\C=C\c2ccc(NC(=O)C3CC3)cc2)c1
COc1cc(OC)c(\C=C\[N+]([O-])=O)c(\C=C\c2ccc(NC(=O)C3CCC3)cc2)c1
COc1cc(OC)c(\C=C\[N+]([O-])=O)c(\C=C\c2ccc(NC(=O)C3CCCCC3)cc2)c1
[H][C@@]12CC[C@]3([H])[C@@]([C@@H]1O)(C(=O)C2=C)[C@@]1(O)OC[C@]32[C@@H](O)CCC(C)(C)[C@@]2([H])[C@@H]1O |r,THB:12:11:7:4.2.3,10:9:7:4.2.3|
COc1cc(cc(c1)OC)/C=C/c2ccc(cc2)O
COc1ccc(cc1OC)\C=C\C(=O)Nc2ccccc2C(=O)O
B([C@H](CC(C)C)NC(=O)CNC(=O)c1cc(ccc1Cl)Cl)(O)O
CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)c1cnccn1)B(O)O |r|
CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)c1cnccn1)C(O)=O |r|
CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)c1cc(Cl)ccc1Cl)C(O)=O |r|
CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)c1cc(Cl)ccc1Cl)B(O)O |r|
CC(C)C[C@H](NC(=O)c1ccc(CNC(=O)c2cc(Cl)ccc2Cl)cc1)B(O)O |r|
CC(C)C[C@H](NC(=O)CN(C)C(=O)c1cc(Cl)ccc1Cl)B(O)O |r|
CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NS(=O)(=O)c1cc(Cl)ccc1Cl)B(O)O |r|
CC(C)C[C@H](NC(=O)c1cc(Cl)ccc1Cl)B(O)O |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)c1cc(Cl)ccc1Cl)C(C)C)B(O)O |r|
CC[C@@H](C)[C@H](NC(=O)c1cc(Cl)ccc1Cl)C(=O)N[C@@H](CC(C)C)B(O)O |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)c1cc(Cl)ccc1Cl)c1ccccc1)B(O)O |r|
CC(C)C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)c1cc(Cl)ccc1Cl)B(O)O |r|
CC(C)C[C@H](NC(=O)[C@H](CO)NC(=O)c1cc(Cl)ccc1Cl)B(O)O |r|
CC(C)C[C@H](NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)c1cc(Cl)ccc1Cl)B(O)O |r|
CC(C)C[C@H](NC(=O)[C@H](Cc1ccc2ccccc2c1)NC(=O)c1cc(Cl)ccc1Cl)B(O)O |r|
CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccccn1)B(O)O |r|
CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)c1cncc(C)n1)B(O)O |r|
CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)c1cnc2ccccc2n1)B(O)O |r|
CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)c1nc(Cl)ccc1Cl)B(O)O |r|
CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)c1cccc(Cl)c1Cl)B(O)O |r|
CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)c1c(Cl)cccc1Cl)B(O)O |r|
CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc(Cl)cc1Cl)B(O)O |r|
COc1ccc(Cl)cc1C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CC(C)C)B(O)O |r|
COc1ccc(F)cc1C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CC(C)C)B(O)O |r|
CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc(F)cc1F)B(O)O |r|
CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)c1cccc(F)c1F)B(O)O |r|
CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)c1cc(F)ccc1F)B(O)O |r|
CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)c1cc(Cl)ccc1F)B(O)O |r|
Clc1ccc(c2nonc12)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
CN(C)c1ccc(c2nonc12)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
CC(C)(C)OC(=O)NC1CN(C1)c1ccc(c2nonc12)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
O=C(Nc1c2CCCc2cc2CCCc12)NS(=O)(=O)c1ccc(N2CCOCC2)c2nonc12
[H][C@@]12CN(C[C@]1([H])[C@H]2CO)c1ccc(c2nonc12)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12 |r|
O=C(Nc1c2CCCc2cc2CCCc12)NS(=O)(=O)c1ccc(N2CC3CCC(C2)O3)c2nonc12
FC1(F)CC(C1)Nc1ccc(c2nonc12)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
OCCN1CCN(CC1)c1ccc(c2nonc12)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
CN(C)[C@@H]1CCCC[C@H]1N(C)c1ccc(c2nonc12)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12 |r|
CSc1ccc(c2nonc12)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
CN(C)c1cccc2c(cccc12)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
CN(C)c1ccc(c2nsnc12)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
CN(C)c1ccc(c2n[se]nc12)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
C[C@@H]1CC[C@@]2(C)C(=C)[C@H](CC[C@@]22C=C(C=O)[C@H](C[C@@]12C)OC(C)=O)OC(C)=O |r,t:13|
Oc1cccc(NC(=O)Cc2ccc3cc[nH]c3c2)c1
Oc1cccc(NC(=O)Cn2ccc3ccccc3c2=O)c1
Oc1cccc(NC(=O)Cc2ccc3ncccc3c2)c1
Oc1cccc(NC(=O)Cc2ccc3OCCc3c2)c1
Oc1cccc(NC(=O)Cc2ccc3OCOc3c2)c1
Oc1cccc(NC(=O)Cc2cccc3ccccc23)c1
Oc1cccc(NC(=O)Cc2ccc3ccccc3c2)c1
CS(=O)(=O)Nc1ccc(CC(=O)Nc2cccc(O)c2)cc1
CC(=O)Nc1ccc(CC(=O)Nc2cccc(O)c2)cc1
Oc1cccc(NC(=O)Cc2ccc(cc2)[N+]([O-])=O)c1
CS(=O)(=O)c1ccc(CC(=O)Nc2cccc(O)c2)cc1
Oc1cccc(NC(=O)Cc2ccc(OC(F)F)cc2)c1
Oc1cccc(NC(=O)Cc2ccc(OC(F)(F)F)cc2)c1
Oc1cccc(NC(=O)Cc2ccc(cc2)C(F)(F)F)c1
Oc1cccc(NC(=O)Cc2ccc(Br)cc2)c1
Oc1cccc(NC(=O)Cc2ccc(Cl)cc2)c1
Oc1cccc(NC(=O)Cc2ccc(F)cc2)c1
Oc1cccc(NC(=O)Cc2ccc(cc2)-c2ccccc2)c1
CCCCCc1ccc(CC(=O)Nc2cccc(O)c2)cc1
COc1ccc(CC(=O)Nc2cccc(N)c2)cc1
COC(=O)c1cccc(NC(=O)Cc2ccc(OC)cc2)c1
COc1ccc(CC(=O)Nc2cccc(c2)C(O)=O)cc1
COc1ccc(CC(=O)Nc2ccccc2)cc1
COc1ccc(CC(=O)Nc2cccc(c2)B(O)O)cc1
CC(C)(C)c1ccc(CC(=O)Nc2cccc(O)c2)cc1
CC(C)c1ccc(CC(=O)Nc2cccc(O)c2)cc1
CCCc1ccc(CC(=O)Nc2cccc(O)c2)cc1
Cc1ccc(CC(=O)Nc2cccc(O)c2)cc1
Oc1cccc(NC(=O)Cc2ccc(OCc3ccccc3)cc2)c1
CCOc1ccc(CC(=O)Nc2cccc(O)c2)cc1
Oc1ccc(CC(=O)Nc2cccc(O)c2)cc1
COc1cccc(CC(=O)Nc2cccc(O)c2)c1
COc1ccccc1CC(=O)Nc1cccc(O)c1
Oc1cccc(NC(=O)Cc2ccccc2)c1
COc1ccc(CC(=O)Nc2ccc3OC(F)(F)Oc3c2)cc1
COc1ccc(CC(=O)Nc2ccc3C(=O)NCc3c2)cc1
COc1ccc(CC(=O)Nc2ccc3CNC(=O)c3c2)cc1
COc1ccc(CC(=O)Nc2ccc3C(=O)OCc3c2)cc1
COc1ccc(CC(=O)Nc2cccc(c2)C(C)=O)cc1
COc1ccc(CC(=O)Nc2ccc3COC(=O)c3c2)cc1
COc1ccc(CC(=O)Nc2ccc3CCC(=O)c3c2)cc1
COc1ccc(CC(=O)Nc2ccc3COCc3c2)cc1
COc1ccc(CC(=O)Nc2ccc3ncoc3c2)cc1
COc1ccc(CC(=O)Nc2cccc(OC(F)F)c2)cc1
COc1ccc(CC(=O)Nc2cccc(OC(F)(F)F)c2)cc1
COc1ccc(CC(=O)Nc2cccc(c2)C(F)(F)F)cc1
COc1ccc(CC(=O)Nc2cccc(Br)c2)cc1
COc1ccc(cc1)CC(=O)Nc2cccc(c2)Cl
COc1ccc(CC(=O)Nc2cccc(F)c2)cc1
COc1ccc(CC(=O)Nc2cccc(c2)[N+]([O-])=O)cc1
COc1ccc(CC(=O)Nc2cccc(C)c2)cc1
COc1ccc(CC(=O)Nc2ccc3COB(O)c3c2)cc1
COc1ccc(CC(=O)Nc2cccc(c2)C(C)(C)O)cc1
COc1ccc(CC(=O)Nc2cccc(CO)c2)cc1
COc1ccc(CC(=O)Nc2cccc(OC)c2)cc1
COc1ccc(CC(=O)Nc2ccc(O)cc2)cc1
COc1ccc(CC(=O)Nc2ccccc2O)cc1
COc1ccc(CC(=O)Nc2cccc(O)c2)cc1
COc1ccc(CC(=O)Nc2cccc(c2)S(N)(=O)=O)cc1
Oc1cccc(NC(=O)Cc2cc3ccccc3[nH]2)c1
Oc1cccc(NC(=O)Cc2cccc3[nH]ccc23)c1
Oc1cccc(NC(=O)Cc2c[nH]c3ccccc23)c1
Oc1cccc(NC(=O)Cn2ccc3ccccc23)c1
Oc1cccc(NC(=O)c2ccc3cc[nH]c3c2)c1
Oc1cccc(CNC(=O)Cc2ccc3cc[nH]c3c2)c1
Oc1cccc(c1)C(=O)NCc1ccc2cc[nH]c2c1
CN(C(=O)Cc1ccc2cc[nH]c2c1)c1cccc(O)c1
CCCOc1ccccc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)Cc1ccsc1
Clc1ccc(OCC#C)c(CN(CCc2ccc(cc2)S(=O)(=O)NCC#C)C(=O)Cc2ccsc2)c1
Oc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)Cc1ccsc1
Nc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)Cc1ccsc1
FC(F)(F)c1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)Cc1ccsc1
[O-][N+](=O)c1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)Cc1ccsc1
O=C(Cc1ccsc1)N(CCc1ccc(cc1)S(=O)(=O)NCC#C)Cc1cccc2OCOc12
O=C(Cc1ccsc1)N(CCc1ccc(cc1)S(=O)(=O)NCC#C)Cc1ccco1
