6919 SMILES Strings for Receptor-interacting serine/threonine-protein kinase 1

Compound Name
SMILES String
CN1C(=S)NC(Cc2c[nH]c3ccccc23)C1=O
CN1C(=O)[C@H](NC1=O)Cc2c[nH]c3c2cccc3Cl
Cc1ccc(F)c(NC(=O)Nc2ccc(cc2)-c2cccc3[nH]nc(N)c23)c1
CCN1CCN(Cc2ccc(NC(=O)Nc3ccc(Oc4cc(NC)ncn4)cc3)cc2C(F)(F)F)CC1
CN1CCN(CC1)c1ccc2nc([nH]c2c1)-c1c(N)c2c(F)cccc2[nH]c1=O
CN(c1ccc2c(C)n(C)nc2c1)c1ccnc(Nc2ccc(C)c(c2)S(N)(=O)=O)n1
c1cc(c(c(c1)F)C(=O)n2c(nc(n2)Nc3ccc(cc3)S(=O)(=O)N)N)F
Cc1[nH]c(\C=C2/C(=O)Nc3ccc(F)cc23)c(C)c1C(=O)NC[C@H](O)CN1CCOCC1
CCN(CC)CCNC(=O)c1c(C)[nH]c(\C=C2/C(=O)Nc3ccc(F)cc23)c1C
CN1CCN(CC1)c1cc(Nc2cc(C)n[nH]2)nc(Sc2ccc(NC(=O)C3CC3)cc2)n1
CCC(C)(C)C(=O)N1CCCC1c1cc(F)cc(F)c1F
CCC(C)(C)C(=O)N1CCC1c1ccccc1
CCC(C)(C)C(=O)N1C(CC1=O)c1cccc(c1)N=[N+]=[N-]
CC(C)(C=C)C(=O)N1[C@@H](CC1=O)c1ccccc1 |r|
CCC(C)(C)C(=O)N1C[C@H](O)C[C@H]1c1ccccc1 |r|
CCC(C)(C)C(=O)N1[C@@H](CC1=O)c1ccccc1 |r|
CCC(C)(C)C(=O)N1[C@@H](CN(C)C1=O)c1ccccc1 |r|
CN1c2cc(Cl)sc2CC[C@H](NC(=O)c2cc(Cc3ccccc3)on2)C1=O |r|
CN1c2cc(Cl)sc2CC[C@@H](NC(=O)c2cc(Cc3ccccc3)on2)C1=O |r|
CN1c2ccccc2C(F)CC(NC(=O)c2cc(Cc3ccccc3)on2)C1=O
CN1c2ccccc2C(=C)C[C@H](NC(=O)c2cc(Cc3ccccc3)on2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2nn(Cc3ccccc3)c(C)c2Cl)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2ncc(Cc3ccccc3)s2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2nn(Cc3ccccc3)c(C)c2F)C1=O |r|
CN1c2ccccc2C2CC2[C@H](NC(=O)c2cc(Cc3ccccc3)on2)C1=O |r|
CN1c2ccccc2[C@@H]2C[C@@H]2[C@H](NC(=O)c2cc(Cc3ccccc3)on2)C1=O |r|
CN1c2ccccc2[C@H]2C[C@H]2[C@@H](NC(=O)c2cc(Cc3ccccc3)on2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2cc(on2)C2(CC2)c2ccccc2)C1=O |r|
CN1c2ccccc2C2(CC2)C[C@H](NC(=O)c2cc(Cc3ccccc3)on2)C1=O |r|
CN1c2ccccc2C(F)(F)CC(NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O
CN1c2ccccc2[C@H](F)C[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2ccccc2[C@@H](F)C[C@@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2ccccc2[C@@H](F)C[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2ccccc2[C@H](F)C[C@@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2cc3[C@H](CCn3n2)c2ccccc2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2cc(CC(F)(F)F)on2)C1=O |r|
O=C(NC1CCc2ccccc2CC1)c1cc(Cc2ccccc2)on1
CN1c2ccccc2OC[C@H](NC(=O)c2cc(C)nn2Cc2ccccc2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2cnn3CC[C@@H](c23)c2ccccc2)C1=O |r|
CN1c2ccccc2OC[C@H](NCC(=O)NCc2ccccc2)C1=O |r|
CCN1c2ccccc2OC[C@H](NC(=O)c2cc(Cc3ccccc3)on2)C1=O |r|
CN1CC(CCc2ccccc12)NC(=O)c1nnc(Cc2ccccc2)[nH]1
O=C(N[C@H]1COC[C@H]2CCCN2C1=O)c1cc(Cc2ccccc2)on1 |r|
O=C(N[C@H]1COC[C@@H]2CCCN2C1=O)c1cc(Cc2ccccc2)on1 |r|
CN1CCCC[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2ccc(C#N)n2C)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2nnc(C)[nH]2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(C)=O)C1=O |r|
O=C(N[C@H]1COC[C@@H]2CCCN2C1=O)c1nnc(Cc2ccccc2)[nH]1 |r|
O=C(N[C@H]1CCc2ccccc2-n2ccnc12)c1cc(Cc2ccccc2)on1 |r|
CN1c2cccc(Cl)c2OC[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)C2CN(Cc3ccccc3)C2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2nnc([nH]2)C2(CC2)c2ccccc2)C1=O |r|
CN1c2nc(C)sc2CC[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2nc(C)sc2CC[C@@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2ccncc2OC[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2ncccc2OC[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)C2CC(Cc3ccccc3)C2)C1=O |r,wU:10.11,(-4.87,2.94,;-4.47,1.46,;-5.68,.49,;-7.01,1.26,;-8.34,.49,;-8.34,-1.05,;-7.01,-1.82,;-5.68,-1.05,;-4.47,-2.01,;-2.97,-1.66,;-2.3,-.28,;-.76,-.28,;.01,-1.61,;-.76,-2.94,;1.55,-1.61,;2.64,-2.7,;3.72,-1.61,;5.26,-1.61,;6.03,-.28,;7.57,-.28,;8.34,1.06,;7.57,2.39,;6.03,2.39,;5.26,1.06,;2.64,-.52,;-2.97,1.11,;-2.2,2.45,)|
CN1c2ccccc2C2(CC2)C[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
Cc1c(F)c(nn1Cc1ccccc1)C(=O)N[C@H]1COc2ccccc2NC1=O |r|
CN1c2ccccc2[C@@H]2C[C@@H]2[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2ccccc2[C@H]2C[C@H]2[C@@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2ncc(s2)S(=O)(=O)c2ccccc2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)C2C[C@H]2Cc2ccccc2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)C2C[C@@H]2Cc2ccccc2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2nnc([nH]2)C2CCc3ccccc23)C1=O |r|
O=C(N[C@H]1CCc2ccccc2-n2ccnc12)c1nnc(Cc2ccccc2)[nH]1 |r|
CN1c2ncccc2OC[C@H](NC(=O)c2nnc([nH]2)C2CCc3ccccc23)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2nn(Cc3ccccn3)cc2F)C1=O |r|
CN1c2cccc(C#N)c2OC[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
Fc1cn(Cc2ccccc2)nc1C(=O)N[C@H]1COc2cccnc2NC1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2nnc(s2)C2(CC2)c2ccccc2)C1=O |r|
CN1c2ccccc2C2(CC2)C[C@H](NC(=O)c2cc(Cc3ccccc3)[nH]n2)C1=O |r|
CN1c2ccccc2[C@@H]2C[C@@H]2[C@H](NC(=O)c2cc(Cc3ccccc3)[nH]n2)C1=O |r|
CN1c2ccccc2[C@H]2C[C@H]2[C@@H](NC(=O)c2cc(Cc3ccccc3)[nH]n2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2coc(n2)C2(CC2)c2ccccc2)C1=O |r|
O=C(N[C@H]1COc2cccnc2NC1=O)c1cc(on1)C1(CC1)c1ccccc1 |r|
CN1c2ncccc2OC[C@H](NC(=O)c2ncc(s2)C2(CC2)c2ccccc2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2nn(Cc3ccccc3)cc2F)C1=O |r|
O=C(N[C@H]1COC[C@H]2CCCN2C1=O)c1nnc(Cc2ccccc2)[nH]1 |r|
CN1c2ncccc2OC[C@H](NC(=O)c2nnc(o2)C2(CC2)c2ccccc2)C1=O |r|
CN1c2ccccc2[C@H]2C[C@H]2[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2ccccc2[C@@H]2C[C@@H]2[C@@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
O=C(N[C@H]1COc2ccccc2-n2ccnc12)c1nnc(Cc2ccccc2)[nH]1 |r|
O=C(N[C@@H]1COc2ccccc2-n2ccnc12)c1nnc(Cc2ccccc2)[nH]1 |r|
O=C(N[C@H]1CCc2ccccc2-n2cnnc12)c1nnc(Cc2ccccc2)[nH]1 |r|
O=C(N[C@@H]1CCc2ccccc2-n2cnnc12)c1nnc(Cc2ccccc2)[nH]1 |r|
O=C(N[C@H]1COc2ccccc2-n2cnnc12)c1cc(Cc2ccccc2)[nH]n1 |r|
O=C(N[C@@H]1COc2ccccc2-n2ccnc12)c1cc(Cc2ccccc2)on1 |r|
O=C(N[C@H]1CCc2ccccc2-n2cnnc12)c1cc(Cc2ccccc2)on1 |r|
O=C(N[C@@H]1CCc2ccccc2-n2cnnc12)c1cc(Cc2ccccc2)on1 |r|
CN1c2ccccc2OC[C@H](NC(=O)c2cc([nH]n2)C2(CC2)c2ccccc2)C1=O |r|
CN1c2ncccc2OC[C@H](NC(=O)c2cc([nH]n2)C2(CC2)c2ccccc2)C1=O |r|
CN1c2ncccc2OC[C@H](NC(=O)c2nn(cc2F)C2(CC2)c2ccccn2)C1=O |r|
CN1c2ncccc2[C@@H]2C[C@@H]2[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2ncccc2[C@H]2C[C@H]2[C@@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2ncccc2OC[C@H](NC(=O)c2nn(Cc3ccccc3)cc2F)C1=O |r|
CN1c2ncccc2OC[C@H](NC(=O)c2cc(on2)C2(CC2)c2ccccc2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2ncc([nH]2)C2(CC2)c2ccccc2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2nc3cccc(-c4ccccc4F)c3s2)C1=O |r|
CN1c2ncccc2[C@@H]2C[C@@H]2[C@H](NC(=O)c2cc(Cc3ccccc3)[nH]n2)C1=O |r|
CN1c2ncccc2[C@H]2C[C@H]2[C@@H](NC(=O)c2cc(Cc3ccccc3)[nH]n2)C1=O |r|
CN1c2ncccc2[C@@H]2C[C@@H]2[C@H](NC(=O)c2cc(Cc3ccccc3)on2)C1=O |r|
CN1c2ncccc2[C@H]2C[C@H]2[C@@H](NC(=O)c2cc(Cc3ccccc3)on2)C1=O |r|
CN1c2ncccc2[C@@H]2C[C@@H]2[C@H](NC(=O)c2nn(Cc3ccccc3)cc2F)C1=O |r|
CN1c2ncccc2[C@H]2C[C@H]2[C@@H](NC(=O)c2nn(Cc3ccccc3)cc2F)C1=O |r|
Fc1cc(F)c2NC(=O)[C@@H](NC(=O)c3nnc(Cc4ccccc4)[nH]3)[C@H]3C[C@H]3c2c1 |r|
Fc1cc(F)c2NC(=O)[C@H](NC(=O)c3nnc(Cc4ccccc4)[nH]3)[C@@H]3C[C@@H]3c2c1 |r|
CN1c2ccccc2OC[C@H](NC(=O)c2nc3cccc(-c4ccccc4)c3s2)C1=O |r|
CN1c2ncccc2OC[C@H](NC(=O)c2nnc(Cc3ccccc3)s2)C1=O |r|
CN1c2ncccc2OC[C@H](NC(=O)c2ncc(Cc3ccccc3)s2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2cn(nn2)C2(CC2)c2ccccc2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2cnc([nH]2)C2(CC2)c2ccccc2)C1=O |r|
Fc1cc(F)c2NC(=O)[C@H](NC(=O)c3nnc(Cc4ccccc4)o3)[C@@H]3C[C@@H]3c2c1 |r|
Fc1cc(F)c2NC(=O)[C@@H](NC(=O)c3nnc(Cc4ccccc4)o3)[C@H]3C[C@H]3c2c1 |r|
Fc1cc(F)c2NC(=O)[C@H](NC(=O)c3cn(Cc4ccccc4)nn3)[C@@H]3C[C@@H]3c2c1 |r|
Fc1cc(F)c2NC(=O)[C@@H](NC(=O)c3cn(Cc4ccccc4)nn3)[C@H]3C[C@H]3c2c1 |r|
O=C(N[C@H]1COc2cccnc2NC1=O)c1cc([nH]n1)C1(CC1)c1ccccc1 |r|
C[C@H]1Oc2cccnc2N(C)C(=O)[C@H]1NC(=O)c1nn(Cc2ccccc2)cc1F |r|
C[C@@H]1Oc2cccnc2N(C)C(=O)[C@H]1NC(=O)c1nn(Cc2ccccc2)cc1F |r|
C[C@H]1Oc2cccnc2N(C)C(=O)[C@H]1NC(=O)c1nnc(Cc2ccccc2)[nH]1 |r|
C[C@@H]1Oc2cccnc2N(C)C(=O)[C@H]1NC(=O)c1nnc(Cc2ccccc2)[nH]1 |r|
C[C@H]1Oc2cccnc2NC(=O)[C@H]1NC(=O)c1nnc(Cc2ccccc2)[nH]1 |r|
O=C(N[C@@H]1CC2(CC2)c2cccnc2NC1=O)c1nnc(Cc2ccccc2)[nH]1 |r|
O=C(N[C@H]1CC2(CC2)c2cccnc2NC1=O)c1nnc(Cc2ccccc2)[nH]1 |r|
CN1c2ncccc2OC[C@H](NC(=O)c2ncc([nH]2)C2(CC2)c2ccccc2)C1=O |r|
CN1c2ncccc2[C@@H]2C[C@@H]2[C@H](NC(=O)c2cc(Oc3ccccc3F)ccn2)C1=O |r|
CN1c2ncccc2[C@H]2C[C@H]2[C@@H](NC(=O)c2cc(Oc3ccccc3F)ccn2)C1=O |r|
CN1c2cnn(C)c2CC[C@@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2cnn(C)c2CC[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
O=C(N[C@H]1COc2cccnc2NC1=O)c1nnc([nH]1)C1CCc2ccccc12 |r|
Fc1cc(F)c2NC(=O)[C@@H](CC3(CC3)c2c1)NC(=O)c1nnc(Cc2ccccc2)[nH]1 |r|
Fc1cc(F)c2NC(=O)[C@H](CC3(CC3)c2c1)NC(=O)c1nnc(Cc2ccccc2)[nH]1 |r|
Cn1cc2NC(=O)[C@@H](CCc2n1)NC(=O)c1nnc(Cc2ccccc2)[nH]1 |r|
Cn1cc2NC(=O)[C@H](CCc2n1)NC(=O)c1nnc(Cc2ccccc2)[nH]1 |r|
CN1c2cn(C)nc2CC[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2cn(C)nc2CC[C@@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2ncccc2OC[C@H](NC(=O)c2nnc([nH]2)C2(CC2)c2ccccc2)C1=O |r|
CN1c2ncccc2CC[C@@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2ncccc2CC[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2ncccc2OC[C@H](NC(=O)c2cnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2cn(C)nc2CC[C@H](NC(=O)c2nn(Cc3ccccc3)cc2F)C1=O |r|
CN1c2cn(C)nc2CC[C@@H](NC(=O)c2nn(Cc3ccccc3)cc2F)C1=O |r|
O=C(N[C@@H]1[C@@H]2C[C@@H]2c2cccnc2NC1=O)c1nnc(Cc2ccccc2)[nH]1 |r|
O=C(N[C@H]1[C@H]2C[C@H]2c2cccnc2NC1=O)c1nnc(Cc2ccccc2)[nH]1 |r|
CN1c2ncccc2CC[C@@H](NC(=O)c2nn(Cc3ccccc3)cc2F)C1=O |r|
CN1c2ncccc2CC[C@H](NC(=O)c2nn(Cc3ccccc3)cc2F)C1=O |r|
C[C@H]1Oc2cccnc2N(C)C(=O)[C@H]1NC(=O)c1cc(Cc2ccccc2)on1 |r|
CN1c2ccncc2OC[C@H](NC(=O)c2cc(on2)C2(CC2)c2ccccc2)C1=O |r|
CN1c2cnn(C)c2OC[C@H](NC(=O)c2nn(Cc3ccccc3)cc2F)C1=O |r|
CN1c2cnn(C)c2CC[C@@H](NC(=O)c2nn(Cc3ccccc3)cc2F)C1=O |r|
CN1c2ncccc2OC[C@H](NC(=O)c2nn(Cc3ccc(F)cc3)cc2F)C1=O |r|
Fc1ccccc1Oc1cnnc(c1)C(=O)N[C@H]1CCc2ccccc2-n2ccnc12 |r|
C[C@H]1Oc2cccnc2N(C)C(=O)[C@H]1NC(=O)c1cc(Oc2ccccc2F)ccn1 |r|
Cn1ncc2NC(=O)[C@@H](CCc12)NC(=O)c1nnc(Cc2ccccc2)[nH]1 |r|
Cn1ncc2NC(=O)[C@H](CCc12)NC(=O)c1nnc(Cc2ccccc2)[nH]1 |r|
CN1c2nccnc2[C@H]2C[C@H]2[C@@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2nccnc2[C@@H]2C[C@@H]2[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2ncccc2[C@@H]2C[C@@H]2[C@H](NC(=O)c2nnc(Cc3ccccc3)s2)C1=O |r|
CN1c2ncccc2[C@H]2C[C@H]2[C@@H](NC(=O)c2nnc(Cc3ccccc3)s2)C1=O |r|
CN1c2ncccc2CC[C@@H](NC(=O)c2cc(Oc3ccc(F)cc3F)ccn2)C1=O |r|
CN1c2ncccc2CC[C@H](NC(=O)c2cc(Oc3ccc(F)cc3F)ccn2)C1=O |r|
C[C@H]1Oc2cccnc2N(C)C(=O)[C@H]1NC(=O)c1cc(Cc2ccccc2)no1 |r|
O=C(N[C@H]1COc2cccnc2NC1=O)c1ncc(Cc2ccccc2)s1 |r|
C[C@H]1Oc2cccnc2N(C)C(=O)[C@H]1NC(=O)c1ncc(Cc2ccccc2)s1 |r|
CN1c2ncccc2C2(CC2)C[C@@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2ncccc2C2(CC2)C[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2ncccc2OC[C@H](NC(=O)c2nc(F)c(Cc3ccccc3)s2)C1=O |r|
C[C@H]1Oc2cccnc2N(C)C(=O)[C@H]1NC(=O)c1nn(Cc2ccc(cc2)C#N)cc1F |r|
C[C@H]1Oc2cccnc2N(C)C(=O)[C@H]1NC(=O)c1nn(Cc2cccc(c2)C#N)cc1F |r|
CN1c2cc(C)nn2CC[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2cc(C)nn2CC[C@@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2ncccc2OC[C@H](NC(=O)c2nn(Cc3cc(F)cc(c3)C#N)cc2F)C1=O |r|
CN1c2c(C)cnn2CC[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2c(C)cnn2CC[C@@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
C[C@H]1Oc2cccnc2N(C)C(=O)[C@H]1NC(=O)c1nn(Cc2ccccc2)cc1Cl |r|
CN1c2ncccc2OC[C@H](NC(=O)c2nn(Cc3ccccc3F)cc2F)C1=O |r|
C[C@H]1Oc2cccnc2N(C)C(=O)[C@H]1NC(=O)c1nnc(Cc2ccccc2)o1 |r|
CN1c2ncccc2OC[C@H](NC(=O)c2nn(Cc3cccc(F)c3)cc2F)C1=O |r|
C[C@H]1Oc2cccnc2N(C)C(=O)[C@H]1NC(=O)c1ncn(Cc2ccccc2)n1 |r|
CN1c2ncccc2OC[C@H](NC(=O)c2nn(Cc3cncc(F)c3)cc2F)C1=O |r|
C[C@H]1Oc2cccnc2N(C)C(=O)[C@H]1NC(=O)c1nnc(o1)C1(CC1)c1ccccc1 |r|
C[C@H]1Oc2cccnc2N(C)C(=O)[C@H]1NC(=O)c1cc(Oc2ccccc2F)cnn1 |r|
C[C@H]1Oc2cccnc2N(C)C(=O)[C@H]1NC(=O)c1cn(Cc2ccccc2)cn1 |r|
O=C(N[C@@H]1COc2cccnc2-n2ccnc12)c1nnc(Cc2ccccc2)[nH]1 |r|
O=C(N[C@H]1COc2cccnc2-n2ccnc12)c1nnc(Cc2ccccc2)[nH]1 |r|
CN1c2ncccc2OC[C@H](NC(=O)c2cc(Cc3ccccc3)on2)C1=O |r|
C[C@H]1Oc2cccnc2N(C)C(=O)[C@H]1NC(=O)c1nn(Cc2ccc(F)cc2)cc1F |r|
CN1c2ncccc2OC[C@H](NC(=O)c2nn(Cc3cccc(c3)C#N)cc2F)C1=O |r|
CN1c2ncccc2CC[C@H](NC(=O)c2nnc(o2)C2(CC2)c2ccccc2)C1=O |r|
CN1c2ncccc2CC[C@@H](NC(=O)c2nnc(o2)C2(CC2)c2ccccc2)C1=O |r|
CN1c2ncccc2OC[C@H](NC(=O)c2nnc(Cc3ccccc3)o2)C1=O |r|
C[C@H]1Oc2cc(cnc2N(C)C(=O)[C@H]1NC(=O)c1nnc(Cc2ccccc2)[nH]1)S(C)(=O)=O |r|
CN1c2ncccc2CC[C@H](NC(=O)c2nnc(Cc3ccccc3)o2)C1=O |r|
CN1c2ncccc2CC[C@@H](NC(=O)c2nnc(Cc3ccccc3)o2)C1=O |r|
CN1c2ncccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3F)cnn2)C1=O |r|
C[C@H]1Oc2cc(cnc2N(C)C(=O)[C@H]1NC(=O)c1nnc(Cc2ccccc2)[nH]1)C#N |r|
CN1c2ncccc2OC[C@H](NC(=O)c2nc(C#N)c(Cc3ccccc3)s2)C1=O |r|
CN1c2ncccc2CC[C@@H](NC(=O)c2nn(Cc3cccc(c3)C#N)cc2F)C1=O |r|
CN1c2ncccc2CC[C@H](NC(=O)c2nn(Cc3cccc(c3)C#N)cc2F)C1=O |r|
CN1c2ncccc2OC[C@H](NC(=O)c2nn(Cc3ccccc3C#N)cc2F)C1=O |r|
Fc1cn(Cc2ccccc2)nc1C(=O)N[C@@H]1COc2cccnc2-n2ccnc12 |r|
Fc1cn(Cc2ccccc2)nc1C(=O)N[C@H]1COc2cccnc2-n2ccnc12 |r|
C[C@H]1Oc2cccnc2N(C)C(=O)[C@H]1NC(=O)c1ccn(Cc2ccccc2)n1 |r|
CN1c2ncccc2[C@H]2C[C@H]2[C@@H](NC(=O)c2nn(Cc3ccc(F)cc3)cc2F)C1=O |r|
CN1c2ncccc2[C@@H]2C[C@@H]2[C@H](NC(=O)c2nn(Cc3ccc(F)cc3)cc2F)C1=O |r|
CN1c2ncccc2[C@H]2C[C@H]2[C@@H](NC(=O)c2nnc(Cc3ccccc3)o2)C1=O |r|
CN1c2ncccc2[C@@H]2C[C@@H]2[C@H](NC(=O)c2nnc(Cc3ccccc3)o2)C1=O |r|
CN1c2ncccc2OC[C@H](NC(=O)c2cc(C#N)n(Cc3ccccc3)n2)C1=O |r|
CN1c2ncccc2OC[C@H](NC(=O)c2cc(C#N)n(Cc3ccc(F)cc3)n2)C1=O |r|
CN1c2ncccc2OC2(CC2)[C@H](NC(=O)c2nnc(Cc3ccccc3)o2)C1=O |r|
CN1c2ncccc2OC2(CC2)[C@@H](NC(=O)c2nnc(Cc3ccccc3)o2)C1=O |r|
CN1c2ncccc2OC[C@H](NC(=O)c2nnc(Cc3cccc(c3)C#N)[nH]2)C1=O |r|
CN1c2ncccc2OC[C@H](NC(=O)c2nnc(Cc3cc(F)cc(c3)C#N)[nH]2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2nnc(Cc3cccc(c3)C#N)[nH]2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2ncc(Cc3cccc(c3)C#N)s2)C1=O |r|
CN1c2ncccc2OC[C@H](NC(=O)c2cc(F)n(Cc3ccccc3)n2)C1=O |r|
CN1c2ncccc2OC[C@H](NC(=O)c2cc(F)n(Cc3ccc(F)cc3)n2)C1=O |r|
CN1c2ncccc2OC[C@H](NC(=O)c2cc(C#N)n(Cc3cccc(c3)C#N)n2)C1=O |r|
CN1c2ncccc2OC[C@H](NC(=O)c2nn(Cc3cncc(c3)C#N)cc2F)C1=O |r|
Fc1cn(Cc2cccc(c2)C#N)nc1C(=O)N[C@H]1[C@H]2C[C@H]2c2cc(F)cc(F)c2NC1=O |r|
Fc1cn(Cc2cccc(c2)C#N)nc1C(=O)N[C@@H]1[C@@H]2C[C@@H]2c2cc(F)cc(F)c2NC1=O |r|
CN1c2ncccc2OC[C@H](NC(=O)c2ncn(Cc3cccc(c3)C#N)n2)C1=O |r|
C[C@H]1Oc2cccnc2N(C)C(=O)[C@H]1NC(=O)c1ncn(Cc2cccc(c2)C#N)n1 |r|
Fc1cc(F)c2NC(=O)[C@@H](NC(=O)c3nnc(Cc4ccccc4)[nH]3)[C@@H]3C[C@@H]3c2c1 |r|
CN1c2nccnc2[C@@H]2C[C@@H]2[C@H](NC(=O)c2nnc(Cc3ccccc3)o2)C1=O |r|
CN1c2nccnc2[C@H]2C[C@H]2[C@@H](NC(=O)c2nnc(Cc3ccccc3)o2)C1=O |r|
CN1c2nccnc2CC[C@H](NC(=O)c2nn(Cc3ccccc3F)cc2F)C1=O |r|
CN1c2nccnc2CC[C@@H](NC(=O)c2nn(Cc3ccccc3F)cc2F)C1=O |r|
CN1c2nccnc2[C@@H]2C[C@@H]2[C@H](NC(=O)c2nn(Cc3ccccc3F)cc2F)C1=O |r|
CN1c2nccnc2[C@H]2C[C@H]2[C@@H](NC(=O)c2nn(Cc3ccccc3F)cc2F)C1=O |r|
CN1c2nccnc2CC[C@H](NC(=O)c2nnc(o2)C2(CC2)c2ccccc2)C1=O |r|
CN1c2nccnc2CC[C@@H](NC(=O)c2nnc(o2)C2(CC2)c2ccccc2)C1=O |r|
Fc1cc(F)c2NC(=O)[C@H](NC(=O)c3nnc(Cc4cccc(c4)C#N)[nH]3)[C@@H]3C[C@@H]3c2c1 |r|
Fc1cc(F)c2NC(=O)[C@@H](NC(=O)c3nnc(Cc4cccc(c4)C#N)[nH]3)[C@H]3C[C@H]3c2c1 |r|
CN1c2nccnc2CC[C@@H](NC(=O)c2nn(Cc3cccnc3C)cc2F)C1=O |r|
CN1c2nccnc2CC[C@H](NC(=O)c2nn(Cc3cccnc3C)cc2F)C1=O |r|
CN1c2ccc(cc2[C@H]2C[C@H]2[C@@H](NC(=O)c2nn(Cc3ccccc3)cc2F)C1=O)S(C)(=O)=O |r|
CN1c2ccc(cc2[C@@H]2C[C@@H]2[C@H](NC(=O)c2nn(Cc3ccccc3)cc2F)C1=O)S(C)(=O)=O |r|
CN1c2ncccc2OC[C@H](NC(=O)c2nn(Cc3cnn(C)c3)cc2F)C1=O |r|
CN1c2nccnc2CC[C@H](NC(=O)c2cc(Cc3ccccc3)on2)C1=O |r|
CN1c2nccnc2CC[C@H](NC(=O)c2nnc(Cc3ccccc3)o2)C1=O |r|
C[C@H]1Oc2cccnc2N(C)C(=O)[C@H]1NC(=O)c1ncc(Cc2ccccc2)o1 |r|
C[C@H]1Oc2ncccc2N(C)C(=O)[C@H]1NC(=O)c1nnc(Cc2ccccc2)o1 |r|
CN1c2nccnc2[C@@H]2C[C@@H]2[C@H](NC(=O)c2ncc(Cc3ccccc3)o2)C1=O |r|
CN1c2nccnc2[C@@H]2C[C@@H]2[C@H](NC(=O)c2cn(Cc3ccccc3)nn2)C1=O |r|
CN1c2nccnc2[C@@H]2C[C@@H]2[C@H](NC(=O)c2cc(Cc3ccccc3)on2)C1=O |r|
CN1c2nccnc2[C@@H]2C[C@@H]2[C@H](NC(=O)c2nnc(Cc3ccccc3)s2)C1=O |r|
CN1c2nc(C)sc2CC[C@H](NC(=O)c2nnc(Cc3ccccc3)o2)C1=O |r|
CN1c2ncccc2OC[C@H](NC(=O)c2cn(Cc3ccccc3)nn2)C1=O |r|
C[C@H]1Oc2cccnc2N(C)C(=O)[C@H]1NC(=O)c1cn(Cc2ccccc2)nn1 |r|
C[C@H]1Oc2cccnc2N(C)C(=O)[C@H]1NC(=O)c1cnn(Cc2ccccc2)n1 |r|
C[C@H]1Oc2ncccc2N(C)C(=O)[C@H]1NC(=O)c1nn(Cc2ccccc2)cc1F |r|
CN1c2ccc(cc2[C@@H]2C[C@@H]2[C@H](NC(=O)c2nn(Cc3ccccc3)cc2F)C1=O)C#N |r|
CN1c2ncccc2CC[C@H](NC(=O)c2cc(on2)C2(CC2)n2nccn2)C1=O |r|
CN1c2nccnc2[C@@H]2C[C@@H]2[C@H](NC(=O)c2cn(Cc3ccccc3)c(C)n2)C1=O |r|
CN1c2ncccc2OC[C@H](NC(=O)c2nn(Cc3cocn3)cc2F)C1=O |r|
CN1c2ncccc2OC[C@H](NC(=O)c2ncc(Cc3ccccn3)s2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2nn(Cc3ccc(F)cn3)cc2F)C1=O |r|
CN1c2ncccc2OC[C@H](NC(=O)c2noc(Cc3ccccc3)n2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2nn(Cc3ccc(Cl)cn3)cc2F)C1=O |r|
C[C@H]1Oc2cccnc2N(C)C(=O)[C@H]1NC(=O)c1nnc(Cc2ccccc2)s1 |r|
CN1c2ncc(cc2[C@@H]2C[C@@H]2[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O)C#N |r|
CN1c2ncccc2CC[C@H](NC(=O)c2ncc(Cc3cccc(c3)C#N)s2)C1=O |r|
COc1cccc(Cn2cc(F)c(n2)C(=O)N[C@H]2COc3ccccc3N(C)C2=O)n1 |r|
C[C@H]1Oc2cccnc2N(C)C(=O)[C@H]1NC(=O)c1nnc(o1)C(F)(F)c1ccccc1 |r|
C[C@H]1Oc2cccnc2N(C)C(=O)[C@H]1NC(=O)c1noc(Cc2ccccc2)n1 |r|
CN1c2nccnc2[C@@H]2C[C@@H]2[C@H](NC(=O)c2nnc(Cc3ccc(F)cc3)o2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2nn(Cc3ncccn3)cc2F)C1=O |r|
CN1c2ccccc2CC[C@H](NC(=O)c2nnc(Cc3ccccc3)o2)C1=O |r|
CN1c2nccnc2[C@@H]2C[C@@H]2[C@H](NC(=O)c2ncc(Cc3ccccn3)o2)C1=O |r|
CN1c2nccnc2[C@@H]2C[C@@H]2[C@H](NC(=O)c2ncc(o2)C(F)(F)c2ccccc2)C1=O |r|
CN1c2ccccc2[C@H](F)CC(NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2ccccc2[C@@H](F)CC(NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
O=C(N[C@H]1COc2ccccc2-n2ccnc12)c1cc(Cc2ccccc2)on1 |r|
CN1c2ncccc2OC[C@H](NC(=O)c2nn(Cc3ccccn3)cc2F)C1=O |r|
C[C@H]1Cc2cccnc2N(C)C(=O)[C@H]1NC(=O)c1cc(Cc2ccccc2)on1 |r|
CN1c2ccncc2OC[C@H](NC(=O)c2nnc([nH]2)C2(CC2)c2ccccc2)C1=O |r|
CN1c2cnn(C)c2CC[C@H](NC(=O)c2nn(Cc3ccccc3)cc2F)C1=O |r|
CN1c2ncccc2[C@H]2CC2[C@@H](NC(=O)c2nnc(Cc3ccccc3)s2)C1=O |r|
C[C@H]1Oc2cccnc2N(C)C(=O)[C@H]1NC(=O)c1cc(Cc2ccccc2F)cnn1 |r|
CN1c2ncccc2OC[C@H](NC(=O)c2nc(C#N)c(Cc3cccc(c3)C#N)s2)C1=O |r|
CN1C(=O)N[C@H](Cc2c[nH]c3c(Cl)c(F)ccc23)C1=O |r|
Fc1ccc2cc[nH]c2c1Cl
Fc1ccc(cc1)-c1ccnc2sc(cc12)C(=O)N1CCOCC1
Fc1ccccc1-c1cccc2sc(cc12)C(=O)N1CCOCC1
Fc1ccc(cc1)-c1cccc2sc(cc12)C(=O)N1CCCC1
Fc1cccc(c1)-c1cccc2sc(cc12)C(=O)N1CCOCC1
Fc1ccc(cc1)-c1cccc2sc(cc12)C(=O)N1CCOCC1
Fc1ccc(cc1)-c1cccc2sc(cc12)C(=O)N1CCSCC1
Fc1ccc(cc1)-c1cccc2sc(cc12)C(=O)N1CCCOCC1
Fc1ccc(c(F)c1)-c1cccc2sc(cc12)C(=O)N1CCOCC1
O=C(N1CCOCC1)c1cc2c(cccc2s1)-c1cccs1
O=C(N1CCOCC1)c1cc2c(cccc2s1)-c1ccoc1
O=C(N1CCOCC1)c1cc2c(cccc2s1)-c1ccsc1
CN1c2ccccc2CC[C@H](NC(=O)c2nnc([nH]2)C2CCc3ccccc23)C1=O |r|
O=C(N[C@H]1COc2ccccc2-n2cnnc12)c1cc(Cc2ccccc2)on1 |r|
O=C(N[C@@H]1COc2ccccc2-n2cnnc12)c1cc(Cc2ccccc2)on1 |r|
CN1c2ncccc2OC[C@@H](NC(=O)c2cc(Oc3ccc(F)cc3F)ccn2)C1=O |r|
CN1c2ncccc2OC[C@H](NC(=O)c2cc(Oc3ccc(F)cc3F)ccn2)C1=O |r|
CN1c2ncccc2OC[C@H](NC(=O)c2nc(F)c(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2ncccc2CC[C@H](NC(=O)c2nc(C#N)c(Cc3ccccc3)s2)C1=O |r|
CN1c2ncccc2CC[C@H](NC(=O)c2nn(Cc3ccccc3C#N)cc2F)C1=O |r|
CN1c2ncccc2OC[C@H](NC(=O)c2cc(on2)C2(CC2)n2nccn2)C1=O |r|
COCC(=O)CCc1ccc2OC[C@H](NC(=O)c3n[nH]c(Cc4ccccc4)n3)C(=O)N(C)c2c1 |r|
CN1c2cc(CCC(=O)Nc3ccc4[nH]ncc4c3)ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O |r|
CN6C(=O)[C@@H](NC(=O)c2n[nH]c(Cc1ccccc1)n2)COc5ccc(CCC(=O)Nc4ccc3cn[nH]c3c4)cc56
COC1Cc2cccc(NC(=O)CCc3ccc4OC[C@H](NC(=O)c5n[nH]c(Cc6ccccc6)n5)C(=O)N(C)c4c3)c2CC1OC |r|
CCOC(=O)CCc1ccc2OC[C@H](NC(=O)c3ncn(Cc4ccccc4F)n3)C(=O)N(C)c2c1 |r|
CN1c2cc(CCC(O)=O)ccc2OC[C@H](NC(=O)c2ncn(Cc3ccccc3F)n2)C1=O |r|
CN1c2cc(CCC(=O)Nc3ccc4[nH]ncc4c3)ccc2OC[C@H](NC(=O)c2ncn(Cc3ccccc3F)n2)C1=O |r|
CCOC(=O)CCc1ccc2OC[C@H](NC(=O)c3ncn(Cc4c(Cl)cccc4Cl)n3)C(=O)N(C)c2c1 |r|
CN1c2cc(CCC(O)=O)ccc2OC[C@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O |r,c:31,t:20|
CN1c2cc(CCC(=O)N3CCCC3)ccc2OC[C@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O |r,c:36,t:25|
CN1c2cc(CCC(=O)N3CCOCC3)ccc2OC[C@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O |r,c:37,t:26|
CN1c2cc(CCC(=O)Nc3ccc4cccnc4c3)ccc2OC[C@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O |r,c:43,t:32|
CN1c2cc(CCC(=O)NC3CC3)ccc2OC[C@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O |r,c:35,t:24|
CN1c2cc(CCCO)ccc2OC[C@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O |r,c:30,t:19|
CN1c2cc(CCCCO)ccc2OC[C@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O |r,c:31,t:20|
CN1c2cc(CCCCOCc3ccccn3)ccc2OC[C@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O |r,c:39,t:28|
CN1c2cc(CCCCNc3ccccn3)ccc2OC[C@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O |r,c:38,t:27|
CN1c2cc(CCC(=O)N3CCCC3)ccc2OC[C@H](NC(=O)c2ncn(Cc3c(Cl)cccc3Cl)n2)C1=O |r|
CN1c2cc(CCC(=O)NC3CC3)ccc2OC[C@H](NC(=O)c2ncn(Cc3c(Cl)cccc3Cl)n2)C1=O |r|
CN1c2cc(CN3CCN(CC3)c3ccncc3)ccc2OC[C@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O |r,c:41,t:30|
CN1c2cc(CN3CCN(CC3)c3ccncc3)ccc2OC[C@H](NC(=O)C2=NC(Cc3c(Cl)cccc3Cl)N=N2)C1=O |r,c:43,t:30|
CN1c2cc(\C=C\C(=O)N3CCCC3)ccc2OC[C@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O |r,c:36,t:25|
CN1c2cc(\C=C\C(=O)NC3CC3)ccc2OC[C@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O |r,c:35,t:24|
CN1c2cc(CN3CCn4ncnc4C3)ccc2OC[C@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O |r,c:38,t:27|
CN1c2cc(CN3CCn4ncnc4C3)ccc2OC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O |r|
CN1c2cc(CCC(=O)NC3CC3)ccc2OC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O |r|
CN1c2cc(CCC(=O)NC3CC3)ccc2OC[C@H](NC(=O)c2ncn(Cc3ccc(F)cc3F)n2)C1=O |r|
CN1c2cc(CCC(C)(C)O)ccc2OC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O)C#CC(C)(C)O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O)C#CC(C)(C)O |r,c:26,t:15|
CN1c2cc(CCC(N)=O)ccc2OC[C@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O |r,c:31,t:20|
CN1c2cc(CCC(N)=O)ccc2OC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O |r|
CN1c2cc(CCC(=O)N3CCCC3)ccc2OC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O |r|
CN1c2cc(CCC(=O)N3CCCC3)ccc2OC[C@H](NC(=O)c2nnn(Cc3cc(F)ccc3F)n2)C1=O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O)C#CCCCO |r,c:26,t:15|
CN1c2cc(ccc2OC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O)C#CCCOc1ccc2ncccc2c1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O)C#CCCOc1ccc2ncccc2c1 |r,c:26,t:15|
CN1c2cc(CN3CCN4N=C(NC4C3)C(F)(F)F)ccc2OC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O |r,c:10|
CN1c2cc(CN3CCN4N=C(NC4C3)C(F)(F)F)ccc2OC[C@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O |r,c:10,42,t:31|
CN1c2cc(ccc2OC[C@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O)C#CCCOc1ccc2cccnc2c1 |r,c:26,t:15|
CN1c2cc(ccc2OC[C@@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O)C#CCCOc1ccc2cccnc2c1 |r,c:26,t:15|
CN1c2cc(ccc2OC[C@H](NC(=O)C2=NC(Cc3ccc(F)cc3F)N=N2)C1=O)C#CC(C)(C)O |r,c:28,t:15|
CN1c2cc(ccc2OC[C@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O)C#CCCOc1cccc2ncccc12 |r,c:26,t:15|
CN1c2cc(ccc2OC[C@@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O)C#CCCOc1cccc2ncccc12 |r,c:26,t:15|
CN1c2cc(CN3CCn4c(C3)nnc4C(F)(F)F)ccc2OC[C@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O |r,c:42,t:31|
CN1c2cc(CN3CCn4c(C3)nnc4C(F)(F)F)ccc2OC[C@@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O |r,c:42,t:31|
CN1c2cc(ccc2OC[C@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O)C#CC(C)(C)C |r,c:26,t:15|
CN1c2cc(ccc2OC[C@@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O)C#CC(C)(C)C |r,c:26,t:15|
CN5C(=O)[C@@H](NC(=O)c2n[nH]c(Cc1ccccc1)n2)COc4ccc(C#CC3(O)CCC3)cc45
CN1c2cc(ccc2OC[C@@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O)C#CC1(O)CCC1 |r,c:26,t:15|
CN1c2cc(ccc2OC[C@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O)C#CC1(O)CCCC1 |r,c:26,t:15|
CN1c2cc(ccc2OC[C@@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O)C#CC1(O)CCCC1 |r,c:26,t:15|
CN1c2cc(ccc2OC[C@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O)C#CC1(O)CCOCC1 |r,c:26,t:15|
CN1c2cc(ccc2OC[C@@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O)C#CC1(O)CCOCC1 |r,c:26,t:15|
CN1c2cc(ccc2OC[C@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O)C#CC1(O)COC1 |r,c:26,t:15|
CN1c2cc(ccc2OC[C@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O)C#CC(C)=C |r,c:26,t:15|
CC(C)CCc1ccc2OC[C@H](NC(=O)C3=NC(Cc4ccccc4)N=N3)C(=O)N(C)c2c1 |r,c:26,t:15|
COC(C)(C)C#Cc1ccc2OC[C@H](NC(=O)C3=NC(Cc4ccccc4)N=N3)C(=O)N(C)c2c1 |r,c:28,t:17|
CN1c2cc(ccc2OC[C@H](NC(=O)C2=NC(Oc3ccccc3)N=N2)C1=O)C#CC(C)(C)O |r,c:26,t:15|
CN1c2cc(ccc2OC[C@H](NC(=O)C2=NC(Cc3c(Cl)cccc3Cl)N=N2)C1=O)C#CC(C)(C)O |r,c:28,t:15|
CN1c2ccc(CN3CCn4nc(nc4C3)C(F)(F)F)cc2OC[C@H](NC(=O)C2=NC(Cc3c(Cl)cccc3Cl)N=N2)C1=O |r,c:44,t:31|
CN1c2ccc(CN3CCn4nc(nc4C3)C(F)(F)F)cc2OC[C@H](NC(=O)c2ncn(Cc3c(Cl)cccc3Cl)n2)C1=O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC(C)(C)O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CC(C)(C)O |r|
CN1c2cc(ccc2OC[C@@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CC(C)(C)O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2nnc(Cc3ccccc3)o2)C1=O)C#CC(C)(C)O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CC1(O)COC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#C[C@@]1(O)COC2[C@H](COC12)OC(=O)c1ccccc1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#C[C@@]1(O)COC2[C@@H](O)COC12 |r|
COC(=O)C(C)(C)C#Cc1ccc2OC[C@H](NC(=O)c3n[nH]c(Cc4ccccc4)n3)C(=O)N(C)c2c1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2ccn(Cc3ccccc3)n2)C1=O)C#CC(C)(C)O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)C2=NC(Cc3cccc(F)c3)N=N2)C1=O)C#CC(C)(C)O |r,c:27,t:15|
CN1c2cc(ccc2OC[C@H](NC(=O)C2=NC(Cc3ccc(F)cc3)N=N2)C1=O)C#CC(C)(C)O |r,c:27,t:15|
CN1c2cc(ccc2OC[C@H](NC(=O)C2=NC(Cc3ccccc3F)N=N2)C1=O)C#CC(C)(C)O |r,c:27,t:15|
CN1c2cc(ccc2OC[C@H](NC(=O)c2ccn(Cc3ccccc3)n2)C1=O)C#C |r|
CN1c2cc(ccc2OC[C@H](NC(=O)C2=NC(Cc3ccccc3C)N=N2)C1=O)C#CC(C)(C)O |r,c:27,t:15|
CN1c2cc(ccc2OC[C@H](NC(=O)C2=NC(Cc3ccc(cc3)-c3ccccc3)N=N2)C1=O)C#CC(C)(C)O |r,c:33,t:15|
CN1c2cc(ccc2OC[C@H](NC(=O)c2ncn(Cc3c(C)cccc3C)n2)C1=O)C#CC(C)(C)O |r|
CC(C)Cn1cnc(n1)C(=O)N[C@H]1COc2ccc(cc2N(C)C1=O)C#CC(C)(C)O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Cc3ccccc3)on2)C1=O)C#CC(C)(C)O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#Cc1ccc2CCNCc2c1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3F)n2)C1=O)C#CC(C)(C)C |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3c(C)cccc3C)n2)C1=O)C#CC(C)(C)C |r|