CCCOc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC(C)(C)C)C(=O)Cc1ccsc1
CCCOc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)N(C)CC#C)C(=O)Cc1ccsc1
CCCOc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)N1CCOCC1)C(=O)Cc1ccsc1
CCCOc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)CC#C)C(=O)Cc1ccsc1
CCCOc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)Cc1ccsc1
CCCOc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)CCCc1ccsc1
CCCOc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)Cc1ccc(F)cc1
CCCOc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)Cc1csc2ccccc12
CCCOc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)c1csc2ccccc12
CCCOc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)c1ccc(F)cc1
CCCOc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)c1ccc(O)cc1
CCCOc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)c1ccc(cc1)[N+]([O-])=O
CCCOc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)c1ccc(cc1)B1OC(C)(C)C(C)(C)O1
CCCOc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)NCC#C)C(=O)c1csc2CCCCc12
CCCOc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)N1CCC1)C(=O)Cc1ccc(F)cc1
CCCOc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)N1CCC1)C(=O)c1csc2ccccc12
Fc1ccc(CC(=O)N(CCc2ccc(cc2)S(=O)(=O)NCC#C)Cc2cccc3OCOc23)cc1
Fc1ccc(cc1)C(=O)N(CCc1ccc(cc1)S(=O)(=O)NCC#C)Cc1cccc2OCOc12
CCCOc1ccc(Cl)cc1CN(CCc1ccc(cc1)S(=O)(=O)CC#C)C(=O)c1csc2ccccc12
CC(C)(C)c1coc(c1)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
Cc1cc(=O)n2nc(Nc3c4CCCc4cc4CCCc34)nc2n1C
Cc1ccn2nc(Nc3c4CCCc4cc4CCCc34)nc2n1
Cc1cc2[nH]c(Nc3c4CCCc4cc4CCCc34)nn2c(=O)n1
Cc1c[nH]c2nc(Nc3c4CCCc4cc4CCCc34)nn2c1=O
Cc1[nH]c2nc(Nc3c4CCCc4cc4CCCc34)nn2c(=O)c1C
Cc1[nH]c2nc(Nc3c4CCCc4cc4CCCc34)nn2c(=O)c1Cc1ccccc1
COc1c(C)[nH]c2nc(Nc3c4CCCc4cc4CCCc34)nn2c1=O
Cc1[nH]c2nc(Nc3c4CCCc4cc4CCCc34)nn2c(=O)c1C#N
CCc1cc(=O)n2nc(Nc3c4CCCc4cc4CCCc34)nc2[nH]1
COCCc1cc(=O)n2nc(Nc3c4CCCc4cc4CCCc34)nc2[nH]1
O=c1cc(Cc2ccccc2)[nH]c2nc(Nc3c4CCCc4cc4CCCc34)nn12
O=c1cc(CCc2ccccc2)[nH]c2nc(Nc3c4CCCc4cc4CCCc34)nn12
O=c1cc([nH]c2nc(Nc3c4CCCc4cc4CCCc34)nn12)C1CCOCC1
O=c1cc([nH]c2nc(Nc3c4CCCc4cc4CCCc34)nn12)C1CCNCC1
CN1CCC(CC1)c1cc(=O)n2nc(Nc3c4CCCc4cc4CCCc34)nc2[nH]1
O=c1cc([nH]c2nc(Nc3c4CCCc4cc4CCCc34)nn12)C1CCCNC1
CN1CCCC(C1)c1cc(=O)n2nc(Nc3c4CCCc4cc4CCCc34)nc2[nH]1
O=c1cc(CC2CCCCC2)[nH]c2nc(Nc3c4CCCc4cc4CCCc34)nn12
COc1ccc(Cc2cc(=O)n3nc(Nc4c5CCCc5cc5CCCc45)nc3[nH]2)cc1
Clc1cccc(Cc2cc(=O)n3nc(Nc4c5CCCc5cc5CCCc45)nc3[nH]2)c1
Clc1ccc(Cc2cc(=O)n3nc(Nc4c5CCCc5cc5CCCc45)nc3[nH]2)cc1
O=c1cc(Cc2cccc(c2)C#N)[nH]c2nc(Nc3c4CCCc4cc4CCCc34)nn12
O=c1cc(Cc2ccc(cc2)C#N)[nH]c2nc(Nc3c4CCCc4cc4CCCc34)nn12
Cc1ccccc1Cc1cc(=O)n2nc(Nc3c4CCCc4cc4CCCc34)nc2[nH]1
Fc1ccccc1Cc1cc(=O)n2nc(Nc3c4CCCc4cc4CCCc34)nc2[nH]1
O=c1cc(Cc2ccccn2)[nH]c2nc(Nc3c4CCCc4cc4CCCc34)nn12
O=c1cc(Cc2cccnc2)[nH]c2nc(Nc3c4CCCc4cc4CCCc34)nn12
O=c1cc(Cc2ccncc2)[nH]c2nc(Nc3c4CCCc4cc4CCCc34)nn12
O=c1cc(Cc2ncccn2)[nH]c2nc(Nc3c4CCCc4cc4CCCc34)nn12
O=c1cc(CC2CCOC2)[nH]c2nc(Nc3c4CCCc4cc4CCCc34)nn12
O=c1cc(CC2CCCCO2)[nH]c2nc(Nc3c4CCCc4cc4CCCc34)nn12
O=c1cc(CC2CCOCC2)[nH]c2nc(Nc3c4CCCc4cc4CCCc34)nn12
O=c1cc(CN2CCOCC2)[nH]c2nc(Nc3c4CCCc4cc4CCCc34)nn12
O=c1cc(CC2CNCCO2)[nH]c2nc(Nc3c4CCCc4cc4CCCc34)nn12
CN1CCOC(Cc2cc(=O)n3nc(Nc4c5CCCc5cc5CCCc45)nc3[nH]2)C1
O=c1cc(CC2COCCN2)[nH]c2nc(Nc3c4CCCc4cc4CCCc34)nn12
CN1CCOCC1Cc1cc(=O)n2nc(Nc3c4CCCc4cc4CCCc34)nc2[nH]1
CN1CCN(Cc2cc(=O)n3nc(Nc4c5CCCc5cc5CCCc45)nc3[nH]2)CC1
Cn1nccc1Cc1cc(=O)n2nc(Nc3c4CCCc4cc4CCCc34)nc2[nH]1
Cn1ccc(Cc2cc(=O)n3nc(Nc4c5CCCc5cc5CCCc45)nc3[nH]2)n1
Cn1cc(Cc2cc(=O)n3nc(Nc4c5CCCc5cc5CCCc45)nc3[nH]2)cn1
Cn1cnc(Cc2cc(=O)n3nc(Nc4c5CCCc5cc5CCCc45)nc3[nH]2)c1
Cn1cncc1Cc1cc(=O)n2nc(Nc3c4CCCc4cc4CCCc34)nc2[nH]1
Cc1cc(=S)n2nc(Nc3c4CCCc4cc4CCCc34)nc2[nH]1
S=c1cc(Cc2ccccn2)[nH]c2nc(Nc3c4CCCc4cc4CCCc34)nn12
S=c1cc(CC2CCCCO2)[nH]c2nc(Nc3c4CCCc4cc4CCCc34)nn12
Cc1cc(C)cc(NC(=O)[N-]S(=O)(=O)c2cc(co2)C(C)(C)O)c1
COc1cc(OC)c(\C=C\[N+]([O-])=O)c(\C=C\c2ccc(NC(=O)c3ccccc3)cc2)c1
COc1cc(OC)c(\C=C\[N+]([O-])=O)c(\C=C\c2ccc(NC(=O)c3ccc4ccccc4c3)cc2)c1
COc1cc(OC)c(\C=C\[N+]([O-])=O)c(\C=C\c2ccc(NC(=O)\C=C\c3ccccc3)cc2)c1
COc1ccc(cc1)C(=O)Nc1ccc(\C=C\c2cc(OC)cc(OC)c2\C=C\[N+]([O-])=O)cc1
COc1cc(OC)c(\C=C\[N+]([O-])=O)c(\C=C\c2ccc(NC(=O)c3ccc(F)cc3)cc2)c1
COc1cc(OC)c(\C=C\[N+]([O-])=O)c(\C=C\c2ccc(NC(=O)c3ccccc3Br)cc2)c1
COc1cc(OC)c(\C=C\[N+]([O-])=O)c(\C=C\c2ccc(NC(=O)c3ccco3)cc2)c1
COc1cc(OC)c(\C=C\[N+]([O-])=O)c(\C=C\c2ccc(NC(=O)c3cccs3)cc2)c1
[H][C@@]12CC[C@]3([H])[C@@]([C@@H]1O)(C(=O)C2=C)[C@]1(O)OC[C@]32[C@@H](O)CCC(C)(C)[C@@]2([H])[C@@H]1O |r,THB:10:9:7:4.3.2,12:11:7:4.3.2|
O=C(Nc1c2CCCc2cc2CCCc12)NS(=O)(=O)c1nccs1
O=C(Nc1c2CCCc2cc2CCCc12)NS(=O)(=O)c1cnccn1
O=C(Nc1c2CCCc2cc2CCCc12)NS(=O)(=O)c1ccncc1
O=C(Nc1c2CCCc2cc2CCCc12)NS(=O)(=O)c1cccnc1
O=C(Nc1c2CCCc2cc2CCCc12)NS(=O)(=O)c1ccccn1
O=C(Nc1c2CCCc2cc2CCCc12)NS(=O)(=O)c1ccco1
Cc1ncc(s1)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
Cc1nc(cn1C)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
Cn1nccc1S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
Cn1ccc(n1)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
Cn1cc(cn1)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
CC(C)n1cc(cn1)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
Cc1c(cnn1C)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
O=C(Nc1c2CCCc2cc2CCCc12)NS(=O)(=O)c1cnn2CCCCc12
O=C(Nc1c2CCCc2cc2CCCc12)NS(=O)(=O)c1cnn2CCCOc12
O=C(Nc1c2CCCc2cc2CCCc12)NS(=O)(=O)c1cnn2cccnc12
CN1CCn2ncc(c2C1=O)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
CN[C@H]1Cn2c(c(cn2)S(=O)(=O)NC(=O)Nc3c4c(cc5c3CCC5)CCC4)OC1
CN[C@H]1COc2c(cnn2C1)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12 |r|
CN(C)[C@@H]1COc2c(cnn2C1)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12 |r|
COC1CN(C1)[C@@H]1COc2c(cnn2C1)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12 |r|
CN(C)CC1COc2c(cnn2C1)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
CN1CCC[C@H](C1)Nc1nnc(c(C)n1)-c1ccc(cc1O)C(F)(F)F |r|
CN1CCC[C@H](C1)Nc1nnc(c(C)n1)-c1ccc(cc1O)C1CC1 |r|
COc1ccc(c(O)c1)-c1nnc(N[C@@H]2CCCN(C)C2)nc1C |r|
CN1CCC[C@H](C1)Nc1nnc(c(C)n1)-c1ccc(Cl)cc1O |r|
CN1CCC[C@H](C1)Nc1nnc(c(C)n1)-c1c(O)cc(C)cc1F |r,wD:5.7,(1.33,-5,;2.66,-4.23,;4,-5,;5.33,-4.23,;5.33,-2.69,;4,-1.92,;2.66,-2.69,;4,-.38,;2.66,.39,;1.34,-.38,;-0,.38,;-0,1.92,;1.33,2.69,;1.33,4.23,;2.66,1.93,;-1.33,2.69,;-2.66,1.93,;-2.66,.39,;-4,2.69,;-4,4.23,;-5.33,5,;-2.66,5,;-1.33,4.23,;-0,5,)|