CCN1c2cc(ccc2OC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O)C#CC(C)(C)O |r|
CCN1c2cc(ccc2OC[C@H](NC(=O)c2ncn(Cc3cccc(F)c3)n2)C1=O)C#CC(C)(C)O |r|
CC(=C)C#Cc1ccc2OC[C@H](NC(=O)c3ncn(Cc4ccccc4)n3)C(=O)Nc2c1 |r|
CN1c2cc(\C=C(/Cl)C(C)(C)O)ccc2OC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O)C#CCN1CCCC1 |r,c:26,t:15|
CN1c2cc(ccc2OC[C@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O)C#CCN1CCOCC1 |r,c:26,t:15|
CN1c2cc(ccc2OC[C@H](NC(=O)C2=NC(Cc3ccccc3)N=N2)C1=O)C#C[Si](C)(C)C |r,c:26,t:15|
CN1c2ccc(=O)n(C)c2CC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O |r|
CN1c2ccc(=O)n(C)c2CC[C@H](NC(=O)c2ncn(Cc3ccccc3F)n2)C1=O |r|
CN1c2cccc(=O)n2CC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O |r|
CN1c2cccc(=O)n2CC[C@H](NC(=O)c2ncn(Cc3ccccc3F)n2)C1=O |r|
CN1c2cc(=O)n(C)cc2CC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O |r|
CN1c2cc(=O)n(C)cc2CC[C@H](NC(=O)c2ncn(Cc3ccccc3F)n2)C1=O |r|
CN1c2cn(C)c(=O)cc2CC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O |r|
CN1c2cn(C)c(=O)cc2CC[C@@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O |r|
CN1c2cn(C)c(=O)cc2CC[C@H](NC(=O)c2ncn(Cc3ccccc3F)n2)C1=O |r|
CN1c2cn(C)c(=O)cc2CC[C@@H](NC(=O)c2ncn(Cc3ccccc3F)n2)C1=O |r|
CN1c2cn(C)c(=O)cc2CC[C@H](NC(=O)c2nc3CC[C@@H](c4ccccc4F)n3n2)C1=O |r|
CN1c2cn(C)c(=O)cc2CC[C@@H](NC(=O)c2nc3CC[C@@H](c4ccccc4F)n3n2)C1=O |r|
CN1c2cc(=O)n(C)cc2CC[C@H](NC(=O)c2nc3CC[C@@H](c4ccccc4F)n3n2)C1=O |r|
CN1c2cc(=O)n(CC3CC3)cc2CC[C@H](NC(=O)c2nc3CC[C@@H](c4ccccc4F)n3n2)C1=O |r|
CN1c2cc(=O)n(CC3CC3)cc2CC[C@H](NC(=O)c2ncn(Cc3ccccc3F)n2)C1=O |r|
CN1c2cc(=O)n(CC3CC3)cc2CC[C@@H](NC(=O)c2nc3CC[C@@H](c4ccccc4F)n3n2)C1=O |r|
CN1c2cc(=O)n(CC3CC3)cc2CC[C@@H](NC(=O)c2ncn(Cc3ccccc3F)n2)C1=O |r|
CCn1cc2CC[C@H](NC(=O)c3nc4CC[C@@H](c5ccccc5F)n4n3)C(=O)N(C)c2cc1=O |r|
CCn1cc2CC[C@H](NC(=O)c3ncn(Cc4ccccc4F)n3)C(=O)N(C)c2cc1=O |r|
CCn1cc2CC[C@@H](NC(=O)c3nc4CC[C@@H](c5ccccc5F)n4n3)C(=O)N(C)c2cc1=O |r|
CCn1cc2CC[C@@H](NC(=O)c3ncn(Cc4ccccc4F)n3)C(=O)N(C)c2cc1=O |r|
CN1c2ccc(=O)n(C)c2CC[C@@H](NC(=O)c2ncn(Cc3ccccc3F)n2)C1=O |r|
CN1c2ccc(=O)n(C)c2CC[C@@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2ncn(Cc3ccc(F)cc3)n2)C1=O)N1CCC(CO)(CCl)CC1
CN1c2cc(ccc2OC[C@H](NC(=O)c2ncn(Cc3ccc(F)cc3)n2)C1=O)N1CC2(C1)CCOCC2
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Cc3ccccc3)on2)C1=O)N1CC2(C1)CCOCC2
CN1c2cc(ccc2OC[C@H](NC(=O)c2ncn(Cc3ccc(F)cc3)n2)C1=O)N1CCC2(COC2)CC1
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)N1CC2(C1)CCOCC2
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Cc3ccccc3)on2)C1=O)N1C[C@@H]2C[C@H]1CO2
CN1c2cc(ccc2OC[C@H](NC(=O)c2ncn(Cc3ccc(F)cc3)n2)C1=O)N1C[C@@H]2C[C@H]1CO2
CN1c2cc(ccc2OC[C@H](NC(=O)c2ncn(Cc3ccc(F)cc3)n2)C1=O)N1CCCOCC1
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Cc3ccccc3)on2)C1=O)N1CCCOCC1
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccc(F)cc3)n2)C1=O)N1CCCOCC1
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccc(F)cc3)n2)C1=O)N1CC2(C1)CCOCC2
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)N1CCCOCC1
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Cc3ccccc3)on2)C1=O)N1CC2CCC(C1)O2
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Cc3ccccc3)on2)C1=O)N1CCN2CCC1CC2 |wD:10.11,(5.39,-5.08,;5.16,-3.56,;3.69,-3.11,;2.73,-4.31,;1.21,-4.08,;.64,-2.65,;1.6,-1.44,;3.13,-1.67,;3.9,-.34,;5.42,-.11,;6.55,-1.16,;7.98,-.6,;9.19,-1.56,;8.96,-3.08,;10.62,-.99,;11.92,-1.82,;13.11,-.84,;14.6,-1.23,;15.01,-2.72,;16.5,-3.1,;16.91,-4.59,;15.83,-5.68,;14.34,-5.3,;13.93,-3.81,;12.55,.59,;11.01,.5,;6.43,-2.69,;7.77,-3.46,;.25,-5.29,;.92,-6.67,;.25,-8.06,;-1.25,-8.4,;-2.46,-7.44,;-2.46,-5.9,;-1.25,-4.94,;-.97,-6.1,;-.97,-7.25,)|
CN1c2ccc(cc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)N1CCC2(CCOCC2)CC1
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)N1CCN2CCC1CC2 |wD:10.11,(5.39,-5.08,;5.16,-3.56,;3.69,-3.11,;2.73,-4.31,;1.21,-4.08,;.64,-2.65,;1.6,-1.44,;3.13,-1.67,;3.9,-.34,;5.42,-.11,;6.55,-1.16,;7.98,-.6,;9.19,-1.56,;8.96,-3.08,;10.62,-.99,;11.01,.5,;12.55,.59,;13.11,-.84,;14.6,-1.23,;15.01,-2.72,;16.5,-3.1,;16.91,-4.59,;15.83,-5.68,;14.34,-5.3,;13.93,-3.81,;11.92,-1.82,;6.43,-2.69,;7.77,-3.46,;.25,-5.29,;.92,-6.67,;.25,-8.06,;-1.25,-8.4,;-2.46,-7.44,;-2.46,-5.9,;-1.25,-4.94,;-.97,-6.1,;-.97,-7.25,)|
CN1c2cc(NCCCCl)ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)N1CCC2(CCCO2)CC1
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccc(F)cc3)n2)C1=O)N1CCC2(CCCO2)CC1
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)N1CCC1
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)N1CCC2(CCOC2)CC1
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)N1CCC2(C1)CCOCC2
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)N1CCC2(CCN(Cc3ccccc3)C2=O)CC1
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)N1CCC2(CCCN(Cc3ccccc3)C2=O)CC1
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)N1CCC2(CCOCC2)CC1
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)N1CC(F)(F)C1
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)N1CC(F)C1
FC1(F)CN(C1)C(=O)c1nc2n(n1)C(CC2(F)F)c1ccccc1
FC1(F)CN(C1)C(=O)c1nc2n(n1)[C@H](CC2(F)F)c1ccccc1 |r|
FC1(F)CN(C1)C(=O)c1nc2n(n1)[C@@H](CC2(F)F)c1ccccc1 |r|
F[C@H]1C[C@H](c2ccccc2)n2nc(nc12)C(=O)N1CC(F)(F)C1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)N1CC(F)(F)C1 |r|
FC1(F)CN(C1)C(=O)c1nc2C(CCn2n1)c1ccccc1
FC1(F)CN(C1)C(=O)c1nc2C(OCCn2n1)c1ccccc1
Fc1ccccc1C1OCCn2nc(nc12)C(=O)N1CC(F)(F)C1
CC[C@@]1(C)OCc2cnc(cc12)C(=O)N1CC(F)(F)C1 |r|
CC(F)(F)C1CCc2nc(nn12)C(=O)N1CC(F)(F)C1
FC1(F)CN(C1)C(=O)c1cc2[C@H](CCn2n1)c1ccccc1 |r|
Fc1ccccc1[C@@H]1CCc2nc(nn12)C(=O)N1CC(F)(F)C1 |r|
Fc1ccccc1[C@H]1CCc2nc(nn12)C(=O)N1CC(F)(F)C1 |r|
Fc1ccccc1[C@H]1CCc2nc(nn12)C(=O)N1CCC1 |r|
Fc1ccccc1C1CCn2nc(nc12)C(=O)N1CC(F)(F)C1
FC1(F)CN(C1)C(=O)c1nc2[C@@H](CCn2n1)c1ccccc1 |r|
FC1(F)CN(C1)C(=O)c1nc2CCC(c3ccccc3)n2n1
COC1CN(C1)C(=O)c1nc2CCC(c3ccccc3)n2n1
FC1CN(C1)C(=O)c1nc2CCC(c3ccccc3)n2n1
CC1CN(C1)C(=O)c1nc2CCC(c3ccccc3)n2n1
CC1(F)CN(C1)C(=O)c1nc2CCC(c3ccccc3)n2n1
CCC1CN(C1)C(=O)c1nc2CCC(c3ccccc3)n2n1
Fc1ccccc1C1CCc2nc(nn12)C(=O)N1CCC1
Fc1ccccc1C1CCc2nc(nn12)C(=O)N1CC(F)(F)C1
FC1CN(C1)C(=O)c1nc2CCC(c3ccccc3F)n2n1
CNC(=O)c1nc2CCC(c3ccccc3)n2n1
O=C(N1CCC1)c1nc2CCC(c3ccccc3)n2n1
CN(C)C(=O)c1nc2CCC(c3ccccc3)n2n1
O=C(N1CC2CC1C2)c1nc2CCC(c3ccccc3)n2n1 |(3.24,-1.79,;2.84,-.31,;3.93,.78,;3.93,2.32,;5.39,2.8,;6.3,1.55,;5.39,.31,;4.14,1.55,;1.35,.09,;1.11,1.61,;-.41,1.85,;-1.5,2.94,;-2.87,2.24,;-2.63,.72,;-3.72,-.37,;-3.32,-1.85,;-4.41,-2.94,;-5.9,-2.54,;-6.3,-1.06,;-5.21,.03,;-1.11,.48,;-.02,-.61,)|
O=C(N1CCCCC1)c1nc2CCC(c3ccccc3)n2n1
O=C(N1CCCC1)c1nc2CCC(c3ccccc3)n2n1
FC1(F)CN(C1)C(=O)c1nc2CC[C@@H](c3ccccc3)n2n1 |r|
FC1(F)CN(C1)C(=O)c1nc2CC[C@H](c3ccccc3)n2n1 |r|
CN(C)C(=O)c1nc2CCC(c3ccccc3F)n2n1
Fc1ccccc1C1CCc2nc(nn12)C(=O)N1CCCC1
FC1CN(C1)C(=O)c1nc2[C@H](F)C[C@@H](c3ccccc3)n2n1 |r|
CC1(F)CN(C1)C(=O)c1nc2n(n1)[C@H](CC2(F)F)c1ccccc1 |r|
FC1CN(C1)C(=O)c1nc2[C@H](F)C[C@H](c3ccccc3)n2n1 |r|
CCC(F)(F)C1CCc2nc(nn12)C(=O)N1CC(F)(F)C1
CN(C)C(=O)c1nc2C(OCCn2n1)c1ccccc1
FC1CN(C1)C(=O)c1nc2C(OCCn2n1)c1ccccc1
CN(C)C(=O)c1nc2C(OCCn2n1)c1ccccc1F
CCN(CC)C(=O)c1nc2C(OCCn2n1)c1ccccc1F
FC1CN(C1)C(=O)c1nc2C(OCCn2n1)c1ccccc1F
FC1CN(C1)C(=O)c1nc2C3CC3C(c3ccccc3)n2n1
FC1(F)CN(C1)C(=O)c1nc2C3CC3C(c3ccccc3)n2n1
FC1CN(C1)C(=O)c1nc2n(n1)[C@H](CC2(F)F)c1ccccc1 |r|
FC(F)(F)[C@@H]1CCc2nc(nn12)C(=O)N1CC(F)(F)C1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)N1CC(C1)C(F)(F)F |r|
FC(F)C1CN(C1)C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
FC(F)[C@H]1CCN1C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
F[C@@H]1C[C@H](c2ccccc2)n2nc(nc12)C(=O)N1CCC(F)(F)C1 |r|
COCCN(CC(F)(F)F)C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
COCCN(CC(F)F)C(=O)c1nc2[C@H](F)C[C@H](c3ccccc3)n2n1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)N(CC(F)(F)F)C1COC1 |r|
FC(F)CN(C1CC1)C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)N(CC(F)(F)F)C1CC1 |r|
FC(F)C1CCN1C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)N(C1CC1)C1CC1 |r|
CC1CN(Cc2ccnn12)C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
Cc1cc2CN(CCn2n1)C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
FC(F)[C@@H]1CCCN1C(=O)c1nc2[C@H](F)C[C@H](c3ccccc3)n2n1 |r|
F[C@@H]1C[C@H](c2ccccc2)n2nc(nc12)C(=O)N1CCn2nccc2C1 |r|
F[C@@H]1C[C@H](c2ccccc2)n2nc(nc12)C(=O)N1CCc2cccnc2C1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)N1CCn2ccnc2C1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)N1CCn2nccc2C1 |r|
C[C@@H]1C[C@H](F)CN1C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
OC[C@H]1CCCN1C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
OCC1CC(F)(F)CN1C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
FC[C@@H]1CC(F)(F)CN1C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)N1CCc2cccnc2C1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)N1CCc2cnccc2C1 |r|
F[C@@H]1C[C@H](c2ccccc2)n2nc(nc12)C(=O)N1CCc2ccccc2C1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)N1CCC(C1)Oc1ccccc1 |r|
FC(F)C1CCCN1C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)N1CCCC(F)(F)C1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)N1CCCn2nccc12 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)N1CCC(n2nccc12)C(F)(F)F |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)N1CCC[C@H]1C(F)(F)F |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)N1CCC[C@@H]1C(F)(F)F |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)N1CCCC1C(F)(F)F |r|
C[C@H]1[C@@H](CCN1C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1)C(F)(F)F |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)N1CC2CC1CC2(F)F |r,TLB:15:17:22.23:20|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)N1CCc2ccncc2C1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)N1CCc2ncccc2C1 |r|
CN(C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1)c1ccccc1 |r|
CN(CC(F)F)C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
CN(CC(F)(F)F)C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)N1CCC(Cc2ccccc2)C1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)N1CCCc2ccccc2C1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)N1CCc2cccc(F)c2C1 |r|
CC1N(CCc2cccc(F)c12)C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
CC1N(CCc2ccccc12)C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)N1CCC(F)(F)C1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)N1CCc2ccccc2C1 |r|
F[C@@H]1C[C@H](c2ccccc2)n2nc(nc12)C(=O)N1CC2C(C1)C2(F)F |r|
F[C@@H]1C[C@H](c2ccccc2)n2nc(nc12)C(=O)N1CC2CC2C1 |r|
FC1(F)CN(C1)C(=O)c1cc2CCC(c3ccccc3)n2n1
CCC(F)(F)n1ncc2cnc(cc12)C(=O)N1CC(F)(F)C1
F[C@@H]1C[C@H](c2ccccc2)n2nc(nc12)C(=O)N1CCC1 |r|
CN(C)C(=O)c1nc2[C@H](F)C[C@H](c3ccccc3)n2n1 |r|
CCC(F)(F)[C@H]1CCc2nc(nn12)C(=O)N[C@H]1CCc2cc(F)cc(F)c2NC1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2nc3[C@@H](F)C[C@H](c4ccccc4)n3n2)C1=O |r|
F[C@H]1C[C@H](c2ccccc2)n2nc(nc12)C(=O)N[C@H]1CCc2cc(F)cc(F)c2NC1=O |r|
F[C@@H]1C[C@H](c2ccccc2)n2nc(nc12)C(=O)N[C@H]1CCc2cc(F)cc(F)c2NC1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2ncc3cnn(CC(C)(F)F)c3n2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2ncc3cnn(C4CC4)c3n2)C1=O |r|
COc1cc2CC[C@H](NC(=O)c3nc4CC[C@H](c5ccccc5)n4n3)C(=O)N(C)c2cn1 |r|
O=C(N[C@H]1CCc2ncccc2NC1=O)c1nc2CC[C@H](c3ccccc3)n2n1 |r|
CN1c2ccccc2OC[C@H](NC(=O)c2nc3[C@@H](F)C[C@@H](c4ccccc4)n3n2)C1=O |r|
CN1c2ccnn2CC[C@H](NC(=O)c2nc3[C@@H](F)C[C@@H](c4ccccc4)n3n2)C1=O |r|
COc1cc2CC[C@H](NC(=O)c3nc4CC[C@@H](c5ccccc5F)n4n3)C(=O)N(C)c2cn1 |r|
Fc1ccccc1[C@@H]1CCc2nc(nn12)C(=O)N[C@H]1CCc2ncccc2NC1=O |r|
CN1c2cccnc2CC[C@H](NC(=O)c2nc3CC[C@H](c4ccccc4F)n3n2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2cc3[C@@H](OCCn3n2)c2ccccc2)C1=O |r|
Fc1cc(F)c2NC(=O)[C@H](CCc2c1)NC(=O)c1cc2C(OCCn2n1)c1ccccc1 |r|
CN1c2ccccc2OC[C@H](NC(=O)c2cc3n(CC(C)(F)F)ncc3cn2)C1=O |r|
CN1c2cccnc2CC[C@H](NC(=O)c2nc3[C@@H](CCn3n2)c2ccccc2F)C1=O |r|
CN1c2cccnc2CC[C@H](NC(=O)c2nc3[C@@H](CCn3n2)c2ccccc2)C1=O |r|
CN1c2cccnc2CC[C@H](NC(=O)c2nc3CC[C@@H](c4ccccc4)n3n2)C1=O |r|
F[C@@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)N[C@H]1CCc2cc(F)cc(F)c2NC1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2nc3[C@H](F)C[C@@H](c4ccccc4)n3n2)C1=O |r|
CN1c2cc(C)nn2CC[C@H](NC(=O)c2nc3[C@@H](F)C[C@H](c4ccccc4)n3n2)C1=O |r|
CN1c2ccnn2CC[C@H](NC(=O)c2nc3[C@@H](F)C[C@H](c4ccccc4)n3n2)C1=O |r|
Fc1cc(F)c2NC(=O)[C@H](CCc2c1)NC(=O)c1nc2n(n1)C(CC2(F)F)c1ccccc1 |r|
CN1c2ccccc2OC[C@H](NC(=O)c2nc3n(n2)C(CC3(F)F)c2ccccc2)C1=O |r|
FC1CC(c2ccccc2)n2nc(nc12)C(=O)N[C@H]1CCc2cc(F)cc(F)c2NC1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2nc3C(F)CC(c4ccccc4)n3n2)C1=O |r|
CN1c2ccnn2CC[C@H](NC(=O)c2nc3C(F)CC(c4ccccc4)n3n2)C1=O |r|
CN1c2ccnn2CC[C@H](NC(=O)c2nc3[C@@H](CCn3n2)c2ccccc2F)C1=O |r|
CN1c2cc(C)nn2CC[C@H](NC(=O)c2nc3[C@@H](CCn3n2)c2ccccc2F)C1=O |r|
CN1c2cn(C)nc2CC[C@H](NC(=O)c2ncn(Cc3ccccc3F)n2)C1=O |r|
CN1c2cn(C)nc2CC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O |r|
CN1c2cnn(C)c2CC[C@H](NC(=O)c2ncn(Cc3ccccc3F)n2)C1=O |r|
CN1c2cnn(C)c2CC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O |r|
CN1c2cc(CC3CCOC3)nn2CC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O |r|
CN1c2cc(C)nn2CC[C@H](NC(=O)c2nc3[C@@H](F)C[C@@H](c4ccccc4)n3n2)C1=O |r|
CN1c2cc(C)nn2CC[C@H](NC(=O)c2nc3n(n2)[C@H](CC3(F)F)c2ccccc2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2nc3n(n2)[C@H](CC3(F)F)c2ccccc2)C1=O |r|
CN1c2ccnn2CC[C@H](NC(=O)c2nc3n(n2)[C@H](CC3(F)F)c2ccccc2)C1=O |r|
CCC(F)(F)[C@@H]1CCc2nc(nn12)C(=O)N[C@H]1COc2ccccc2N(C)C1=O |r|
F[C@@H]1C[C@@H]1C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
F[C@H]1C[C@H]1C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
F[C@@H]1C[C@@H]1C(=O)c1nc2[C@H](F)C[C@H](c3ccccc3)n2n1 |r|
F[C@H]1C[C@H]1C(=O)c1nc2[C@H](F)C[C@H](c3ccccc3)n2n1 |r|
CC(C)(O)C(=O)c1nc2[C@H](F)C[C@H](c3ccccc3)n2n1 |r|
CC(C)(O)C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)Cc1ccccc1 |r|
F[C@H]1C[C@@H]1C(=O)c1nc2[C@H](F)C[C@H](c3ccccc3)n2n1 |r|
F[C@@H]1C[C@H]1C(=O)c1nc2[C@H](F)C[C@H](c3ccccc3)n2n1 |r|
F[C@H]1C[C@H]1C(=O)c1nc2C(F)CC(c3ccccc3)n2n1 |r|
FC1CC(c2ccccc2)n2nc(nc12)C(=O)C1CC1(F)F
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)c1ccccc1 |r|
CCC(=O)c1nc2[C@@H](F)C[C@H](c3ccccc3)n2n1 |r|
FC1CC(c2ccccc2)n2nc(nc12)C(=O)C1(CC1)C(F)(F)F
CC1(COC1)C(=O)c1nc2C(F)CC(c3ccccc3)n2n1
F[C@@H]1C[C@H]1C(=O)c1nc2C(F)CC(c3ccccc3)n2n1 |r|
CCC(=O)c1cn2CCC(c2n1)c1ccccc1
F[C@H]1C[C@H](c2ccccc2)n2nc(nc12)C(=O)C1CC1 |r|
CCC(=O)c1cc2CCC(c3ccccc3)n2n1
CCC(=O)c1cc2[C@H](OCCn2n1)c1ccccc1F |r|
CCC(=O)c1cc2[C@@H](OCCn2n1)c1ccccc1F |r|
CC(C)(C#N)C(=O)c1nc2C(F)CC(c3ccccc3)n2n1
CCC(=O)c1cc2[C@@H](CCn2n1)c1ccccc1 |r|
CCC(=O)c1cc2[C@H](CCn2n1)c1ccccc1 |r|
CC(C)(O)C(=O)c1nc2C(F)CC(c3ccccc3)n2n1
CC1(CC1)C(=O)c1nc2C(F)CC(c3ccccc3)n2n1
CCC(=O)c1cc2[C@H](OCCn2n1)c1ccccc1 |r|
CCC(=O)c1cc2[C@@H](OCCn2n1)c1ccccc1 |r|
F[C@@H]1C[C@H](c2ccccc2)n2nc(nc12)C(=O)CC(F)(F)F |r|
CCC(=O)c1nc2CC[C@@H](c3ccccc3)n2n1 |r|
CCC(=O)c1nc2CC[C@@H](c3ccccc3F)n2n1 |r|
CCC(=O)c1nc2C[C@H](F)[C@@H](c3ccccc3)n2n1 |r|
FC1CC(c2ccccc2)n2nc(nc12)C(=O)c1ccccn1
c1ccc(cc1)[C@@H]2C[C@@H](c3n2nc(n3)C(=O)C4CC4)F
F[C@@H]1C[C@H](c2ccccc2)n2nc(nc12)C(=O)C1CC1 |r|
FC1CC(c2ccccc2)n2nc(nc12)C(=O)C1CCCC1
CC(C)(C)C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
CC(C)(C)C(=O)c1nc2[C@H](F)C[C@H](c3ccccc3)n2n1 |r|
Cn1cc(cn1)C(=O)c1nc2[C@H](F)C[C@H](c3ccccc3)n2n1 |r|
Cn1cc(cn1)C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
FC1CC(c2ccccc2)n2nc(nc12)C(=O)c1cccs1
FC1CC(c2ccccc2)n2nc(nc12)C(=O)C1CC1
F[C@@H]1C[C@H](c2ccccc2)n2nc(nc12)C(=O)C1CCC1 |r|
CC(C)(C)C(=O)c1nc2C(F)CC(c3ccccc3)n2n1
CC(C)C(=O)c1nc2C(F)CC(c3ccccc3)n2n1
CCC(=O)c1nc2[C@H](F)C[C@H](c3ccccc3)n2n1 |r|
CCC(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
CC(=O)c1nc2[C@H](F)C[C@H](c3ccccc3)n2n1 |r|
F[C@H]1C[C@@H]1C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
F[C@@H]1C[C@H]1C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
FC1CC(c2ccccc2)n2nc(nc12)C(=O)C1(F)CC1
CC1(COC1)C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
CC1(COC1)C(=O)c1nc2[C@H](F)C[C@H](c3ccccc3)n2n1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)C1C2COCC12 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)C1COC1 |r|
OCC1(CC1)C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)[C@H]1CC1(F)F |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)[C@@H]1CC1(F)F |r|
OC(c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1)C1(F)CC1 |r|
F[C@H]1C[C@@H](c2ccccc2F)n2nc(nc12)C(=O)C1CC1 |r|
Fc1ccccc1[C@@H]1CCc2nc(nn12)C(=O)C1CC1 |r|
F[C@@H]1C[C@H](c2ccccc2)n2nc(nc12)C(=O)C1CC(F)(F)C1 |r|
F[C@@H]1C[C@H]1C(=O)c1nc2n(n1)[C@@H](CC2(F)F)c1ccccc1 |r|
F[C@H]1C[C@@H]1C(=O)c1nc2n(n1)[C@@H](CC2(F)F)c1ccccc1 |r|
FC1(F)C[C@@H](c2ccccc2)n2nc(nc12)C(=O)C1CC1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)C1CC2(CC2(F)F)C1 |r,wU:1.0,3.3,(4.68,4.14,;3.91,2.81,;4.82,1.56,;3.91,.32,;4.31,-1.17,;3.22,-2.26,;3.62,-3.75,;5.11,-4.14,;6.2,-3.05,;5.8,-1.57,;2.45,.79,;.98,.32,;.08,1.56,;.98,2.81,;2.45,2.33,;-1.46,1.56,;-2.23,2.9,;-2.23,.23,;-3.72,-.17,;-3.32,-1.66,;-3.32,-3.2,;-4.66,-2.43,;-6.2,-2.43,;-5.43,-1.09,;-1.83,-1.26,)|
CCC(=O)c1nc2CC[C@@H](c3ccccc3Cl)n2n1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)C1CC(F)(F)C1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)C1CC1c1ccccn1 |r|
C[C@H]1C[C@@H]1C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)C1CC2(CC2)C1 |r|
Clc1ccccc1[C@@H]1CCc2nc(nn12)C(=O)C1CC1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(cc12)C(=O)C1CC1 |r|
FCC1(CC1)C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)C1C2CC(F)(F)CC12 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)C1CC1C(F)(F)F |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)C1CC2C(C1)C2(F)F |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)C1(CC#N)CC1 |r|
CO[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)C1CC1 |r|
F[C@H]1C[C@@H](c2ccc(F)cc2)n2nc(nc12)C(=O)C1CC1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)C1CC1C#N |r|
O[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)C1CC1 |r|
O[C@@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)C1CC1 |r|
F[C@H]1C[C@@H]1C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3F)n2n1 |r|
C[C@@H]1C[C@H]1C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
CC[C@@H]1C[C@H](F)c2nc(nn12)C(=O)C1CC1 |r|
CCC[C@@H]1C[C@H](F)c2nc(nn12)C(=O)C1CC1 |r|
F[C@H]1C[C@@H](c2c(F)cccc2F)n2nc(nc12)C(=O)C1CC1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)C1(CC1)C#N |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)C1CC11CC1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)C1CC11CCC1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)C1(CC1)c1ccccn1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)C1(CC1)C1CC1 |r|
F[C@H]1C[C@@H](c2ccccc2Cl)n2nc(nc12)C(=O)C1CC1 |r|
F[C@H]1C[C@@H](c2cc(F)ccc2F)n2nc(nc12)C(=O)C1CC1 |r|
F[C@H]1C[C@@H](c2c(F)ccc(F)c2F)n2nc(nc12)C(=O)C1CC1 |r|
F[C@@H]1C[C@H]1C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3F)n2n1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)[C@@H]1C[C@H]1C#N |r|
F[C@H]1C[C@@H](c2cccc(F)c2F)n2nc(nc12)C(=O)C1CC1 |r|
F[C@H]1C[C@@H](c2cc(F)cc(F)c2F)n2nc(nc12)C(=O)C1CC1 |r|
CC(C)[C@@H]1C[C@H](F)c2nc(nn12)C(=O)C1CC1 |r|
F[C@H]1C[C@@H](C2CC2)n2nc(nc12)C(=O)C1CC1 |r|
O=C(C1CC1)c1nc2CC[C@@H](c3ccccc3)n2n1 |r|
CCC(F)(F)[C@@H]1C[C@H](F)c2nc(nn12)C(=O)C1CC1 |r|
F[C@H]1C[C@@H](CC2CC2)n2nc(nc12)C(=O)C1CC1 |r|
Cl[C@@H]1C[C@H](c2ccccc2)n2nc(nc12)C(=O)C1CC1 |r|
Cl[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)C1CC1 |r|
Cl[C@@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)C1CC1 |r|
F[C@H]1C[C@@H](c2ncccc2Cl)n2nc(nc12)C(=O)C1CC1 |r|
CC(F)(F)[C@@H]1C[C@H](F)c2nc(nn12)C(=O)C1CC1 |r|
F[C@H]1C[C@@H](c2ccccc2C#N)n2nc(nc12)C(=O)C1CC1 |r|
CCC1(CC1)C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)C1CCOCC1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)C1CCCOC1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)[C@H]1CCCN1 |r|
CC1(CCCO1)C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)C1CCOC1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)[C@H]1CCOC1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)[C@@H]1CCOC1 |r|
COCC(C)(C)C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
O[C@@H](C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1)C(F)(F)F |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)CC1CCCCO1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)CC1CCOCC1 |r|
C[C@]1(CCOC1)C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
C[C@@]1(CCOC1)C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)[C@@H]1C[C@@H]2CC[C@H]1O2 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)[C@@H]1C[C@H]2CC[C@@H]1O2 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)[C@H]1C[C@@H]2CC[C@H]1O2 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)COC(F)(F)F |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)[C@]12C[C@H]1COC2 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)[C@@]12C[C@@H]1COC2 |r|
O=C(C1CC1)c1nc2CCCC(c3ccccc3)n2n1
O=C(C1CC1)c1nc2CCC[C@@H](c3ccccc3)n2n1 |r|
Cc1ccccc1[C@@H]1C[C@@H](O)c2nc(nn12)C(=O)C1CC1 |r|
Cc1ccccc1[C@@H]1C[C@@H](F)c2nc(nn12)C(=O)C1CC1 |r|
Cc1ccccc1[C@@H]1C[C@H](F)c2nc(nn12)C(=O)C1CC1 |r|
F[C@H]1C[C@@H](c2ncccc2F)n2nc(nc12)C(=O)C1CC1 |r|
F[C@@H]1C[C@@H](c2ncccc2F)n2nc(nc12)C(=O)C1CC1 |r|
Cn1cc(cn1)[C@@H]1C[C@H](F)c2nc(nn12)C(=O)C1CC1 |r|
Cc1oncc1C1CC(F)c2nc(nn12)C(=O)C1CC1
Cn1cc(Cl)c(n1)[C@@H]1C[C@H](F)c2nc(nn12)C(=O)C1CC1 |r|
Cn1cc(Cl)c(n1)[C@@H]1C[C@@H](F)c2nc(nn12)C(=O)C1CC1 |r|
COc1cccc(c1)[C@@H]1C[C@H](F)c2nc(nn12)C(=O)C1CC1 |r|
F[C@H]1C[C@@H](c2cc(F)cc(c2)C(F)(F)F)n2nc(nc12)C(=O)C1CC1 |r|
O=C(c1nc2CCC(c3ccccc3)n2n1)C1(Cn2cccn2)CC1
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)[C@H]1C[C@@H]1C(F)(F)F |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)[C@@H]1C[C@H]1C(F)(F)F |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)[C@H]1CC11CC1 |r|
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)[C@@H]1CC11CC1 |r|
CC1(C)CCCN2CCC(N2C1=O)c1cncc(F)c1
Cc1cnc(cn1)C1CCN2CCCC(C)(C)C(=O)N12
CC1(C)CCCN2CCC(N2C1=O)c1cc(F)cc(F)c1
CC1(C)CCCN2CCC(N2C1=O)c1ccc(F)c(F)c1
CC1(C)CCCN2CCC(N2C1=O)c1cccc(F)c1
CC1(C)CCCN2CCC(N2C1=O)c1cc(F)cc(c1)C#N
CC1(C)CCCN2CCC(N2C1=O)c1ccc(cc1)C#N
CCC1(C)COC[C@H]2CC[C@H](N2C1=O)c1cccc(F)c1 |r|
CC1(C)CCCN2CCC(N2C1=O)c1cncc(c1)C#N
C[C@@]1(CCCN2CCC(N2C1=O)c1cncc(F)c1)C(F)F |r|
C[C@]1(CCCN2CCC(N2C1=O)c1cncc(F)c1)C(F)F |r|
Cc1cnc(cn1)C1CCN2CCC[C@](C)(C(F)F)C(=O)N12 |r|
Cc1cnc(cn1)C1CCN2CCC[C@@](C)(C(F)F)C(=O)N12 |r|
C[C@@]1(CCCN2CCC(N2C1=O)c1cncc(c1)C#N)C(F)F |r|
C[C@]1(CCCN2CCC(N2C1=O)c1cncc(c1)C#N)C(F)F |r|
Fc1cncc(c1)C1CCN2CCCC3(CC3)C(=O)N12
CC[C@@]1(CCCN2CCC(N2C1=O)c1cnc(C)cn1)C(F)F |r|
CC[C@]1(CCCN2CCC(N2C1=O)c1cnc(C)cn1)C(F)F |r|
Cc1cc(F)c(cc1C(=O)NCC[C@H](O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1cc(F)c(cc1C(=O)NCCC(O)c1ccc(cc1)C(F)(F)F)-c1ccn2nc(N)nc2c1
Cc1cc(F)c(cc1C(=O)NCC[C@@H](O)c1ccc(cc1)C(F)(F)F)-c1ccn2nc(N)nc2c1 |r|
Cc1cc(F)c(cc1C(=O)NCC[C@H](O)c1ccc(cc1)C(F)(F)F)-c1ccn2nc(N)nc2c1 |r|
Cc1cc(F)c(cc1C(=O)NCCC(O)c1ccc(Cl)cn1)-c1ccn2nc(N)nc2c1
Cc1cc(F)c(cc1C(=O)NCC[C@@H](O)c1ccc(Cl)cn1)-c1ccn2nc(N)nc2c1 |r|
Cc1cc(F)c(cc1C(=O)NCC[C@H](O)c1ccc(Cl)cn1)-c1ccn2nc(N)nc2c1 |r|
Cc1cc(F)c(cc1C(=O)NCCC(O)c1ccc(F)cc1)-c1ccn2nc(N)nc2c1
Cc1cc(F)c(cc1C(=O)NCC[C@@H](O)c1ccc(F)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1cc(F)c(cc1C(=O)NCC[C@H](O)c1ccc(F)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCCC(c1ccccc1)C(F)(F)F
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCC[C@H](c1ccccc1)C(F)(F)F |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCC[C@@H](c1ccccc1)C(F)(F)F |r|
Cc1ccc(c(F)c1C(=O)NCCC(O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1
Cc1ccc(c(F)c1C(=O)NCCC(C)(C)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1
Cc1ccc(c(F)c1C(=O)NCCC1(CC1)c1ccc(F)cc1)-c1ccn2nc(N)nc2c1
Cc1ccc(c(F)c1C(=O)NCCC(C)(O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1
C[C@H](C[C@H](O)c1ccc(Cl)cc1)NC(=O)c1c(C)ccc(c1F)-c1ccn2nc(N)nc2c1 |r|
C[C@@H](C[C@@H](O)c1ccc(Cl)cc1)NC(=O)c1c(C)ccc(c1F)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(c(F)c1C(=O)N[C@H](CF)C[C@H](O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(c(F)c1C(=O)N[C@H](CF)C[C@@H](O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(c(F)c1C(=O)N[C@@H](CF)C[C@H](O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(c(F)c1C(=O)N[C@@H](CF)C[C@@H](O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)N[C@H](CF)C[C@H](O)c1ccc(F)cc1 |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)N[C@H](CF)C[C@@H](O)c1ccc(F)cc1 |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)N[C@@H](CF)C[C@H](O)c1ccc(F)cc1 |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)N[C@@H](CF)C[C@@H](O)c1ccc(F)cc1 |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCC(F)(F)C(O)c1ccc(F)cc1
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCC(F)(F)[C@@H](O)c1ccc(F)cc1 |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCC(F)(F)[C@H](O)c1ccc(F)cc1 |r|
Cc1ccc(c(F)c1C(=O)NCC[C@@H](O)c1ccc(Cl)c(Cl)c1)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(c(F)c1C(=O)NCC[C@H](O)c1ccc(Cl)c(Cl)c1)-c1ccn2nc(N)nc2c1 |r|
CC(CC(O)c1ccc(F)cc1)NC(=O)c1c(C)ccc(-c2ccn3nc(N)nc3c2)c1F
C[C@H](C[C@H](O)c1ccc(F)cc1)NC(=O)c1c(C)ccc(-c2ccn3nc(N)nc3c2)c1F |r|
C[C@H](C[C@@H](O)c1ccc(F)cc1)NC(=O)c1c(C)ccc(-c2ccn3nc(N)nc3c2)c1F |r|
C[C@@H](C[C@H](O)c1ccc(F)cc1)NC(=O)c1c(C)ccc(-c2ccn3nc(N)nc3c2)c1F |r|
C[C@@H](C[C@@H](O)c1ccc(F)cc1)NC(=O)c1c(C)ccc(-c2ccn3nc(N)nc3c2)c1F |r|
Cc1ccc(c(F)c1C(=O)NCCC(O)C1CCCCC1)-c1ccn2nc(N)nc2c1
Cc1ccc(c(F)c1C(=O)NCC[C@@H](O)C1CCCCC1)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(c(F)c1C(=O)NCC[C@H](O)C1CCCCC1)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(c(F)c1C(=O)NCCC(O)c1cccc(Cl)c1)-c1ccn2nc(N)nc2c1
Cc1ccc(c(F)c1C(=O)NCC[C@@H](O)c1cccc(Cl)c1)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(c(F)c1C(=O)NCC[C@H](O)c1cccc(Cl)c1)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(c(F)c1C(=O)NCCC(O)c1ccc(Cl)cn1)-c1ccn2nc(N)nc2c1
Cc1ccc(c(F)c1C(=O)NCC[C@@H](O)c1ccc(Cl)cn1)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(c(F)c1C(=O)NCC[C@H](O)c1ccc(Cl)cn1)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCCC(O)c1ccc(F)cc1
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCC[C@@H](O)c1ccc(F)cc1 |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCC[C@H](O)c1ccc(F)cc1 |r|