COc1cc(O)c(c(F)c1)-c1nnc(N[C@@H]2CCCN(C)C2)nc1C |r,wD:15.15,(-6,4.23,;-4.66,5,;-3.33,4.23,;-3.33,2.69,;-1.99,1.93,;-1.99,.39,;-.67,2.69,;-.67,4.23,;.67,5,;-2,5,;.67,1.92,;.67,.38,;2,-.38,;3.33,.39,;4.66,-.38,;4.66,-1.92,;6,-2.69,;6,-4.24,;4.66,-5,;3.33,-4.24,;2,-5,;3.33,-2.69,;3.33,1.93,;2,2.69,;2,4.23,)|
CCOC(=O)Cn1nc(Cc2ccccc2Cl)oc1=O
OC(=O)Cn1nc(Cc2ccccc2Cl)oc1=O
COC(=O)c1ccc(cc1)-c1cn(Cc2cc(Cl)ccc2OC)nn1
CCCOc1ccc(Cl)cc1Cn1cc(nn1)-c1ccc(cc1)C(=O)OC
COc1ccc(cc1)-c1cn(Cc2cc(Cl)ccc2OC)nn1
COC(=O)[C@H]1CCCN1C(=O)Nc1c2CCCc2cc2CCCc12 |r|
COC(=O)[C@@H]1CCCN1C(=O)Nc1c2CCCc2cc2CCCc12 |r|
COC(=O)CN1CC(=O)N(C1=O)c1c2CCCc2cc2CCCc12
CCOC(=O)c1cnc(Nc2c3CCCc3cc3CCCc23)[nH]1
CCOC(=O)c1cnc(Nc2c3CCCc3cc3CCCc23)o1
CCOC(=O)c1coc(Nc2c3CCCc3cc3CCCc23)n1
CCOC(=O)c1nnc(Nc2c3CCCc3cc3CCCc23)o1
CCOC(=O)c1cnc(Nc2c3CCCc3cc3CCCc23)s1
COC(=O)c1ccnc(Nc2c3CCCc3cc3CCCc23)n1
OC(=O)c1cnc(Nc2c3CCCc3cc3CCCc23)o1
NC(=O)c1cnc(Nc2c3CCCc3cc3CCCc23)o1
CNC(=O)c1cnc(Nc2c3CCCc3cc3CCCc23)o1
CS(=O)(=O)NC(=O)c1cnc(Nc2c3CCCc3cc3CCCc23)o1
CN1CCN(C(=O)c2cnc(Nc3c4CCCc4cc4CCCc34)o2)S1(=O)=O
CSc1ccc(cc1)C(=O)\C=C\c1cc(O)cc(O)c1
COc1ccc(cc1)C(=O)\C=C\c1cc(C)c(O)c(C)c1
CCOC(=O)CSc1ccc(cc1)C(=O)\C=C\c1cc(C)c(O)c(C)c1
CCN(CC)C(=S)Sc1ccc(cc1)C(=O)\C=C\c1cc(C)c(O)c(C)c1
COC(=O)C1(CC1)C(=O)Nc1ccc(cc1)C(=O)\C=C\c1cc(C)c(O)c(C)c1
CN(C)CCC(=O)Nc1ccc(cc1)C(=O)\C=C\c1cc(C)c(O)c(C)c1
CCN(CC)C(=S)SCCC(=O)Nc1ccc(cc1)C(=O)\C=C\c1cc(C)c(O)c(C)c1
Cc1cc(\C=C\C(=O)c2ccc(cc2)C(O)=O)cc(C)c1O
CCOC(=O)c1ccc(cc1)C(=O)\C=C\c1cc(C)c(O)c(C)c1
COC(=O)CNC(=O)c1ccc(cc1)C(=O)\C=C\c1cc(C)c(O)c(C)c1
Cc1cc(\C=C\C(=O)c2ccc(cc2)C(=O)NCC(O)=O)cc(C)c1O
COC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc(cc1)C(=O)\C=C\c1cc(C)c(O)c(C)c1 |r|
Cc1cc(\C=C\C(=O)c2ccc(cc2)C(=O)N[C@@H](Cc2ccccc2)C(O)=O)cc(C)c1O |r|
CNC(=O)CNC(=O)c1ccc(cc1)C(=O)\C=C\c1cc(C)c(O)c(C)c1
CCNC(=O)CNC(=O)c1ccc(cc1)C(=O)\C=C\c1cc(C)c(O)c(C)c1
Cc1cc(\C=C\C(=O)c2ccc(cc2)C(=O)NCC(=O)Nc2ccccc2)cc(C)c1O
CN(C)C(=O)CNC(=O)c1ccc(cc1)C(=O)\C=C\c1cc(C)c(O)c(C)c1
CCN(CC)C(=O)CNC(=O)c1ccc(cc1)C(=O)\C=C\c1cc(C)c(O)c(C)c1
Cc1cc(\C=C\C(=O)c2ccc3c(COC33CNC3)c2)cc(C)c1O
CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc(cc1)C(=O)\C=C\c1cc(C)c(O)c(C)c1)B(O)O |r|
CCN1CCC[C@H](C1)Nc1nc2nc(ccc2o1)-c1c(C)cc(Cl)cc1O |r|
[H][C@@]12CCN(c3nc4nc(ccc4o3)-c3c(C)cc(Cl)cc3O)[C@]1([H])CN(C)CC2 |r|
CCN1CCC[C@@H](C1)Nc1nc2nc(ccc2o1)-c1c(C)cc(Cl)c(F)c1O
[H][C@]12CCCN1CCC[C@@H]2Nc1nc2nc(ccc2o1)-c1c(C)cc(Cl)cc1O |r|
COC(=O)CCN1CCC[C@@H](C1)Nc1nc2nc(ccc2o1)-c1c(C)cc(Cl)cc1O |r|
CCN1CCC[C@@H](C1)Nc1nc2nc(ccc2o1)-c1c(C)cc(Cl)cc1O
CCN1CCC[C@H](C1)Nc1cc(C)c(nn1)-c1ccc(cc1O)C#N
CCN1CCC[C@H](C1)Nc1ccc(nn1)-c1c(C)cc(cc1O)C#N |r|
[H][C@@]12CCN(c3ccc(nn3)-c3c(C)cc(cc3O)C#N)[C@]1([H])CN(C)CC2 |r|
CN1CCC2CCN(C2C1)c1cc(C)c(nn1)-c1ccc(cc1O)C#N
[H][C@@]12CCN(c3cc(C)c(nn3)-c3ccc(cc3O)C#N)[C@]1([H])CN(C)CC2 |r|
CCN1CCC[C@H](C1)Nc1cc(CC)c(nn1)-c1ccc(cc1O)C#N |r|
CC(C)(O)c1cccc(c1)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
CC(C)(O)c1cc(Br)cc(c1)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
CC(=O)c1cccc(c1)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
CNC(=O)c1cccc(c1)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
CN(C)C(=O)c1cccc(c1)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
CN(C)Cc1cccc(c1)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
COC1CN(Cc2cccc(c2)S(=O)(=O)NC(=O)Nc2c3CCCc3cc3CCCc23)C1
CN(C)Cc1cc(ccn1)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
CN(C)Cc1cc(F)cc(c1)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
CN(C)Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
CN(C)c1ccc(cc1)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
CCN(C)Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
CCCN(C)Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
CCCCN(C)Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
CCCCCN(C)Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
O=C(Nc1c2CCCc2cc2CCCc12)NS(=O)(=O)c1ccc(CN2CCCCC2)cc1
O=C(Nc1c2CCCc2cc2CCCc12)NS(=O)(=O)c1ccc(CN2CCOCC2)cc1
CN1CCN(Cc2ccc(cc2)S(=O)(=O)NC(=O)Nc2c3CCCc3cc3CCCc23)CC1
CN(C)Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc1cc(C)cc(C)c1
CN(C)Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc1c(C)cccc1C
CCc1cccc(CC)c1NC(=O)NS(=O)(=O)c1ccc(CN(C)C)cc1
CC(C)c1cccc(C(C)C)c1NC(=O)NS(=O)(=O)c1ccc(CN(C)C)cc1
CN(C)Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc1c(cccc1-c1ccccc1)-c1ccccc1
CC(C)c1cccc(C(C)C)c1CC(=O)NS(=O)(=O)c1ccc(CN(C)C)cc1
CC(C)(C)OC(=O)Nc1ccc(cc1)-c1c2CCCc2c(NC(=O)NS(=O)(=O)c2cc(co2)C(C)(C)O)c2CCCc12
CN(C)c1ccc(cc1)-c1c2CCCc2c(NC(=O)NS(=O)(=O)c2cc(co2)C(C)(C)O)c2CCCc12
COC(=O)c1ccc(cc1)-c1c2CCCc2c(NC(=O)NS(=O)(=O)c2cc(co2)C(C)(C)O)c2CCCc12
CC(C)(O)c1coc(c1)S(=O)(=O)NC(=O)Nc1c2CCCc2c(c2CCCc12)-c1ccc(C=O)cc1
CC(C)(O)c1coc(c1)S(=O)(=O)NC(=O)Nc1c2CCCc2c(c2CCCc12)-c1cccc(c1)C#N
CC(C)(C)OC(=O)N1CCC(=CC1)c1c2CCCc2c(NC(=O)NS(=O)(=O)c2cc(co2)C(C)(C)O)c2CCCc12 |c:10|
CC(C)(C)OC(=O)N1CCCC(=C1)c1c2CCCc2c(NC(=O)NS(=O)(=O)c2cc(co2)C(C)(C)O)c2CCCc12 |c:11|
CC(C)c1nn(CC(=O)NC2CCOCC2)c(=O)c2cccn12
CC(C)c1nn(CC(=O)NC2CCOCC2)c(=O)c2ccc(-c3ccsc3)n12
CC(C)c1nn(CC(=O)NC2CCOCC2)c(=O)c2ccc(-c3ccc(Cl)s3)n12
CC(C)c1nn(CC(=O)NC2CCOCC2)c(=O)c2cc(NC3COC3)cn12
CC(C)c1nn(CC(=O)NC2CCOCC2)c(=O)c2cc(Nc3ccccc3)cn12
CC(C)c1nn(CC(=O)NC2CCOCC2)c(=O)c2cc3ccccc3n12
CC(C)c1nn(CC(=O)NC2CCOCC2)c(=O)c2cc3cc(Cl)ccc3n12
O=C(CN1CCn2c(cc3sccc23)C1=O)NC1CCOCC1
O=C(CNC(=O)c1cc2sccc2[nH]1)NC1CCOCC1
CC(C)c1nn(Cc2nnc(o2)C2CCOCC2)c(=O)c2cc3sccc3n12
CC(C)c1nn(Cc2nnc(o2)C2CCOCC2)c(=O)c2cc3sc(Cl)cc3n12
CC(C)c1nn(Cc2nnc(o2)-c2cccnc2)c(=O)c2cc3sc(Cl)cc3n12
CC(C)c1nn(Cc2nnc([nH]2)-c2cccnc2)c(=O)c2cc3sc(Cl)cc3n12
CC(C)c1nn(Cc2nnc(o2)C2CCC2)c(=O)c2cc3sc(Cl)cc3n12
CC(C)c1nn(Cc2nnc(o2)C2CCCC2)c(=O)c2cc3sc(Cl)cc3n12
CC(C)c1nn(Cc2nnc(o2)C2CCOC2)c(=O)c2cc3sc(Cl)cc3n12
CC(C)c1nn(Cc2nnc(o2)C2CCCCC2)c(=O)c2cc3sc(Cl)cc3n12
CC(C)c1nn(Cc2nnc(o2)-c2cccc(c2)C#N)c(=O)c2cc3sc(Cl)cc3n12
CC(C)c1nn(Cc2nnc(o2)-c2cccc(F)c2)c(=O)c2cc3sc(Cl)cc3n12
CC(C)c1nn(Cc2nnc(o2)-c2cccc(c2)C(F)(F)F)c(=O)c2cc3sc(Cl)cc3n12
COc1cccc(c1)-c1nnc(Cn2nc(C(C)C)n3c4cc(Cl)sc4cc3c2=O)o1
CC(C)c1nn(Cc2nnc(o2)-c2cccc(C)c2)c(=O)c2cc3sc(Cl)cc3n12
CC(C)c1nn(Cc2nnc(o2)-c2cnccc2Cl)c(=O)c2cc3sc(Cl)cc3n12
CC(C)c1nn(Cc2nnc(o2)-c2ncccc2Cl)c(=O)c2cc3sc(Cl)cc3n12
CC(C)c1nn(Cc2nnc(o2)-c2ccncc2Cl)c(=O)c2cc3sc(Cl)cc3n12
CC(C)c1nn(Cc2nnc(o2)-c2cccnc2Cl)c(=O)c2cc3sc(Cl)cc3n12
CC(C)c1nn(Cc2nnc(o2)-c2cnccc2C(F)(F)F)c(=O)c2cc3sc(Cl)cc3n12
CC(C)c1nn(Cc2nnc(o2)-c2cncc(c2)C(F)(F)F)c(=O)c2cc3sc(Cl)cc3n12
CC(C)c1nn(Cc2nnc(o2)-c2ccc(nc2)C(F)(F)F)c(=O)c2cc3sc(Cl)cc3n12
CC(C)c1nn(Cc2nnc(o2)-c2ccc(C)nc2)c(=O)c2cc3sc(Cl)cc3n12
CC(C)c1nn(Cc2nnc(o2)-c2cnccn2)c(=O)c2cc3sc(Cl)cc3n12
CC(C)c1nn(Cc2nnc(o2)-c2ccncn2)c(=O)c2cc3sc(Cl)cc3n12