Cc1ccc(c(F)c1C(=O)NCCCC1CCCCC1)-c1ccn2nc(N)nc2c1
Cc1ccc(c(F)c1C(=O)NCC[C@@H](O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(c(F)c1C(=O)NCC[C@H](O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCCC(O)c1ccc(cc1)C(F)(F)F
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCC[C@@H](O)c1ccc(cc1)C(F)(F)F |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCC[C@H](O)c1ccc(cc1)C(F)(F)F |r|
Cc1ccc(c(F)c1C(=O)NCCC(C)(C)c1ccccc1)-c1ccn2nc(N)nc2c1
Cc1ccc(c(F)c1C(=O)NCC[C@](C)(O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(c(F)c1C(=O)NCC[C@@](C)(O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCC(F)(F)[C@](C)(O)c1ccc(F)cc1 |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCC(F)(F)[C@@](C)(O)c1ccc(F)cc1 |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCC[C@@H](O)c1cccc(F)c1 |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCC[C@H](O)c1cccc(F)c1 |r|
COc1cc(Cl)ccc1[C@H](O)CCNC(=O)c1c(C)ccc(c1F)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCC[C@@H](O)c1ccc(F)c(F)c1 |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCC[C@H](O)c1ccc(F)c(F)c1 |r|
Cc1ccc(c(F)c1C(=O)NCC[C@@H](O)c1ccc(Cl)cc1F)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(c(F)c1C(=O)NCC[C@H](O)c1ccc(Cl)cc1F)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCC[C@H](O)c1ccccc1F |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCC[C@@H](O)c1ccccc1F |r|
COc1c(F)cccc1[C@H](O)CCNC(=O)c1c(C)ccc(c1F)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCC[C@@H](O)c1c(F)cccc1F |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCC[C@H](O)c1c(F)cccc1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCCC(O)c2ccc(Cl)cc2)c1F
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC[C@@H](O)c2ccc(Cl)cc2)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC[C@H](O)c2ccc(Cl)cc2)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCCC(O)c2ccc(F)cc2)c1F
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC[C@@H](O)c2ccc(F)cc2)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC[C@H](O)c2ccc(F)cc2)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCCC(O)c2ccc(Cl)cn2)c1F
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC[C@@H](O)c2ccc(Cl)cn2)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC[C@H](O)c2ccc(Cl)cn2)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCCC2(CC2)c2ccc(F)cc2)c1F
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC[C@@H](O)c2ccc(cc2)C(F)(F)F)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC[C@H](O)c2ccc(cc2)C(F)(F)F)c1F |r|
C[C@](O)(c1ccc(F)cc1)C(F)(F)CNC(=O)c1c(Cl)ccc(c1F)-c1ccn2nc(N)nc2c1 |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(c1)C(=O)NCC[C@@H](O)c1ccc(Cl)cc1 |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(c1)C(=O)NCC[C@H](O)c1ccc(Cl)cc1 |r|
CC(CCNC(=O)c1cc(ccc1Cl)-c1ccn2nc(N)nc2c1)c1ccccc1
CC(O)(CCNC(=O)c1cc(ccc1Cl)-c1ccn2nc(N)nc2c1)c1ccccc1
Cc1c(F)cc(cc1C(=O)NCC[C@@H](O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1c(F)cc(cc1C(=O)NCCC(O)c1ccccc1)-c1ccn2nc(N)nc2c1
Cc1c(F)cc(cc1C(=O)NCCC(C)(O)c1ccccc1)-c1ccn2nc(N)nc2c1
Cc1cc(F)c(cc1C(=O)NCC(F)(F)[C@@H](O)c1ccc(F)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1cc(F)c(cc1C(=O)NCC(F)(F)[C@H](O)c1ccc(F)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1c(F)c(F)c(cc1C(=O)NCC[C@H](O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
C[C@@H](C[C@@H](O)c1ccc(Cl)cc1)NC(=O)c1cc(c(F)c(F)c1C)-c1ccn2nc(N)nc2c1 |r|
C[C@H](C[C@H](O)c1ccc(Cl)cc1)NC(=O)c1cc(c(F)c(F)c1C)-c1ccn2nc(N)nc2c1 |r|
CC[C@H](C[C@H](O)c1ccc(Cl)cc1)NC(=O)c1cc(c(F)c(F)c1C)-c1ccn2nc(N)nc2c1 |r|
CC[C@@H](C[C@@H](O)c1ccc(Cl)cc1)NC(=O)c1cc(c(F)c(F)c1C)-c1ccn2nc(N)nc2c1 |r|
Cc1c(F)c(F)c(cc1C(=O)NCC(F)(F)[C@@H](O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1c(F)c(F)c(cc1C(=O)NCC(F)(F)[C@H](O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1c(F)c(F)c(cc1C(=O)NCC(F)(F)[C@@H](O)c1ccc(F)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1c(F)c(F)c(cc1C(=O)NCC(F)(F)[C@H](O)c1ccc(F)cc1)-c1ccn2nc(N)nc2c1 |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@@H](O)c2ccc(F)cc2)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@H](O)c2ccc(F)cc2)c1F |r|
Cc1ccc(c(F)c1C(=O)NCC(F)(F)[C@@H](O)c1ccc(Cl)c(Cl)c1)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(c(F)c1C(=O)NCC(F)(F)[C@H](O)c1ccc(Cl)c(Cl)c1)-c1ccn2nc(N)nc2c1 |r|
COc1ccc(c(F)c1C(=O)NCC(F)(F)C(O)c1ccc(Cl)c(Cl)n1)-c1ccn2nc(N)nc2c1
Cc1ccc(c(F)c1C(=O)NCC(F)(F)C(O)c1ccc(Cl)c(Cl)n1)-c1ccn2nc(N)nc2c1
CCc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCC(F)(F)C(O)c1ccc(F)cc1
COc1ccc(c(F)c1C(=O)NCC(F)(F)[C@@H](O)c1ccc(F)cc1)-c1ccn2nc(N)nc2c1 |r|
COc1ccc(c(F)c1C(=O)NCC(F)(F)[C@H](O)c1ccc(F)cc1)-c1ccn2nc(N)nc2c1 |r|
Nc1nc2cc(ccn2n1)-c1cc(C(=O)NCC(F)(F)[C@H](O)c2ccc(F)cc2)c(Cl)cc1Cl |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NC[C@@H](F)[C@H](O)c2ccc(Cl)cc2)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NC[C@H](F)[C@@H](O)c2ccc(Cl)cc2)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NC[C@H](F)[C@@H](O)c2ccc(F)cc2)c1F |r|
Cc1ccc(c(F)c1C(=O)NCC[C@H](O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1C |r|
COc1c(ccn2nc(N)nc12)-c1ccc(C)c(C(=O)NCC(F)(F)[C@@H](O)c2ccc(F)cc2)c1F |r|
COc1c(ccn2nc(N)nc12)-c1ccc(C)c(C(=O)NCC(F)(F)[C@H](O)c2ccc(F)cc2)c1F |r|
Cc1ccc(c(F)c1C(=O)NCC(F)(F)[C@@H](O)c1ccc(F)cc1)-c1ccn2nc(N)nc2c1F |r|
Cc1ccc(c(F)c1C(=O)NCC(F)(F)[C@H](O)c1ccc(F)cc1)-c1ccn2nc(N)nc2c1F |r|
Cc1ccc(c(F)c1C(=O)NCC[C@H](O)c1ccc(cc1)C#N)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(c(F)c1C(=O)NCCC(O)c1cccc(c1)C#N)-c1ccn2nc(N)nc2c1
Cc1ccc(c(F)c1C(=O)NCCC(C)(O)c1ccc(cc1)C#N)-c1ccn2nc(N)nc2c1
Cc1ccc(c(F)c1C(=O)NCC[C@H](O)c1ccc(cc1)C#C)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(c(F)c1C(=O)NCCC(=O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1
Cc1cc(Cl)c(cc1C(=O)NCC[C@H](O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(Cl)c1C(=O)NCC[C@H](O)c1ccc(Cl)cc1 |r|
Cc1cc(C)c(cc1C(=O)NCC[C@H](O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
COc1ccc(c(F)c1C(=O)NCC[C@H](O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
COc1ccc(c(F)c1C(=O)NCC[C@@H](O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(cc1C(=O)NCC[C@H](O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
CCc1ccc(cc1C(=O)NCC[C@H](O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
CCc1ccc(c(F)c1C(=O)NCC[C@H](O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
CCc1ccc(c(F)c1C(=O)NCC[C@@H](O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
CCc1cc(F)c(cc1C(=O)NCC[C@H](O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1c(F)cc(cc1C(=O)NCC[C@H](O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(cc1C(=O)NCC[C@@H](O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(c(F)c1C(=O)NCCC(F)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1
Cc1ccc(c(F)c1C(=O)NCC(F)(F)C(OP(O)(O)=O)c1ccc(F)cc1)-c1ccn2nc(N)nc2c1
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@@H](O)c2ccc(Cl)cc2F)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@H](O)c2ccc(Cl)cc2F)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@@H](O)c2ccc(cc2F)C(F)(F)F)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@H](O)c2ccc(cc2F)C(F)(F)F)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@@H](O)c2cccc(F)c2F)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@H](O)c2cccc(F)c2F)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@@H](O)c2cccc(F)c2)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@H](O)c2cccc(F)c2)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@@H](O)c2cccc(Cl)c2F)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@H](O)c2cccc(Cl)c2F)c1F |r|
Cc1ccc(cc1)[C@@H](O)C(F)(F)CNC(=O)c1c(Cl)ccc(c1F)-c1ccn2nc(N)nc2c1 |r|
Cc1cccc(c1)[C@H](O)C(F)(F)CNC(=O)c1c(Cl)ccc(c1F)-c1ccn2nc(N)nc2c1 |r|
Cc1cccc(c1)[C@@H](O)C(F)(F)CNC(=O)c1c(Cl)ccc(c1F)-c1ccn2nc(N)nc2c1 |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@@H](O)c2cc(F)ccc2F)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@H](O)c2cc(F)ccc2F)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@@H](O)c2ccc(F)cc2F)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@H](O)c2ccc(F)cc2F)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@@H](O)c2cc(Cl)ccc2F)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@H](O)c2cc(Cl)ccc2F)c1F |r|
Cc1ccc([C@H](O)C(F)(F)CNC(=O)c2c(Cl)ccc(c2F)-c2ccn3nc(N)nc3c2)c(F)c1 |r|
Cc1ccc([C@@H](O)C(F)(F)CNC(=O)c2c(Cl)ccc(c2F)-c2ccn3nc(N)nc3c2)c(F)c1 |r|
COc1ccc(cc1)[C@H](O)C(F)(F)CNC(=O)c1c(Cl)ccc(c1F)-c1ccn2nc(N)nc2c1 |r|
COc1ccc(cc1)[C@@H](O)C(F)(F)CNC(=O)c1c(Cl)ccc(c1F)-c1ccn2nc(N)nc2c1 |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@@H](O)c2ccc(OC(F)F)cc2)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@H](O)c2ccc(OC(F)F)cc2)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@@H](O)c2cc(F)cc(F)c2)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@H](O)c2cc(F)cc(F)c2)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@@H](O)c2ccc(Cl)c(F)c2)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@H](O)c2ccc(Cl)c(F)c2)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@@H](O)c2cccc(Cl)c2)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@H](O)c2cccc(Cl)c2)c1F |r|
C[C@@](O)([C@@H](F)CNC(=O)c1c(F)c(ccc1C(F)F)-c1ccn2nc(N)nc2c1)c1ccc(F)cc1 |r|
C[C@](O)([C@@H](F)CNC(=O)c1c(F)c(ccc1C(F)F)-c1ccn2nc(N)nc2c1)c1ccc(F)cc1 |r|
C[C@@](O)([C@H](F)CNC(=O)c1c(F)c(ccc1C(F)F)-c1ccn2nc(N)nc2c1)c1ccc(F)cc1 |r|
C[C@](O)([C@H](F)CNC(=O)c1c(F)c(ccc1C(F)F)-c1ccn2nc(N)nc2c1)c1ccc(F)cc1 |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCC(F)(F)[C@@H](O)c1ccc(F)c(F)c1 |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCC(F)(F)[C@H](O)c1ccc(F)c(F)c1 |r|
Cc1ccc(cc1)[C@H](O)C(F)(F)CNC(=O)c1c(C)ccc(-c2ccn3nc(N)nc3c2)c1F |r|
Cc1ccc(cc1)[C@@H](O)C(F)(F)CNC(=O)c1c(C)ccc(-c2ccn3nc(N)nc3c2)c1F |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NC[C@](C)(F)[C@@H](O)c1ccc(F)cc1 |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NC[C@@](C)(F)[C@@H](O)c1ccc(F)cc1 |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NC[C@](C)(F)[C@H](O)c1ccc(F)cc1 |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NC[C@@](C)(F)[C@H](O)c1ccc(F)cc1 |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)Cc2ccc(F)cc2)c1F
Cc1ccc(c(F)c1C(=O)NCC(F)(F)Cc1ccc(F)cc1)-c1ccn2nc(N)nc2c1
C[C@@](O)([C@@H](F)CNC(=O)c1c(Cl)ccc(c1F)-c1ccn2nc(N)nc2c1)c1ccc(F)cc1 |r|
C[C@](O)([C@H](F)CNC(=O)c1c(Cl)ccc(c1F)-c1ccn2nc(N)nc2c1)c1ccc(F)cc1 |r|
C[C@](O)([C@@H](F)CNC(=O)c1c(Cl)ccc(c1F)-c1ccn2nc(N)nc2c1)c1ccc(F)cc1 |r|
C[C@@](O)([C@H](F)CNC(=O)c1c(Cl)ccc(c1F)-c1ccn2nc(N)nc2c1)c1ccc(F)cc1 |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NC[C@H](F)[C@@](C)(O)c1ccc(F)cc1 |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NC[C@@H](F)[C@](C)(O)c1ccc(F)cc1 |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NC[C@H](F)[C@](C)(O)c1ccc(F)cc1 |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NC[C@@H](F)[C@@](C)(O)c1ccc(F)cc1 |r|
Nc1nc2cc(ccn2n1)-c1cccc(C(=O)NCC[C@H](O)c2ccc(Cl)cc2)c1F |r|
Nc1nc2cc(ccn2n1)-c1cccc(C(=O)NCC[C@@H](O)c2ccc(Cl)cc2)c1F |r|
Nc1nc2cc(ccn2n1)-c1c(F)ccc(C(=O)NCC[C@H](O)c2ccc(Cl)cc2)c1F |r|
Nc1nc2cc(ccn2n1)-c1c(F)ccc(C(=O)NCC[C@@H](O)c2ccc(Cl)cc2)c1F |r|
Cc1ccc(c(F)c1C(=O)NCC(F)(F)[C@](C)(O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(c(F)c1C(=O)NCC(F)(F)[C@@](C)(O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
C[C@@](O)(c1ccc(Cl)cc1)C(F)(F)CNC(=O)c1c(Cl)ccc(c1F)-c1ccn2nc(N)nc2c1 |r|
C[C@](O)(c1ccc(Cl)cc1)C(F)(F)CNC(=O)c1c(Cl)ccc(c1F)-c1ccn2nc(N)nc2c1 |r|
Cc1cc(F)c(cc1C(=O)NCC(F)(F)[C@](C)(O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1cc(F)c(cc1C(=O)NCC(F)(F)[C@@](C)(O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCC(F)(F)C(C)(O)c1ccc(cc1)C(F)(F)F
Cc1ccc(c(F)c1C(=O)NCCC(C)(F)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1
Cc1c(F)cc(cc1C(=O)NCC(F)(F)[C@@H](O)c1ccc(F)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1c(F)cc(cc1C(=O)NCC(F)(F)[C@H](O)c1ccc(F)cc1)-c1ccn2nc(N)nc2c1 |r|
CO[C@@H](c1ccc(F)cc1)C(F)(F)CNC(=O)c1c(C)ccc(c1F)-c1ccn2nc(N)nc2c1 |r|
CO[C@H](c1ccc(F)cc1)C(F)(F)CNC(=O)c1c(C)ccc(c1F)-c1ccn2nc(N)nc2c1 |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)C2(COC2)c2ccc(F)cc2)c1F
Cc1ccc(c(F)c1C(=O)NCC(F)(F)C1(COC1)c1ccc(F)cc1)-c1ccn2nc(N)nc2c1
Cc1ccc(c(F)c1C(=O)NCC[C@@H](O)C1CCCC1)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(c(F)c1C(=O)NCC[C@H](O)C1CCCC1)-c1ccn2nc(N)nc2c1 |r|
Nc1nc2cc(ccn2n1)-c1ccc(F)c(C(=O)NCCC2(CC2)c2ccc(F)cc2)c1F
Nc1nc2cc(ccn2n1)-c1ccc(F)c(C(=O)NCC[C@@H](O)c2ccc(Cl)cc2)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@@H](O)c2cccc(n2)C(F)(F)F)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@H](O)c2cccc(n2)C(F)(F)F)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@H](O)C2CCC(F)(F)CC2)c1F |r|
Cc1ccc(c(F)c1C(=O)NCC(F)(F)[C@@H](O)C1CC(F)(F)C1)-c1ccn2nc(N)nc2c1
Cc1ccc(c(F)c1C(=O)NCC(F)(F)[C@H](O)C1CC(F)(F)C1)-c1ccn2nc(N)nc2c1
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCC(F)(F)[C@@H](O)c1ccnc(c1)C(F)(F)F |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCC(F)(F)[C@H](O)c1ccnc(c1)C(F)(F)F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@@H](O)c2cccc(Cl)n2)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@H](O)c2cccc(Cl)n2)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@@H](O)c2ccc(Cl)c(Cl)c2)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@H](O)c2ccc(Cl)c(Cl)c2)c1F |r|
CCc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCC(F)(F)[C@@H](O)c1ccc(F)cn1 |r|
COc1ccc(c(F)c1C(=O)NCC(F)(F)[C@@H](O)c1ccc(Cl)c(Cl)c1)-c1ccn2nc(N)nc2c1 |r|
COc1ccc(c(F)c1C(=O)NCC(F)(F)[C@H](O)c1ccc(Cl)c(Cl)c1)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCC(F)(F)[C@@H](O)c1ccc(F)cn1 |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCC(F)(F)[C@H](O)c1ccc(F)cn1 |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@@H](O)c2ccc(Cl)c(Cl)n2)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@H](O)c2ccc(Cl)c(Cl)n2)c1F |r|
COC(=O)c1ccc(CCCNC(=O)c2c(Cl)ccc(c2F)-c2ccn3nc(N)nc3c2)cc1
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCC(F)(F)C(O)(C(F)F)c1ccc(F)cc1
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCC(F)(F)C(N)c1ccc(F)cc1
Cc1ccc(c(F)c1C(=O)NCC(F)(F)[C@@H](OC(N)=O)c1ccc(F)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1cc(F)c(c(F)c1C(=O)NCC[C@H](O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1cc(F)c(c(F)c1C(=O)NCC[C@@H](O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCC(C)(O)C(=O)c1ccc(F)cc1
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)C(=O)c2ccc(F)cc2)c1F
Cc1ccc(c(F)c1C(=O)NCC(F)(F)C(=O)c1ccc(F)cc1)-c1ccn2nc(N)nc2c1
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCC(F)(F)[C@@H](F)c1ccc(F)cc1 |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCC(F)(F)[C@@H](O)c1c(F)cc(F)cc1F |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NCC(F)(F)[C@H](O)c1c(F)cc(F)cc1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(F)c(C(=O)NCC(F)(F)[C@@H](F)c2ccc(F)cc2)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(c(C(=O)NCC(F)(F)[C@@H](F)c2ccc(F)cc2)c1F)C(F)(F)F |r|
Nc1nc2cc(ccn2n1)-c1ccc(F)c(C(=O)NCC(F)(F)[C@H](F)c2ccc(F)cc2)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(c(C(=O)NCC(F)(F)[C@H](F)c2ccc(F)cc2)c1F)C(F)(F)F |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NC[C@@H](O)C(F)(F)c1ccc(F)cc1 |r|
Cc1ccc(-c2ccn3nc(N)nc3c2)c(F)c1C(=O)NC[C@H](O)C(F)(F)c1ccc(F)cc1 |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NC[C@H](O)C(F)(F)c2ccc(F)cc2)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NC[C@@H](O)C(F)(F)c2ccc(F)cc2)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(CF)c(C(=O)NCC(F)(F)[C@@H](O)c2ccc(F)cc2)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(C(F)F)c(C(=O)NCC(F)(F)[C@@H](O)c2ccc(F)cc2)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NC[C@@H](F)[C@H](O)c2ccc(F)cc2)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NC[C@@H](F)[C@@H](O)c2ccc(F)cc2)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NC[C@H](F)[C@H](O)c2ccc(F)cc2)c1F |r|
Cc1ccc(c(F)c1C(=O)NC[C@@H](F)[C@@H](O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(c(F)c1C(=O)NC[C@H](F)[C@H](O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(c(F)c1C(=O)NC[C@@H](F)[C@H](O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
Nc1nc2cc(ccn2n1)-c1ccc(C2CC2)c(C(=O)NCC(F)(F)[C@@H](O)c2ccc(F)cc2)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(C2CC2)c(C(=O)NCC(F)(F)[C@H](O)c2ccc(F)cc2)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(OC(F)F)c(C(=O)NCC(F)(F)[C@H](O)c2ccc(F)cc2)c1F |r|
Cc1ccc(c(F)c1C(=O)NCC1(CC1)[C@@H](O)c1ccc(F)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1ccc(c(F)c1C(=O)NCC1(CC1)[C@H](O)c1ccc(F)cc1)-c1ccn2nc(N)nc2c1 |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@@H](O)c2ccc(cc2)C(F)F)c1F |r|
Nc1nc2cc(ccn2n1)-c1ccc(Cl)c(C(=O)NCC(F)(F)[C@H](O)c2ccc(cc2)C(F)F)c1F |r|
CC[C@@](O)(c1ccc(F)cc1)C(F)(F)CNC(=O)c1c(Cl)ccc(c1F)-c1ccn2nc(N)nc2c1 |r|
CC[C@](O)(c1ccc(F)cc1)C(F)(F)CNC(=O)c1c(Cl)ccc(c1F)-c1ccn2nc(N)nc2c1 |r|
Nc1nc2cc(ccn2n1)-c1ccc(c(C(=O)NCC(F)(F)[C@@H](O)c2ccc(F)cc2)c1F)C(F)(F)F |r|
CC(CCNC(=O)c1cccc(c1)-c1ccn2nc(N)nc2c1)c1ccccc1
COc1ncc(cc1C(=O)NCCC(O)c1ccc(Cl)cn1)-c1ccn2nc(N)nc2c1
COc1ncc(cc1C(=O)NCCC(O)c1ccc(F)c(F)c1)-c1ccn2nc(N)nc2c1
CC(CCNC(=O)c1cc(cnc1C)-c1ccn2nc(N)nc2c1)c1ccccc1
Cc1nc(C)c(cc1C(=O)NCC[C@H](O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
COc1ncc(cc1C(=O)NCC[C@H](O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
COc1nc(C)c(cc1C(=O)NCC[C@H](O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1ncc(cc1C(=O)NCC[C@H](O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1ncc(cc1C(=O)NCC[C@@H](O)c1ccc(Cl)cc1)-c1ccn2nc(N)nc2c1 |r|
Cc1ncc(cc1C(=O)NCC(C)(O)Cc1ccc(F)cc1)-c1ccn2nc(N)nc2c1
Cc1ncc(cc1C(=O)NCC(O)Cc1ccccc1)-c1ccn2nc(N)nc2c1
CC(CCNC(=O)c1cncc(c1)-c1ccn2nc(N)nc2c1)c1ccccc1
CCOC(=O)CCc1ccc2OC[C@H](NC(=O)c3n[nH]c(Cc4ccccc4)n3)C(=O)N(C)c2c1
CN1c2cc(CCC(=O)Nc3ccc4cn[nH]c4c3)ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
COc1cc2ncnc(NC(=O)CCc3ccc4OC[C@H](NC(=O)c5n[nH]c(Cc6ccccc6)n5)C(=O)N(C)c4c3)c2cc1OC
CN1c2cc(CCC(=O)Nc3ccc4cn[nH]c4c3)ccc2OC[C@H](NC(=O)c2ncn(Cc3ccccc3F)n2)C1=O
CN1c2cc(CCC(O)=O)ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2cc(CCC(=O)N3CCCC3)ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2cc(CCC(=O)N3CCOCC3)ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2cc(CCC(=O)Nc3ccc4cccnc4c3)ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2cc(CCC(=O)NC3CC3)ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2cc(CCCO)ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2cc(CCCCO)ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2cc(CCCCOCc3ccccn3)ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2cc(CCCCNc3ccccn3)ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2cc(CN3CCN(CC3)c3ccncc3)ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2cc(CN3CCN(CC3)c3ccncc3)ccc2OC[C@H](NC(=O)c2ncn(Cc3c(Cl)cccc3Cl)n2)C1=O
CN1c2cc(\C=C\C(=O)N3CCCC3)ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2cc(\C=C\C(=O)NC3CC3)ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2cc(CN3CCn4ncnc4C3)ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2cc(CCC(=O)NC3CC3)ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccc(F)cc3F)n2)C1=O
CN1c2cc(CCC(C)(C)O)ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2cc(CCC(N)=O)ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2cc(CCC(=O)N3CCCC3)ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccc(F)cc3F)n2)C1=O
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CCCCO
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[n-]c(Cc3ccccc3)n2)C1=O)C#CC(C)(C)O
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CCCOc1ccc2ncccc2c1
CN1c2cc(CN3CCn4nc(nc4C3)C(F)(F)F)ccc2OC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O
CN1c2cc(CN3CCn4nc(nc4C3)C(F)(F)F)ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CCCOc1ccc2cccnc2c1
CN1c2cc(ccc2OC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O)C#CCCOc1ccc2cccnc2c1
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccc(F)cc3F)n2)C1=O)C#CC(C)(C)O
CN1c2cc(ccc2OC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O)C#CCCOc1cccc2ncccc12
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CCCOc1cccc2ncccc12
CN1c2cc(CN3CCn4c(C3)nnc4C(F)(F)F)ccc2OC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O
CN1c2cc(CN3CCn4c(C3)nnc4C(F)(F)F)ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2cc(ccc2OC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O)C#CC(C)(C)C
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CC(C)(C)C
CN1c2cc(ccc2OC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O)C#CC1(O)CCC1
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CC1(O)CCC1
CN1c2cc(ccc2OC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O)C#CC1(O)CCCC1
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CC1(O)CCCC1
CN1c2cc(ccc2OC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O)C#CC1(O)CCOCC1
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CC1(O)CCOCC1
CN1c2cc(ccc2OC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O)C#CC1(O)COC1
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CC(C)=C
CC(C)CCc1ccc2OC[C@H](NC(=O)c3n[nH]c(Cc4ccccc4)n3)C(=O)N(C)c2c1
COC(C)(C)C#Cc1ccc2OC[C@H](NC(=O)c3n[nH]c(Cc4ccccc4)n3)C(=O)N(C)c2c1
CN1c2ccc(cc2OC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O)C#CC(C)(C)O
CN1c2ccc(cc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CC(C)(C)O
CN1c2ccc(cc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC(C)(C)O
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3c(Cl)cccc3Cl)n2)C1=O)C#CC(C)(C)O
CN1c2ccc(CN3CCn4nc(nc4C3)C(F)(F)F)cc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2ccc(CN3CCn4nc(nc4C3)C(F)(F)F)cc2OC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O
CN1c2ccc(cc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CC1(O)COC1
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#C[C@@]1(O)CO[C@@H]2[C@H](CO[C@H]12)OC(=O)c1ccccc1
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#C[C@@]1(O)CO[C@@H]2[C@@H](O)CO[C@H]12
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3cccc(F)c3)n2)C1=O)C#CC(C)(C)O
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccc(F)cc3)n2)C1=O)C#CC(C)(C)O
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3F)n2)C1=O)C#CC(C)(C)O
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#C
CN1c2cc(ccc2OC[C@H](NC(=O)c2ncn(Cc3ccccc3C)n2)C1=O)C#CC(C)(C)O
CN1c2cc(ccc2OC[C@H](NC(=O)c2ncn(Cc3ccc(cc3)-c3ccccc3)n2)C1=O)C#CC(C)(C)O
CCN([C@H]1COc2ccc(cc2N(C)C1=O)C#CC(C)(C)O)C(=O)c1n[nH]c(Cc2ccccc2)n1
CN1c2cc(ccc2OC[C@H](NC(=O)c2ncn(Cc3c(C)cccc3C)n2)C1=O)C#CC(C)(C)C
CCN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CC(C)(C)O
CCN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3cccc(F)c3)n2)C1=O)C#CC(C)(C)O
CC(=C)C#Cc1ccc2OC[C@H](NC(=O)c3n[nH]c(Cc4ccccc4)n3)C(=O)Nc2c1
CN1c2cc(\C=C(/Cl)C(C)(C)O)ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CCN1CCCC1
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CCN1CCOCC1
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#C[Si](C)(C)C
CN1c2cc(\C=C\C(=O)NC3CC3)ccc2OC[C@H](NC(=O)c2n[nH]c(n2)-c2ccccc2)C1=O
CN1c2cc(CCC(=O)N3CCCC3)ccc2OC[C@H](NC(=O)c2ncn(n2)-c2ccccc2)C1=O
CN1c2cc(CN3CCn4nc(nc4C3)C(F)(F)F)ccc2OC[C@H](NC(=O)c2nncn2Cc2ccccc2)C1=O
CN1c2cc(CN3CCn4nc(nc4C3)C(F)(F)F)ccc2OC[C@H](NC(=O)C2N=NC(Cc3ccccc3)=N2)C1=O |c:32,42|
CCOC(=O)CCc1ccc2OCC(NC(=O)c3n[nH]c(Cc4ccccc4)n3)C(=O)N(C)c2c1
CN1c2cc(CCC(=O)Nc3ccc4[nH]ncc4c3)ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O |$;;;;;;;;;N;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;$|
CN1c2cc(CCC(=O)Nc3ccc4cn[nH]c4c3)ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O |$;;;;;;;;;N;;;;;;;N;;;;;;;;;;;;;;;;;;;;;;;;;$|
COc1cc2ncnc(NC(=O)CCc3ccc4OCC(NC(=O)c5n[nH]c(Cc6ccccc6)n5)C(=O)N(C)c4c3)c2cc1OC |$;;;;;;;;;N;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;$|
CCOC(=O)CCc1ccc2OCC(NC(=O)c3ncn(Cc4ccccc4F)n3)C(=O)N(C)c2c1
CN1c2cc(CCC(O)=O)ccc2OCC(NC(=O)c2ncn(Cc3ccccc3F)n2)C1=O
CN1c2cc(CCC(=O)Nc3ccc4cn[nH]c4c3)ccc2OCC(NC(=O)c2ncn(Cc3ccccc3F)n2)C1=O |$;;;;;;;;;N;;;;;;;N;;;;;;;;;;;;;;;;;;;;;;;;;;$|
CCOC(=O)CCc1ccc2OCC(NC(=O)c3ncn(Cc4c(Cl)cccc4Cl)n3)C(=O)N(C)c2c1
CN1c2cc(CCC(O)=O)ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2cc(CCC(=O)Nc3ccc4cccnc4c3)ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O |$;;;;;;;;;N;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;$|
CN1c2cc(CCC(=O)N3CCOCC3)ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2cc(CCC(=O)NC3CC3)ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O |$;;;;;;;;;N;;;;;;;;;;;;;;;;;;;;;;;;;;$|
CN1c2cc(CCCO)ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2cc(CCCCO)ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2cc(CCCCOCc3ccccn3)ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2cc(CCCCNc3ccccn3)ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2cc(CCC(=O)N3CCCC3)ccc2OCC(NC(=O)c2ncn(Cc3c(Cl)cccc3Cl)n2)C1=O
CN1c2cc(CCC(=O)NC3CC3)ccc2OCC(NC(=O)c2ncn(Cc3c(Cl)cccc3Cl)n2)C1=O |$;;;;;;;;;N;;;;;;;;;;;;;;;;;;;;;;;;;;;;$|
CN1c2cc(CN3CCN(CC3)c3ccncc3)ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2cc(CN3CCN(CC3)c3ccncc3)ccc2OCC(NC(=O)c2ncn(Cc3c(Cl)cccc3Cl)n2)C1=O
CN1c2cc(\C=C\C(=O)N3CCCC3)ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2cc(\C=C\C(=O)NC3CC3)ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O |$;;;;;;;;;N;;;;;;;;;;;;;;;;;;;;;;;;;;$|
CN1c2cc(CN3CCn4ncnc4C3)ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2cc(CN3CCn4ncnc4C3)ccc2OCC(NC(=O)c2ncn(Cc3ccccc3)n2)C1=O
CN1c2cc(CCC(=O)NC3CC3)ccc2OCC(NC(=O)c2ncn(Cc3ccccc3)n2)C1=O |$;;;;;;;;;N;;;;;;;;;;;;;;;;;;;;;;;;;;$|
CN1c2cc(CCC(=O)NC3CC3)ccc2OCC(NC(=O)c2n[nH]c(Cc3ccc(F)cc3F)n2)C1=O |$;;;;;;;;;N;;;;;;;;;;;;;;;;;;;;;;;;;;;;$|
CN1c2cc(CCC(C)(C)O)ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2cc(ccc2OCC(NC(=O)c2ncn(Cc3ccccc3)n2)C1=O)C#CC(C)(C)O
CN1c2cc(ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CC(C)(C)O
CN1c2cc(CCC(N)=O)ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2cc(CCC(N)=O)ccc2OCC(NC(=O)c2ncn(Cc3ccccc3)n2)C1=O
CN1c2cc(CCC(=O)N3CCCC3)ccc2OCC(NC(=O)c2ncn(Cc3ccccc3)n2)C1=O
CN1c2cc(CCC(=O)N3CCCC3)ccc2OCC(NC(=O)c2n[nH]c(Cc3ccc(F)cc3F)n2)C1=O |$;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;F;;;;;;$|
CN1c2cc(ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CCCCO
CN1c2cc(ccc2OCC(NC(=O)c2n[n-]c(Cc3ccccc3)n2)C1=O)C#CC(C)(C)O
CN1c2cc(ccc2OCC(NC(=O)c2ncn(Cc3ccccc3)n2)C1=O)C#CCCOc1ccc2ncccc2c1
CN1c2cc(ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CCCOc1ccc2ncccc2c1
CN1c2cc(CN3CCn4nc(nc4C3)C(F)(F)F)ccc2OCC(NC(=O)c2ncn(Cc3ccccc3)n2)C1=O
CN1c2cc(CN3CCn4nc(nc4C3)C(F)(F)F)ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2cc(ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CCCOc1ccc2cccnc2c1
CN1c2cc(ccc2OCC(NC(=O)c2ncn(Cc3ccccc3)n2)C1=O)C#CCCOc1ccc2cccnc2c1
CN1c2cc(ccc2OCC(NC(=O)c2n[nH]c(Cc3ccc(F)cc3F)n2)C1=O)C#CC(C)(C)O |$;;;;;;;;;;;;;;;;;;;;;;;F;;;;;;;;;;;;$|
CN1c2cc(ccc2OCC(NC(=O)c2ncn(Cc3ccccc3)n2)C1=O)C#CCCOc1cccc2ncccc12
CN1c2cc(ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CCCOc1cccc2ncccc12
CN1c2cc(CN3CCn4c(C3)nnc4C(F)(F)F)ccc2OCC(NC(=O)c2ncn(Cc3ccccc3)n2)C1=O
CN1c2cc(CN3CCn4c(C3)nnc4C(F)(F)F)ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2cc(ccc2OCC(NC(=O)c2ncn(Cc3ccccc3)n2)C1=O)C#CC(C)(C)C
CN1c2cc(ccc2OCC(NC(=O)c2ncn(Cc3ccccc3)n2)C1=O)C#CC1(O)CCC1
CN1c2cc(ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CC1(O)CCC1
CN1c2cc(ccc2OCC(NC(=O)c2ncn(Cc3ccccc3)n2)C1=O)C#CC1(O)CCCC1
CN1c2cc(ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CC1(O)CCCC1
CN1c2cc(ccc2OCC(NC(=O)c2ncn(Cc3ccccc3)n2)C1=O)C#CC1(O)CCOCC1
CN1c2cc(ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CC1(O)CCOCC1
CN1c2cc(ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CC1(O)COC1
CN1c2cc(ccc2OCC(NC(=O)c2ncn(Cc3ccccc3)n2)C1=O)C#CC1(O)COC1
CN1c2cc(ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CC(C)=C
CC(C)CCc1ccc2OCC(NC(=O)c3n[nH]c(Cc4ccccc4)n3)C(=O)N(C)c2c1
COC(C)(C)C#Cc1ccc2OCC(NC(=O)c3n[nH]c(Cc4ccccc4)n3)C(=O)N(C)c2c1
CN1c2ccc(cc2OCC(NC(=O)c2ncn(Cc3ccccc3)n2)C1=O)C#CC(C)(C)O
CN1c2ccc(cc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CC(C)(C)O
CN1c2ccc(cc2OCC(NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC(C)(C)O
CN1c2cc(ccc2OCC(NC(=O)c2n[nH]c(Cc3c(Cl)cccc3Cl)n2)C1=O)C#CC(C)(C)O
CN1c2ccc(CN3CCn4nc(nc4C3)C(F)(F)F)cc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2ccc(CN3CCn4nc(C)nc4C3)cc2OCC(NC(=O)c2ncn(Cc3ccccc3)n2)C1=O
CN1c2cc(ccc2OCC(NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC(C)(C)O
CN1c2cc(ccc2OCC(NC(=O)c2nnc(Cc3ccccc3)o2)C1=O)C#CC(C)(C)O
CN1c2ccc(cc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CC1(O)COC1
CN1c2cc(ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#C[C@@]1(O)CO[C@@H]2[C@H](CO[C@H]12)OC(=O)c1ccccc1 |r|
CN1c2cc(ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#C[C@@]1(O)CO[C@@H]2[C@@H](O)CO[C@H]12 |r|
CN1c2cc(ccc2OCC(NC(=O)c2n[nH]c(Cc3cccc(F)c3)n2)C1=O)C#CC(C)(C)O
CN1c2cc(ccc2OCC(NC(=O)c2n[nH]c(Cc3ccc(F)cc3)n2)C1=O)C#CC(C)(C)O
CN1c2cc(ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3F)n2)C1=O)C#CC(C)(C)O
CN1c2cc(ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#C
CN1c2cc(ccc2OCC(NC(=O)c2ncn(Cc3ccccc3C)n2)C1=O)C#CC(C)(C)O
CN1c2cc(ccc2OCC(NC(=O)c2ncn(Cc3ccc(cc3)-c3ccccc3)n2)C1=O)C#CC(C)(C)O
CN1c2cc(ccc2OCC(NC(=O)c2ncn(Cc3c(C)cccc3C)n2)C1=O)C#CC(C)(C)O
CC(C)Cn1cnc(n1)C(=O)NC1COc2ccc(cc2N(C)C1=O)C#CC(C)(C)O
CCN(C1COc2ccc(cc2N(C)C1=O)C#CC(C)(C)O)C(=O)c1n[nH]c(Cc2ccccc2)n1
CCN(C1COc2ccc(cc2N(C)C1=O)C#CC(C)(C)O)C(=O)c1cc(Cc2ccccc2)on1
CN1c2cc(ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#Cc1ccc2CCNCc2c1
CN1c2cc(ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3F)n2)C1=O)C#CC(C)(C)C
CN1c2cc(ccc2OCC(NC(=O)c2ncn(Cc3c(C)cccc3C)n2)C1=O)C#CC(C)(C)C
CCN1c2cc(ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CC(C)(C)O
CCN1c2cc(ccc2OCC(NC(=O)c2n[nH]c(Cc3cccc(F)c3)n2)C1=O)C#CC(C)(C)O
CC(=C)C#Cc1ccc2OCC(NC(=O)c3n[nH]c(Cc4ccccc4)n3)C(=O)Nc2c1
CN1c2cc(\C=C(/Cl)C(C)(C)O)ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2cc(ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CCN1CCOCC1
CN1c2cc(ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#C[Si](C)(C)C
CN1c2cc(ccc2OCC(NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC1(O)CCCC1
CN1c2cc(ccc2OCC(NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC(C)=C
CN1c2cc(ccc2OCC(NC(=O)c2cc(Oc3ccc(F)cc3)ccn2)C1=O)C#CC(C)(C)O
CN1c2cc(ccc2OCC(NC(=O)c2cc(Oc3ccc(F)cc3)ccn2)C1=O)C#CC(C)(C)C
CN1c2cc(ccc2OCC(NC(=O)c2cc(Oc3ccccc3F)ccn2)C1=O)C#CC(C)(C)C
CN1c2cc(ccc2OCC(NC(=O)c2cc(Oc3ccccc3F)ccn2)C1=O)C#CC(C)(C)O
CN1c2cc(ccc2OCC(NC(=O)c2cc(Oc3ccc(F)cc3F)ccn2)C1=O)C#CC(C)(C)C
CN1c2cc(ccc2OCC(NC(=O)c2cc(Oc3ccc(F)cc3F)ccn2)C1=O)C#CC(C)(C)O
CN1c2cc(ccc2OCC(NC(=O)c2cc(Oc3cccc(F)c3)ccn2)C1=O)C#CC(C)(C)C
CN1c2cc(ccc2OCC(NC(=O)c2cc(Oc3cccc(F)c3)ccn2)C1=O)C#CC(C)(C)O
CC(C)CCc1ccc2OCC(NC(=O)c3cc(Oc4ccccc4)ccn3)C(=O)N(C)c2c1
CN1c2cc(ccc2OCC(NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC(C)(C)CO
CN1c2cc(ccc2OCC(NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC1(O)COC1
CN1c2cc(ccc2OCC(NC(=O)c2cc(Oc3ccc(F)cc3)ccn2)C1=O)C#CC1(O)COC1
CN1c2cc(ccc2OCC(NC(=O)c2cc(Oc3ccccc3F)ccn2)C1=O)C#CC1(O)COC1
CN1c2cc(ccc2OC[C@@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC(C)(C)O |r|
CN1c2cc(ccc2OCC(NC(=O)c2cc(Oc3ccc(F)cc3F)ccn2)C1=O)C#CC1(O)COC1
CN1c2cc(ccc2OCC(NC(=O)c2cc(Oc3cccc(F)c3)ccn2)C1=O)C#CC1(O)COC1
CN1c2cc(ccc2OCC(NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CCN1CCCC1
CN1c2cc(ccc2OCC(NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CCN1CCOCC1
CN1c2cc(ccc2OCC(NC(=O)c2cc(Oc3c(F)cccc3F)ccn2)C1=O)C#CC(C)(C)O
CN1c2cc(ccc2OCC(NC(=O)c2cc(Oc3ccccc3)cc(C)n2)C1=O)C#CC(C)(C)O
CN1c2cc(ccc2OCC(NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC1(O)CCC1
CN1c2cc(ccc2OCC(NC(=O)c2ccc(Oc3ccccc3)cn2)C1=O)C#CC(C)(C)O
CN1c2cc(ccc2OCC(NC(=O)c2ccc(Oc3ccc(F)cc3)cn2)C1=O)C#CC(C)(C)O
CN1c2cc(ccc2OCC(NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC1(O)CCOCC1
CN1c2cc(ccc2OCC(NC(=O)c2cc(Oc3c(C)cccc3C)ccn2)C1=O)C#CC(C)(C)O
CN1c2cc(ccc2OCC(NC(=O)c2cc(Cc3ccc(F)cc3)ccn2)C1=O)C#CC(C)(C)O
CN1c2cc(ccc2OCC(NC(=O)c2cc(Cc3ccc(F)cc3)ccn2)C1=O)C#CC1(O)COC1
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC1(C)COC1 |r|
COC1(COC1)C#Cc1ccc2OC[C@H](NC(=O)c3cc(Oc4ccccc4)ccn3)C(=O)N(C)c2c1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC1(F)COC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC1(COC1)OC(=O)NCCCN1CCOCC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC1(O)CCN(CC1)C(=O)c1cc(Oc2ccccc2)ccn1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC1(O)CCNCC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccc(F)cc3)ccn2)C1=O)C#CC1(O)CCNCC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccc(F)cc3)ccn2)C1=O)C#CC1(O)CCN(CC1)C(C)=O |r|
CN1CCC(O)(CC1)C#Cc1ccc2OC[C@H](NC(=O)c3cc(Oc4ccc(F)cc4)ccn3)C(=O)N(C)c2c1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC1(O)CNC1 |r|
CN1CC(O)(C1)C#Cc1ccc2OC[C@H](NC(=O)c3cc(Oc4ccccc4)ccn3)C(=O)N(C)c2c1 |r|
CNCCC(=C)C#Cc1ccc2OC[C@H](NC(=O)c3cc(Oc4ccc(F)cc4)ccn3)C(=O)N(C)c2c1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC(C)(C)N |r,$;;;;;;;;;;;N;;;;;;;;;;;;;;;;;;;;;;;$|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC(C)(C)CN1CCOCC1 |r|
C[C@H](NC(=O)OC(C)(C)C)C(=O)OCC(C)(C)C#Cc1ccc2OC[C@H](NC(=O)c3cc(Oc4ccccc4)ccn3)C(=O)N(C)c2c1 |r|
C[C@H](N)C(=O)OCC(C)(C)C#Cc1ccc2OC[C@H](NC(=O)c3cc(Oc4ccccc4)ccn3)C(=O)N(C)c2c1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC1(F)CNC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC(C)(C)COC(=O)CCC(O)=O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC(C)(C)COC(=O)[C@H](OC(C)=O)[C@@H](OC(C)=O)C(O)=O |r|
CN1CC(F)(C1)C#Cc1ccc2OC[C@H](NC(=O)c3cc(Oc4ccccc4)ccn3)C(=O)N(C)c2c1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC1(COC1)OC(=O)CCC(O)=O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccc(F)cc3)ccn2)C1=O)C#CC(C)(C)CO |r,$;;;;;;;;;;;;;;;;;;;;;;F;;;;;;;;;;;;;;$|
CN1c2cc(CN3CCC4(CCOCC4)CC3)ccc2NC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O |r|
CN1c2cc(CN3CC4(C3)CCOCC4)ccc2NC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC1(O)CN(C1)C(=O)C(F)(F)F |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(OC3CCC3)ccn2)C1=O)C#CC(C)(C)O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(OC3CCC3)ccn2)C1=O)C#CC1(O)COC1 |r|
COC1(CNC1)C#Cc1ccc2OC[C@H](NC(=O)c3cc(Oc4ccccc4)ccn3)C(=O)N(C)c2c1 |r|
COC1(CN(C)C1)C#Cc1ccc2OC[C@H](NC(=O)c3cc(Oc4ccccc4)ccn3)C(=O)N(C)c2c1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(OC3CCCC3)ccn2)C1=O)C#CC(C)(C)O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(OC3CCCC3)ccn2)C1=O)C#CC1(O)COC1 |r|
COC(=O)C#Cc1ccc2OC[C@H](NC(=O)c3cc(Oc4ccccc4)ccn3)C(=O)N(C)c2c1 |r|
CC(C)[C@H](N)C(=O)OC1(COC1)C#Cc1ccc2OC[C@H](NC(=O)c3cc(Oc4ccccc4)ccn3)C(=O)N(C)c2c1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC(O)=O |r|
COc1ccnc(c1)C(=O)N[C@H]1COc2ccc(cc2N(C)C1=O)C#CC1(O)COC1 |r|
COc1ccnc(c1)C(=O)N[C@H]1COc2ccc(cc2N(C)C1=O)C#CC(C)(C)O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC(C)(C)N |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3ccc(F)cc3)cn2)C1=O)C#CC1(O)CCOCC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC1(O)COC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC1(F)CN(C1)C(C)=O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC(C)(C)NCc1ccc(F)cc1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC1(O)CCS(=O)(=O)CC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC1(O)CS(=O)C1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC1(O)CS(=O)(=O)C1 |r|
CN[C@@H](C)C(=O)OC1(COC1)C#Cc1ccc2OC[C@H](NC(=O)c3cc(Oc4ccccc4)ccn3)C(=O)N(C)c2c1 |r|
C[C@H](N)C(=O)OC1(COC1)C#Cc1ccc2OC[C@H](NC(=O)c3cc(Oc4ccccc4)ccn3)C(=O)N(C)c2c1 |r|
CC(C)N1CC(O)(C1)C#Cc1ccc2OC[C@H](NC(=O)c3cc(Oc4ccccc4)ccn3)C(=O)N(C)c2c1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC(C)(C)N1CCCC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#Cc1cn(C)cn1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3ccccc3)cn2)C1=O)C#CC(C)(C)C |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3ccccc3)cn2)C1=O)C#CC(C)(C)O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3ccccc3)cn2)C1=O)C#Cc1cccnc1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3ccccc3)cn2)C1=O)C#Cc1ccccn1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3ccccc3)cn2)C1=O)C#CC1(O)COC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3ccccc3)cn2)C1=O)C#CC1CC2(C1)CCOCC2 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3ccc(F)cc3)cn2)C1=O)C#CC(C)(C)O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3ccccc3)cn2)C1=O)C#CC1(O)CCC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2ncc(Cc3ccccc3)c2C)C1=O)C#CC(C)(C)O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3ccc(F)cc3)cn2)C1=O)C#CC1(O)CCC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3ccc(F)cc3)cn2)C1=O)C#CC1(O)COC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2ccc(Cc3ccc(F)cc3)n2)C1=O)C#CC1(O)CCC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3ccc(F)cc3)cn2)C1=O)C#CC1(O)CC2(CCC2)C1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3ccc(F)cc3)cn2)C1=O)C#CC1(O)CC2(COC2)C1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3ccc(F)cc3)cn2)C1=O)C#CC(C)(C)N |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2nnc(o2)C2(CC2)c2ccccc2)C1=O)N1CC2(C1)CCOCC2 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2nnc(Cc3ccccc3)o2)C1=O)N1CC2(C1)CCOCC2 |r|
CN1c2cc(Br)ccc2OC[C@H](NC(=O)N\C=C(\Cc2ccc(F)cc2F)C=N)C1=O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)N\C=C(\Cc2ccc(F)cc2F)C=N)C1=O)C#CC(C)(C)CNC(=O)OC(C)(C)C |r|
CN1c2cc(ccc2OC[C@H](NC(=O)N\C=C(\Cc2ccc(F)cc2F)C=N)C1=O)C#CC(C)(C)CN |r|
CN1c2ccc(cc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#Cc1ccccn1 |r|
CN1c2ccc(cc2OC[C@H](NC(=O)c2cc(Oc3ccc(cc3)C#N)ccn2)C1=O)C#CC(C)(C)O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccc(cc3)C#N)ccn2)C1=O)C#CC(C)(C)O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccc(cc3)C#N)ccn2)C1=O)C#CC1(O)COC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(ccn2)-c2ccccc2)C1=O)C#CC(C)(C)O |r|
CN1c2ccc(cc2OC[C@H](NC(=O)c2cc(Oc3cccc(c3)C#N)ccn2)C1=O)C#CC(C)(C)O |r|
COc1ccc(cc1)-c1ccnc(c1)C(=O)N[C@H]1COc2ccc(cc2N(C)C1=O)C#CC(C)(C)O |r|
COc1cccc(c1)-c1ccnc(c1)C(=O)N[C@H]1COc2ccc(cc2N(C)C1=O)C#CC(C)(C)O |r|
CN1c2cc(CCC(N)=O)ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC(C)(C)C |r|
COc1ccc(cc1)-c1ccnc(c1)C(=O)N[C@H]1COc2cc(ccc2N(C)C1=O)N1CCC2(CCOCC2)CC1 |r|
CN1CCC2(CC1)CCN(CC2)c1ccc2OC[C@H](NC(=O)c3cc(Oc4ccccc4)ccn3)C(=O)N(C)c2c1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)N1CC2(C1)CCOCC2 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)N1CCC2(C1)CCOCC2 |r|
COC(C)(C)C#Cc1ccc2OC[C@H](NC(=O)c3cc(Oc4ccccc4)ccn3)C(=O)N(C)c2c1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#Cc1cccc(n1)C#N |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CCO |r|
CN(C)CC#Cc1ccc2OC[C@H](NC(=O)c3cc(Oc4ccccc4)ccn3)C(=O)N(C)c2c1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC1CCCN1 |r|
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(CNC(=O)c2cc(OC(F)(F)F)ccc2F)c1
COc1ncc(cc1C(=O)NCc1cc(F)cc(F)c1OC1CCOCC1)-c1ccc2nc(NC(=O)CO)cn2n1
COCC(=O)Nc1cn2nc(ccc2n1)-c1cnc(OC)c(c1)C(=O)NCc1ccccc1OC(F)(F)F
CCC(=O)Nc1cn2nc(ccc2n1)-c1cnc(OC)c(c1)C(=O)NCc1cc(F)cc(F)c1OCC1CC1
COc1ncc(cc1C(=O)NCc1cc(F)cc(F)c1OCC1CC1)-c1ccc2nc(NC(=O)C(C)C)cn2n1
COc1ncc(cc1C(=O)NCc1cc(OC(F)(F)F)ccc1F)-c1ccc2nc(NC(C)=O)c(C)n2n1
COc1ncc(cc1C(=O)NCc1cc(F)cc(F)c1OCC1CC1)-c1ccc2nc(NC(=O)CC#N)cn2n1
COc1ncc(cc1C(=O)NCc1cc(F)cc(F)c1OCC1CC1)-c1ccc2nc(NC(=O)C(C)(C)C#N)cn2n1
C[C@H](NC(=O)c1cc(cnc1C)-c1ccc2nc(NC(C)=O)cn2n1)c1cc(OC(F)(F)F)ccc1F |r|
C[C@@H](NC(=O)c1cc(cnc1C)-c1ccc2nc(NC(C)=O)cn2n1)c1cc(OC(F)(F)F)ccc1F |r|
CCC(=O)Nc1cn2nc(ccc2n1)-c1cnc(OC)c(c1)C(=O)NCc1cc(OC(F)(F)F)ccc1F
COc1ncc(cc1C(=O)NCc1cc(OC(F)(F)F)ccc1F)-c1ccc2nc(NC(=O)C(C)C)cn2n1
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(Cl)c(c1)C(=O)NCc1cc(OC(F)(F)F)ccc1F
COc1nc(C)c(cc1C(=O)N[C@@H](C)c1ccccc1OC(F)(F)F)-c1ccc2nc(NC(C)=O)cn2n1 |r|
COc1nc(C)c(cc1C(=O)N[C@H](C)c1ccccc1OC(F)(F)F)-c1ccc2nc(NC(C)=O)cn2n1 |r|
COc1ncc(cc1C(=O)NCc1ccccc1OC(F)(F)F)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1cccc(F)c1OCC1CC1)-c1ccc2nc(NC(=O)C(C)(C)O)cn2n1
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(cnc1C)C(=O)NCc1cc(F)cc(F)c1OCC1CC1
COc1nc(C)c(cc1C(=O)NCc1ccccc1OC(C)CO)-c1ccc2nc(NC(C)=O)cn2n1
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(c(c1)C(=O)NCc1cc(OC(F)(F)F)ccc1F)C(F)(F)F
COc1nc(C)c(cc1C(=O)NCc1ccccc1OC(F)(F)F)-c1ccc2nc(NC(C)=O)cn2n1
CC(C)Oc1ccccc1CNC(=O)c1cc(cnc1C)-c1ccc2nc(NC(C)=O)cn2n1
CC(=O)Nc1cn2nc(ccc2n1)-c1cncc(c1)C(=O)NCc1ccccc1OC1CCCC1
COc1ncc(cc1C(=O)NCc1ccccc1OCC1CC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCCC(O)c1ccc(Cl)cc1)-c1ccc2nc(NC(C)=O)cn2n1
CC(CCNC(=O)c1cccc(c1)-c1ccc2nc(NC(=O)c3ccnc(F)c3)cn2n1)c1ccccc1
COc1ncc(cc1C(=O)NCCC(C)c1ccccc1)-c1ccc2nc(NC(C)=O)cn2n1
Cc1ncc(cc1C(=O)NCc1ccccc1Sc1ccccc1CO)-c1ccc2nc(NC(=O)C(C)(C)C#N)cn2n1
C[C@@H](NC(=O)c1cc(cnc1C)-c1ccc2nc(NC(=O)C(C)(C)C#N)cn2n1)c1cc(OC(F)(F)F)ccc1F |r|
COc1ncc(cc1C(=O)NCc1cc(OC(F)(F)F)ccc1F)-c1ccc2nc(NC(=O)C(C)(C)C#N)cn2n1
COc1ncc(cc1C(=O)NCc1cc(OCC2CC2)ccc1F)-c1ccc2nc(NC(=O)C(C)(C)C#N)cn2n1
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(c(c1)C(=O)NCc1cc(ccc1F)C(F)(F)F)C(F)(F)F
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(c(c1)C(=O)NCc1c(F)ccc(F)c1OCC1CC1)C(F)(F)F
COc1ncc(cc1C(=O)NCc1ccccc1OC(F)(F)F)-c1ccc2nc(NC(=O)CC#N)cn2n1
COc1ncc(cc1C(=O)NCc1cc(OC(F)(F)F)ccc1F)-c1ccc2nc(NC(=O)CC#N)cn2n1
COc1ncc(cc1C(=O)NCc1cc(ccc1F)C(F)(F)F)-c1ccc2nc(NC(=O)CO)cn2n1
COc1ncc(cc1C(=O)NCc1cc(OC(F)(F)F)ccc1F)-c1ccc2nc(NC(=O)CO)cn2n1
COc1ncc(cc1C(=O)NCc1cc(OC(F)(F)F)ccc1F)-c1ccc2nc(NC(=O)C(C)(C)O)cn2n1
COc1ccc(F)c(CNC(=O)c2cc(c(C)nc2C)-c2ccc3nc(NC(C)=O)cn3n2)c1
Cc1nc(C)c(cc1C(=O)NCc1cc(OC(F)(F)F)ccc1F)-c1ccc2nc(NC(=O)CO)cn2n1
Cc1ncc(cc1C(=O)NCc1cc(OC(F)(F)F)ccc1F)-c1ccc2nc(NC(=O)CO)cn2n1
COc1ccc(F)c(CNC(=O)c2cc(cnc2OC)-c2ccc3nc(NC(C)=O)cn3n2)c1
COc1ncc(cc1C(=O)N[C@@H](C)c1cc(OC(F)(F)F)ccc1F)-c1ccc2nc(NC(C)=O)cn2n1 |r|
COc1ncc(cc1C(=O)NCc1c(F)cccc1OCC(F)(F)F)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1cc(F)cc(F)c1OC1CCCOC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1cc(F)cc(F)c1O[C@@H]1CCOC1)-c1ccc2nc(NC(C)=O)cn2n1 |r|
COc1ncc(cc1C(=O)NCc1cc(F)cc(F)c1O[C@H]1CCOC1)-c1ccc2nc(NC(C)=O)cn2n1 |r|
COc1ncc(cc1C(=O)N[C@H](C)c1cc(OC(F)(F)F)ccc1F)-c1ccc2nc(NC(C)=O)cn2n1 |r|
COc1ncc(cc1C(=O)NCc1cc(F)cc(F)c1OC1COC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1cc(F)cc(F)c1OCC1CC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1cc(F)cc(F)c1OC1CCOCC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NC(C)c1cc(ccc1F)C(F)(F)F)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1ccc(F)c(F)c1OCC1CC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NC(C)c1ccccc1OC(F)(F)F)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1cc(OCC2CC2)ccc1F)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1c(F)cccc1OC(F)(F)F)-c1ccc2nc(NC(C)=O)cn2n1
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(C(=O)NCc2cc(F)cc(F)c2OC2CCCOC2)c(C)nc1C
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(C(=O)NCc2cc(F)cc(F)c2O[C@H]2CCOC2)c(C)nc1C
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(C(=O)NCc2cc(F)cc(F)c2O[C@@H]2CCOC2)c(C)nc1C
CC1CC(CCO1)Oc1c(F)cc(F)cc1CNC(=O)c1cc(c(C)nc1C)-c1ccc2nc(NC(C)=O)cn2n1
C[C@H]1CC(C[C@@H](C)O1)Oc1c(F)cccc1CNC(=O)c1cc(c(C)nc1C)-c1ccc2nc(NC(C)=O)cn2n1
CC1CC(CC(C)O1)Oc1c(F)cc(F)cc1CNC(=O)c1cc(c(C)nc1C)-c1ccc2nc(NC(C)=O)cn2n1
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(C(=O)NCc2ncccc2OCC(F)(F)F)c(C)nc1C
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(C(=O)NCc2cc(F)cc(F)c2OC2CCOCC2)c(C)nc1C
CC(NC(=O)c1cc(c(C)nc1C)-c1ccc2nc(NC(C)=O)cn2n1)c1cc(ccc1F)C(F)(F)F
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(C(=O)NCc2ccccc2OCC(F)(F)F)c(C)nc1C
C[C@@H](NC(=O)c1cc(c(C)nc1C)-c1ccc2nc(NC(C)=O)cn2n1)c1cc(ccc1F)C(F)(F)F
CC(NC(=O)c1cc(c(C)nc1C)-c1ccc2nc(NC(C)=O)cn2n1)c1cc(OC(F)(F)F)ccc1F
C[C@@H](NC(=O)c1cc(c(C)nc1C)-c1ccc2nc(NC(C)=O)cn2n1)c1cc(OC(F)(F)F)ccc1F
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(C(=O)NCc2cc(F)ccc2OCC(F)(F)F)c(C)nc1C
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(C(=O)NCc2cccc(OCC(F)(F)F)c2)c(C)nc1C
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(C(=O)NCc2cccc(c2)C(F)(F)F)c(C)nc1C
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(C(=O)NCc2cc(ccc2F)C(F)(F)F)c(C)nc1C
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(C(=O)NCc2cc(OC(F)(F)F)ccc2F)c(C)nc1C
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(C(=O)NCc2cc(F)cc(F)c2OC2COC2)c(C)nc1C
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(C(=O)NCc2cc(F)cc(OC(F)(F)F)c2)c(C)nc1C
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(C(=O)NCC[C@H](O)c2ccc(Cl)cc2)c(C)nc1C
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(C(=O)NCc2ccccc2OCC2CC2)c(C)nc1C
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(C(=O)NCc2cccnc2OCC2CCCC2)c(C)nc1C
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(C(=O)NCc2ccccc2OCC2CCCC2)c(C)nc1C
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(C(=O)NCc2cc(F)cc(F)c2OCC2CC2)c(C)nc1C
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(C(=O)NCc2cccc(OC(F)(F)F)c2)c(C)nc1C
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(C(=O)NCc2ccccc2OC(F)(F)F)c(C)nc1C
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(C(=O)NCc2cc(F)cc(F)c2OCC2CCCC2)c(C)nc1C
Cc1nc(C)c(cc1C(=O)NCc1cc(F)cc(F)c1O[C@H]1CCOC1)-c1ccc2nc(NC(=O)CO)cn2n1
C[C@@H](NC(=O)c1cc(c(C)nc1C)-c1ccc2nc(NC(=O)CO)cn2n1)c1cc(ccc1F)C(F)(F)F
Cc1nc(C)c(cc1C(=O)NCc1cc(ccc1F)C(F)(F)F)-c1ccc2nc(NC(=O)CO)cn2n1
C[C@@H](NC(=O)c1cc(c(C)nc1C)-c1ccc2nc(NC(=O)CO)cn2n1)c1cc(OC(F)(F)F)ccc1F
COc1ncc(cc1C(=O)NCc1cc(F)cc(F)c1OC1CCOC(C)C1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1cc(F)cc(F)c1OCC1CCC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1cc(F)cc(F)c1O[C@H]1CCOC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1cc(F)cc(F)c1OC1CC(C)OC(C)C1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)N[C@H](C)c1ccccc1C(F)(F)F)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1cc(F)ccc1OCC(F)(F)F)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)N[C@H](C)c1cc(ccc1F)C(F)(F)F)-c1ccc2nc(NC(C)=O)cn2n1 |r|
COc1ncc(cc1C(=O)N[C@@H](C)c1cc(ccc1F)C(F)(F)F)-c1ccc2nc(NC(C)=O)cn2n1 |r|
COc1ncc(cc1C(=O)NCc1ccccc1OCC(F)(F)F)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1cccc(c1)C(F)(F)F)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1cc(ccc1F)C(F)(F)F)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)N[C@H](C)c1cccc(OC(F)(F)F)c1)-c1ccc2nc(NC(C)=O)cn2n1 |r|
COc1ncc(cc1C(=O)NCc1ccccc1CN1CCOCC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1ccccc1COC(C)C)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1cc(F)cc(F)c1OCC(C)C)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1ccccc1OCC(C)C)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1cc(F)cc(F)c1OC1CC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCC[C@H](O)c1ccc(Cl)cc1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1ccc(F)cc1OC(F)(F)F)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NC(C)c1c(F)cccc1OCC1CC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)N[C@@H](C)c1cccc(OC(F)(F)F)c1)-c1ccc2nc(NC(C)=O)cn2n1 |r|
COc1ncc(cc1C(=O)NCc1cccc(OC(F)(F)F)c1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1c(F)ccc(F)c1OCC1CC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1c(F)cccc1OC1CCOCC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NC(C)c1cc(F)cc(F)c1OCC1CC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1ccc(F)c(F)c1OC(C)C1CC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1cccc(F)c1OC(C)C1CC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1ncccc1OC(C)C1CC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1cc(F)cc(OC(F)(F)F)c1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1cc(F)cc(OCC2CC2)c1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1c(F)ccc(F)c1OC)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1ccc(F)c(OCC2CC2)c1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)N(C)Cc1cccc(OC(F)(F)F)c1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1cc(OC(F)(F)F)ccc1F)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1cc(ccc1Cl)C(F)(F)F)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1c(F)cc(F)cc1OCC1CC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1cccc(F)c1OCC1CC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1ccc(F)cc1OC1CCOCC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1ccccc1OCC1CCC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1c(F)cccc1OC1CCCC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1ccccc1S(=O)(=O)C1CC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1ccccc1OC1CCCC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1ccccc1-n1cccc1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NC[C@H]1C[C@@H]1c1ccc(F)cc1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1ccccc1N1CCOCC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1ncccc1OC1CCCC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1ccccc1OCC1CCCC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1ccccc1OC(C)C)-c1ccc2nc(NC(C)=O)cn2n1
COc1ncc(cc1C(=O)NCc1cc(F)ccc1OC1CCCC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCc1cc(F)cc(F)c1OC1CC(C)OC(C)C1)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCc1cccc(F)c1OC1C[C@H](C)O[C@H](C)C1)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCc1cc(F)cc(F)c1O[C@@H]1CCOC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCc1cc(F)cc(F)c1OC1CCCOC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCc1cc(F)cc(F)c1O[C@H]1CCOC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCc1cc(F)cc(F)c1OC1CCOC(C)C1)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCc1c(F)cccc1OCC(F)(F)F)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCc1cc(F)cc(F)c1OCC1CC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCc1cc(OC(F)(F)F)ccc1F)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCc1ccc(F)c(F)c1OCC1CC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCc1cc(OCC2CC2)ccc1F)-c1ccc2nc(NC(C)=O)cn2n1
C[C@H](NC(=O)c1cc(cnc1C)-c1ccc2nc(NC(=O)CO)cn2n1)c1cc(OC(F)(F)F)ccc1F
C[C@@H](NC(=O)c1cc(cnc1C)-c1ccc2nc(NC(=O)CO)cn2n1)c1cc(ccc1F)C(F)(F)F
Cc1ncc(cc1C(=O)NCc1cc(ccc1F)C(F)(F)F)-c1ccc2nc(NC(=O)CO)cn2n1
Cc1ncc(cc1C(=O)NCc1cc(F)cc(F)c1OC1CCOCC1)-c1ccc2nc(NC(=O)CO)cn2n1
C[C@@H](NC(=O)c1cc(cnc1C)-c1ccc2nc(NC(=O)CO)cn2n1)c1cc(OC(F)(F)F)ccc1F
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)NCc1cc(F)cc(F)c1OC1CCCOC1
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)NCc1cc(F)cc(F)c1O[C@H]1CCOC1
CC1CC(CCO1)Oc1c(F)cc(F)cc1CNC(=O)c1cc(cnc1C)-c1ccc2nc(NC(C)=O)cn2n1
CC1CC(CC(C)O1)Oc1c(F)cc(F)cc1CNC(=O)c1cc(cnc1C)-c1ccc2nc(NC(C)=O)cn2n1
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)NCc1c(F)cccc1OCC(F)(F)F
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)NCc1cc(ccn1)C(F)(F)F
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)NCc1cc(F)cc(F)c1OC1CCOCC1
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)NCc1ccccc1OCC(F)(F)F
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)NCc1cccc(OCC(F)(F)F)c1
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)NCc1cc(F)ccc1OCC(F)(F)F
C[C@H](NC(=O)c1cc(cnc1C)-c1ccc2nc(NC(C)=O)cn2n1)c1cc(ccc1F)C(F)(F)F |r|
C[C@@H](NC(=O)c1cc(cnc1C)-c1ccc2nc(NC(C)=O)cn2n1)c1cc(ccc1F)C(F)(F)F |r|
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)NCc1cc(ccc1F)C(F)(F)F
CC(NC(=O)c1cc(cnc1C)-c1ccc2nc(NC(C)=O)cn2n1)c1ccccc1OC(F)(F)F
CC(NC(=O)c1cc(cnc1C)-c1ccc2nc(NC(C)=O)cn2n1)c1cc(ccc1F)C(F)(F)F
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)NCc1cc(F)cc(OC(F)(F)F)c1
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)NCc1cc(OC(F)(F)F)ccc1F
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)NCc1ccc(F)c(F)c1OCC1CC1
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)NCc1cc(F)cc(F)c1OCC1CCC1
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)NCC[C@@H](O)c1ccc(Cl)cc1
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)NCc1cccc(F)c1OCC1CC1
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)NCc1cc(F)cc(F)c1OCC1CC1
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)NCc1cc(OCC2CC2)ccc1F
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)NCC[C@H](O)c1ccc(Cl)cc1
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)NCc1cccnc1OCC1CCCC1
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)NCc1cc(F)ccc1OCC1CCCC1
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)NCc1c(F)cccc1OCC1CCC1
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)NCc1ccccc1OC(F)(F)F