CC(C)c1nn(Cc2nnc(o2)-c2ccnc(Cl)n2)c(=O)c2cc3sc(Cl)cc3n12
CC(C)c1nn(Cc2nnc(o2)-c2ccc(C)nc2Cl)c(=O)c2cc3sc(Cl)cc3n12
CC(C)c1nn(Cc2nnc(o2)-c2ccc(F)nc2F)c(=O)c2cc3sc(Cl)cc3n12
CC(C)c1nn(Cc2nnc(o2)-c2cc(F)cnc2Cl)c(=O)c2cc3sc(Cl)cc3n12
CC(C)c1nn(Cc2nnc(o2)-c2cc(cnc2Cl)C(F)(F)F)c(=O)c2cc3sc(Cl)cc3n12
CC(C)c1nn(Cc2nnc(o2)-c2ccc(nc2Cl)C(F)(F)F)c(=O)c2cc3sc(Cl)cc3n12
CC(C)c1nn([C@H](C)c2nnc(o2)-c2ccc(nc2Cl)C(F)(F)F)c(=O)c2cc3sc(Cl)cc3n12 |r|
CC(C)c1nn([C@@H](C)c2nnc(o2)-c2ccc(nc2Cl)C(F)(F)F)c(=O)c2cc3sc(Cl)cc3n12 |r|
CC(C)c1nn(CC(=O)NC2CCOCC2)c(=O)c2cc3sc(Cl)cc3n12
COC(=O)CN(C)C(=O)Nc1c2CCCc2cc2CCCc12
CCOC(=O)COC(=O)Nc1c2CCCc2cc2CCCc12
CCOC(=O)COC(=O)N(C)c1c2CCCc2cc2CCCc12
CCOC(=O)CNC(=O)Oc1c2CCCc2cc2CCCc12
CCOC(=O)COC(=O)Nc1ccccc1C#N
CCOC(=O)COC(=O)Nc1ccccc1C(C)C
CCOC(=O)COC(=O)Nc1ccccc1C(F)(F)F
CCOC(=O)COC(=O)Nc1ccccc1OC(F)(F)F
CCOC(=O)COC(=O)Nc1cc(C)ccc1C
CCOC(=O)COC(=O)Nc1cccc(C)c1C
CCOC(=O)COC(=O)Nc1c(C)cccc1C
CCOC(=O)COC(=O)Nc1c(C)cc(C)cc1C
CCOC(=O)COC(=O)Nc1c(C)cccc1CC
CCOC(=O)COC(=O)Nc1c(C)cccc1C(C)C
CCOC(=O)COC(=O)Nc1c(C)cccc1C(C)(C)C
CCOC(=O)COC(=O)Nc1c(CC)cccc1CC
CCOC(=O)COC(=O)Nc1c(cccc1C(C)C)C(C)C
CCOC(=O)COC(=O)Nc1c(Cl)cccc1Cl
CCOC(=O)COC(=O)Nc1c(F)cccc1F
CCOC(=O)C(Cn1cccn1)OC(=O)Nc1c2CCCc2cc2CCCc12
CCOC(=O)C(Cn1cccn1)OC(=O)Nc1c(C)cccc1C
CCOC(=O)C(Cc1ncccn1)OC(=O)Nc1c2CCCc2cc2CCCc12
CCOC(=O)C(Cc1ncccn1)OC(=O)Nc1c(C)cccc1C
CCOC(=O)C(Cc1cnccn1)OC(=O)Nc1c2CCCc2cc2CCCc12
CCOC(=O)C(Cn1cc(cn1)C#N)OC(=O)Nc1c2CCCc2cc2CCCc12
CCOC(=O)C(Cn1cncn1)OC(=O)Nc1c2CCCc2cc2CCCc12
CC(C)OC(=O)[C@@H](Cn1cc(cn1)C#N)OC(=O)Nc1c2CCCc2cc2CCCc12 |r|
CC(C)OC(=O)[C@@H](Cn1cncn1)OC(=O)Nc1c2CCCc2cc2CCCc12 |r|
CC(C)OC(=O)[C@@H](Cc1cnccn1)OC(=O)Nc1c2CCCc2cc2CCCc12 |r|
O=C(Nc1c2CCCc2cc2CCCc12)O[C@H](Cc1ncccn1)C(=O)OC1CCCC1 |r|
CC(C)OC(=O)[C@H](Cc1ncccn1)OC(=O)Nc1c2CCCc2cc2CCCc12 |r|
CC(C)OC(=O)[C@@H](Cc1ncccn1)OC(=O)Nc1c2CCCc2cc2CCCc12 |r|
OC(=O)[C@@H](Cc1ncccn1)OC(=O)Nc1c2CCCc2cc2CCCc12 |r|
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)NC(=O)c1cc(Cl)ccc1OC
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)NC(=O)c1cc(Cl)ccc1OCCC
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)NC(=O)c1cc(Cl)ccc1OCCOC
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)NC(=O)c1cc(Cl)ccc1OCCN(C)C
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)NC(=O)c1cc(Cl)ccc1Cl
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)NC(=O)c1ncc(cc1O)-c1cccc(Cl)c1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)NC(=O)c1ncc(cc1OCCC)-c1cccc(Cl)c1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)NC(=O)c1ncc(cc1OCCOC)-c1cccc(Cl)c1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)NS(=O)(=O)c1cccs1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)NS(=O)(=O)c1ccc(Cl)s1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)NS(=O)(=O)c1ccc(Br)s1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)NC(=O)NCc1cc(Cl)ccc1OC
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)NC(=S)NCc1cc(Cl)ccc1OC
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCC)C(=O)Cc1ccsc1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)Cc1ccsc1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)c1cccs1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)C1CCOC1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)CC1CCOC1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)C1CCCCC1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)C1CCOCC1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)CC1CCOCC1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)c1ccccc1OC(C)=O
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)c1ccccc1O
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)c1csc(n1)-c1cccnc1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)c1ccc(cc1)N1CCN(CC1)C(=O)OC(C)(C)C
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)c1ccc(cc1)N1CCNCC1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)c1ccc2OCOc2c1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)C(C)(C)C
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)C(F)(F)F
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)CBr
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)C1CC1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)S(=O)(=O)C1CC1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)\C=C\CN1CCCCC1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)\C=C\c1ccccc1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)\C=C\c1ccc(O)cc1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)\C=C\c1ccc(O)c(O)c1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)\C=C\c1ccc(O)c(OC)c1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)\C=C/c1ccc(O)cc1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)\C=C/c1ccc(O)c(OC)c1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)c1cc2ccccc2o1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)c1cc2ccccc2[nH]1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)c1cc2ccccc2s1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)c1nc2ccccc2s1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)c1cc2cc(F)ccc2o1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)c1cc2cc(Cl)ccc2o1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)c1cc2cc(Br)ccc2o1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)c1cc2cc(OC)ccc2o1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)c1cc2cc(O)ccc2o1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)c1cc2cc(OC(=O)C(C)(C)C)ccc2o1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)c1ccc2ccccc2c1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)c1ccc2ccccc2n1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)c1ccc2cnccc2n1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)S(=O)(=O)c1ccc2CCN(Cc2c1)C(=O)C(F)(F)F
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)S(=O)(=O)c1ccc2CCNCc2c1
CCC(=O)NS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)c1cc2ccccc2o1
CCCCN(CCCC)S(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)c1cc2ccccc2o1
COCCOc1ccc(Cl)cc1CN(C1Cc2ccc(cc2C1)S(=O)(=O)Nc1c2CCCc2cc2CCCc12)C(=O)c1cc2ccccc2o1
COCCOc1ccc(Cl)cc1CN(C1Cc2ccc(cc2C1)S(=O)(=O)NCC#C)C(=O)c1cc2ccccc2o1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(Cl)ccc1OCCN(C)C)C(=O)c1cc2ccccc2o1
CCCNS(=O)(=O)c1ccc2CC(Cc2c1)N(Cc1cc(F)ccc1OCCOC)C(=O)c1cc2ccccc2o1
CCCNS(=O)(=O)c1ccc2C[C@@H](Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)c1cc2ccccc2o1 |r|
CCCNS(=O)(=O)c1ccc2C[C@H](Cc2c1)N(Cc1cc(Cl)ccc1OCCOC)C(=O)c1cc2ccccc2o1 |r|
Cc1cccc2c3C(=O)C(=O)c4c5CCN(CCCN6CCOCC6)Cc5oc4-c3ccc12
CC(C)[C@H](NS(=O)(=O)c1ccc(cc1)[N+]([O-])=O)C(=O)Nc1c2CCCc2cc2CCCc12 |r|