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)NCc1cccc(OC(F)(F)F)c1
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)NCc1cc(F)ccc1OC1CCCC1
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)NCc1c(F)cccc1OC1CCCC1
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)NCc1ccccc1OC1CCOC1
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)NCc1ccccc1OC1CCCC1
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)NCc1c(F)cccc1OCC1CC1
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)NCc1ccccc1OCC1CC1
C[C@H](NC(=O)c1cnc(C)c(c1)-c1ccc2nc(NC(C)=O)cn2n1)c1cc(OC(F)(F)F)ccc1F
C[C@@H](NC(=O)c1cnc(C)c(c1)-c1ccc2nc(NC(C)=O)cn2n1)c1cc(OC(F)(F)F)ccc1F
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(cnc1C)C(=O)NCc1cc(OC(F)(F)F)ccc1F
CC(CCNC(=O)c1cnc(C)c(c1)-c1ccc2nc(NC(C)=O)cn2n1)c1ccccc1
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(cnc1C)C(=O)NCc1cccc(F)c1OCC1CC1
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(cnc1C)C(=O)NCc1ccccc1OC(F)(F)F
C[C@@H](NC(=O)c1cncc(c1)-c1ccc2nc(NC(C)=O)cn2n1)c1cc(OC(F)(F)F)ccc1F
CC(=O)Nc1cn2nc(ccc2n1)-c1cncc(c1)C(=O)NCc1cc(OCC2CC2)ccc1F
CC(=O)Nc1cn2nc(ccc2n1)-c1cncc(c1)C(=O)NCc1cc(OC(F)(F)F)ccc1F
CC(CCNC(=O)c1cncc(c1)-c1ccc2nc(NC(C)=O)cn2n1)c1ccccc1
CC(=O)Nc1cn2nc(ccc2n1)-c1cncc(c1)C(=O)NCc1ccccc1OCC1CC1
CC(=O)Nc1cn2nc(ccc2n1)-c1cncc(c1)C(=O)NCc1c(F)cccc1OC1CCCC1
CC(=O)Nc1cn2nc(ccc2n1)-c1cncc(c1)C(=O)NCc1ncccc1OC1CCCC1
CC(=O)Nc1cn2nc(ccc2n1)-c1cncc(c1)C(=O)NCc1cc(F)ccc1OC1CCCC1
CCC(=O)Nc1cn2nc(ccc2n1)-c1cnc(OC)c(c1)C(=O)N[C@H](C)c1cc(OC(F)(F)F)ccc1F
CCC(=O)Nc1cn2nc(ccc2n1)-c1cnc(OC)c(c1)C(=O)NCC[C@H](O)c1ccc(Cl)cc1
CCC(=O)Nc1cn2nc(ccc2n1)-c1cnc(OC)c(c1)C(=O)NCc1cc(F)cc(F)c1OC1CCOCC1
CCC(=O)Nc1cn2nc(ccc2n1)-c1cnc(OC)c(c1)C(=O)NCc1ccccc1OC(F)(F)F
CCC(=O)Nc1cn2nc(ccc2n1)-c1cnc(OC)c(c1)C(=O)NCc1ccc(F)c(F)c1OCC1CC1
CCC(=O)Nc1cn2nc(ccc2n1)-c1cnc(OC)c(c1)C(=O)NCc1cc(OCC2CC2)ccc1F
CC(=O)Nc1nc2ccc(nn2c1C)-c1cnc(C)c(c1)C(=O)NCc1cccc(OC(F)(F)F)c1
CC(=O)Nc1nc2ccc(nn2c1C)-c1cnc(C)c(c1)C(=O)NCc1cc(ccc1F)C(F)(F)F
CC(=O)Nc1nc2ccc(nn2c1C)-c1cnc(C)c(c1)C(=O)NCc1cc(OC(F)(F)F)ccc1F
COc1ncc(cc1C(=O)NCc1cc(ccc1F)C(F)(F)F)-c1ccc2nc(NC(C)=O)c(C)n2n1
COc1ncc(cc1C(=O)NCc1ccc(F)c(OC(F)(F)F)c1)-c1ccc2nc(NC(C)=O)c(C)n2n1
COc1ncc(cc1C(=O)NCCC(C)c1ccccc1)-c1ccc2nc(NC(C)=O)c(C)n2n1
COc1ncc(cc1C(=O)NCc1cccc(OC(F)(F)F)c1)-c1ccc2nc(NC(C)=O)c(C)n2n1
COc1ncc(cc1C(=O)NCc1ccccc1OC(F)(F)F)-c1ccc2nc(NC(C)=O)c(C)n2n1
COc1ncc(cc1C(=O)NCc1cc(F)cc(F)c1OCC1CC1)-c1ccc2nc(NC(C)=O)c(C)n2n1
COCC(=O)Nc1cn2nc(ccc2n1)-c1cnc(OC)c(c1)C(=O)NCc1cc(OCC2CC2)ccc1F
COCC(=O)Nc1cn2nc(ccc2n1)-c1cnc(OC)c(c1)C(=O)NCc1cc(F)cc(F)c1OCC1CC1
COCC(=O)Nc1cn2nc(ccc2n1)-c1cnc(OC)c(c1)C(=O)NCc1cc(OC(F)(F)F)ccc1F
COc1ncc(cc1C(=O)NCc1ccccc1OC(F)(F)F)-c1ccc2nc(NC(=O)C(C)C)cn2n1
COc1ncc(cc1C(=O)NCc1ccc(F)c(F)c1OCC1CC1)-c1ccc2nc(NC(=O)C(C)C)cn2n1
COc1ncc(cc1C(=O)NCc1cc(F)cc(F)c1OC1CCOCC1)-c1ccc2nc(NC(=O)C(C)C)cn2n1
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(Cl)c(c1)C(=O)NCc1cc(F)cc(F)c1OCC1CC1
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(Cl)c(c1)C(=O)NCC[C@H](O)c1ccc(Cl)cc1
CC(NC(=O)c1cc(cnc1Cl)-c1ccc2nc(NC(C)=O)cn2n1)c1ccccc1OC(F)(F)F
CC(NC(=O)c1cc(cnc1Cl)-c1ccc2nc(NC(C)=O)cn2n1)c1cc(ccc1F)C(F)(F)F
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(Cl)c(c1)C(=O)NCc1cccc(OC(F)(F)F)c1
CC(Oc1c(F)cc(F)cc1CNC(=O)c1cc(cnc1Cl)-c1ccc2nc(NC(C)=O)cn2n1)C1CCC1
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(Cl)c(c1)C(=O)NCc1cc(ccc1Cl)C(F)(F)F
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(Cl)c(c1)C(=O)NCc1cc(ccc1F)C(F)(F)F
COc1nc(C)c(cc1C(=O)NC(C)c1cc(ccc1F)C(F)(F)F)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NC(C)c1cc(OC(F)(F)F)ccc1F)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCc1cc(F)cc(OC(F)(F)F)c1)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)N(C)Cc1cccc(OC(F)(F)F)c1)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)N(C)Cc1ccccc1OC(F)(F)F)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCc1cc(F)c(F)cc1OCC1CC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCc1c(F)ccc(F)c1OC)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCc1cccc(F)c1OCC1CCC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NC(C)c1cccc(OC(F)(F)F)c1)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NC(C)c1ccccc1OC(F)(F)F)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCc1cc(F)cc(c1)C(F)(F)F)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCc1cc(F)cc(F)c1OCC1CCC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCc1cc(ccc1F)C(F)(F)F)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCc1c(F)cc(F)cc1OCC1CC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCc1cccc(F)c1OCC1CC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCC[C@H](O)c1ccc(Cl)cc1)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCc1ccccc1OC(C)C1CCCC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCCc1cccc(OC(F)(F)F)c1)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCc1cccc(c1)C(F)(F)F)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCc1ccccc1OC1CCOC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCc1c(F)cc(F)cc1OCC1CCCC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCc1cccc(OCC2CC2)c1)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCc1ccccc1OCC1CCC(F)(F)CC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCc1ncccc1OCC1CCCC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCc1cccnc1OCC1CCCC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCc1cccnc1OCC1CCC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCc1cc(F)ccc1OCC1CCCC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCc1ccccc1OCC1CCCC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCc1ccc(F)cc1OCC1CC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCc1ccccc1OCC1CC1)-c1ccc2nc(NC(C)=O)cn2n1
COc1nc(C)c(cc1C(=O)NCc1cccc(OC(F)(F)F)c1)-c1ccc2nc(NC(C)=O)cn2n1
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(cnc1Cl)C(=O)NCc1cc(F)ccc1OC(F)(F)F
COc1nc(C)c(cc1C(=O)NCc1cc(OC(F)(F)F)ccc1F)-c1ccc2nc(NC(=O)COC(C)=O)cn2n1
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(C(=O)NCc2c(F)cccc2OCC(F)(F)F)c(C)nc1C
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(C(=O)NCc2cc(OCC3CC3)ccc2F)c(C)nc1C
CC(=O)OCC(=O)Nc1cn2nc(ccc2n1)-c1cc(C(=O)NCc2cc(OC(F)(F)F)ccc2F)c(C)nc1C
CCc1ncc(cc1C(=O)N[C@H](C)c1cc(OC(F)(F)F)ccc1F)-c1ccc2nc(NC(C)=O)cn2n1 |r|
CCc1ncc(cc1C(=O)NCc1cc(ccc1F)C(F)(F)F)-c1ccc2nc(NC(C)=O)cn2n1
C[C@@H](N(C)C(=O)c1cc(cnc1C)-c1ccc2nc(NC(C)=O)cn2n1)c1cc(OC(F)(F)F)ccc1F |r|
C[C@@H](NC(=O)c1cc(cnc1C)-c1ccc2nc(NC(=O)CN3CCC(CC3)C(F)(F)F)cn2n1)c1cc(ccc1F)C(F)(F)F
C[C@@H](NC(=O)c1cc(cnc1C)-c1ccc2nc(NC(=O)CN3CCN(C)CC3)cn2n1)c1cc(ccc1F)C(F)(F)F
C[C@@H](NC(=O)c1cc(cnc1C)-c1ccc2nc(NC(=O)CN3CCCC3)cn2n1)c1cc(ccc1F)C(F)(F)F
C[C@@H](NC(=O)c1cc(cnc1C)-c1ccc2nc(NC(=O)CN3CCC(F)(F)CC3)cn2n1)c1cc(OC(F)(F)F)ccc1F
C[C@@H](NC(=O)c1cc(cnc1C)-c1ccc2nc(NC(=O)CN3CC(F)(F)C3)cn2n1)c1cc(OC(F)(F)F)ccc1F
C[C@@H](NC(=O)c1cc(cnc1C)-c1ccc2nc(NC(=O)CN3CCN(C)CC3)cn2n1)c1cc(OC(F)(F)F)ccc1F
C[C@@H](NC(=O)c1cc(cnc1C)-c1ccc2nc(NC(=O)CN(C)C)cn2n1)c1cc(OC(F)(F)F)ccc1F
C[C@H](O)C(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)N[C@H](C)c1cc(OC(F)(F)F)ccc1F
CNCC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)N[C@H](C)c1cc(OC(F)(F)F)ccc1F
C[C@@H](NC(=O)c1cc(cnc1C)-c1ccc2nc(NC(=O)CN)cn2n1)c1cc(OC(F)(F)F)ccc1F
C[C@@H](NC(=O)c1cc(cnc1C)-c1ccc2nc(NC(=O)COC(C)=O)cn2n1)c1cc(OC(F)(F)F)ccc1F
Cc1ncc(cc1C(=O)NCC[C@@H](O)c1ccc(Cl)cc1)-c1ccc2nc(NC(=O)CN3CCC(F)(F)CC3)cn2n1
Cc1ncc(cc1C(=O)NCC[C@@H](O)c1ccc(Cl)cc1)-c1ccc2nc(NC(=O)CN3CC(F)(F)C3)cn2n1
CN(C)CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)NCC[C@H](O)c1ccc(Cl)cc1
CC(c1ccc(F)cc1)n1cc(NC(=O)c2cc(cnc2C)-c2ccc3nc(NC(C)=O)cn3n2)cn1
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)Nc1cn(Cc2ccc(Cl)cc2)cn1
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)Nc1cn(Cc2ccc(F)cc2)cn1
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)Nc1cn(Cc2ccccc2)cn1
CN\C=C(/C=N)c1ccc(F)c(CNC(=O)c2cc(cnc2C)-c2ccc3nc(NC(C)=O)cn3n2)c1
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)N1CCCC(C1)C(O)c1ccc(F)cc1
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)NCC(C)(O)Cc1ccc(F)cc1
CC(=O)Nc1cn2nc(ccc2n1)-c1cnc(C)c(c1)C(=O)N1CCCC(O)(Cc2ccc(F)cc2)C1
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(F)c(C)c(c1)C(=O)NCc1cc(ccc1F)-c1cnn(C)c1
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(F)c(C)c(c1)C(=O)NCc1cc(OC(F)(F)F)ccc1F
C[C@H](NC(=O)c1cc(cc(F)c1C)-c1ccc2nc(NC(C)=O)cn2n1)c1cc(OC(F)(F)F)ccc1F |r|
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(F)c(C)c(c1)C(=O)NCc1cccc(OC(F)(F)F)c1F
CN(C)CC(=O)Nc1cn2nc(ccc2n1)-c1cc(F)c(C)c(c1)C(=O)NCC[C@H](O)c1ccc(Cl)cc1 |r|
CNCC(=O)Nc1cn2nc(ccc2n1)-c1cc(F)c(C)c(c1)C(=O)NCC[C@H](O)c1ccc(Cl)cc1 |r|
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(F)c(C)c(c1)C(=O)NCc1ccccc1Oc1ccccc1
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(F)c(C)c(c1)C(=O)NCc1c(F)cccc1C(=O)N1CCC(F)(F)C1
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(F)c(F)c(c1)C(=O)NCc1cc(OC(F)(F)F)ccc1F
C[C@@H](NC(=O)c1cc(cc(F)c1F)-c1ccc2nc(NC(C)=O)cn2n1)c1cc(OC(F)(F)F)ccc1F |r|
CC(=O)Nc1cn2nc(ccc2n1)-c1c(F)c(F)cc(C(=O)NCc2cc(OC(F)(F)F)ccc2F)c1F
CC(=O)Nc1cn2nc(ccc2n1)-c1c(F)c(F)cc(C(=O)NCc2cc(ccc2F)C(F)(F)F)c1F
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(F)cc(c1)C(=O)NCC[C@@H](O)c1ccc(Cl)cc1 |r|
COc1c(F)cc(cc1C(=O)NCc1cc(OC(F)(F)F)ccc1F)-c1ccc2nc(NC(C)=O)cn2n1
COc1c(F)cc(cc1C(=O)NCc1cc(ccc1F)C(F)(F)F)-c1ccc2nc(NC(C)=O)cn2n1
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(cc(F)c1C)C(=O)NCC[C@@H](O)c1ccc(Cl)cc1 |r|
COc1ccc(c(F)c1C(=O)N[C@@H](C)c1cc(OC(F)(F)F)ccc1F)-c1ccc2nc(NC(C)=O)cn2n1 |r|
COc1ccc(c(F)c1C(=O)NCc1cc(F)ccc1C(=O)N1CCC(F)(F)C1)-c1ccc2nc(NC(C)=O)cn2n1
COc1ccc(c(F)c1C(=O)NCc1cccc2CCCOc12)-c1ccc2nc(NC(C)=O)cn2n1
COc1ccc(c(F)c1C(=O)N[C@H](C)c1cc(OC(F)(F)F)ccc1F)-c1ccc2nc(NC(C)=O)cn2n1 |r|
C[C@H](NC(=O)c1c(F)ccc(c1F)-c1ccc2nc(NC(C)=O)cn2n1)c1cc(OC(F)(F)F)ccc1F |r|
C[C@@H](NC(=O)c1c(F)ccc(c1F)-c1ccc2nc(NC(C)=O)cn2n1)c1cc(OC(F)(F)F)ccc1F |r|
CC(=O)Nc1cn2nc(ccc2n1)-c1ccc(F)c(C(=O)NCc2cc(F)ccc2C(=O)N2CCC(F)(F)CC2)c1F
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(C(=O)NCC[C@@H](O)c2ccc(Cl)cc2)c(C)cc1C |r|
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(C(=O)NCC[C@H](O)c2ccc(Cl)cc2)c(C)cc1C |r|
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(C(=O)NCc2cc(cc(Cl)c2F)C(F)(F)F)c(C)cc1C
CC(=O)Nc1cn2nc(ccc2n1)-c1ccc(c(c1)C(=O)NCc1cc(ccc1F)C(F)(F)F)C(F)(F)F
CC(=O)Nc1cn2nc(ccc2n1)-c1ccc(Cl)c(c1)C(=O)NCC[C@@H](O)c1ccc(Cl)cc1 |r|
CC(=O)Nc1cn2nc(ccc2n1)-c1ccc(Cl)c(c1)C(=O)NCc1cc(F)ccc1C(=O)N1CCC(F)(F)C1
C[C@@H](NC(=O)c1c(Cl)ccc(c1F)-c1ccc2nc(NC(C)=O)cn2n1)c1cc(OC(F)(F)F)ccc1F |r|
CC(=O)Nc1cn2nc(ccc2n1)-c1ccc(Cl)c(C(=O)NCc2cc(ccc2F)-c2cnn(C)c2)c1F
CC(=O)Nc1cn2nc(ccc2n1)-c1ccc(Cl)c(C(=O)NCC[C@H](O)c2ccc(Cl)cc2)c1F |r|
CC(=O)Nc1cn2nc(ccc2n1)-c1ccc(Cl)c(C(=O)NCc2ccc(OC(F)(F)F)cc2)c1F
C[C@@H](NC(=O)c1cc(c(F)cc1Cl)-c1ccc2nc(NC(C)=O)cn2n1)c1cc(OC(F)(F)F)ccc1F |r|
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(C(=O)NCc2cc(OC(F)(F)F)ccc2F)c(Cl)cc1C
CC(=O)Nc1cn2nc(ccc2n1)-c1ccc(C)c(c1)C(=O)NCc1cc(OC(F)(F)F)ccc1F
COc1ccc(c(F)c1C(=O)NCC[C@@H](O)c1ccc(Cl)cc1)-c1ccc2nc(NC(C)=O)cn2n1 |r|
C[C@@H](NC(=O)c1cc(ccc1C)-c1ccc2nc(NC(C)=O)cn2n1)c1cc(OC(F)(F)F)ccc1F |r|
CC(=O)Nc1cn2nc(ccc2n1)-c1ccc(C)c(c1)C(=O)NCC[C@@H](O)c1ccc(Cl)cc1 |r|
CC(=O)Nc1cn2nc(ccc2n1)-c1ccc(C)c(c1)C(=O)NCC[C@H](O)c1ccc(Cl)cc1 |r|
CC(=O)Nc1cn2nc(ccc2n1)-c1ccc(C)c(c1)C(=O)NCC(O)COc1ccccc1
CC(=O)Nc1cn2nc(ccc2n1)-c1ccc(C)c(c1)C(=O)NC[C@H]1C[C@@H]1c1ccc(F)cc1 |r|
CC(=O)Nc1cn2nc(ccc2n1)-c1ccc(C)c(c1)C(=O)NCc1c(F)cccc1-c1cnn(C)c1
CC(=O)Nc1cn2nc(ccc2n1)-c1ccc(C)c(c1)C(=O)NCc1cc(F)ccc1-c1cnn(C)c1
CC(=O)Nc1cn2nc(ccc2n1)-c1ccc(C)c(c1)C(=O)NCc1cc(ccc1F)C(=O)N1CC(F)(F)C1
CC(=O)Nc1cn2nc(ccc2n1)-c1ccc(C)c(c1)C(=O)NCc1ccc(F)cc1C(=O)N1CCC(F)(F)C1
CC(=O)Nc1cn2nc(ccc2n1)-c1ccc(C)c(c1)C(=O)NCc1cc(ccc1F)C(=O)N1CCC(C)(C)C1
CC(=O)Nc1cn2nc(ccc2n1)-c1ccc(C)c(c1)C(=O)NCc1cc(F)cc(F)c1C(=O)N1CC[C@H](O)C1 |r|
CC(=O)Nc1cn2nc(ccc2n1)-c1ccc(C)c(c1)C(=O)NCc1cc(F)ccc1C(=O)N1CCCCC1
CC(=O)Nc1cn2nc(ccc2n1)-c1ccc(C)c(C(=O)NCc2cc(ccc2F)-c2cnn(c2)C2CC2)c1F
CC(=O)Nc1cn2nc(ccc2n1)-c1ccc(C)c(C(=O)NCc2cc(F)ccc2-c2cnn(c2)C2CC2)c1F
CC(=O)Nc1cn2nc(ccc2n1)-c1ccc(C)c(C(=O)NCc2ccc(F)c(F)c2C(=O)N2CCC(F)(F)C2)c1F
C[C@@H](NC(=O)c1c(C)ccc(c1F)-c1ccc2nc(NC(C)=O)cn2n1)c1cc(OC(F)(F)F)ccc1F |r|
C[C@@H](NC(=O)c1c(C)ccc(-c2ccc3nc(NC(C)=O)cn3n2)c1F)c1cc(ccc1F)C(F)(F)F |r|
COc1c(F)cc(F)cc1CNC(=O)c1c(C)ccc(c1F)-c1ccc2nc(NC(C)=O)cn2n1
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(C(=O)NCc2cc(ccc2F)C(=O)N2CCCC2(C)C)c(C)cc1F
COc1cc(C)c(cc1C(=O)NCc1cc(OC(F)(F)F)ccc1F)-c1ccc2nc(NC(C)=O)cn2n1
COc1cc(F)c(cc1C(=O)NCc1cc(F)ccc1C(=O)N1CCCC1(C)C)-c1ccc2nc(NC(C)=O)cn2n1
COc1cccc(F)c1CNC(=O)c1cc(c(F)cc1OC)-c1ccc2nc(NC(C)=O)cn2n1
COc1cc(C)c(cc1C(=O)NCc1cc(OC(F)(F)F)ccc1F)-c1ccc2nc(NC(=O)CO)cn2n1
CC(=O)Nc1cn2nc(ccc2n1)-c1cccc(C(=O)NCc2cc(OC(F)(F)F)ccc2F)c1F
CC(=O)Nc1cn2nc(ccc2n1)-c1cccc(C(=O)NCc2cc(ccc2F)C(=O)N2CCC2(C)C)c1F
Fc1ccc(OC(F)(F)F)cc1CNC(=O)c1cccc(c1F)-c1ccc2nc(NC(=O)CN3CCC(F)(F)CC3)cn2n1
Cc1ccc(cc1)[C@H](O)CCNC(=O)c1cccc(c1F)-c1ccc2nc(NC(=O)CN3CCC(CC3)C(F)(F)F)cn2n1 |r|
C[C@H](NC(=O)c1ccc(C)c(c1F)-c1ccc2nc(NC(C)=O)cn2n1)c1cc(OC(F)(F)F)ccc1F |r|
CC(=O)Nc1cn2nc(ccc2n1)-c1c(C)ccc(C(=O)NCc2cc(OC(F)(F)F)ccc2F)c1F
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(ccc1Cl)C(=O)NCc1cc(OC(F)(F)F)ccc1F
CC(=O)Nc1cn2nc(ccc2n1)-c1cc(ccc1F)C(=O)NCc1cc(OC(F)(F)F)ccc1F
CN1c2cc(CCC(=O)N3CCCC3)ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O
CN1c2cc(ccc2OCC(NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O)C#CC(C)(C)O
CN1c2cc(ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CC(C)(C)C
CN1c2ccc(CN3CCn4nc(nc4C3)C(F)(F)F)cc2OCC(NC(=O)c2ncn(Cc3ccccc3)n2)C1=O |$;;;;;;;;;;;;;;;;C;;;;;;;;;;;;;;;;;;;;;;;;;$|
COC(=O)C(C)(C)C#Cc1ccc2OCC(NC(=O)c3n[nH]c(Cc4ccccc4)n3)C(=O)N(C)c2c1
CN1c2cc(ccc2OCC(NC(=O)c2ccn(Cc3ccccc3)n2)C1=O)C#CC(C)(C)O
CN1c2cc(ccc2OCC(NC(=O)c2cc(Cc3ccccc3)on2)C1=O)C#CC(C)(C)O
CN1c2cc(ccc2OCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CCN1CCCC1
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3cccc(F)n3)cn2)C1=O)C#CC(C)(C)O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3cccc(C)n3)cn2)C1=O)C#CC(C)(C)O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccc(C)nc3)ccn2)C1=O)C#CC1(O)COC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccc(C)nc3)ccn2)C1=O)C#CC(C)(C)O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccc(F)nc3)ccn2)C1=O)C#CC1(O)COC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccc(F)nc3)ccn2)C1=O)C#CC(C)(C)O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Cc3cccc(F)n3)ccn2)C1=O)C#CC1(O)COC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3ccccn3)cn2)C1=O)C#CC(C)(C)O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3cccc(n3)C(F)(F)F)cn2)C1=O)C#CC(C)(C)O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Cc3cccc(O)n3)ccn2)C1=O)C#CC1(O)COC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Cc3cccc(C)n3)ccn2)C1=O)C#CC(C)(C)O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Cc3cccc(C)n3)ccn2)C1=O)C#CC1(O)COC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Cc3cccc(F)n3)ccn2)C1=O)C#CC(C)(C)O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3cccnc3)cn2)C1=O)C#CC(C)(C)O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3ccc(C)nc3)cn2)C1=O)C#CC(C)(C)O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3ccc(F)nc3)cn2)C1=O)C#CC(C)(C)O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3cccnn3)cn2)C1=O)C#CC(C)(C)O |r|
CN1c2cc(Br)ccc2OC[C@H](NC(=O)n2cc(Cc3ccccn3)cn2)C1=O |r|
CN1c2cc(Br)ccc2OC[C@H](NC(=O)n2cc(Cc3cccc(C)n3)cn2)C1=O |r|
CN1c2cc(Br)ccc2OC[C@H](NC(=O)n2cc(Cc3cccc(F)n3)cn2)C1=O |r|
CN1c2cc(Br)ccc2OC[C@H](NC(=O)n2cc(Cc3cccc(n3)C(F)(F)F)cn2)C1=O |r|
CN1c2cc(Br)ccc2OC[C@H](NC(=O)n2cc(Cc3cccnc3)cn2)C1=O |r|
CN1c2cc(Br)ccc2OC[C@H](NC(=O)n2cc(Cc3ccc(C)nc3)cn2)C1=O |r|
CN1c2cc(Br)ccc2OC[C@H](NC(=O)n2cc(Cc3ccc(F)nc3)cn2)C1=O |r|
CN1c2cc(Br)ccc2OC[C@H](NC(=O)n2cc(Cc3cccnn3)cn2)C1=O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Cc3cccnc3F)ccn2)C1=O)C#CC1(O)COC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Cc3cccnc3F)ccn2)C1=O)C#CC(C)(C)O |r|
CN1c2cc(Br)ccc2OC[C@H](NC(=O)n2cc(Cc3ccncc3)cn2)C1=O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3ccncc3)cn2)C1=O)C#CC(C)(C)O |r|
CN1c2cc(Br)ccc2OC[C@H](NC(=O)n2cc(Cc3ncccn3)cn2)C1=O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3ncccn3)cn2)C1=O)C#CC(C)(C)O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3cccc(F)n3)cn2)C1=O)C#CC1(O)COC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3cccc(F)n3)cn2)C1=O)C#CC1(O)CCOCC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3cccc(F)n3)cn2)C1=O)C#CC1CCOCC1 |r|
CN1c2cc(Br)ccc2CC[C@H](NC(=O)n2cc(Cc3cccc(F)n3)cn2)C1=O |r|
CN1c2cc(ccc2CC[C@H](NC(=O)n2cc(Cc3cccc(F)n3)cn2)C1=O)C#CC1(O)COC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3cccc(F)n3)cn2)C1=O)C#CC(C)(C)CO |r|
CN1c2cc(ccc2CC[C@H](NC(=O)n2cc(Cc3cccc(F)n3)cn2)C1=O)C#CC(C)(C)O |r|
CN1c2cc(ccc2CC[C@H](NC(=O)n2cc(Cc3cccc(F)n3)cn2)C1=O)C#CC(C)(C)CO |r|
CN1c2cc(ccc2CC[C@H](NC(=O)n2cc(Cc3cccc(F)n3)cn2)C1=O)C#CC1(O)CCOCC1 |r|
CN1c2cc(Br)ccc2OC[C@H](NC(=O)n2cc(Cc3cccnc3F)cn2)C1=O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3cccnc3F)cn2)C1=O)C#CC(C)(C)O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3cccnc3F)cn2)C1=O)C#CC1(O)CCOCC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3cccnc3F)cn2)C1=O)C#CC1CCOCC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3cccnc3F)cn2)C1=O)C#CC(C)(C)CO |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3cccnc3F)cn2)C1=O)C#CC1(O)COC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3cccnc3F)cn2)C1=O)C#CC1(O)CCC1 |r|
CN1c2cc(Br)ccc2OC[C@H](NC(=O)n2cc(Cc3ccc(F)nc3F)cn2)C1=O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3ccc(F)nc3F)cn2)C1=O)C#CC(C)(C)O |r|
CN1c2cc(ccc2OC[C@H](N2CCc3c(Cl)n(Cc4ccccc4)nc3C2=O)C1=O)C#CC(C)(C)O
CN1c2cc(ccc2OC[C@H](N2CCc3c(Cl)n(Cc4ccccc4)nc3C2=O)C1=O)C#CC(C)(C)C
CN1c2ccc(cc2OC[C@H](N2CCc3c(Cl)n(Cc4ccccc4)nc3C2=O)C1=O)C#CC1(O)CCCC1
CN1c2ccc(cc2OC[C@H](N2CCc3c(Cl)n(Cc4ccccc4)nc3C2=O)C1=O)C#Cc1ccncc1
CN1c2ccc(cc2OC[C@H](N2CCc3c(Cl)n(Cc4ccccc4)nc3C2=O)C1=O)C#Cc1cccnc1
CN1c2ccc(cc2OC[C@H](N2CCc3c(Cl)n(Cc4ccccc4)nc3C2=O)C1=O)C#Cc1ccccn1
CN1c2ccc(cc2OC[C@H](N2CCc3c(Cl)n(Cc4ccccc4)nc3C2=O)C1=O)C#CCOC(C)(C)C
CN1c2ccc(cc2OC[C@H](N2CCc3c(Cl)n(Cc4ccccc4)nc3C2=O)C1=O)C#CC1(O)COC1
COCC#Cc1ccc2N(C)C(=O)[C@H](COc2c1)N1CCc2c(Cl)n(Cc3ccccc3)nc2C1=O
COC(C)(C)C#Cc1ccc2N(C)C(=O)[C@H](COc2c1)N1CCc2c(Cl)n(Cc3ccccc3)nc2C1=O
CN1c2ccc(cc2OC[C@H](N2Cc3c(Cl)n(Cc4ccccc4)nc3C2=O)C1=O)C#CC(C)(C)O
CN1c2ccc(cc2OC[C@H](N2CCc3c(Cl)n(Cc4ccccc4)nc3C2=O)C1=O)C#CC(C)(C)CO
CN1c2ccc(cc2OC[C@H](N2Cc3c(Cl)n(Cc4ccccc4)nc3C2=O)C1=O)C#Cc1cccc(n1)C(F)(F)F
CN1c2ccc(cc2OC[C@H](N2Cc3c(Cl)n(Cc4ccccc4)nc3C2=O)C1=O)C#Cc1ccccn1
CN1c2ccc(cc2OC[C@H](N2CCc3c(Cl)n(Cc4ccccc4)nc3C2=O)C1=O)C#Cc1cccc(n1)C#N
CN1c2cc(ccc2OC[C@H](N2Cc3c(Cl)n(Cc4ccccc4)nc3C2=O)C1=O)N1CC2(C1)CCOCC2
CN1c2cc(ccc2OC[C@H](N2CCc3c(Cl)n(Cc4ccccc4)nc3C2=O)C1=O)N1CC2(C1)CCOCC2
CN1c2cc(ccc2OC[C@H](N2CCc3c(Cl)n(Cc4ccccc4)nc3C2=O)C1=O)C#Cc1ccccn1
CN1c2cc(ccc2OC[C@H](N2CCc3c(Cl)n(Cc4ccccc4)nc3C2=O)C1=O)C#CCO
CN1c2cc(ccc2OC[C@H](N2CCc3c(Cl)n(Cc4ccccc4)nc3C2=O)C1=O)C#CC1CCCN1
CN1c2cc(ccc2OC[C@H](N2CCc3c(Cl)n(Cc4ccccc4)nc3C2=O)C1=O)C#Cc1cccc(C)n1
CN1c2ccc(cc2OC[C@H](N2CCc3c(Cl)n(Cc4ccccc4)nc3C2=O)C1=O)C#Cc1cccc(n1)C(F)(F)F
CN1c2ccc(cc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)N1CCC2(CCOCC2)CC1
CN1c2cc(ccc2CC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)-c1ccc(nc1)C#CC(C)(C)O
O=C(NC1CCc2ccc(cc2NC1=O)N1CC2(C1)CCOCC2)c1n[nH]c(Cc2ccccc2)n1
CN1c2cc(ccc2CCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)N1CCN2CCC1CC2 |(-3.01,2.04,;-2.67,.53,;-3.88,-.43,;-5.21,.34,;-6.54,-.43,;-6.54,-1.97,;-5.21,-2.74,;-3.88,-1.97,;-2.67,-2.93,;-1.17,-2.58,;-.5,-1.2,;1.04,-1.2,;1.81,.14,;1.04,1.47,;3.35,.14,;4.25,-1.11,;5.72,-.63,;5.72,.91,;6.96,1.81,;8.37,1.19,;9.62,2.09,;11.02,1.46,;11.18,-.07,;9.94,-.97,;8.53,-.35,;4.25,1.38,;-1.17,.19,;-.21,1.39,;-7.88,.34,;-7.76,1.88,;-8.89,2.93,;-10.41,2.7,;-9.18,2.07,;-8.67,.78,;-9.15,-.52,;-10.62,-.07,;-11.18,1.36,)|
CN1c2cc(ccc2CCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)N1CC2(C1)CCCCC2
CN1c2cc(ccc2CCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)N1CCC2(CCOCC2)CC1
CN1c2cc(ccc2CCC(NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)N1CC2(C1)CCOCC2
CN1c2cc(ccc2CC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)N1CC2(C1)CCOCC2
CN1c2cc(ccc2CCC(NC(=O)n2cc(Cc3ccccc3)cn2)C1=O)N1CC2(C1)CCOCC2
CN1c2cc(ccc2CCC(NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)N1CCC2(CCOCC2)CC1
CN1c2cc(ccc2CCC(NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)N1CC2(C1)CCOCC2
CN1c2cc(ccc2CCC(NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)N1CC2(C1)CCCCC2
CN1c2cc(ccc2CC[C@H](NC(=O)c2ccn(Cc3ccccc3)n2)C1=O)N1CC2(C1)CCOCC2
CN1c2cc(ccc2OC[C@H](NC(=O)n2cc(Cc3ccccc3)cn2)C1=O)N1CC2(C1)CCOCC2
CN1CCC2(CC1)CCN(CC2)c1ccc2OC[C@H](NC(=O)n3cc(Cc4ccc(F)cc4)cn3)C(=O)N(C)c2c1
CN1c2ncc(cc2OC[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O)C#CC(C)(C)O |r|
C[C@H]1Oc2cccnc2N(C)C(=O)[C@H]1N1CCc2c(Cl)n(Cc3ccccc3)nc2C1=O |r|
CN1c2ncc(cc2OC[C@H](NC(=O)c2nnc(Cc3ccccc3)o2)C1=O)C#CCN1CCOCC1 |r|
CN1c2ncc(Br)cc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O |r|
CN1c2ncc(cc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC(C)(C)O |r|
CN1c2ncc(cc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC(C)(C)CO |r|
CN1c2ncc(cc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#Cc1ccccn1 |r|
C[C@H]1Oc2cc(Br)cnc2N(C)C(=O)[C@H]1N1CCc2c(Cl)n(Cc3ccccc3)nc2C1=O |r|
CCOC(=O)c1nn(Cc2ccccc2)c(Cl)c1CCN[C@H]1[C@@H](C)Oc2cc(cnc2N(C)C1=O)C#N |r|
CN1c2nc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)N1CCC2(C1)CCOCC2 |r|
CN1c2nc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)N1CC2(C1)CCOCC2 |r|
CN1c2nccc(C#CC(C)(C)O)c2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O |r|
CN1c2nccc(C#CC3(O)COC3)c2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O |r|
CN1c2nccc(C#CC3(O)CCOCC3)c2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O |r|
CN1c2nc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC1(O)COC1 |r|
CN1c2nc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC(C)(C)O |r|
CN1c2nc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccc(F)cc3)ccn2)C1=O)C#CC1(O)COC1 |r|
CN1c2nc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC1(F)COC1 |r|
CN1c2nc(ccc2OC[C@H](NC(=O)c2cc(Oc3cccc(F)c3)ccn2)C1=O)C#CC(C)(C)O |r|
CN1c2nc(ccc2OC[C@H](NC(=O)c2cc(Oc3cccc(F)c3)ccn2)C1=O)C#CC1(O)COC1 |r|
CN1c2nc(ccc2OC[C@H](NC(=O)c2cc(Oc3cccc(F)c3)ccn2)C1=O)C#CC1(F)COC1 |r|
CN1c2nc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CC(C)(C)O |r|
CN1c2nc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CC1(O)COC1 |r|
CN1c2nc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3F)ccn2)C1=O)C#CC(C)(C)O |r|
CN1c2nc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC1(O)CC(F)(F)C1 |r|
CN1c2nc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC(C)(C)CO |r|
CN1c2nc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC(C)(C)C(F)F |r|
CN1c2nc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC(O)C(F)(F)F |r|
CN1c2nc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3F)n2)C1=O)C#CC(C)(C)O |r|
CN1c2nc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccc(F)cc3)n2)C1=O)C#CC(C)(C)O |r|
CN1c2nc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CC1(O)CC(F)(F)C1 |r|
CN1c2nc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CC(O)C(F)(F)F |r|
CN1c2nc(ccc2OC[C@H](NC(=O)c2nn(Cc3ccc(F)cc3)cc2F)C1=O)C#CC(C)(C)O |r|
CN1c2nc(ccc2OC[C@H](NC(=O)c2cc(Oc3cccc(F)c3)ccn2)C1=O)C#C |r|
CN1c2nc(ccc2OC[C@H](NC(=O)c2nn(Cc3ccc(F)cc3)cc2F)C1=O)C#C |r|
CC#Cc1ccc2OC[C@H](NC(=O)c3nn(Cc4ccc(F)cc4)cc3F)C(=O)N(C)c2n1 |r|
CC#Cc1ccc2OC[C@H](NC(=O)c3nn(Cc4cccc(F)n4)cc3F)C(=O)N(C)c2n1 |r|
CN1c2nc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC(C)(O)C(F)(F)F |r|
CN1c2nc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC1COC1 |r|
CN1c2nc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC(F)(F)C1COC1 |r|
CN1c2nc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC(C)(N)C(F)(F)F |r|
CN1c2nc(ccc2OC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC1CCOCC1 |r|
CN1c2ncc(Br)cc2CCC(NC(=O)c2cc(Oc3ccc(F)cc3)ccn2)C1=O |w:11.12|
CN1c2ncc(cc2CCC(NC(=O)c2cc(Oc3ccc(F)cc3)ccn2)C1=O)C#CC(C)(C)O
CN1c2ncc(CN3CC4(C3)CCOCC4)cc2CCC(NC(=O)c2cc(Oc3ccc(F)cc3)ccn2)C1=O
COc1ccc2CC[C@H](NC(=O)c3cc(Oc4ccccc4)ccn3)C(=O)N(C)c2n1 |r|
CN1c2nc(ccc2CC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC(C)(C)O |r|
CN1c2nc(ccc2CC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC1(O)COC1 |r|
CN1c2nc(ccc2CC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CC(C)(C)O |r|
CN1c2nc(ccc2CC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC(O)C(F)(F)F |r|
CN1c2nc(ccc2CC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC(C)(O)C(F)(F)F |r|
CN1c2nc(ccc2CC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC1(O)CC(F)(F)C1 |r|
CN1c2nc(ccc2CC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC1COC1 |r|
CN1c2nc(ccc2CC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC(F)(F)C1COC1 |r|
CN1c2nc(ccc2CC[C@H](NC(=O)c2cc(Oc3ccccc3)ccn2)C1=O)C#CC(C)(N)C(F)(F)F |r|
FC1(F)CN(C1)C(=O)c1cc2C(OCCn2n1)c1ccccc1
Fc1ccccc1C1OCCn2nc(cc12)C(=O)N1CC(F)(F)C1
FC(F)[C@@H]1CCN1C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
FC(F)CN(C1COC1)C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1 |r|
FC(F)[C@H]1CCCN1C(=O)c1nc2[C@H](F)C[C@H](c3ccccc3)n2n1 |r|
C[C@H]1[C@H](CCN1C(=O)c1nc2[C@@H](F)C[C@@H](c3ccccc3)n2n1)C(F)(F)F |r|
CC(CCNC(=O)c1cccc(c1)-c1ccc2c(N)ncnn12)c1ccccc1
CC(CCNC(=O)c1cccc(c1)-c1cc(c2c(N)ncnn12)C(F)(F)F)c1ccccc1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(F)c(c1)C(=O)Nc1cnn(Cc2ccccc2)c1
Nc1ncnn2c(c(F)cc12)-c1cccc(c1)C(=O)NCc1ccccc1Oc1ccccc1
Nc1ncnn2c(cc(C#N)c12)-c1cccc(c1)C(=O)NCCC(O)c1ccccc1
Nc1ncnn2c(cc(C#N)c12)-c1cccc(c1)C(=O)Nc1cnn(Cc2ccccc2)c1
CC(CCNC(=O)c1cccc(c1)-c1cc(C#N)c2c(N)ncnn12)c1ccccc1
COc1ncc(cc1C(=O)Nc1cnn(Cc2ccccc2)c1)-c1cc(F)c2c(N)ncnn12
COc1ncc(cc1C(=O)NCC[C@H](O)c1ccc(Cl)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1ncc(cc1C(=O)NC1CCN(C1)C(=O)OC(C)(C)C)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CCN(C1)C(=O)c1ccc(C)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)NCCC(O)(c1ccccc1)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@H]1CN(C[C@H]1C)C(=O)c1ccccc1)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1ncc(cc1C(=O)NC1CN(CC1C)C(=O)CC(C)(C)C)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@H]1CN(C[C@H]1C)C(=O)C1CCCCC1)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cnc(F)c(c1)C(=O)NCC[C@H](O)c1ccc(Cl)cc1 |r|
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cncc(c1)C(=O)NCCC(O)c1ccc(F)cc1
COc1ncc(cc1C(=O)NC1CN(C[C@@H]1C)C(=O)C1CCCC1)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1nc(C)c(cc1C(=O)NCC[C@H](O)c1ccc(Cl)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
C[C@H]1CN(CC1NC(=O)c1cc(cnc1C)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(=O)C1CCCCC1 |r|
Cc1ncc(cc1C(=O)NC1CN(C[C@@H]1CF)C(=O)C1CCC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
C[C@H]1CN(CC1NC(=O)c1cc(cnc1C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(=O)C1CCC(F)(F)C1 |r|
C[C@H]1CN(CC1NC(=O)c1cc(cnc1C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(=O)C1CCC(F)(F)CC1 |r|
Cc1ncc(cc1C(=O)NC1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)CC1)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
Nc1ncc(cc1C(=O)NCC[C@@H](O)c1ccc(Cl)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1ncc(cc1C(=O)NC1CN(C[C@@H]1F)C(=O)C1CCC(F)CC1)-c1cc(c2c(N)ncnn12)C(F)(F)F |r,wU:15.17,(.44,-3.61,;.44,-2.07,;-.89,-1.3,;-2.22,-2.07,;-3.56,-1.3,;-3.56,.24,;-2.22,1.01,;-.89,.24,;.44,1.01,;.44,2.55,;1.78,.24,;3.11,1.01,;4.52,.38,;5.55,1.52,;4.78,2.86,;3.27,2.54,;2.13,3.57,;7.08,1.36,;7.99,2.61,;7.71,-.04,;6.8,-1.29,;7.43,-2.7,;8.96,-2.86,;9.59,-4.26,;9.86,-1.61,;9.24,-.2,;-4.89,1.01,;-5.05,2.54,;-6.56,2.86,;-7.33,1.52,;-8.83,1.2,;-9.86,2.35,;-9.31,-.26,;-8.28,-1.41,;-6.77,-1.09,;-6.3,.38,;-7.18,4.26,;-6.28,5.51,;-8.72,4.43,;-7.81,5.67,)|
CO[C@H](CCNC(=O)c1cc(cnc1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F)c1ccc(Cl)cc1 |r|
CO[C@@H](CCNC(=O)c1cc(cnc1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F)c1ccc(Cl)cc1 |r|
CNc1ncc(cc1C(=O)NCC[C@H](O)c1ccc(Cl)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1ncc(cc1C(=O)NC1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1ncc(cc1C(=O)NCC[C@H](O)c1ccc(Cl)cc1)-c1cc(Cl)c2c(N)ncnn12 |r|
COc1ncc(cc1C(=O)Nc1cnn(Cc2ccccc2)c1)-c1cc(Cl)c2c(N)ncnn12
COc1ncc(cc1C(=O)NC1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
CC(C)(C)n1cc(NC(=O)c2cc(cnc2N)-c2cc(c3c(N)ncnn23)C(F)(F)F)cn1
COc1ncc(cc1C(=O)NCC[C@@H](O)c1ccc(Cl)cc1)-c1cc(Cl)c2c(N)ncnn12 |r|
COc1ncc(cc1C(=O)NC1CN(CC1F)C(=O)C1CC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)C1=C[C@H](NC1)C(=O)NCc1cc(OC(F)(F)F)ccc1F |r,t:16|
COc1ncc(cc1C(=O)NCC[C@H](O)c1ccc(Cl)cc1)-c1cc(C)c2c(N)ncnn12 |r|
COc1ncc(cc1C(=O)NC1CN(CC2CCCCC2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)NC1CN(C[C@@H]1F)C(=O)c1ccc(F)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1ncc(cc1C(=O)Nc1cnn(Cc2ccccc2)c1)-c1cc(C)c2c(N)ncnn12
COc1ncc(cc1C(=O)NC1CN(C[C@@H]1F)C(=O)c1ccc(F)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1ncc(cc1C(=O)NC1CN(CC(O)C(F)(F)F)C[C@@H]1F)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1ncc(cc1C(=O)N[C@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1nc(C)c(cc1C(=O)NC1CN(C[C@@H]1F)C(=O)c1ccc(F)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1ncc(cc1C(=O)Nc1cnn(CC(C)(C)C)c1)-c1cc(Cl)c2c(N)ncnn12
COc1ncc(cc1C(=O)Nc1cnn(CC(C)(C)C)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COCc1cc(-c2cnc(OC)c(c2)C(=O)Nc2cnn(Cc3ccccc3)c2)n2ncnc(N)c12
COCc1cc(-c2cnc(O)c(c2)C(=O)NCC[C@H](O)c2ccc(Cl)cc2)n2ncnc(N)c12 |r|
COc1ncc(cc1C(=O)Nc1cnn(Cc2ccccc2)c1)-c1cc(CO)c2c(N)ncnn12
Nc1ncnn2c(cc(CO)c12)-c1cnc(O)c(c1)C(=O)NCC[C@H](O)c1ccc(Cl)cc1 |r|
OCCNc1ncnn2c(ccc12)-c1cnc(O)c(c1)C(=O)NCC[C@H](O)c1ccc(Cl)cc1 |r|
COc1ncc(cc1C(=O)Nc1cnn(Cc2ccccc2)c1)-c1ccc2c(NCCO)ncnn12
COCCNc1ncnn2c(ccc12)-c1cnc(OC)c(c1)C(=O)Nc1cnn(Cc2ccccc2)c1
Nc1ncnn2c(cc(CNCCO)c12)-c1cnc(O)c(c1)C(=O)NCC[C@H](O)c1ccc(Cl)cc1 |r|
COc1ncc(cc1C(=O)Nc1cnn(Cc2ccccc2)c1)-c1cc(CNCCO)c2c(N)ncnn12
Nc1ncnn2c(ccc12)-c1cccc(c1)C(=O)NCCC(O)c1ccccc1
Nc1ncnn2c(ccc12)-c1cccc(c1)C(=O)Nc1cnn(Cc2ccccc2)c1
COc1ncc(cc1C(=O)NCCC(C)c1ccccc1)-c1c(F)cc2c(N)ncnn12
COc1ncc(cc1C(=O)Nc1cnn(Cc2ccccc2)c1)-c1c(F)cc2c(N)ncnn12
COc1ccc(cc1C(=O)Nc1cnn(Cc2ccccc2)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(F)c2c(N)ncnn12 |r|
Cc1cc(F)c(cc1C(=O)NC1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1ncc(cc1C(=O)NCC[C@H](O)c1ccc(Cl)cc1)-c1cc(C(=O)NCCNC(C)=O)c2c(N)ncnn12 |r|
CC(CCNC(=O)c1cccc(c1)-c1c(F)cc2c(N)ncnn12)c1ccccc1
Nc1ncnn2c(c(F)cc12)-c1cccc(c1)C(=O)NCCC(O)c1ccccc1
Nc1ncnn2c(c(F)cc12)-c1cccc(c1)C(=O)Nc1cnn(Cc2ccccc2)c1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(c1)C(=O)NCCC(O)c1ccccc1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(c1)C(=O)NCC[C@@H](O)c1ccc(Cl)cc1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(c1)C(=O)NCCC(O)c1ccc(F)cc1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(c1)C(=O)Nc1cnn(CC2CC2)c1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(C(=O)Nc2cnn(Cc3ccccc3)c2)c1C(=O)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(c1)C(=O)NCC[C@H](O)c1ccc(Cl)cc1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(c1)C(=O)N[C@H]1CCN(Cc2ccccc2)C1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(c1)C(=O)N[C@H]1CCN(C1)C(=O)c1ccccc1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(c1)C(=O)N[C@H]1CCCN(Cc2ccccc2)C1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(c1)C(=O)N1CCC[C@H](Cc2ccc(F)cc2)C1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(c1)C(=O)N1CCC[C@@H](Cc2ccc(F)cc2)C1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1(O)CCOCC1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccc(F)c(F)c1
CC(C)(O)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cccc(c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
CC(C)(CF)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cccc(c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
CC(C)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cccc(c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
CC(C)(C)CC(=O)N1C[C@H](F)[C@@H](C1)N(C(=O)c1cccc(c1)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(=O)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccccc1F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1cccc(F)c1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1(F)CCC1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1c(F)cncc1F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1(CCC1)C(F)(F)F
CC(C)(F)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cccc(c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1(F)CC1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(c1)C(=O)N([C@@H]1CN(C[C@@H]1F)C(=O)CC(F)(F)F)C(=O)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(c1)C(=O)N([C@@H]1CN(C[C@@H]1F)C(=O)C1(CCCC1)C(F)(F)F)C(=O)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@H]1C[C@H](F)C1 |wU:31.34,wD:23.25,27.31,33.37,(6.12,3.85,;6.12,2.31,;7.45,1.54,;7.45,,;6.12,-.77,;4.79,,;3.32,-.48,;2.42,.77,;3.32,2.02,;4.79,1.54,;2.85,3.48,;2.37,4.95,;4.31,3.96,;1.38,3,;2.85,-1.94,;3.88,-3.09,;3.4,-4.55,;1.89,-4.87,;.86,-3.73,;1.34,-2.26,;-.64,-4.05,;-1.67,-2.9,;-1.12,-5.51,;-2.62,-5.83,;-3.25,-7.24,;-4.78,-7.08,;-5.1,-5.57,;-3.77,-4.8,;-3.61,-3.27,;-5.81,-8.22,;-7.32,-7.9,;-5.34,-9.69,;-4.09,-10.59,;-5,-11.84,;-4.76,-13.36,;-6.24,-10.93,)|
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@H]1C[C@H](F)C1 |wU:31.34,33.37,wD:23.25,27.31,(6.12,3.85,;6.12,2.31,;7.45,1.54,;7.45,,;6.12,-.77,;4.79,,;3.32,-.48,;2.42,.77,;3.32,2.02,;4.79,1.54,;2.85,3.48,;2.37,4.95,;4.31,3.96,;1.38,3,;2.85,-1.94,;3.88,-3.09,;3.4,-4.55,;1.89,-4.87,;.86,-3.73,;1.34,-2.26,;-.64,-4.05,;-1.67,-2.9,;-1.12,-5.51,;-2.62,-5.83,;-3.25,-7.24,;-4.78,-7.08,;-5.1,-5.57,;-3.77,-4.8,;-3.61,-3.27,;-5.81,-8.22,;-7.32,-7.9,;-5.34,-9.69,;-6.24,-10.93,;-5,-11.84,;-4.76,-13.36,;-4.09,-10.59,)|
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)CC1 |wU:27.31,23.25,(-8.42,-4.35,;-8.42,-2.81,;-9.75,-2.04,;-9.75,-.5,;-8.42,.27,;-7.08,-.5,;-5.62,-.02,;-4.71,-1.27,;-5.62,-2.51,;-7.08,-2.04,;-5.14,-3.98,;-6.23,-5.07,;-4.74,-5.46,;-3.66,-4.38,;-5.14,1.44,;-6.17,2.59,;-5.7,4.05,;-4.19,4.37,;-3.16,3.23,;-3.64,1.76,;-1.65,3.55,;-1.18,5.01,;-.62,2.4,;.88,2.72,;2.03,1.69,;3.36,2.46,;3.04,3.97,;1.51,4.13,;.74,5.46,;4.77,1.84,;4.93,.31,;6.01,2.74,;5.85,4.27,;7.1,5.18,;8.51,4.55,;9.75,5.46,;8.67,3.02,;7.42,2.12,)|
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccc(F)cc1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)CC1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)C1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC1(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1
COc1ncc(cc1C(=O)NCCC(C)c1ccccc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)Nc1cnn(Cc2ccccc2)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NCCCOCC(C)C)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NCCCOC(C)(C)C)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NCCCOc1ccc(F)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)Nc1cnn(CC2CC2)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)Nc1cnn(CC(F)(F)F)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NCCC(O)c1ccccc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC[C@H]1C[C@@H]1c1cc(cc(c1)C(F)(F)F)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@H]1CCN(Cc2ccccc2)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CCN(Cc2ccccc2)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@H]1CCN(C1)C(=O)c1ccccc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N1CCC[C@@H](Cc2ccc(F)cc2)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N1CCC[C@H](Cc2ccc(F)cc2)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N1CCC(Cc2ccccc2)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NCCC(O)c1ccc(F)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NCC1CCCOC1c1ccccc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N1CCCC(Cc2cccc(F)c2)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N1CCCC(Cc2ccc(C)cc2)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ccc(CC2CCCN(C2)C(=O)c2cc(cnc2OC)-c2cc(c3c(N)ncnn23)C(F)(F)F)cc1
COc1ncc(cc1C(=O)N1CCCC(Cc2ccc(Cl)cc2)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N1CCC[C@@H](Cc2cccc(F)c2)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NCCC(O)c1ccc(F)c(F)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CCN(Cc2ccccc2)C1=O)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2ccccc2)C(=O)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N1CCC(F)(F)C(Cc2ccccc2)C1)-c1cc(c2c(N)nc(nn12)C(=O)C(F)(F)F)C(F)(F)F
COc1ncc(cc1C(=O)N1CCOC(Cc2ccccc2)C1)-c1cc(c2c(NC(=O)C(F)(F)F)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NCC[C@@H](O)c1ccc(Cl)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NCCC(O)(c1ccccc1)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NCCNc1ccccc1C)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)Nc1cnn(c1)C(C)(C)C)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NCCC(C)(O)c1ccc(Cl)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NCCC(O)(C(C)C)c1ccc(Cl)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCC(O)(CCNC(=O)c1cc(cnc1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F)c1ccc(Cl)cc1
COc1ncc(cc1C(=O)NCCC(=O)c1ccc(Cl)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NCCC(=O)c1ccc(F)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N1CCCN(Cc2ccccc2)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NCCC(C)c1ccccc1)-c1ccc2c(N)ncnn12
COc1ncc(cc1C(=O)NCCC(O)c1ccccc1)-c1ccc2c(N)ncnn12
COc1ncc(cc1C(=O)Nc1cnn(Cc2ccccc2)c1)-c1ccc2c(N)ncnn12
COc1ncc(cc1C(=O)N([C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)C(=O)C(F)(F)F)-c1ccc2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCOCC1)-c1ccc2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC1(F)F)-c1ccc2c(N)ncnn12
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)C1 |wD:23.25,27.31,(6.12,3.85,;6.12,2.31,;7.45,1.54,;7.45,,;6.12,-.77,;4.79,,;3.32,-.48,;2.42,.77,;3.32,2.02,;4.79,1.54,;2.85,3.48,;2.37,4.95,;4.31,3.96,;1.38,3,;2.85,-1.94,;3.88,-3.09,;3.4,-4.55,;1.89,-4.87,;.86,-3.73,;1.34,-2.26,;-.64,-4.05,;-1.67,-2.9,;-1.12,-5.51,;-2.62,-5.83,;-3.25,-7.24,;-4.78,-7.08,;-5.1,-5.57,;-3.77,-4.8,;-3.61,-3.27,;-5.81,-8.22,;-7.32,-7.9,;-5.34,-9.69,;-3.93,-10.31,;-4.56,-11.72,;-4,-13.16,;-5.96,-11.09,)|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)CC1)-c1ccc2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccc(F)cc1)-c1ccc2c(N)ncnn12
CC(CCC(C)(C)C)c1ccccc1 |w:4.5,4.6|
CC(C)(C)CCC(O)c1ccccc1 |w:1.1,1.2|
CC(C)(C)Cc1ccccc1Oc1ccccc1 |w:1.1,1.2|
CC(C)(C)Cc1ccccc1OCC1CC1 |w:1.1,1.2|
CC(C)(C)Cc1nccnc1Cl |w:1.1,1.2|
Cc1ncc(cc1C(=O)NCC[C@@H](O)c1ccc(Cl)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)Nc1cnn(Cc2ccccc2)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)NCCC(O)c1ccccc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)NCCC(O)c1ccc(F)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)NCC[C@H](O)c1ccc(Cl)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)Nc1cnn(CC2CC2)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
CC(CCNC(=O)c1cncc(c1)-c1cc(c2c(N)ncnn12)C(F)(F)F)c1ccccc1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cncc(c1)C(=O)N1CCC[C@@H](Cc2ccc(F)cc2)C1 |r|
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cncc(c1)C(=O)N1CCC[C@@H](Cc2cccc(F)c2)C1 |r|
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cncc(c1)C(=O)N1CCC[C@H](Cc2ccc(F)cc2)C1 |r|
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cncc(c1)C(=O)N1CCC[C@H](Cc2cccc(F)c2)C1 |r|
Cc1ncc(cc1C(=O)Nc1cnn(CC(F)(F)F)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
CO[C@@H](CCNC(=O)c1cc(cnc1C)-c1cc(c2c(N)ncnn12)C(F)(F)F)c1ccc(Cl)cc1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cnc(c(c1)C(=O)NCC[C@H](O)c1ccc(Cl)cc1)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cnc(c(c1)C(=O)NCC[C@@H](O)c1ccc(Cl)cc1)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cnc(c(c1)C(=O)N1CCC[C@@H](Cc2ccc(F)cc2)C1)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cnc(c(c1)C(=O)N1CCC[C@H](Cc2ccc(F)cc2)C1)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cnc(c(c1)C(=O)Nc1cnn(Cc2ccccc2)c1)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(CC2CC(F)(F)C2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(CC2CCOC2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COCCCN1CC(F)C(C1)NC(=O)c1cc(cnc1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(CCC2CC2(F)F)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(CC2CCC2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(CCC2CC2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(CC2CCCCO2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCOCCN1CC(F)C(C1)NC(=O)c1cc(cnc1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(CCC(C(F)(F)F)C(F)(F)F)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(CC2CCCC2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(CC2CCCO2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(CC2CC2(F)F)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(CC2CC2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(CCCC(F)(F)F)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(CC1F)C1CCCC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(CC2(C)COC2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2nc3ccccc3o2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2ccnc3ccccc23)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2cccnc2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2cccc(n2)C(F)(F)F)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2cccc(C)n2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2cscn2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2nnc(s2)C2CC2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2csc(C)n2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2c(C)noc2C)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2ccccn2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2ccc(F)c(F)c2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2nnnn2C2CC2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2ccc(F)cc2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2ccccc2C#N)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2ccccc2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2ccc(cc2)C(F)(F)F)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2ccccc2F)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2cnc(Br)s2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2cncn2Cc2ccccc2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCn1cncc1CN1CC(F)C(C1)NC(=O)c1cc(cnc1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2cc(Br)no2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2nc3ccccc3s2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COCCn1cncc1CN1CC(F)C(C1)NC(=O)c1cc(cnc1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2ccc(Cl)cc2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2ccc3ccccc3n2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2cccc3cccnc23)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2cccc(c2)C#N)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2cccc(c2)C(F)(F)F)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2c(Cl)cccc2Cl)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2cncc(F)c2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2ccncc2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2ccccc2C(F)(F)F)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2ccc(C)cc2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2cc(F)ccc2F)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2ccc(F)c(C)c2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2ccc(OC(F)(F)F)c(F)c2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2cccc(C)c2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2cc(F)cc(F)c2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2cncc(Br)c2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2cccc3ccccc23)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2ccc(cc2)C#N)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(Cc2cc(C)on2)CC1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CC(CCNC(=O)c1cc(ccc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F)c1ccccc1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(F)c(c1)C(=O)NCc1ccccc1Oc1ccccc1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(F)c(c1)C(=O)NCCC(O)c1ccccc1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(F)c(c1)C(=O)NCC[C@@H](O)c1ccc(Cl)cc1 |r|
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(F)c(c1)C(=O)NCCC(O)c1ccc(F)cc1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(F)c(c1)C(=O)NCC[C@H](O)c1ccc(F)cc1 |r|
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(F)c(c1)C(=O)NCCC(O)(c1ccccc1)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(F)c(c1)C(=O)NCC1CCCOC1c1ccccc1
CC(C)(C)OC(=O)N1CC[C@@H](C1)NC(=O)c1cc(ccc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(F)c(c1)C(=O)N[C@H]1CCN(C1)C(=O)[C@H]1C[C@H](F)C1 |wU:24.26,33.37,wD:31.34,(6.12,3.85,;6.12,2.31,;7.45,1.54,;7.45,,;6.12,-.77,;4.79,,;3.32,-.48,;2.42,.77,;3.32,2.02,;4.79,1.54,;2.85,3.48,;2.37,4.95,;4.31,3.96,;1.38,3,;2.85,-1.94,;3.88,-3.09,;3.4,-4.55,;1.89,-4.87,;1.42,-6.33,;.86,-3.73,;1.34,-2.26,;-.64,-4.05,;-1.12,-5.51,;-1.67,-2.9,;-3.18,-3.22,;-3.81,-4.63,;-5.34,-4.47,;-5.66,-2.96,;-4.32,-2.19,;-7.06,-2.33,;-8.31,-3.24,;-7.22,-.8,;-6.26,.39,;-7.45,1.36,;-7.61,2.89,;-8.42,.17,)|
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(F)c(c1)C(=O)N[C@H]1CCN(C1)C(=O)[C@@H]1C[C@H](F)C1 |wU:24.26,31.34,33.37,(6.12,3.85,;6.12,2.31,;7.45,1.54,;7.45,,;6.12,-.77,;4.79,,;3.32,-.48,;2.42,.77,;3.32,2.02,;4.79,1.54,;2.85,3.48,;2.37,4.95,;4.31,3.96,;1.38,3,;2.85,-1.94,;3.88,-3.09,;3.4,-4.55,;1.89,-4.87,;1.42,-6.33,;.86,-3.73,;1.34,-2.26,;-.64,-4.05,;-1.12,-5.51,;-1.67,-2.9,;-3.18,-3.22,;-3.81,-4.63,;-5.34,-4.47,;-5.66,-2.96,;-4.32,-2.19,;-7.06,-2.33,;-8.31,-3.24,;-7.22,-.8,;-6.26,.39,;-7.45,1.36,;-7.61,2.89,;-8.42,.17,)|
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(F)c(c1)C(=O)N[C@H]1CCN(C1)C(=O)C1CC(F)(F)C1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)CC1 |r|
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccc(F)cc1 |r|
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)C1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCOCC1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC1(F)F
COc1ncc(cc1C(=O)N1CCOC(Cc2ccccc2)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@H]1CCN(C1)C(=O)CC(C)(C)C)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@H]1CCN(C1)C(=O)C(C)(C(F)(F)F)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@H]1CCN(C1)C(=O)C1CCCCC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@H]1CCN(C1)C(=O)C1CCCC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@H]1CCN(C1)C(=O)C1CCC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@H]1CCN(C1)C(=O)C1CC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@H]1CCN(C1)C(=O)C1CCC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cnc(F)c(c1)C(=O)Nc1cnn(CC2CC2)c1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cnc(F)c(c1)C(=O)NCC[C@@H](O)c1ccc(Cl)cc1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cnc(F)c(c1)C(=O)Nc1cnn(Cc2ccccc2)c1
CC(CCNC(=O)c1cc(cnc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F)c1ccccc1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cnc(F)c(c1)C(=O)NCCC(O)c1ccc(F)cc1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cnc(F)c(c1)C(=O)NCCC(O)(c1ccccc1)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cncc(c1)C(=O)NCC[C@@H](O)c1ccc(Cl)cc1 |r|
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cncc(c1)C(=O)Nc1cnn(Cc2ccccc2)c1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cncc(c1)C(=O)NCC[C@H](O)c1ccc(Cl)cc1 |r|
CC(C)(F)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cncc(c1)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
C[C@@](O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cncc(c1)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F |r|
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cncc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)CC1 |r|
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cncc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC1(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cncc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cncc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)C1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cncc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccc(F)cc1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cncc(c1)C(=O)N1CCOC(Cc2ccccc2)C1
COc1nc(C)c(cc1C(=O)NCCC(O)(c1ccccc1)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1nc(C)c(cc1C(=O)NCC[C@@H](O)c1ccc(Cl)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1nc(C)c(cc1C(=O)Nc1cnn(CC2CC2)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
C[C@H]1CN(C[C@H]1NC(=O)c1cc(cnc1C)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(=O)c1ccccc1
C[C@H]1CN(C[C@H]1NC(=O)c1cc(cnc1C)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(=O)C1CC(F)(F)C1
C[C@H]1CN(C[C@H]1NC(=O)c1cc(cnc1C)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(=O)C1CCC(F)(F)CC1
C[C@H]1CN(C[C@H]1NC(=O)c1cc(cnc1C)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(=O)C1CCC(F)(F)C1
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1C)C(=O)c1ccccc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1C)C(=O)C1CCCCC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1C)C(=O)C1CCC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1C)C(=O)C1CC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1C)C(=O)C1CCC(F)(F)CC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)CC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(CC1F)C(=O)C1CCC(F)CC1)-c1cc(c2c(N)ncnn12)C(F)(F)F |(-2.15,5.8,;-3.66,5.48,;-4.13,4.02,;-5.64,3.69,;-6.12,2.23,;-5.09,1.09,;-3.58,1.41,;-3.1,2.87,;-1.6,3.19,;-1.2,4.68,;-.51,2.1,;.98,2.5,;2.18,1.53,;3.47,2.37,;3.07,3.86,;1.53,3.94,;.76,5.27,;4.91,1.82,;5.15,.3,;6.1,2.79,;5.86,4.31,;7.06,5.28,;8.5,4.73,;9.69,5.69,;8.74,3.2,;7.54,2.24,;-5.56,-.38,;-4.66,-1.62,;-5.56,-2.87,;-7.03,-2.39,;-8.36,-3.16,;-8.36,-4.7,;-9.69,-2.39,;-9.69,-.85,;-8.36,-.08,;-7.03,-.85,;-5.09,-4.34,;-6.12,-5.48,;-4.61,-5.8,;-3.58,-4.66,)|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC1(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1(C)CC1(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccc(F)c(F)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1c(F)cccc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@](C)(O)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CCC(C)C)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccc(F)cn1)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cnc1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N([C@@H]1CN(C[C@@H]1F)C(=O)C1(CCCCC1)C(F)(F)F)C(=O)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccnc(C)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)CF)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N([C@@H]1CN(C[C@@H]1F)C(=O)C1(O)CCC1)C(=O)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C)(C)O)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@H](O)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCC(C)(O)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cnc1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1(O)CC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@H](O)CC(C)C)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@H](O)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@H](O)C(C)(C)C)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@H](O)CC(C)C)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCCO1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCCCO1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCCOC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1(C)CCCC(C)(C)O1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1(C)COC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1(F)CCC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1(F)CC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)N(C)C)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)N1CCCC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C)C)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1cccnc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N([C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)C(F)(F)F)C(=O)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C)(C)C)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N([C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)O)C(=O)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COCCC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cnc1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N(C(=O)C(F)(F)F)[C@]1(CNC[C@@H]1F)C(=O)c1cc(F)ccc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1cccc(F)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccccc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)c1ccccc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)C)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1COC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N([C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)F)C(=O)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(CC1F)C(=O)C1CC(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F |(-1.8,5.8,;-3.31,5.48,;-3.78,4.02,;-5.29,3.69,;-5.77,2.23,;-4.73,1.09,;-3.23,1.41,;-2.75,2.87,;-1.25,3.19,;-.85,4.68,;-.16,2.1,;1.33,2.5,;2.53,1.53,;3.82,2.37,;3.42,3.86,;1.88,3.94,;1.11,5.27,;5.26,1.82,;5.5,.3,;6.45,2.79,;6.61,4.32,;8.15,4.16,;9.34,5.13,;7.98,2.63,;-5.21,-.38,;-4.31,-1.62,;-5.21,-2.87,;-6.68,-2.39,;-8.01,-3.16,;-8.01,-4.7,;-9.34,-2.39,;-9.34,-.85,;-8.01,-.08,;-6.68,-.85,;-4.73,-4.34,;-5.77,-5.48,;-4.26,-5.8,;-3.23,-4.66,)|