Nc1ccc(cc1)S(=O)(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)Nc1c2CCCc2cc2CCCc12 |r|
Nc1ccc(cc1)S(=O)(=O)N1Cc2ccccc2C[C@H]1C(=O)Nc1c2CCCc2cc2CCCc12 |r|
CC(C)(O)c1ccoc1S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
CCCOc1nc(N)nc2nc(ccc12)-c1cc[nH]n1
Nc1nc(NC2CCOCC2)c2ccc(nc2n1)-c1cc[nH]n1
CCNc1nc(N)nc2cc(ccc12)-c1cc[nH]n1
Nc1nc(NCCn2cccn2)c2ccc(nc2n1)-c1cc[nH]n1
CCNc1nc(N)nc2nc(ccc12)-c1cc[nH]n1
CCNc1nc(N)nc2cc(ccc12)-n1cccn1
CCNc1nc(N)nc2cc(cnc12)-n1cccn1
CCNc1nc(N)nc2nc(ccc12)-n1cccn1
CCNc1nc(N)nc2nc(ccc12)-c1ccc[nH]c1=O
CCNc1nc(N)nc2nc(ccc12)-c1ccccc1
CCNc1cc(N)nc2cc(ccc12)-n1cccn1
Nc1cc(NCCn2cccn2)c2ccccc2n1
C(Cn1cccn1)Nc1ccnc2cc(ccc12)-n1cccn1
CCN(Cc1nc2c(N)nc3cc(ccc3c2[nH]1)-c1cc[nH]n1)C(C)=O
Nc1cc(NCCn2cccn2)c2ccc(cc2n1)-n1cccn1
Cn1nccc1CNc1nc(N)nc2nc(ccc12)-c1cc[nH]n1
Cn1ccc(CNc2nc(N)nc3nc(ccc23)-c2cc[nH]n2)n1
Cn1cc(CNc2nc(N)nc3nc(ccc23)-c2cc[nH]n2)cn1
Nc1nc(NC2CC2)c2ccc(nc2n1)-c1cc[nH]n1
CC1(CC1)Nc1nc(N)nc2nc(ccc12)-c1cc[nH]n1
CC1(CC1)Nc1nc(N)nc2cc(ccc12)-c1cc[nH]n1
Cn1ccc(CNc2nc(N)nc3cc(ccc23)-c2cc[nH]n2)n1
CN(C)C\C=C\S(=O)(=O)NC(=O)Nc1c2CCCc2cc2C=CCc12 |c:22|
CC(C)(N)\C=C\[S+]([O-])(NC(=O)Nc1c2CCCc2cc2CCCc12)=NC#N
CN(C)C\C=C\S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
CC1(C)CCc2c1cc1CCCc1c2NC(=O)NS(=O)(=O)c1ccnn1CCCB(O)O
O=C(Nc1c2CCCc2ccc1C1CC1)NS(=O)(=O)c1cc2CN3CCC(CC3)c2o1 |(-1.88,1.81,;-1.88,.27,;-3.22,-.5,;-4.55,.27,;-4.55,1.81,;-3.41,2.84,;-4.03,4.24,;-5.56,4.08,;-5.88,2.58,;-7.21,1.81,;-7.21,.26,;-5.88,-.5,;-5.88,-2.04,;-6.65,-3.38,;-5.11,-3.37,;-.55,-.5,;.79,.27,;-.3,1.36,;1.56,1.6,;2.12,-.5,;3.53,.13,;4.56,-1.02,;6.08,-.78,;7.21,-1.82,;7.11,-3.36,;5.84,-4.24,;4.36,-3.8,;4.61,-2.25,;5.78,-1.4,;3.79,-2.35,;2.28,-2.03,)|
CC(C)c1cc(F)cc(C(C)C)c1NC(=O)NS(=O)(=O)c1cc2c(CCCC2(C)O)o1
CN1CCC(CC1)Oc1cc(ccn1)-c1c(C)cc2CCCc2c1NC(=O)N[S+]([O-])(=N)c1ccccc1
CC(C)c1cc(F)cc(C(C)C)c1NC(=O)N=[S+](N)([O-])c1ccc2ccccc2c1
CC(C)c1cc(F)cc(C(C)C)c1NC(=O)N=[S+](N)([O-])c1ccccc1-c1ccccc1
C[C@H](O)Cn1cc(F)c(n1)[S+](N)([O-])=NC(=O)Nc1c2CCCc2nc2c1CCC21CC1 |r|
N[S+]([O-])(=NC(=O)Nc1c2CCCc2nc(C2CC2)c1C1CC1)c1nn(cc1F)C1CC1
N[S+]([O-])(=NC(=O)Nc1c2CCCc2nc(c1C1CC1)C(F)(F)F)c1nn(cc1F)C1CC1
Fc1cnc(NC(=O)CN2CC3(CC3)c3cc(Br)ccc3C2=O)nc1
C[C@@]1(O)C[C@@H](C1)NC(=O)CN1C[C@@]2(C[C@@H]2F)c2cc(I)ccc2C1=O |r,wD:12.12,4.6,1.1,14.16,(7.09,.85,;6.32,-.48,;7.8,-.88,;5.53,-1.84,;4.2,-1.07,;4.98,.29,;2.86,-1.83,;1.53,-1.06,;1.53,.48,;.19,-1.83,;-1.14,-1.06,;-1.13,.48,;-2.47,1.26,;-3.24,2.59,;-1.7,2.59,;-.36,3.36,;-3.8,.49,;-5.13,1.26,;-6.47,.49,;-7.8,1.26,;-6.47,-1.05,;-5.14,-1.82,;-3.8,-1.05,;-2.47,-1.82,;-2.48,-3.36,)|
CC(C)c1cc(cc(C(C)C)c1CC(=O)NS(=O)(=O)c1sc(nc1CO)C(C)(C)O)-c1ccc2OC(F)(F)Oc2c1
CC(C)c1cc(C#N)c(F)c(C(C)C)c1CC(=O)NS(=O)(=O)c1sc(nc1CCO)C(C)(C)O
CC(C)c1cc(cc(C(C)C)c1CC(=O)NS(=O)(=O)c1ccc(CN(C)C)cc1)-c1cccc2ccccc12
COc1cc(ccn1)-c1ccc2CCCc2c1NC(=O)NS(=O)(=O)c1nc(c[se]1)C(C)(C)O
COc1cc(ccn1)-c1cccc(C(C)C)c1NC(=O)NS(=O)(=O)c1nc(c[se]1)C(C)(C)O
CC(C)(O)c1coc(n1)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
C[C@@H]1CCc2c1nc1CCCc1c2NC(=O)N=[S+]1([O-])NC(=O)c2ccc(cc12)C(C)(C)O |r|
CC(C)c1cc(NC(=O)NS(=O)(=O)C(C2CCCN(C)C2)c2cnn(C)c2)c(s1)C(C)C
CCc1oc(cc1NC(=O)NS(=O)(=O)C(C1CCCN(C)C1)c1cnn(C)c1)C(C)C
CCN1CCC[C@@H](C1)Nc1ccc(nn1)-c1c(C)cc(cc1O)C(F)(F)F |r|
CN1CCC[C@H](C1)Nc1cc(C)c(nn1)-c1ccc(cc1O)C(F)(F)F |r|
CN1CCC[C@H](C1)Nc1cc(c(nn1)-c1ccc(cc1O)C(F)(F)F)C(F)(F)F |r|
CC1(O)CCCc2oc(cc12)S(=O)(=O)NC(=O)Nc1c2CCCc2c(Br)c2CCCc12
C[C@@]1(CO)Cn2ncc(c2O1)[S@@+](N)([O-])=NC(=O)Nc1c2CCCc2cc2CCCc12 |r|
CC(C)(O)c1ccc2C(=O)N=[S+]([O-])(NC(=O)Nc3c4CCCc4cc4CCCc34)c2c1
COC(=O)c1cccc(c1)C(=O)NC1(CC1)C(=O)Nc1c2CCCc2cc2CCCc12
COC(C)(C)Cn1ccc(n1)S(=O)(=O)c1nnc(Nc2c3CCCc3cc3CCCc23)[nH]1
CC(C)OC(=O)c1nc(Nc2c3CCCc3cc3CCCc23)cs1
COc1cc(C)c(cn1)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
CS(C)(=O)=Nc1ccc(s1)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
Cc1cc(NC2CCCN(C2)C2CCC2)nnc1-c1ccc2sccc2c1O
CN1CCC[C@H](C1)Nc1cc(C)c(nn1)-c1ccc2ccccc2c1O |r|
CN1CCC[C@H](C1)Nc1cc(C)c(nn1)-c1ccc(cc1O)-c1ccc(F)cc1 |r|
[O-][N+](=O)C1(CC(C1)C(=O)CBr)[N+]([O-])=O
Nc1ccc(cc1)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
C[C@@]1(O)CCCc2oc(cc12)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12 |r|
O=C(Nc1c2CCCc2cc2CCCc12)NS(=O)(=O)c1cc2CN3CCC(CC3)c2o1 |THB:30:29:24.25:27.28,(-1.31,1.81,;-1.31,.26,;-2.64,-.5,;-3.98,.27,;-3.97,1.82,;-2.83,2.85,;-3.47,4.25,;-5,4.09,;-5.31,2.58,;-6.64,1.81,;-6.64,.27,;-7.79,-.75,;-7.16,-2.16,;-5.64,-2,;-5.31,-.5,;.03,-.51,;1.36,.26,;.59,1.6,;2.13,1.6,;2.69,-.51,;4.1,.11,;5.13,-1.03,;6.65,-.8,;7.79,-1.83,;7.68,-3.38,;6.41,-4.25,;4.93,-3.81,;4.93,-2.27,;6.27,-1.5,;4.36,-2.36,;2.85,-2.04,)|
Cn1ncc2ccc(cc12)S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
CN1C[C@]2(C)CCCN2[C@H](CS(=O)(=O)NC(=O)Nc2c3CCCc3cc3CCCc23)C1(C)C |r|
N[S+]([O-])(=NC(=O)Nc1c2CCCc2cc2CCCc12)c1cnn2cc(CO)oc12
Fc1cn2CCOc3cc(ccn3)-c3ccc4CCCc4c3NC(=O)NS(=O)(=O)c1n2
CC(C)c1nn(CC(=O)N[C@@H]2CCCN(C2)C2CCC2)c(=O)c2cc3sc(Cl)cc3n12 |r|
CN(C)c1nn(CC(=O)N[C@H]2C[C@@](C)(O)C2)c(=O)c2cc3sccc3n12 |r,wU:10.9,12.13,(-2.73,3.67,;-1.64,2.58,;-.15,2.98,;-2.03,1.09,;-1,-.05,;-1.48,-1.52,;-.39,-2.61,;1.1,-2.21,;1.49,-.72,;2.19,-3.3,;3.67,-2.9,;4.46,-1.54,;5.79,-2.31,;7.28,-2.71,;6.56,-.98,;5.01,-3.67,;-2.99,-1.84,;-3.39,-3.32,;-4.02,-.69,;-5.56,-.69,;-6.03,.77,;-7.28,1.68,;-6.8,3.14,;-5.26,3.14,;-4.79,1.68,;-3.54,.77,)|
CC(C)c1nn(CC(=O)Nc2ccc3nncn3c2)c(=O)c2cc3ccccc3n12
CC(C)c1nn(CC(=O)Nc2ccncn2)c(=O)c2cc(I)nn12
CCNc1cc2n(n1)c(nn(CC(=O)Nc1ccc3nncn3c1)c2=O)C(C)C
CC(C)c1nn(CC(=O)N[C@H]2CN(CC[C@H]2O)C2CCC2)c(=O)c2cc(nn12)C1CC1 |r|
CC(C)c1nc2c(nn(CC(=O)Nc3ccc4nncn4c3)c(=O)c2s1)C(C)C
CC(C)c1nn(CC(=O)Nc2ccc3nncn3c2)c(=O)c2sc(nc12)C1CC1
CCNc1nc2c(nn(CC(=O)Nc3ccc4nncn4c3)c(=O)c2s1)C(C)C
CC(C)c1nn(CC(=O)N[C@H]2C[C@](C)(O)C2)c(=O)c2ccc(Br)cc12 |r,wD:10.9,12.12,(-4.89,.95,;-3.35,.95,;-2.58,2.28,;-2.58,-.38,;-1.04,-.22,;-.14,-1.47,;1.4,-1.47,;2.17,-.13,;1.4,1.2,;3.71,-.13,;4.48,1.2,;5.97,1.6,;5.56,3.11,;5.17,4.6,;6.9,3.88,;4.08,2.71,;-.77,-2.87,;0,-4.21,;-2.3,-3.04,;-2.92,-4.44,;-4.45,-4.6,;-5.36,-3.36,;-6.9,-3.36,;-4.74,-1.95,;-3.2,-1.79,)|
CC(C)c1nn(CC(=O)Nc2ncc3nc[nH]c3n2)c(=O)c2ccc(cc12)C(F)(F)F
CC(C)n1nc(CC(=O)Nc2ccc3n(C)c(=O)[nH]c3c2)c(=O)c2ccc(Br)cc12
CC(C)n1nc(CC(=O)Nc2ccncn2)c(=O)c2ccc(Br)cc12
CC(C)c1nn(CC(=O)Nc2ccc3nncn3n2)c(=O)cc1Nc1ccccc1
CC(C)c1nn(CC(=O)Nc2ccc3nncn3n2)c(=O)cc1N1CC2CC2C1
COC(=O)C12CC(C1)(C2)NC(=O)Cn1nc(C(C)C)c(OCC(C)C)cc1=O
CC(C)c1nn(CC(=O)Nc2ccc3nncn3c2)c(=O)cc1Oc1ccccc1