COc1ncc(cc1C(=O)NC1CN(CC1F)C(=O)[C@@H]1C[C@H](F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F |r,wU:19.20,21.23,(-1.8,5.8,;-3.31,5.48,;-3.78,4.02,;-5.29,3.69,;-5.77,2.23,;-4.73,1.09,;-3.23,1.41,;-2.75,2.87,;-1.25,3.19,;-.85,4.68,;-.16,2.1,;1.33,2.5,;2.53,1.53,;3.82,2.37,;3.42,3.86,;1.88,3.94,;1.11,5.27,;5.26,1.82,;5.5,.3,;6.45,2.79,;7.98,2.63,;8.15,4.16,;9.34,5.13,;6.61,4.32,;-5.21,-.38,;-4.31,-1.62,;-5.21,-2.87,;-6.68,-2.39,;-8.01,-3.16,;-8.01,-4.7,;-9.34,-2.39,;-9.34,-.85,;-8.01,-.08,;-6.68,-.85,;-4.73,-4.34,;-5.77,-5.48,;-4.26,-5.8,;-3.23,-4.66,)|
Cc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
CC(C)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cnc1C)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC1(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)NC1CN(CC1F)C(=O)C1CC1(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)NC1CN(CC1F)C(=O)C1CC(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F |(-3.31,5.64,;-3.78,4.18,;-5.29,3.86,;-5.77,2.39,;-4.73,1.25,;-3.23,1.57,;-2.75,3.03,;-1.25,3.35,;-.85,4.84,;-.16,2.26,;1.33,2.66,;2.53,1.69,;3.82,2.53,;3.42,4.02,;1.88,4.1,;1.11,5.43,;5.26,1.98,;5.5,.46,;6.45,2.95,;6.61,4.48,;8.15,4.32,;9.34,5.29,;7.98,2.79,;-5.21,-.22,;-4.31,-1.46,;-5.21,-2.71,;-6.68,-2.23,;-8.01,-3,;-8.01,-4.54,;-9.34,-2.23,;-9.34,-.69,;-8.01,.08,;-6.68,-.69,;-4.73,-4.18,;-5.77,-5.32,;-4.26,-5.64,;-3.23,-4.5,)|
Cc1ncc(cc1C(=O)NC1CN(CC1F)C(=O)C1CCC(F)(F)CC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)NC1CN(CC1F)C(=O)C1CCC(F)CC1)-c1cc(c2c(N)ncnn12)C(F)(F)F |(-3.66,5.53,;-4.13,4.07,;-5.64,3.75,;-6.12,2.28,;-5.09,1.14,;-3.58,1.46,;-3.1,2.92,;-1.6,3.24,;-1.2,4.73,;-.51,2.15,;.98,2.55,;2.18,1.58,;3.47,2.42,;3.07,3.91,;1.53,3.99,;.76,5.32,;4.91,1.87,;5.15,.35,;6.1,2.84,;5.86,4.36,;7.06,5.33,;8.5,4.78,;9.69,5.75,;8.74,3.26,;7.54,2.29,;-5.56,-.33,;-4.66,-1.57,;-5.56,-2.82,;-7.03,-2.34,;-8.36,-3.11,;-8.36,-4.65,;-9.69,-2.34,;-9.69,-.8,;-8.36,-.03,;-7.03,-.8,;-5.09,-4.28,;-6.12,-5.43,;-4.61,-5.75,;-3.58,-4.6,)|
Cc1ncc(cc1C(=O)NC1CN(CC1F)C(=O)C1(O)CCC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
CC(C)CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cnc1C)-c1cc(c2c(N)ncnn12)C(F)(F)F
CC(C)C[C@H](O)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cnc1C)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1cc(F)ccc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CC(C)C[C@@H](O)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cnc1C)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1(F)CC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@H](O)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1(F)CCC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)N([C@@H]1CN(C[C@@H]1F)C(=O)[C@](C)(O)C(F)(F)F)C(=O)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@H](O)C(C)(C)C)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccc(F)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
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Cc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H](O)C(F)(F)F)C[C@@H]1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
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COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(C)c1ccccc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(C)c1cccc(c1)C#N)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)[C@H](C)c1ccc(F)cc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)[C@@H](C)c1ccc(F)cc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(C)c1ccncc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(C)c1cncc(F)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)[C@H](C)c1cncc(F)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)[C@@H](C)c1cncc(F)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(C)c1csc(C)n1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(C)c1cncs1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(CC(F)(F)F)c1ccccc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(C)c1ccccc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(C)c1ncccc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(Cc2ccccc2)C[C@@H]1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(C)c1ccncn1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(C)c1ccncc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(C)c1cccnc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)[C@H](C)c1cccnc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)[C@@H](C)c1cccnc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)[C@H](C)c1ccc(F)c(F)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)[C@@H](C)c1ccc(F)c(F)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(C)c1ccc(F)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(Cc2ccc(F)cn2)C[C@@H]1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(CC(O)c2ccccc2)C[C@@H]1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N1CCC[C@@H](Cc2ccc(F)cc2)C1)-c1cc(C(=O)N2CC3(COC3)C2)c2c(N)ncnn12
CCNC(=O)c1cc(-c2cnc(OC)c(c2)C(=O)N2CCC[C@@H](Cc3ccc(F)cc3)C2)n2ncnc(N)c12
COc1ncc(cc1C(=O)N1CCC[C@@H](Cc2ccc(F)cc2)C1)-c1cc(C(=O)NCC#N)c2c(N)ncnn12
COc1ncc(cc1C(=O)N1CCC[C@@H](Cc2ccc(F)cc2)C1)-c1cc(C(=O)NCCO)c2c(N)ncnn12
COc1ncc(cc1C(=O)N1CCC[C@@H](Cc2ccc(F)cc2)C1)-c1cc(C(=O)N(C)C)c2c(N)ncnn12
COc1ncc(cc1C(=O)N1CCC[C@@H](Cc2ccc(F)cc2)C1)-c1cc(C(=O)NCCNC(C)=O)c2c(N)ncnn12
CCNC(=O)c1cc(-c2cnc(OC)c(c2)C(=O)NCC[C@H](O)c2ccc(Cl)cc2)n2ncnc(N)c12
COc1ncc(cc1C(=O)NCC[C@H](O)c1ccc(Cl)cc1)-c1cc(C(=O)NCC#N)c2c(N)ncnn12
COc1ncc(cc1C(=O)NCC[C@H](O)c1ccc(Cl)cc1)-c1cc(C(=O)NCCO)c2c(N)ncnn12
CCCNC(=O)c1cc(-c2cnc(OC)c(c2)C(=O)NCC[C@H](O)c2ccc(Cl)cc2)n2ncnc(N)c12
COc1ncc(cc1C(=O)NCC[C@H](O)c1ccc(Cl)cc1)-c1cc(C(=O)N(C)C)c2c(N)ncnn12
CNC(=O)c1cc(-c2cnc(OC)c(c2)C(=O)N(CC[C@H](O)c2ccc(Cl)cc2)C(=O)C(F)(F)F)n2ncnc(N)c12
COc1ncc(cc1C(=O)N[C@@H]1CN(CC(O)C(F)(F)F)C[C@@H]1F)-c1cc(CNCCO)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(CC(O)C(F)(F)F)C[C@@H]1F)-c1cc(CN(C)C)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(CC(O)C(F)(F)F)C[C@@H]1F)-c1cc(CN2CC3(COC3)C2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(CC(O)C(F)(F)F)C[C@@H]1F)-c1cc(CN2CCOCC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(CC(O)C(F)(F)F)C[C@@H]1F)-c1cc(CN2CC(N)C2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(CC(O)C(F)(F)F)C[C@@H]1F)-c1cc(CN2CCC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(CC(O)C(F)(F)F)C[C@@H]1F)-c1cc(CN2CCS(=O)(=O)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(CN(C)C)c2c(N)ncnn12
CNCc1cc(-c2cnc(OC)c(c2)C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)C2CC(F)(F)C2)n2ncnc(N)c12
COc1ncc(cc1C(=O)N([C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)C(=O)C(F)(F)F)-c1cc(CN2CCOCC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N([C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)C(=O)C(F)(F)F)-c1cc(CN2CC(O)C2)c2c(N)ncnn12
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COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(CN2CC3(COC3)C2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(CN2CC(N)C2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(CN2CCC2)c2c(N)ncnn12
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COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(CNCCO)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(CN2CCN(C)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)c1ccccc1C#N)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)c1cnc(C)s1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)c1cccc(F)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)c1ccc(F)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)c1cccnc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1c(F)cc2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCOCC1)-c1c(F)cc2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)CC1)-c1c(F)cc2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)C1)-c1c(F)cc2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccc(F)cc1)-c1c(F)cc2c(N)ncnn12
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COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC1(F)F)-c1c(F)cc2c(N)ncnn12
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COc1nc(C)c(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)C2CCC(F)(F)C2)c(F)cc1Cl
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)C2CC(F)(F)C2)c(F)cc1Cl
Cc1nc(C)c(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC1(F)F)-c1cc(c2c(NC(=O)C(F)(F)F)ncnn12)C(F)(F)F |r|
Cc1nc(C)c(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@H]1CCC(F)(F)C1)-c1cc(c2c(NC(=O)C(F)(F)F)ncnn12)C(F)(F)F |r|
Cc1nc(C)c(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@H]1CCC(F)(F)C1)-c1cc(c2c(NC(=O)C(F)(F)F)ncnn12)C(F)(F)F |r|
Cc1nc(C)c(cc1C(=O)N1CCOC(Cc2ccccc2)C1)-c1cc(c2c(NC(=O)C(F)(F)F)ncnn12)C(F)(F)F
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Cc1cc(C)c(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)CC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1cc(C)c(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC1(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1cc(C)c(cc1C(=O)N1CCC[C@H](Cc2ccc(F)cc2)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1c(cc2c(N)ncnn12)C#N |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1c(cc2c(N)ncnn12)-c1nnn[nH]1 |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1c(cc2c(N)ncnn12)-c1nnn(C)n1 |r|
COc1ncc(cc1C(=O)NCC[C@H](O)c1ccc(Cl)cc1)-c1c(cc2c(N)ncnn12)C#N |r|
COc1ncc(cc1C(=O)NCC[C@@H](O)c1ccc(Cl)cc1)-c1c(cc2c(N)ncnn12)C#N |r|
COc1ncc(cc1C(=O)N[C@H](C)c1cc(OC(F)(F)F)ccc1F)-c1c(cc2c(N)ncnn12)C#N |r|
COc1ncc(cc1C(=O)N[C@H](C)c1cc(ccc1F)C(F)(F)F)-c1c(cc2c(N)ncnn12)C#N |r|
COc1ncc(cc1C(=O)Nc1cnn(Cc2ccccc2)c1)-c1c(cc2c(N)ncnn12)C#N
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC1(F)F)-c1c(cc2c(N)ncnn12)C#N
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1c(cc2c(N)ncnn12)C#N
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COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(O)(C1)C(F)(F)F)-c1c(cc2c(N)ncnn12)C#N |wD:11.11,15.17,(1.25,-9.55,;.22,-8.41,;.7,-6.94,;-.33,-5.8,;.14,-4.33,;1.65,-4.01,;2.68,-5.16,;2.2,-6.62,;3.23,-7.77,;4.74,-7.45,;2.76,-9.23,;3.79,-10.38,;5.32,-10.21,;5.95,-11.62,;4.8,-12.65,;3.47,-11.88,;2.06,-12.51,;7.45,-11.94,;8.48,-10.8,;7.93,-13.41,;9.3,-14.11,;8.6,-15.48,;9.97,-16.18,;7.23,-14.78,;7.9,-16.85,;7.2,-18.22,;9.28,-17.55,;6.53,-16.15,;2.13,-2.55,;1.22,-1.3,;2.13,-.06,;3.59,-.53,;4.92,.24,;4.92,1.78,;6.26,-.53,;6.26,-2.07,;4.92,-2.84,;3.59,-2.07,;-.32,-1.3,;-1.86,-1.3,)|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)C(F)(F)F)-c1c(cc2c(N)ncnn12)C#N
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)F)-c1c(cc2c(N)ncnn12)C#N
Cc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(O)(C(F)(F)F)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
C[C@@](O)(C(=O)Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(F)c(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)C(F)(F)F |r|
COc1cc(F)c(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(O)(C(F)(F)F)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
CNc1ccc(cc1C(=O)NC1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
CCc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(O)(C(F)(F)F)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1cc(F)c(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
Cc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(F)c(CF)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(O)(C(F)(F)F)C(F)(F)F |r|
CCc1ccc(-c2cc(c3c(N)ncnn23)C(F)(F)F)c(F)c1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(O)(C(F)(F)F)C(F)(F)F |r|
COc1cc(cc(c1)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1(F)CC1 |r|
COc1cc(cc(c1)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C(F)(F)F)C(F)(F)F
COc1cc(cc(C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)CC(C)C(F)(F)F)c1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1cc(cc(C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)[C@@](C)(O)C(F)(F)F)c1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1cc(cc(C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)C(O)(C(F)(F)F)C(F)(F)F)c1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1cc(cc(C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)c2ccccc2F)c1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1cc(cc(C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)C(C(F)(F)F)C(F)(F)F)c1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(F)cc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@H](O)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(F)cc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)C1 |wU:28.32,24.26,(-8.05,-4.35,;-8.05,-2.81,;-9.39,-2.04,;-9.39,-.5,;-8.05,.27,;-6.72,-.5,;-5.25,-.02,;-4.35,-1.27,;-5.25,-2.51,;-6.72,-2.04,;-4.78,-3.98,;-5.87,-5.07,;-4.38,-5.46,;-3.29,-4.38,;-4.78,1.44,;-5.81,2.59,;-5.33,4.05,;-6.36,5.2,;-3.83,4.37,;-2.8,3.23,;-3.27,1.76,;-1.29,3.55,;-.81,5.01,;-.26,2.4,;1.25,2.72,;2.39,1.69,;3.73,2.46,;3.41,3.97,;1.87,4.13,;1.1,5.46,;5.13,1.84,;5.29,.31,;6.38,2.74,;6.62,4.26,;8.14,4.02,;9.39,4.93,;7.9,2.5,)|
CC(C)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(F)cc(c1)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
CC(C)(F)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(F)cc(c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
CC(C)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(F)cc(c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
CC(C)CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(F)cc(c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
CC(C)(O)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(F)cc(c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(F)cc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(F)(F)F
CC(C)(C)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(F)cc(c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(F)cc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(F)cc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccc(F)cc1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(F)cc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccccc1F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(F)cc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC1(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(F)cc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)CC1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(F)cc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)C1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(F)c(CF)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1(F)CC1
CC(C)(F)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cc(F)c1CF)-c1cc(c2c(N)ncnn12)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(F)c(CF)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC1(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(F)c(CF)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(F)c(CF)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)C1 |wU:30.34,26.28,(-8.05,-4.69,;-8.05,-3.15,;-9.39,-2.38,;-9.39,-.84,;-8.05,-.07,;-6.72,-.84,;-5.25,-.37,;-4.35,-1.61,;-5.25,-2.86,;-6.72,-2.38,;-4.78,-4.32,;-5.87,-5.41,;-4.38,-5.81,;-3.29,-4.72,;-4.78,1.1,;-5.81,2.24,;-5.33,3.71,;-6.36,4.85,;-3.83,4.03,;-3.35,5.49,;-1.84,5.81,;-2.8,2.88,;-3.27,1.42,;-1.29,3.2,;-.81,4.67,;-.26,2.06,;1.25,2.38,;2.39,1.35,;3.73,2.12,;3.41,3.62,;1.87,3.78,;1.1,5.12,;5.13,1.49,;5.29,-.04,;6.38,2.4,;6.62,3.92,;8.14,3.68,;9.39,4.58,;7.9,2.16,)|
C[C@@](O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cc(F)c1CF)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(F)c(CF)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)C1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(F)c(CF)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)CC1
CC(CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cc(F)c1CF)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
CC(O)(CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cc(F)c1CF)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(F)c(CF)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C(F)(F)F)C(F)(F)F
CC(C)(O)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cc(F)c1CF)-c1cc(c2c(N)ncnn12)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(F)c(CF)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(F)(F)F
CC(C)CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cc(F)c1CF)-c1cc(c2c(N)ncnn12)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(F)c(CF)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccccc1F
CC(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cc(F)c1CF)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
CCC(O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cc(F)c1CF)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
CC(O)(CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cc(F)c1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
CC(C)(F)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cc(F)c1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(F)c(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC1(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(F)c(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C(F)(F)F)C(F)(F)F
CC(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cc(F)c1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
CC(CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cc(F)c1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(F)c(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(F)c(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1(F)CC1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(F)c(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(O)(C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(F)c(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)C1 |wU:29.33,25.27,(-8.05,-4.53,;-8.05,-2.99,;-9.39,-2.22,;-9.39,-.68,;-8.05,.09,;-6.72,-.68,;-5.25,-.21,;-4.35,-1.45,;-5.25,-2.7,;-6.72,-2.22,;-4.78,-4.16,;-5.87,-5.25,;-4.38,-5.65,;-3.29,-4.56,;-4.78,1.26,;-5.81,2.4,;-5.33,3.87,;-6.36,5.01,;-3.83,4.19,;-3.35,5.65,;-2.8,3.04,;-3.27,1.58,;-1.29,3.36,;-.81,4.83,;-.26,2.22,;1.25,2.54,;2.39,1.51,;3.73,2.28,;3.41,3.78,;1.87,3.95,;1.1,5.28,;5.13,1.65,;5.29,.12,;6.38,2.56,;6.62,4.08,;8.14,3.84,;9.39,4.74,;7.9,2.32,)|
CC(C)(O)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cc(F)c1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(F)c(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(F)(F)F
CC(C)CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cc(F)c1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(F)c(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccccc1F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(F)c(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)CC1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(F)c(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)C1
CCc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccccc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C)C)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)O)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC1(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(O)(CC)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C)(O)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C(F)(F)F)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F |wU:16.18,12.12,(-1.84,5.81,;-3.35,5.49,;-3.83,4.03,;-5.33,3.71,;-6.36,4.85,;-5.81,2.24,;-4.78,1.1,;-3.27,1.42,;-2.8,2.88,;-1.29,3.2,;-.81,4.67,;-.26,2.06,;1.25,2.38,;2.39,1.35,;3.73,2.12,;3.41,3.62,;1.87,3.78,;1.1,5.12,;5.13,1.49,;5.29,-.04,;6.38,2.4,;6.62,3.92,;8.14,3.68,;9.39,4.58,;7.9,2.16,;-5.25,-.37,;-4.35,-1.61,;-5.25,-2.86,;-6.72,-2.38,;-8.05,-3.15,;-8.05,-4.69,;-9.39,-2.38,;-9.39,-.84,;-8.05,-.07,;-6.72,-.84,;-4.78,-4.32,;-5.87,-5.41,;-4.38,-5.81,;-3.29,-4.72,)|
CCc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1(F)CC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)CC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CC(CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cc(F)c1C)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
Cc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)O)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)C)-c1cc(c2c(N)ncnn12)C(F)(F)F
CC(C)CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cc(F)c1C)-c1cc(c2c(N)ncnn12)C(F)(F)F
CC(C)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cc(F)c1C)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccccc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccc(F)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1(O)CCC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@H](O)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)CC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC1(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F |wU:15.17,11.11,(-3.35,5.65,;-3.83,4.19,;-5.33,3.87,;-6.36,5.01,;-5.81,2.4,;-4.78,1.26,;-3.27,1.58,;-2.8,3.04,;-1.29,3.36,;-.81,4.83,;-.26,2.22,;1.25,2.54,;2.39,1.51,;3.73,2.28,;3.41,3.78,;1.87,3.95,;1.1,5.28,;5.13,1.65,;5.29,.12,;6.38,2.56,;6.62,4.08,;8.14,3.84,;9.39,4.74,;7.9,2.32,;-5.25,-.21,;-4.35,-1.45,;-5.25,-2.7,;-6.72,-2.22,;-8.05,-2.99,;-8.05,-4.53,;-9.39,-2.22,;-9.39,-.68,;-8.05,.09,;-6.72,-.68,;-4.78,-4.16,;-5.87,-5.25,;-4.38,-5.65,;-3.29,-4.56,)|
Cc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C)C)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccccc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccc(F)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F |wU:16.18,12.12,(-1.84,5.81,;-3.35,5.49,;-3.83,4.03,;-5.33,3.71,;-6.36,4.85,;-5.81,2.24,;-4.78,1.1,;-3.27,1.42,;-2.8,2.88,;-1.29,3.2,;-.81,4.67,;-.26,2.06,;1.25,2.38,;2.39,1.35,;3.73,2.12,;3.41,3.62,;1.87,3.78,;1.1,5.12,;5.13,1.49,;5.29,-.04,;6.38,2.4,;6.62,3.92,;8.14,3.68,;9.39,4.58,;7.9,2.16,;-5.25,-.37,;-4.35,-1.61,;-5.25,-2.86,;-6.72,-2.38,;-8.05,-3.15,;-8.05,-4.69,;-9.39,-2.38,;-9.39,-.84,;-8.05,-.07,;-6.72,-.84,;-4.78,-4.32,;-5.87,-5.41,;-4.38,-5.81,;-3.29,-4.72,)|
COc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1(F)CC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)CC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(O)(C(F)(F)F)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C(F)(F)F)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCC(O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cc(F)c1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
COc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)CC1)-c1cc(c2c(N)ncnn12)C(F)(F)F |wU:16.18,12.12,(-2.21,5.81,;-3.72,5.49,;-4.19,4.03,;-5.7,3.71,;-6.73,4.85,;-6.17,2.24,;-5.14,1.1,;-3.64,1.42,;-3.16,2.88,;-1.65,3.2,;-1.18,4.67,;-.62,2.06,;.88,2.38,;2.03,1.35,;3.36,2.12,;3.04,3.62,;1.51,3.78,;.74,5.12,;4.77,1.49,;4.93,-.04,;6.01,2.4,;5.85,3.93,;7.1,4.83,;8.51,4.21,;9.75,5.11,;8.67,2.68,;7.42,1.77,;-5.62,-.37,;-4.71,-1.61,;-5.62,-2.86,;-7.08,-2.38,;-8.42,-3.15,;-8.42,-4.69,;-9.75,-2.38,;-9.75,-.84,;-8.42,-.07,;-7.08,-.84,;-5.14,-4.32,;-6.23,-5.41,;-4.74,-5.81,;-3.66,-4.72,)|
COc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C)(O)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC1(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)O)-c1cc(c2c(N)ncnn12)C(F)(F)F
CC(CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cc(C)c1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
Cc1cc(cc(C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)CC(O)(C(F)(F)F)C(F)(F)F)c1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCC(O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cc(C)c1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
Cc1cc(cc(C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)C2CC2(F)F)c1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1cc(cc(C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)C(C)(C)F)c1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1cc(cc(C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)C2CC(F)(F)C2)c1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1cc(cc(C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)C(C)(C)O)c1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1cc(cc(C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)c2ccccc2F)c1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1cc(cc(C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)CC(C(F)(F)F)C(F)(F)F)c1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1cc(cc(C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)C2CCC(F)(F)C2)c1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1cc(cc(C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)CC(C)(O)C(F)(F)F)c1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1cc(cc(C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)C2CCC(F)(F)CC2)c1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1cc(cc(C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)C2(F)CC2)c1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F