CC(C)c1nn(CC(=O)N[C@H]2C[C@@](C)(O)C2)c(=O)c2cc3ccsc3n12 |r,wU:10.9,12.13,(-4.82,.77,;-3.28,.77,;-2.51,2.1,;-2.51,-.57,;-.97,-.41,;-.07,-1.65,;1.47,-1.65,;2.24,-.32,;1.47,1.01,;3.78,-.32,;4.55,1.01,;4.14,2.53,;5.63,2.93,;6.97,3.7,;5.63,4.47,;6.04,1.41,;-.7,-3.06,;.07,-4.39,;-2.23,-3.22,;-3.13,-4.47,;-4.6,-3.99,;-6.06,-4.47,;-6.97,-3.22,;-6.06,-1.97,;-4.6,-2.45,;-3.13,-1.97,)|
CC(C)c1nn(CC(=O)N[C@H]2C[C@@](C)(O)C2)c(=O)c2cc3CC(C)(C)Cc3n12 |r,wD:10.9,12.13,(-4.07,.77,;-2.53,.77,;-1.76,2.1,;-1.76,-.57,;-.23,-.41,;.67,-1.65,;2.21,-1.65,;2.98,-.32,;2.21,1.01,;4.52,-.32,;5.29,1.01,;6.78,1.41,;6.38,2.93,;7.71,3.7,;6.38,4.47,;4.89,2.53,;.05,-3.06,;.82,-4.39,;-1.48,-3.22,;-2.39,-4.47,;-3.85,-3.99,;-5.32,-4.47,;-6.22,-3.22,;-7.31,-2.13,;-7.71,-3.62,;-5.32,-1.97,;-3.85,-2.45,;-2.39,-1.97,)|
CC(C)Sc1cc2n(c1)c(nn(CC(=O)N[C@H]1C[C@@](C)(O)C1)c2=O)C(C)C |r,wD:16.16,18.20,(-7.12,-5.77,;-5.78,-5,;-4.45,-5.77,;-5.78,-3.46,;-4.45,-2.69,;-2.98,-3.16,;-2.08,-1.92,;-2.98,-.67,;-4.45,-1.15,;-2.36,.73,;-.82,.9,;.08,-.35,;1.62,-.35,;2.39,.98,;1.62,2.32,;3.93,.98,;4.7,2.32,;6.19,2.72,;5.78,4.23,;7.12,5,;5.78,5.77,;4.29,3.83,;-.55,-1.76,;.22,-3.09,;-3.13,2.07,;-4.67,2.07,;-2.36,3.4,)|
CC(C)c1nn(CC(=O)Nc2ccncn2)c(=O)c2cccn12
CC(C)c1nn(CC(=O)Nc2ccncn2)c(=O)c2cc(I)cn12
CC(C)c1cc2n(c1)c(nn(CC(=O)N[C@@H]1CCCN(C1)C1CCC1)c2=O)C(C)C |r|
CN1CCC[C@H](C1)Nc1nnc(c2COCc12)-c1ccc(cc1O)C(F)(F)F |r|
C[C@@]1(O)C[C@@H](C1)Nc1nnc(c2COCc12)-c1ccc(cc1O)C(F)(F)F |r,wU:1.0,wD:4.6,(7.71,-1.58,;6.17,-1.58,;6.57,-.1,;5.77,-3.1,;4.28,-2.7,;4.69,-1.19,;2.95,-3.47,;1.61,-2.7,;.28,-3.46,;-1.05,-2.69,;-1.05,-1.15,;.28,-.38,;.6,1.12,;2.13,1.28,;2.76,-.12,;1.61,-1.15,;-2.38,-.38,;-2.38,1.17,;-3.72,1.93,;-5.05,1.16,;-5.05,-.38,;-3.72,-1.15,;-3.72,-2.69,;-6.38,1.93,;-7.71,1.16,;-6.38,3.47,;-7.71,2.7,)|
CN1CCC[C@H](C1)Nc1cc(C)c(nn1)-c1ccc(cc1O)C1CC1 |r|
CC(C)c1nn(CC(=O)Nc2ncc(F)cn2)c(=O)c2ccc(Br)cc12
CC(C)c1nn(C(C)C(=O)Nc2ncc(F)cn2)c(=O)c2ccc(Br)cc12
CC(C)c1nn(CC(=O)Nc2ncncc2F)c(=O)c2ccc(cc12)C(F)(F)F
CC(C)c1nn(CC(=O)Nc2ncncc2F)c(=O)c2cc(ccc12)C(F)(F)F
Fc1c(Br)ccc2C(=O)N(CC(=O)Nc3ncc(Cl)cn3)C(=O)C3(CC3)c12
CCc1c(-c2cccc(F)c2)c(nn(CC(=O)Nc2ncncc2F)c1=O)C(C)C
CC(C)c1nn(CC(=O)Nc2ncccn2)c(=O)cc1-c1cc(F)cc(F)c1
CC(C)c1nn(c(=O)cc1-c1cc(F)cc(F)c1)C1(CC1)C(=O)Nc1ncccn1
CC(C)c1nn(CC(=O)N[C@@H]2CCCN(C2)C2CCC2)c(=O)cc1-c1cccc(Cl)c1 |r|
C[C@@H](O)CNc1nnc(c(C)c1C#N)-c1ccc(cc1O)C(F)(F)F |r|
Cc1c(C)c(nnc1N[C@@H]1CCCC[C@H]1O)-c1ccc(cc1O)C(F)(F)F |r|
CC(Nc1nnc(c(C)n1)-c1ccc(cc1O)C(F)(F)F)c1cccc(O)c1
Clc1ccc(cc1)-c1nnc(NCC2CCCO2)c2ccccc12
Clc1ccc(cc1)-c1nnc(NCC2CCCO2)c2cnccc12
C[C@@]1(O)C[C@@H](C1)Nc1nnc(c2CCCCc12)-c1ccc(cc1O)C#N |r,wD:4.6,1.1,(7.71,-1.2,;6.17,-1.2,;6.57,.29,;5.77,-2.71,;4.28,-2.31,;4.69,-.8,;2.95,-3.08,;1.61,-2.31,;.28,-3.08,;-1.05,-2.31,;-1.05,-.77,;.28,0,;.28,1.54,;1.61,2.31,;2.95,1.54,;2.95,0,;1.61,-.77,;-2.38,0,;-2.38,1.55,;-3.72,2.31,;-5.05,1.54,;-5.05,0,;-3.72,-.77,;-3.72,-2.31,;-6.38,2.31,;-7.71,3.08,)|
CN1CCC[C@H](C1)Nc1nnc(-c2ccc(C)cc2O)c2cscc12 |r|
CN1CCC[C@H](C1)Nc1nnc(-c2ccc(C)cc2O)c2C3CCC(C=C3)c12 |r,c:27|
CN1CCC[C@H](C1)Nc1nnc(-c2ncc(C)cc2O)c2ccccc12 |r|
CCN1CCC[C@H](C1)Nc1nnc(-c2ccc(Cl)cc2O)n(C)c1=O |r|
CCN1CCC[C@@H](C1)Nc1nnc(-c2ccc3OCCc3c2O)n(C)c1=O |r|
CCN1CCC[C@H](C1)Nc1ccc(nn1)-c1c(C)cc(cc1O)C(F)(F)F |r|
Cc1cc(cc(O)c1-c1ccc(Nc2cccnc2)nn1)C(F)(F)F
Cc1cc(cc(O)c1-c1ccc(Nc2cncnc2)nn1)C(F)(F)F
NS(=O)(=O)c1cccc(\C=C2/SC(=S)N(CC3CCCCC3)C2=O)c1
CCC(CC)CN1C(=S)S\C(=C/c2ccccc2S(C)(=O)=O)C1=O
C=CCN1C(=S)S\C(C1=O)=C1/C(=O)Nc2ccccc12
COCCN1C(=S)S\C(C1=O)=C1/C(=O)Nc2ccccc12
CCCCCN1C(=O)\C(=C2/SC(=S)N(Cc3ccco3)C2=O)c2cc(Br)ccc12
Clc1ccccc1S(=O)(=O)\C=C\C(=O)NCCc1ccccc1
[H][C@]12CC[C@]3([H])[C@@]([C@@H]1O)(C(=O)C2=C)[C@@]1(O)OC[C@]32[C@@H](O)CCC(C)(C)[C@@]2([H])[C@@H]1O |r,THB:12:11:4.3.2:7,10:9:4.3.2:7|
[H][C@@]12CCC3[C@@]([C@@H]1OC(=O)Nc1cccc(Cl)c1)(C(=O)C2=C)[C@]1(O)OC[C@]32[C@@H](O)CCC(C)(C)[C@@]2([H])[C@@H]1O |r,THB:21:20:4.3.2:6,19:18:4.3.2:6|
COCCCNC(=O)c1ccc(Cn2c(SCc3ccc(F)cc3)nc3ccncc32)cc1
COCCCNC(=O)c1ccc(Cn2c(SCc3ccc(Br)cc3)nc3ccncc32)cc1
COCCCNC(=O)c1ccc(Cn2c(SCc3ccc(C#N)cc3)nc3ccncc32)cc1
COCCCNC(=O)c1ccc(Cn2c(SCc3ccc([N+](=O)[O-])cc3)nc3ccncc32)cc1
COCCCNC(=O)c1ccc(Cn2c(SCc3ccc(C(F)(F)F)cc3)nc3ccncc32)cc1
COCCCNC(=O)c1ccc(Cn2c(SCc3ccc(F)nc3)nc3ccncc32)cc1
COCCCNC(=O)c1ccc(Cn2c(SCC3CCCCC3)nc3ccncc32)cc1
COCCCNC(=O)c1ccc(Cn2c(SCC3CCCC3)nc3ccncc32)cc1
COCCCNC(=O)c1ccc(Cn2c(SCC=C(C)C)nc3ccncc32)cc1
O=C(c1ccc(Cn2c(SCC3CCCCC3)nc3ccncc32)cc1)N1CCNCC1
CC(=O)Nc1ccc(Cn2c(SCC3CCCCC3)nc3ccncc32)cc1
COC(=O)c1ccc(Cn2c(SCC3CCCCC3)nc3ccncc32)cc1
CCOC(=O)c1ccc(Cn2c(SCC3CCCCC3)nc3ccncc32)cc1
CC(C)n1ccc(S(=O)(=O)NC(=O)Nc2c3c(cc4c2CCC4)CCC3)n1
C=C1C(=O)[C@]23[C@H](O)[C@H]1CC[C@H]2[C@]12C=CCC(C)(C)[C@H]1[C@H](O)[C@@]3(OCc1cccnc1)OC2
C=C1C(=O)[C@]23[C@H](O)[C@H]1CC[C@H]2[C@]12C=CCC(C)(C)[C@H]1[C@H](O)[C@@]3(OCc1ccncc1)OC2
C=C1C(=O)[C@]23[C@H](O)[C@H]1CC[C@H]2[C@]12C=CCC(C)(C)[C@H]1[C@H](O)[C@@]3(OCc1cocn1)OC2
C=C1C(=O)[C@]23[C@H](O)[C@H]1CC[C@H]2[C@]12C=CCC(C)(C)[C@H]1[C@H](O)[C@@]3(OCc1cnco1)OC2
C=C1C(=O)[C@]23[C@H](O)[C@H]1CC[C@H]2[C@]12C=CCC(C)(C)[C@H]1[C@H](O)[C@@]3(OCc1cncs1)OC2
C=C1C(=O)[C@]23[C@H](O)[C@H]1CC[C@H]2[C@]12C=CCC(C)(C)[C@H]1[C@H](O)[C@@]3(OCc1nccs1)OC2
C=C1C(=O)[C@]23[C@H](O)[C@H]1CC[C@H]2[C@]12C=CCC(C)(C)[C@H]1[C@H](O)[C@@]3(OCc1nc(-c3ccccc3)cs1)OC2
C=C1C(=O)[C@]23[C@H](O)[C@H]1CC[C@H]2[C@]12C=CCC(C)(C)[C@H]1[C@H](O)[C@@]3(OCC(=O)O)OC2
C=C1C(=O)[C@]23[C@H](O)[C@H]1CC[C@H]2[C@]12C=CCC(C)(C)[C@H]1[C@H](O)[C@@]3(OCCC(=O)O)OC2
C=C1C(=O)[C@]23[C@H](O)[C@H]1CC[C@H]2[C@]12C=CCC(C)(C)[C@H]1[C@H](O)[C@@]3(OCCCC(=O)O)OC2
C=C1C(=O)[C@]23[C@H](O)[C@H]1CC[C@H]2[C@]12C=CCC(C)(C)[C@H]1[C@H](O)[C@@]3(OCCC(=O)NC)OC2
C=C1C(=O)[C@]23[C@H](O)[C@H]1CC[C@H]2[C@]12C=CCC(C)(C)[C@H]1[C@H](O)[C@@]3(OCCC(=O)NCCC)OC2
C=C1C(=O)[C@]23[C@H](O)[C@H]1CC[C@H]2[C@]12C=CCC(C)(C)[C@H]1[C@H](O)[C@@]3(OCCC(=O)NCCOC)OC2
C=C1C(=O)[C@]23[C@H](O)[C@H]1CC[C@H]2[C@]12C=CCC(C)(C)[C@H]1[C@H](O)[C@@]3(OCCC(=O)NC(C)C)OC2
C=C1C(=O)[C@]23[C@H](O)[C@H]1CC[C@H]2[C@]12C=CCC(C)(C)[C@H]1[C@H](O)[C@@]3(OCCC(=O)NCC(C)C)OC2
C=CCNC(=O)CCO[C@@]12OC[C@]3(C=CCC(C)(C)[C@H]3[C@@H]1O)[C@@H]1CC[C@H]3C(=C)C(=O)[C@]12[C@@H]3O
C=C1C(=O)[C@]23[C@H](O)[C@H]1CC[C@H]2[C@]12C=CCC(C)(C)[C@H]1[C@H](O)[C@@]3(OCCC(=O)N(C)C)OC2
C=C1C(=O)[C@]23[C@H](O)[C@H]1CC[C@H]2[C@]12C=CCC(C)(C)[C@H]1[C@H](O)[C@@]3(OCCC(=O)N(CCC)CCC)OC2
C=C1C(=O)[C@]23[C@H](O)[C@H]1CC[C@H]2[C@]12C=CCC(C)(C)[C@H]1[C@H](O)[C@@]3(OCCC(=O)NC1CC1)OC2
C=C1C(=O)[C@]23[C@H](O)[C@H]1CC[C@H]2[C@]12C=CCC(C)(C)[C@H]1[C@H](O)[C@@]3(OCCC(=O)NC1CCCC1)OC2
C=C1C(=O)[C@]23[C@H](O)[C@H]1CC[C@H]2[C@]12C=CCC(C)(C)[C@H]1[C@H](O)[C@@]3(OCCC(=O)NC1CCCCC1)OC2
C=C1C(=O)[C@]23[C@H](O)[C@H]1CC[C@H]2[C@]12C=CCC(C)(C)[C@H]1[C@H](O)[C@@]3(OCCC(=O)NC1CCOCC1)OC2
C=C1C(=O)[C@]23[C@H](O)[C@H]1CC[C@H]2[C@]12C=CCC(C)(C)[C@H]1[C@H](O)[C@@]3(OCCC(=O)N1CCCC1)OC2
C=C1C(=O)[C@]23[C@H](O)[C@H]1CC[C@H]2[C@]12C=CCC(C)(C)[C@H]1[C@H](O)[C@@]3(OCCC(=O)N1CCCCC1)OC2
C=C1C(=O)[C@]23[C@H](O)[C@H]1CC[C@H]2[C@]12C=CCC(C)(C)[C@H]1[C@H](O)[C@@]3(OCCC(=O)N1CCOCC1)OC2
C=C1C(=O)[C@]23[C@H](O)[C@H]1CC[C@H]2[C@]12C=CCC(C)(C)[C@H]1[C@H](O)[C@@]3(OCCC(=O)N1CCN(C)CC1)OC2
CS(=O)(=O)/C=C/C#N
CS(=O)(=O)N1CCCc2ccc(NS(=O)(=O)c3ccccc3F)cc21
CC(=O)c1ccc(S(=O)(=O)Nc2ccc3c(c2)N(S(C)(=O)=O)CCC3)cc1
CS(=O)(=O)N1CCCc2ccc(NS(=O)(=O)c3ccc(-c4ccccc4)cc3)cc21
CS(=O)(=O)N1CCCc2ccc(NS(=O)(=O)c3ccc4ccccc4c3)cc21
COc1ccc(S(=O)(=O)Nc2ccc3c(c2)N(S(C)(=O)=O)CCC3)cc1
COC(=O)c1ccc(S(=O)(=O)Nc2ccc3c(c2)N(S(C)(=O)=O)CCC3)cc1
C#CCCC1(CCN2CCCc3ccc(NS(=O)(=O)c4ccc(-c5ccccc5)cc4)cc32)N=N1
CN1CCC[C@]1(C)\C=C\S(=O)(=O)NC(=O)Nc1c2CCCc2cc2CCCc12
NS(=O)(=O)c1ccc(CCNC(=O)/C=C/S(=O)(=O)c2ccccc2Cl)cc1
O=C(/C=C/S(=O)(=O)c1ccccc1Cl)OCCc1ccccc1
O=C(CBr)NCc1ccc(C(F)(F)F)cc1
CCOCCOc1ccc(/C=C/c2cc(OC)cc(OC)c2/C=C/[N+](=O)[O-])cc1
COc1c(O)cc2c(c1C)C(=O)C=C1[C@@]2(C)CC[C@@]2(C)[C@@H]3C[C@@H](C)C(=O)[C@@H](O)[C@]3(C)CC[C@]12C
CC1=C(O)C(=O)C=C2C1=CC=C1[C@@]2(C)[C@@H](Br)C[C@@]2(C)[C@@H]3C[C@@H](C)C(=O)C[C@]3(C)CC[C@]12C
CC1(C)OC(=O)C=C[C@@]2(C)[C@H]1CC(=O)[C@@]1(C)C3=CC[C@@H](C4=CC(=O)O[C@@H]4O)[C@]3(C)CC[C@@H]12
CC(=O)O[C@@H]1C[C@H]2C(C)(C)OC(=O)C=C[C@]2(C)[C@H]2CC[C@]3(C)C(=CC[C@H]3C3=CC(=O)O[C@@H]3O)[C@@]21C
CC(=O)O[C@H]1[C@@H](OC(C)=O)[C@@]2(C)C3=CC[C@@H](C4=CC(=O)O[C@@H]4O)[C@]3(C)CC[C@@H]2[C@@]2(C)C=CC(=O)OC(C)(C)[C@H]12
CC1(C)OC(=O)C=C[C@]2(C)[C@H]3CC[C@@]4(C)[C@H](C5=CC(=O)NC5=O)C[C@H]5O[C@]54[C@]3(C)OC(=O)C[C@@H]12
CCCOc1ccc(Cl)cc1Cn1cc(-c2ccc(S(N)(=O)=O)cc2)nn1
CCCOc1ccc(Cl)cc1Cn1cc(-c2ccc(C(F)(F)F)cc2)nn1
CCCOc1ccc(Cl)cc1Cn1cc(-c2ccc(F)cc2)nn1
CCCOc1ccc(Cl)cc1Cn1cc(-c2ccc(C)cc2)nn1
CCCOc1ccc(Cl)cc1Cn1cc(-c2ccc(C(=O)O)cc2)nn1
COC(=O)c1cccc(-c2cn(Cc3cc(Cl)ccc3OC)nn2)c1
COc1ccc(Cl)cc1Cn1cc(-c2ccc(C(=O)O)cc2)nn1
CNC(=O)c1ccc(-c2cn(Cc3cc(Cl)ccc3OC)nn2)cc1
COC(=O)c1ccc(-c2cn(Cc3cc(Cl)ccc3OC)nn2)c(C)c1
COC(=O)c1ccc(-c2cn(Cc3cc(Cl)ccc3OC)nn2)c(F)c1
COC(=O)c1ccc(-c2cn(Cc3ccccc3OC)nn2)cc1
COC(=O)c1ccc(-c2cn(Cc3cccc(Cl)c3)nn2)cc1
COC(=O)c1ccc(-c2cn(Cc3cc(Cl)ccc3O)nn2)cc1
COC(=O)c1ccc(-c2cn(Cc3cc(Cl)cc(OC)c3)nn2)cc1
COC(=O)c1ccc(-c2cn(Cc3ccccc3OC(F)F)nn2)cc1
COC(=O)c1ccc(-c2cn(Cc3cc(F)ccc3OC)nn2)cc1
COC(=O)c1ccc(-c2cn(Cc3cc(Br)ccc3OC)nn2)cc1
COC(=O)c1ccc(-c2cn(Cc3cc(C(F)(F)F)ccc3OC)nn2)cc1
COC(=O)c1ccc(-c2cn(Cc3c(OC)ccc(F)c3F)nn2)cc1
COC(=O)c1ccc(-c2cn(Cc3cc(F)c(F)cc3OC)nn2)cc1
CCc1nn(CC(=O)Nc2cccc(C(C)=O)c2)c(=O)c2cc3sccc3n12
CCc1nn(CC(=O)Nc2ccccc2)c(=O)c2cc3sccc3n12
CCc1nn(CC(=O)NC)c(=O)c2cc3sccc3n12
CCc1nn(CC(=O)N(C)c2ccccc2)c(=O)c2cc3sccc3n12
CCc1nn(CC(=O)Nc2cccnc2)c(=O)c2cc3sccc3n12
CCC1=NN(C(=O)c2n1c3ccsc3c2)CC(=O)Nc4ccncn4
CCc1nn(CC(=O)Nc2cccc(O)c2)c(=O)c2cc3sccc3n12
CCc1nn(CC(=O)NC2CCCNC2)c(=O)c2cc3sccc3n12
O=C(Cn1ncn2c(cc3sccc32)c1=O)Nc1cccnc1
CCCc1nn(CC(=O)Nc2cccnc2)c(=O)c2cc3sccc3n12
CC(C)c1nn(CC(=O)Nc2cccnc2)c(=O)c2cc3sccc3n12
O=C(Cn1nc(C2CC2)n2c(cc3sccc32)c1=O)Nc1cccnc1
CC(C)(O)c1nn(CC(=O)Nc2cccnc2)c(=O)c2cc3sccc3n12
CC(C)c1nn(CC(=O)Nc2cccnc2)c(=O)c2cc3sc(F)cc3n12
CC(C)c1nn(CC(=O)Nc2cccnc2)c(=O)c2cc3sc(Cl)cc3n12
CC(C)c1nn(CC(=O)N[C@@H]2CCCNC2)c(=O)c2cc3sc(Cl)cc3n12
CC(C)c1nn(CC(=O)N[C@@H]2CCCN(C)C2)c(=O)c2cc3sc(Cl)cc3n12
CC(C)(C1=NN(C(=O)c2n1c3cc(sc3c2)Cl)CC(=O)N[C@@H]4CCCN(C4)C)O
CC(C)(O)c1nn(CC(=O)N[C@H]2C[C@@](C)(O)C2)c(=O)c2cc3sc(Cl)cc3n12
CC(C)c1nn(CC(=O)N[C@@H]2CCCN(C)C2)c(=O)c2cc3scnc3n12
C=C1C(=O)O[C@@H]2C[C@@]3(C)CC[C@@H](OC(=O)CCC)C(=C)[C@@H]3C[C@H]12
C=C1C(=O)O[C@@H]2C[C@@]3(C)CC[C@@H](OC(=O)CCCCC)C(=C)[C@@H]3C[C@H]12
C=C1C(=O)O[C@@H]2C[C@@]3(C)CC[C@@H](OC(=O)CCCCCCC)C(=C)[C@@H]3C[C@H]12
C=C1C(=O)O[C@@H]2C[C@@]3(C)CC[C@@H](OC(=O)C(CC)CC)C(=C)[C@@H]3C[C@H]12
C=C1C(=O)O[C@@H]2C[C@@]3(C)CC[C@@H](OC(=O)C4CC4)C(=C)[C@@H]3C[C@H]12
C=C1C(=O)O[C@@H]2C[C@@]3(C)CC[C@@H](OC(=O)CCCCl)C(=C)[C@@H]3C[C@H]12
C=C1C(=O)O[C@@H]2C[C@@]3(C)CC[C@@H](OC(=O)CCCCCCl)C(=C)[C@@H]3C[C@H]12
C=CCCC(=O)O[C@@H]1CC[C@]2(C)C[C@H]3OC(=O)C(=C)[C@H]3C[C@H]2C1=C
C=C1C(=O)O[C@@H]2C[C@@]3(C)CC[C@@H](OC(=O)/C=C/C(=O)OCC)C(=C)[C@@H]3C[C@H]12
C[C@]12CCCC(=C)[C@@H]1C[C@H]1[C@@H](C2)OC(=O)C1=C |r|
C=C1C(=O)O[C@@H]2C[C@@]3(C)CC[C@@H](OC(=O)c4ccccc4)C(=C)[C@@H]3C[C@H]12
C=C1C(=O)O[C@@H]2C[C@@]3(C)CC[C@@H](OC(=O)c4ccc(F)cc4)C(=C)[C@@H]3C[C@H]12
C=C1C(=O)O[C@@H]2C[C@@]3(C)CC[C@@H](OC(=O)c4ccc(C(F)(F)F)cc4)C(=C)[C@@H]3C[C@H]12
C=C1C(=O)O[C@@H]2C[C@@]3(C)CC[C@@H](OC(=O)Cc4ccc5ccccc5c4)C(=C)[C@@H]3C[C@H]12
C=C1C(=O)O[C@@H]2C[C@@]3(C)CC[C@@H](OC(=O)c4ccco4)C(=C)[C@@H]3C[C@H]12
C=C1C(=O)O[C@@H]2C[C@@]3(C)CC[C@@H](OC(=O)c4cccs4)C(=C)[C@@H]3C[C@H]12
C=C1C(=O)O[C@@H]2C[C@@]3(C)CC[C@@H](OC(=O)c4cccnc4)C(=C)[C@@H]3C[C@H]12
C=C1C(=O)O[C@@H]2C[C@@]3(C)CC[C@@H](OC(=O)c4ccc(F)nc4)C(=C)[C@@H]3C[C@H]12
C=C1C(=O)O[C@@H]2C[C@@]3(C)CC[C@@H](OC(=O)c4ccc(Cl)nc4)C(=C)[C@@H]3C[C@H]12
C=C1C(=O)O[C@@H]2C[C@@]3(C)CC[C@@H](OC(=O)c4ccc(C(F)(F)F)nc4)C(=C)[C@@H]3C[C@H]12
C=C1C(=O)O[C@@H]2C[C@@]3(C)CC[C@@H](OC(=O)c4c(Cl)ccnc4Cl)C(=C)[C@@H]3C[C@H]12
C=C1C(=O)O[C@@H]2C[C@@]3(C)CC[C@@H](OC(=O)c4cnc(Cl)cc4Cl)C(=C)[C@@H]3C[C@H]12
C=C1C(=O)O[C@@H]2C[C@@]3(C)CC[C@@H](OC(=O)c4cc(Cl)cnc4Cl)C(=C)[C@@H]3C[C@H]12
C=C1C(=O)O[C@@H]2C[C@@]3(C)CC[C@@H](OC(=O)/C=C/c4ccccc4)C(=C)[C@@H]3C[C@H]12
C=C1C(=O)O[C@@H]2C[C@@]3(C)CC[C@@H](OC(=O)/C=C/C(=O)c4ccccc4)C(=C)[C@@H]3C[C@H]12
C=C1C(=O)O[C@@H]2C[C@@]3(C)CC[C@@H](OC(=O)/C=C/C(=O)c4ccc(F)cc4)C(=C)[C@@H]3C[C@H]12
C=C1C(=O)O[C@@H]2C[C@@]3(C)CC[C@@H](OC(=O)/C=C/C(=O)c4ccc(C(F)(F)F)cc4)C(=C)[C@@H]3C[C@H]12
C=C1C(=O)O[C@@H]2C[C@@]3(C)CC[C@@H](OC(=O)/C=C/C(=O)c4ccc(C)cc4)C(=C)[C@@H]3C[C@H]12
C=C1C(=O)O[C@@H]2C[C@@]3(C)CC[C@@H](OC(=O)/C=C/C(=O)c4ccc(OC)cc4)C(=C)[C@@H]3C[C@H]12
C=C1C(=O)O[C@@H]2C[C@@]3(C)CC[C@@H](NC(=O)/C=C/C(=O)OCC)C(=C)[C@@H]3C[C@H]12
C=C1C(=O)O[C@@H]2C[C@@]3(C)CC[C@@H](NC(=O)c4ccc(C(F)(F)F)cc4)C(=C)[C@@H]3C[C@H]12
C=C1C(=O)O[C@@H]2C[C@@]3(C)CC[C@@H](NC(=O)/C=C/C(=O)c4ccccc4)C(=C)[C@@H]3C[C@H]12
C=C1C(=O)O[C@@H]2C[C@@]3(C)CC[C@@H](NC(=O)/C=C/C(=O)c4ccc(F)cc4)C(=C)[C@@H]3C[C@H]12
COc1ccc(-c2cc(=O)c3c(O)cc(O)c(CC=C(C)C)c3o2)cc1
COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)C=CC(C)(C)O4)cc1
COc1cc(C2CC(=O)c3c(O)cc(O)c(CC=C(C)C)c3O2)c(O)cc1O
COc1cc(-c2cc(=O)c3c(O)cc(O)c(CC=C(C)C)c3o2)ccc1O
COc1cc(-c2cc(=O)c3c(O)cc4c(c3o2)C=CC(C)(C)O4)ccc1O
CC(C)=CCc1c(O)cc2oc(-c3ccc(O)cc3)c(O)c(=O)c2c1O
CC(C)=CCc1c(O)cc2oc(-c3ccc(O)c(O)c3)c(O)c(=O)c2c1O
[#6]\[#6](-[#6])=[#6]\[#6]-[#6]\[#6](-[#6])=[#6]\[#6]-c1c(-[#8])cc2oc(-c3ccc(-[#8])cc3)c(-[#8])c(=O)c2c1-[#8]
c1cc(ccc1C2=C(C(=O)c3c(cc(cc3O2)O)O)O)O
c1cc(c(cc1C2=C(C(=O)c3c(cc(cc3O2)O)O)O)O)O
CC(C)c1cccc(C(C)C)c1NC(=O)NS(=O)(=O)c1ccc(Br)s1
Cc1cccc(S(=O)(=O)NC(=O)Nc2c(C(C)C)cccc2C(C)C)c1
Cc1ccc(S(=O)(=O)NC(=O)Nc2c(C(C)C)cccc2C(C)C)cc1
CC(C)(C)c1ccc(S(=O)(=O)NC(=O)Nc2cccc3ccccc23)cc1
CC(C)c1cc(Br)cc(C(C)C)c1NC(=O)NS(=O)(=O)c1ccc2ccccc2c1
COc1ccc(-c2ccc3c(c2NC(=O)NS(=O)(=O)c2ccc(C(C)(C)C)cc2)CCC3)cc1
COc1cccc(-c2ccc3c(c2NC(=O)NS(=O)(=O)c2ccc(C(C)(C)C)cc2)CCC3)c1
COc1ccc(-c2ccc3c(c2NC(=O)NS(=O)(=O)c2ccc(Br)s2)CCC3)cc1
COc1ccc(-c2ccc(S(=O)(=O)NC(=O)Nc3c(-c4cccc(OC)c4)ccc4c3CCC4)s2)cc1
CCOc1cc(C(=O)N(C)Cc2cccc3cn[nH]c23)ccc1-c1ccccc1
CCOc1cc(C(=O)N(C)Cc2cccc3cn[nH]c23)ccc1-c1cccc(F)c1
CCOc1cc(C(=O)N(C)Cc2cccc3cn[nH]c23)ccc1-c1cccc(C(F)(F)F)c1
CCOc1cc(C(=O)N(C)Cc2cccc3cn[nH]c23)ccc1-c1cccc(C#N)c1
CCOc1cc(C(=O)N(C)Cc2cccc3cn[nH]c23)ccc1-c1cccc(N)c1
CCOc1cc(C(=O)N(C)Cc2cccc3cn[nH]c23)ccc1-c1cccc([S+](C)[O-])c1
CCOc1cc(C(=O)N(C)Cc2cccc3cn[nH]c23)ccc1-c1cccc(C(=O)NC)c1
CCOc1cc(C(=O)N(C)Cc2cccc3cn[nH]c23)ccc1-c1ccccc1F
CCOc1cc(C(=O)N(C)Cc2cccc3cn[nH]c23)ccc1-c1ccc(F)cc1
CCOc1cc(C(=O)N(C)Cc2cccc3cn[nH]c23)ccc1-c1c(F)cccc1F
CCOc1cc(C(=O)N(C)Cc2cccc3cn[nH]c23)ccc1-c1cc(F)cc(C#N)c1
CCOc1cc(C(=O)N(C)Cc2cccc3cn[nH]c23)ccc1-c1ccc(F)c(F)c1
CCCOc1cc(C(=O)N(C)Cc2cccc3cn[nH]c23)ccc1-c1cccc(F)c1
CN(Cc1cccc2cn[nH]c12)C(=O)c1ccc(-c2cccc(F)c2)c(OCCO)c1
CN(Cc1cccc2cn[nH]c12)C(=O)c1ccc(-c2cccc(F)c2)c(OCC(F)F)c1
CC(C)Oc1cc(C(=O)N(C)Cc2cccc3cn[nH]c23)ccc1-c1cccc(F)c1
CN(Cc1cccc2cn[nH]c12)C(=O)c1ccc(-c2cccc(F)c2)c(OC2CC2)c1
CN(Cc1cccc2cn[nH]c12)C(=O)c1ccc(-c2cccc(F)c2)c(OC2CCC2)c1
CN(Cc1cccc2cn[nH]c12)C(=O)c1ccc(-c2cccc(F)c2)c(OC2COC2)c1
CCOc1cc(C(=O)N(C)Cc2ccc(F)c3cn[nH]c23)ccc1-c1cccc(F)c1
CCOc1cc(C(=O)N(C)Cc2ccc(C(=O)NC)c3cn[nH]c23)ccc1-c1cccc(F)c1
CCOc1cc(C(=O)N(C)Cc2ccc(C#N)c3cn[nH]c23)ccc1-c1cccc(F)c1
CCOc1cc(C(=O)N(C)Cc2ccc(Cl)c3cn[nH]c23)ccc1-c1cccc(F)c1
CCOc1cc(C(=O)N(C)Cc2ccc(OC)c3cn[nH]c23)ccc1-c1cccc(F)c1
CCOc1cc(C(=O)N(C)Cc2ccc(C(=O)N(C)C)c3cn[nH]c23)ccc1-c1cccc(F)c1
CCOc1cc(C(=O)N(C)Cc2ccc(OCF)c3cn[nH]c23)ccc1-c1cccc(F)c1
CCOc1cc(C(=O)N(C)Cc2ccc(C)c3cn[nH]c23)ccc1-c1cccc(F)c1
O=C(Nc1c2c(cc3c1CCC3)CCC2)NS(=O)(=O)c1ccc(OCCOCCOCCOCCN2C(=O)/C(=C/c3cc(Br)c(O)c(Br)c3)c3cc(I)ccc32)cc1
Cc1nc(N[C@H]2CCCN(CC(C)O)C2)nnc1-c1ccc2c(c1O)CCO2
Cc1nc(N[C@@H]2CCCN(CCO)C2)nnc1-c1ccc2c(c1O)CCO2
Cc1nc(N[C@@H]2CCCN(CCCO)C2)nnc1-c1ccc2c(c1O)CCO2
Cc1nc(N[C@@H]2CCCN(CCCC(=O)O)C2)nnc1-c1ccc2c(c1O)CCO2
Cc1nc(N[C@H]2CCCN(CCc3ncco3)C2)nnc1-c1ccc2c(c1O)CCO2
Cc1nc(N[C@H]2CCCN(CCCC(=O)N3CCCC3)C2)nnc1-c1ccc2c(c1O)CCO2
N#CCCS(=O)(=O)C/C(=Cc1ccc(Cl)cc1)C(=O)NCCc1ccccc1
CNC(=O)/C(=C/c1ccc(Cl)cc1)CS(=O)(=O)CCC#N
CN(C)C(=O)/C(=C/c1ccc(Cl)cc1)CS(=O)(=O)CCC#N
CCCNC(=O)/C(=C/c1ccc(Cl)cc1)CS(=O)(=O)CCC#N
N#CCCS(=O)(=O)C/C(=Cc1ccc(Cl)cc1)C(=O)NC1CC1
N#CCCS(=O)(=O)C/C(=Cc1ccc(Cl)cc1)C(=O)NCC1CC1
N#CCCS(=O)(=O)C/C(=Cc1ccc(Cl)cc1)C(=O)N1CC(O)C1
N#CCCS(=O)(=O)C/C(=Cc1ccc(Cl)cc1)C(=O)N1CCCC1
N#CCCS(=O)(=O)C/C(=Cc1ccc(Cl)cc1)C(=O)NC1CCCC1
N#CCCS(=O)(=O)C/C(=Cc1ccc(Cl)cc1)C(=O)N1CCOCC1
N#CCCS(=O)(=O)C/C(=Cc1ccc(Cl)cc1)C(=O)NCCc1ccc(S(N)(=O)=O)cc1
CCCNC(=O)/C(=C/c1ccc(Br)cc1)CS(=O)(=O)CCC#N
N#CCCS(=O)(=O)C/C(=Cc1ccc(Br)cc1)C(=O)NC1CC1
N#CCCS(=O)(=O)C/C(=Cc1ccc(Br)cc1)C(=O)NC1CCCC1
N#CCCS(=O)(=O)C/C(=Cc1ccc(Br)cc1)C(=O)NCCc1ccccc1
N#CCCS(=O)(=O)C/C(=Cc1ccc(Br)cc1)C(=O)NCCc1ccc(S(N)(=O)=O)cc1
CCCNC(=O)/C(=C/c1cccc(Cl)c1)CS(=O)(=O)CCC#N
N#CCCS(=O)(=O)C/C(=Cc1cccc(Cl)c1)C(=O)NC1CC1
N#CCCS(=O)(=O)C/C(=Cc1cccc(Cl)c1)C(=O)NC1CCCC1
N#CCCS(=O)(=O)C/C(=Cc1cccc(Cl)c1)C(=O)NCCc1ccccc1
N#CCCS(=O)(=O)C/C(=Cc1cccc(Cl)c1)C(=O)NCCc1ccc(S(N)(=O)=O)cc1
CCCNC(=O)/C(=C/c1cccc(Br)c1)CS(=O)(=O)CCC#N
N#CCCS(=O)(=O)C/C(=Cc1cccc(Br)c1)C(=O)NC1CC1
N#CCCS(=O)(=O)C/C(=Cc1cccc(Br)c1)C(=O)NC1CCCC1
N#CCCS(=O)(=O)C/C(=Cc1cccc(Br)c1)C(=O)NCCc1ccccc1
N#CCCS(=O)(=O)C/C(=Cc1cccc(Br)c1)C(=O)NCCc1ccc(S(N)(=O)=O)cc1
CCCNC(=O)/C(=C/c1ccc2ccccc2c1)CS(=O)(=O)CCC#N
N#CCCS(=O)(=O)C/C(=Cc1ccc2ccccc2c1)C(=O)NC1CC1
N#CCCS(=O)(=O)C/C(=Cc1ccc2ccccc2c1)C(=O)NC1CCCC1
N#CCCS(=O)(=O)C/C(=Cc1ccc2ccccc2c1)C(=O)NCCc1ccccc1
N#CCCS(=O)(=O)C/C(=Cc1ccc2ccccc2c1)C(=O)NCCc1ccc(S(N)(=O)=O)cc1
CCCNC(=O)/C(=C/c1cc2ccccc2s1)CS(=O)(=O)CCC#N
N#CCCS(=O)(=O)C/C(=Cc1cc2ccccc2s1)C(=O)NC1CC1
N#CCCS(=O)(=O)C/C(=Cc1cc2ccccc2s1)C(=O)NC1CCCC1
N#CCCS(=O)(=O)C/C(=Cc1cc2ccccc2s1)C(=O)NCCc1ccccc1
CCCNC(=O)/C(=C/c1cc2ccccc2o1)CS(=O)(=O)CCC#N
N#CCCS(=O)(=O)C/C(=Cc1cc2ccccc2o1)C(=O)NC1CC1
N#CCCS(=O)(=O)C/C(=Cc1cc2ccccc2o1)C(=O)NC1CCCC1
N#CCCS(=O)(=O)C/C(=Cc1cc2ccccc2o1)C(=O)NCCc1ccccc1
N#CCCS(=O)(=O)C/C(=Cc1ccc(Br)cc1)C(=O)NCc1ccc(Oc2ccccc2)cc1
N#CCCS(=O)(=O)C/C(=Cc1ccc(Br)cc1)C(=O)N1CCC2(CC1)OCCO2
N#CCCS(=O)(=O)C/C(=Cc1ccc(Br)cc1)C(=O)NC1CCC(F)(F)CC1
N#CCCS(=O)(=O)C/C(=Cc1ccc(Br)cc1)C(=O)NCCc1cccnc1
N#CCCS(=O)(=O)C/C(=Cc1ccc(Br)cc1)C(=O)NCCc1ccncc1
N#CCCS(=O)(=O)C/C(=Cc1ccc(Br)cc1)C(=O)NCCc1ccccc1F
N#CCCS(=O)(=O)C/C(=Cc1ccc(Br)cc1)C(=O)NCCc1ccccc1Cl
N#CCCS(=O)(=O)C/C(=Cc1ccc(Br)cc1)C(=O)NCCc1ccccc1Br
COc1ccccc1CCNC(=O)/C(=C/c1ccc(Br)cc1)CS(=O)(=O)CCC#N
N#CCCS(=O)(=O)C/C(=Cc1ccc(Br)cc1)C(=O)NCCc1cccc(F)c1
N#CCCS(=O)(=O)C/C(=Cc1ccc(Br)cc1)C(=O)NCCc1cccc(Cl)c1
N#CCCS(=O)(=O)C/C(=Cc1ccc(Br)cc1)C(=O)NCCc1cccc(Br)c1
COc1cccc(CCNC(=O)/C(=C/c2ccc(Br)cc2)CS(=O)(=O)CCC#N)c1
N#CCCSC/C(=Cc1ccc(Cl)cc1)C(=O)NCCc1ccccc1
Clc1ccc(\C=C\C(=O)NCCc2ccccc2)cc1
OCCN1CCC[C@@H](Nc2nnc(-c3ccc4occc4c3O)c3c2C2CCC3CC2)C1
CCN1CCC[C@@H](N2CCOc3cc(-c4c(C)cc(C#N)cc4O)nnc32)C1
CCN1CCC[C@@H](N2CCCc3cc(-c4c(C)cc(C#N)cc4O)nnc32)C1
Cc1cc2c(c(O)c1-c1cc3c(nn1)N([C@@H]1CCCC[C@H]1O)CCO3)CCC2
Cc1cc2c(c(O)c1-c1cc3c(nn1)N([C@@H]1CCCC[C@H]1O)CCO3)CCO2
Cc1c(-c2ccc3c(c2O)CCC3)nnc2c1OCCN2[C@@H]1CCCC[C@H]1O
Cc1c(-c2ccc3c(c2O)CC3)nnc2c1OCCN2[C@@H]1CCCC[C@H]1O
Cc1coc-2c1C(=O)C(=O)c1c3CCCC(C)(C)c3ccc-21
Cc1c(S(=O)(=O)O)oc2c1C(=O)C(=O)c1c-2ccc2c1CCCC2(C)C
Cc1c(Br)oc-2c1C(=O)C(=O)c1c3CCCC(C)(C)c3ccc-21
Cc1c(-c2ccccc2)oc2c1C(=O)C(=O)c1c-2ccc2c1CCCC2(C)C
Cc1coc2c3ccc4c(c3c3ocnc3c12)CCCC4(C)C
Cc1coc-2c1C(=O)C(=O)c1c-2ccc2c1C=CCC2(C)C |c:19|
CC(=O)OC1CCC(C)(C)c2ccc3c(c21)C(=O)C(=O)c1c(C)coc1-3
COc1cc(/C=C/C(=O)OC2CCC(C)(C)c3ccc4c(c32)C(=O)C(=O)c2c(C)coc2-4)cc(OC)c1OC
Cc1coc2c1C(=O)C(=O)c1c-2ccc2c1C(OC(=O)CCCCC1CCSS1)CCC2(C)C
Cc1coc2c1C(=O)C(=O)c1c-2ccc2c1C(OC(=O)c1cc(Cl)ccc1Cl)CCC2(C)C
Cc1coc2c1C(=O)C(=O)c1c-2ccc2c1C(OC(=O)c1ccccc1O)CCC2(C)C
Cc1coc2c1C(=O)C(=O)c1c-2ccc2c1C(OC(=O)c1ccc(O)cc1)CCC2(C)C
Cc1coc2c1C(=O)C(=O)c1c-2ccc2c1C(OC(=O)c1cccc(O)c1)CCC2(C)C
OC(=O)CCCCCN1C(=S)S\C(=C/c2c[nH]c3ccccc23)C1=O
COc1ccc(N2C(=O)/C(=Cc3ccccc3C(F)(F)F)SC2=S)cc1
CCn1c(NC(=O)Cn2nc(C(F)(F)F)c(Cl)c2C)nc2ccccc21
Cc1cccc(C(=O)Nc2ncn(Cc3ccc(Cl)c(Cl)c3)n2)c1
Nc1nonc1-c1nc2ccccc2n1Cc1ccncc1
Nc1nonc1-c1nc2cccc(F)c2n1Cc1cccnn1