CC(C)CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cc(C)c1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1cc(cc(C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)CC(F)(F)F)c1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F
CC(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cc(C)c1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
C[C@@](O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1c(F)ccc(-c2cc(c3c(N)ncnn23)C(F)(F)F)c1F)C(F)(F)F
CCc1ccc(-c2cc(c3c(N)ncnn23)C(F)(F)F)c(F)c1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C)(O)C(F)(F)F
CCc1ccc(-c2cc(c3c(N)ncnn23)C(F)(F)F)c(F)c1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(F)(F)F
CCc1ccc(-c2cc(c3c(N)ncnn23)C(F)(F)F)c(F)c1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C(F)(F)F)C(F)(F)F
CCc1ccc(-c2cc(c3c(N)ncnn23)C(F)(F)F)c(F)c1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F
CCc1ccc(-c2cc(c3c(N)ncnn23)C(F)(F)F)c(F)c1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C)C
CCc1ccc(-c2cc(c3c(N)ncnn23)C(F)(F)F)c(F)c1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)CC1
CCc1ccc(-c2cc(c3c(N)ncnn23)C(F)(F)F)c(F)c1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC1(F)F
CCc1ccc(-c2cc(c3c(N)ncnn23)C(F)(F)F)c(F)c1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1
CCc1ccc(-c2cc(c3c(N)ncnn23)C(F)(F)F)c(F)c1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)C1 |wU:30.34,26.28,(-1.84,5.81,;-3.35,5.49,;-3.83,4.03,;-5.33,3.71,;-5.81,2.24,;-4.78,1.1,;-5.25,-.37,;-4.35,-1.61,;-5.25,-2.86,;-6.72,-2.38,;-8.05,-3.15,;-8.05,-4.69,;-9.39,-2.38,;-9.39,-.84,;-8.05,-.07,;-6.72,-.84,;-4.78,-4.32,;-5.87,-5.41,;-4.38,-5.81,;-3.29,-4.72,;-3.27,1.42,;-2.24,.27,;-2.8,2.88,;-1.29,3.2,;-.81,4.67,;-.26,2.06,;1.25,2.38,;2.39,1.35,;3.73,2.12,;3.41,3.62,;1.87,3.78,;1.1,5.12,;5.13,1.49,;5.29,-.04,;6.38,2.4,;6.62,3.92,;8.14,3.68,;9.39,4.58,;7.9,2.16,)|
CCc1ccc(-c2cc(c3c(N)ncnn23)C(F)(F)F)c(F)c1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)C1
CCc1ccc(-c2cc(c3c(N)ncnn23)C(F)(F)F)c(F)c1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccccc1F
Cc1ccc(-c2cc(c3c(N)ncnn23)C(F)(F)F)c(F)c1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)C1 |wU:29.33,25.27,(-3.35,5.65,;-3.83,4.19,;-5.33,3.87,;-5.81,2.4,;-4.78,1.26,;-5.25,-.21,;-4.35,-1.45,;-5.25,-2.7,;-6.72,-2.22,;-8.05,-2.99,;-8.05,-4.53,;-9.39,-2.22,;-9.39,-.68,;-8.05,.09,;-6.72,-.68,;-4.78,-4.16,;-5.87,-5.25,;-4.38,-5.65,;-3.29,-4.56,;-3.27,1.58,;-2.24,.43,;-2.8,3.04,;-1.29,3.36,;-.81,4.83,;-.26,2.22,;1.25,2.54,;2.39,1.51,;3.73,2.28,;3.41,3.78,;1.87,3.95,;1.1,5.28,;5.13,1.65,;5.29,.12,;6.38,2.56,;6.62,4.08,;8.14,3.84,;9.39,4.74,;7.9,2.32,)|
Cc1ccc(-c2cc(c3c(N)ncnn23)C(F)(F)F)c(F)c1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(O)(C(F)(F)F)C(F)(F)F
Cc1ccc(-c2cc(c3c(N)ncnn23)C(F)(F)F)c(F)c1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)C2CCC2)c1F
CC(C)CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cccc(-c2cc(c3c(N)ncnn23)C(F)(F)F)c1F
CC(C)(C)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cccc(-c2cc(c3c(N)ncnn23)C(F)(F)F)c1F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)c2ccc(F)cc2)c1F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)c2ccccc2F)c1F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)C2CC(F)(F)C2)c1F
CC(C)(F)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cccc(-c2cc(c3c(N)ncnn23)C(F)(F)F)c1F
CC(C)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cccc(-c2cc(c3c(N)ncnn23)C(F)(F)F)c1F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)C2CC(F)C2)c1F |wU:26.29,22.23,(-8.05,-4.35,;-8.05,-2.81,;-9.39,-2.04,;-9.39,-.5,;-8.05,.27,;-6.72,-.5,;-5.25,-.02,;-4.35,-1.27,;-5.25,-2.51,;-6.72,-2.04,;-4.78,-3.98,;-5.87,-5.07,;-4.38,-5.46,;-3.29,-4.38,;-4.78,1.44,;-5.81,2.59,;-5.33,4.05,;-3.83,4.37,;-2.8,3.23,;-1.29,3.55,;-.81,5.01,;-.26,2.4,;1.25,2.72,;2.39,1.69,;3.73,2.46,;3.41,3.97,;1.87,4.13,;1.1,5.46,;5.13,1.84,;5.29,.31,;6.38,2.74,;6.62,4.26,;8.14,4.02,;9.39,4.93,;7.9,2.5,;-3.27,1.76,;-2.24,.62,)|
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)C2CCC(F)(F)C2)c1F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cccc(C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)C2CC2(F)F)c1F
C[C@@](O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cccc(-c2cc(c3c(N)ncnn23)C(F)(F)F)c1F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)CC(F)(F)F)c(F)cc1F
CC(C)(O)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(-c2cc(c3c(N)ncnn23)C(F)(F)F)c(F)cc1F
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Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)CC(C(F)(F)F)C(F)(F)F)c(Cl)cc1F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)CC(O)(C(F)(F)F)C(F)(F)F)c(Cl)cc1F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)C2CC(F)C2)c(Cl)cc1F |wU:24.27,20.21,(-8.05,-4.53,;-8.05,-2.99,;-9.39,-2.22,;-9.39,-.68,;-8.05,.09,;-6.72,-.68,;-5.25,-.21,;-4.35,-1.45,;-5.25,-2.7,;-6.72,-2.22,;-4.78,-4.16,;-5.87,-5.25,;-4.38,-5.65,;-3.29,-4.56,;-4.78,1.26,;-3.27,1.58,;-2.8,3.04,;-1.29,3.36,;-.81,4.83,;-.26,2.22,;1.25,2.54,;2.39,1.51,;3.73,2.28,;3.41,3.78,;1.87,3.95,;1.1,5.28,;5.13,1.65,;5.29,.12,;6.38,2.56,;6.62,4.08,;8.14,3.84,;9.39,4.74,;7.9,2.32,;-3.83,4.19,;-3.35,5.65,;-5.33,3.87,;-5.81,2.4,;-7.31,2.08,)|
CCC(O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1ccc(F)c(c1)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1(F)CC1)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(O)(C(F)(F)F)C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)C1)C(F)(F)F |wU:27.31,23.25,(-8.05,-5.27,;-8.05,-3.73,;-9.39,-2.96,;-9.39,-1.42,;-8.05,-.65,;-6.72,-1.42,;-5.25,-.94,;-4.35,-2.19,;-5.25,-3.43,;-6.72,-2.96,;-4.78,-4.9,;-5.87,-5.98,;-4.38,-6.38,;-3.29,-5.29,;-4.78,.53,;-5.81,1.67,;-5.33,3.13,;-3.83,3.45,;-2.8,2.31,;-3.27,.85,;-1.29,2.63,;-.81,4.09,;-.26,1.49,;1.25,1.81,;2.39,.78,;3.73,1.55,;3.41,3.05,;1.87,3.21,;1.1,4.55,;5.13,.92,;5.29,-.61,;6.38,1.82,;6.62,3.35,;8.14,3.1,;9.39,4.01,;7.9,1.58,;-3.35,4.92,;-2.87,6.38,;-4.38,6.06,;-1.84,5.24,)|
CC(C)(F)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CC(CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC1(F)F)C(F)(F)F
CC(C)(O)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CC(O)(CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
CCC(O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)C1)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(F)(F)F)C(F)(F)F
CC(C)CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)CC1)C(F)(F)F
C[C@@](O)(CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C(F)(F)F)C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccccc1F)C(F)(F)F
CC(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
CC(C)(O)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1CF)-c1cc(c2c(N)ncnn12)C(F)(F)F
CC(C)CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1CF)-c1cc(c2c(N)ncnn12)C(F)(F)F
C[C@@](O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1CF)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(CF)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(CF)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(O)(C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(CF)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccccc1F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(CF)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC1(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(CF)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(CF)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1(F)CC1
CC(CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1CF)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(CF)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)CC1
CC(O)(CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1CF)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(CF)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)C1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(CF)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(F)(F)F
CCC(O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1CF)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(CF)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)C1 |wU:29.33,25.27,(-8.05,-4.69,;-8.05,-3.15,;-9.39,-2.38,;-9.39,-.84,;-8.05,-.07,;-6.72,-.84,;-5.25,-.37,;-4.35,-1.61,;-5.25,-2.86,;-6.72,-2.38,;-4.78,-4.32,;-5.87,-5.41,;-4.38,-5.81,;-3.29,-4.72,;-4.78,1.1,;-5.81,2.24,;-5.33,3.71,;-3.83,4.03,;-3.35,5.49,;-1.84,5.81,;-2.8,2.88,;-3.27,1.42,;-1.29,3.2,;-.81,4.67,;-.26,2.06,;1.25,2.38,;2.39,1.35,;3.73,2.12,;3.41,3.62,;1.87,3.78,;1.1,5.12,;5.13,1.49,;5.29,-.04,;6.38,2.4,;6.62,3.92,;8.14,3.68,;9.39,4.58,;7.9,2.16,)|
CC(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1CF)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)C1 |wU:28.32,24.26,(-8.05,-4.53,;-8.05,-2.99,;-9.39,-2.22,;-9.39,-.68,;-8.05,.09,;-6.72,-.68,;-5.25,-.21,;-4.35,-1.45,;-5.25,-2.7,;-6.72,-2.22,;-4.78,-4.16,;-5.87,-5.25,;-4.38,-5.65,;-3.29,-4.56,;-4.78,1.26,;-5.81,2.4,;-5.33,3.87,;-3.83,4.19,;-3.35,5.65,;-2.8,3.04,;-3.27,1.58,;-1.29,3.36,;-.81,4.83,;-.26,2.22,;1.25,2.54,;2.39,1.51,;3.73,2.28,;3.41,3.78,;1.87,3.95,;1.1,5.28,;5.13,1.65,;5.29,.12,;6.38,2.56,;6.62,4.08,;8.14,3.84,;9.39,4.74,;7.9,2.32,)|
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C(F)(F)F)C(F)(F)F
CCC(O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(F)(F)F
CC(C)(O)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)C1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(O)(C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccccc1F
CC(C)(F)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1(F)CC1
C[C@@](O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
CC(O)(CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC1(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)CC1
CC(C)CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F
CC(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
CC(CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1cc(ccn1)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccc(F)cc1F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ncc(F)cc1F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1cscn1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccc(Cl)cc1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccc(F)c(F)c1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ncccc1F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccncc1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1cccc(F)c1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccc(F)cc1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1cnccc1C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccccc1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1c(F)cncc1F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccccn1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1cc(F)ccc1F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccc(F)cn1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1cnccc1Cl
Cc1cc(ccn1)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccncc1F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1cc(Cl)ccn1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccccc1Cl
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1c(F)cccc1F
CCc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1(F)CC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCC(O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1C)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC1(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)O)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)CC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
CC(C)CC(=O)N1CC(F)[C@@H](C1)NC(=O)c1cc(ccc1C)-c1cc(c2c(N)ncnn12)C(F)(F)F
CC(CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1C)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(O)(C(F)(F)F)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C)(O)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C(F)(F)F)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F |wU:14.16,10.10,(-3.35,5.65,;-3.83,4.19,;-5.33,3.87,;-5.81,2.4,;-4.78,1.26,;-3.27,1.58,;-2.8,3.04,;-1.29,3.36,;-.81,4.83,;-.26,2.22,;1.25,2.54,;2.39,1.51,;3.73,2.28,;3.41,3.78,;1.87,3.95,;1.1,5.28,;5.13,1.65,;5.29,.12,;6.38,2.56,;6.62,4.08,;8.14,3.84,;9.39,4.74,;7.9,2.32,;-5.25,-.21,;-4.35,-1.45,;-5.25,-2.7,;-6.72,-2.22,;-8.05,-2.99,;-8.05,-4.53,;-9.39,-2.22,;-9.39,-.68,;-8.05,.09,;-6.72,-.68,;-4.78,-4.16,;-5.87,-5.25,;-4.38,-5.65,;-3.29,-4.56,)|
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccccc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CC(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1C)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1cc(ccn1)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccc(F)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1cccc(F)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1cscn1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1c(F)cncc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccncc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ncc(F)cc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccc(F)c(F)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1cnccc1C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ncccc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccc(Cl)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccc(F)cn1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1cnccc1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1c(F)cccc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1cc(Cl)ccn1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1cc(F)ccc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccccc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccncc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccccn1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccccc1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1cc(ccn1)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1C)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccc(F)cc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC1CCCC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC1CC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(OC(F)(F)F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccccc1F
CC(C)CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1OC(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CC(C)(O)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1OC(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(OC(F)(F)F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(F)(F)F
CC(CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1OC(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
CCC(O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1OC(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(OC(F)(F)F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1(F)CC1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(OC(F)(F)F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)C1 |wU:32.36,28.30,(-8.05,-5.84,;-8.05,-4.3,;-9.39,-3.53,;-9.39,-1.99,;-8.05,-1.22,;-6.72,-1.99,;-5.25,-1.51,;-4.35,-2.76,;-5.25,-4,;-6.72,-3.53,;-4.78,-5.47,;-5.87,-6.56,;-4.38,-6.96,;-3.29,-5.87,;-4.78,-.05,;-5.81,1.1,;-5.33,2.56,;-3.83,2.88,;-3.35,4.35,;-4.38,5.49,;-5.89,5.17,;-5.41,6.64,;-3.91,6.96,;-2.8,1.74,;-3.27,.27,;-1.29,2.06,;-.81,3.52,;-.26,.91,;1.25,1.23,;2.39,.2,;3.73,.97,;3.41,2.48,;1.87,2.64,;1.1,3.97,;5.13,.35,;5.29,-1.18,;6.38,1.25,;6.62,2.77,;8.14,2.53,;9.39,3.44,;7.9,1.01,)|
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(OC(F)(F)F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(OC(F)(F)F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)C1
CC(C)(F)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1OC(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(OC(F)(F)F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)CC1
CC(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1OC(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(OC(F)(F)F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC1(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(OC(F)(F)F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(O)(C(F)(F)F)C(F)(F)F
C[C@@](O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1OC(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
CC(O)(CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1OC(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(OCC(F)(F)F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)C1
CC(CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1OCC(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
C[C@@](O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1OCC(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(OCC(F)(F)F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C(F)(F)F)C(F)(F)F
CC(O)(CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1OCC(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(OCC(F)(F)F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC1(F)F
CCC(O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1OCC(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(OCC(F)(F)F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)C1 |wU:33.37,29.31,(-8.05,-6.16,;-8.05,-4.62,;-9.39,-3.85,;-9.39,-2.31,;-8.05,-1.54,;-6.72,-2.31,;-5.25,-1.83,;-4.35,-3.08,;-5.25,-4.32,;-6.72,-3.85,;-4.78,-5.79,;-5.87,-6.88,;-4.38,-7.28,;-3.29,-6.19,;-4.78,-.37,;-5.81,.78,;-5.33,2.24,;-3.83,2.56,;-3.35,4.03,;-1.84,4.35,;-1.37,5.81,;-.89,7.28,;-2.4,6.96,;.14,6.13,;-2.8,1.42,;-3.27,-.05,;-1.29,1.74,;-.81,3.2,;-.26,.59,;1.25,.91,;2.39,-.12,;3.73,.65,;3.41,2.16,;1.87,2.32,;1.1,3.65,;5.13,.03,;5.29,-1.51,;6.38,.93,;6.62,2.45,;8.14,2.21,;9.39,3.12,;7.9,.69,)|
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(OCC(F)(F)F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(OCC(F)(F)F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)CC1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(OCC(F)(F)F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1(F)CC1
CC(C)CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1OCC(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(OCC(F)(F)F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccccc1F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(OCC(F)(F)F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(O)(C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(OC(F)F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1(F)CC1
C[C@@](O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1OC(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(OC(F)F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(OC(F)F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(F)(F)F
CC(C)CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1OC(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CC(CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1OC(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
CC(C)(O)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1OC(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(OC(F)F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC1(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(OC(F)F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)C1 |wU:31.35,27.29,(-8.05,-5.84,;-8.05,-4.3,;-9.39,-3.53,;-9.39,-1.99,;-8.05,-1.22,;-6.72,-1.99,;-5.25,-1.51,;-4.35,-2.76,;-5.25,-4,;-6.72,-3.53,;-4.78,-5.47,;-5.87,-6.56,;-4.38,-6.96,;-3.29,-5.87,;-4.78,-.05,;-5.81,1.1,;-5.33,2.56,;-3.83,2.88,;-3.35,4.35,;-4.38,5.49,;-5.89,5.17,;-3.91,6.96,;-2.8,1.74,;-3.27,.27,;-1.29,2.06,;-.81,3.52,;-.26,.91,;1.25,1.23,;2.39,.2,;3.73,.97,;3.41,2.48,;1.87,2.64,;1.1,3.97,;5.13,.35,;5.29,-1.18,;6.38,1.25,;6.62,2.77,;8.14,2.53,;9.39,3.44,;7.9,1.01,)|
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(OC(F)F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(O)(C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(OC(F)F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccccc1F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(OC(F)F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)CC1
CC(O)(CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1OC(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
CC(C)(F)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1OC(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CC(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1OC(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(OC(F)F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)C1
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1ccc(OC(F)F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1
CCC(O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1OC(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
CCOc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCOc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C)(O)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCOc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccccc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCOc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)O)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCOc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCOc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCOc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCOc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1(F)CC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCOc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCOc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(O)(C(F)(F)F)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCOc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCOc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)CC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCOc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(O)(CC)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCOc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C(F)(F)F)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCOc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCOc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC1(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCOc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C)C)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCOc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F |wU:16.18,12.12,(-1.37,6.54,;-1.84,5.08,;-3.35,4.76,;-3.83,3.29,;-5.33,2.97,;-5.81,1.51,;-4.78,.36,;-3.27,.69,;-2.8,2.15,;-1.29,2.47,;-.81,3.93,;-.26,1.33,;1.25,1.65,;2.39,.62,;3.73,1.39,;3.41,2.89,;1.87,3.05,;1.1,4.39,;5.13,.76,;5.29,-.77,;6.38,1.66,;6.62,3.19,;8.14,2.94,;9.39,3.85,;7.9,1.42,;-5.25,-1.1,;-4.35,-2.35,;-5.25,-3.59,;-6.72,-3.12,;-8.05,-3.89,;-8.05,-5.43,;-9.39,-3.12,;-9.39,-1.58,;-8.05,-.81,;-6.72,-1.58,;-4.78,-5.06,;-5.87,-6.15,;-4.38,-6.54,;-3.29,-5.45,)|
COc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)O)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C)C)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCC(O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
COc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccccc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(O)(C(F)(F)F)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1(F)CC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)CC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C)(O)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C(F)(F)F)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC1(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F |wU:15.17,11.11,(-1.84,5.81,;-3.35,5.49,;-3.83,4.03,;-5.33,3.71,;-5.81,2.24,;-4.78,1.1,;-3.27,1.42,;-2.8,2.88,;-1.29,3.2,;-.81,4.67,;-.26,2.06,;1.25,2.38,;2.39,1.35,;3.73,2.12,;3.41,3.62,;1.87,3.78,;1.1,5.12,;5.13,1.49,;5.29,-.04,;6.38,2.4,;6.62,3.92,;8.14,3.68,;9.39,4.58,;7.9,2.16,;-5.25,-.37,;-4.35,-1.61,;-5.25,-2.86,;-6.72,-2.38,;-8.05,-3.15,;-8.05,-4.69,;-9.39,-2.38,;-9.39,-.84,;-8.05,-.07,;-6.72,-.84,;-4.78,-4.32,;-5.87,-5.41,;-4.38,-5.81,;-3.29,-4.72,)|
CCC(O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cccc(c1)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
CNc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C(F)(F)F)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CNc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CNc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(O)(C(F)(F)F)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Nc1ncnn2c(cc(CN3CCC(F)(F)CC3)c12)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(CN3CCC(F)(F)CC3)c12)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(O)(C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(CN3CCC(F)(F)CC3)c12)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1
C[C@@](O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1Cl)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12)C(F)(F)F
Nc1ncnn2c(cc(CN3CCC(F)(F)CC3)c12)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)C1 |wU:33.38,29.32,(-8.05,-4.22,;-8.05,-2.68,;-9.39,-1.91,;-9.39,-.37,;-8.05,.4,;-6.72,-.37,;-5.25,.1,;-4.35,-1.14,;-5.25,-2.39,;-4.78,-3.86,;-3.27,-4.18,;-2.24,-3.03,;-.73,-3.35,;-.26,-4.82,;.89,-5.85,;1.21,-4.34,;-1.29,-5.96,;-2.8,-5.64,;-6.72,-1.91,;-4.78,1.57,;-5.81,2.71,;-5.33,4.18,;-3.83,4.5,;-3.35,5.96,;-2.8,3.35,;-3.27,1.89,;-1.29,3.67,;-.81,5.14,;-.26,2.53,;1.25,2.85,;2.39,1.82,;3.73,2.59,;3.41,4.09,;1.87,4.25,;1.1,5.59,;5.13,1.96,;5.29,.43,;6.38,2.87,;6.62,4.39,;8.14,4.15,;9.39,5.05,;7.9,2.62,)|
Nc1ncnn2c(cc(CN3CCC(F)(F)CC3)c12)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1(F)CC1
CC(C)(F)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1Cl)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
Nc1ncnn2c(cc(CN3CCC(F)(F)CC3)c12)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(F)(F)F
CC(C)CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1Cl)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
Nc1ncnn2c(cc(CN3CCC(F)(F)CC3)c12)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)CC1
Nc1ncnn2c(cc(CN3CCC(F)(F)CC3)c12)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)C1
Nc1ncnn2c(cc(CN3CCC(CC3)C(F)(F)F)c12)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1(F)CC1
CC(CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1Cl)-c1cc(CN2CCC(CC2)C(F)(F)F)c2c(N)ncnn12)C(F)(F)F
Nc1ncnn2c(cc(CN3CCC(CC3)C(F)(F)F)c12)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)C1 |wU:35.40,31.34,(-8.05,-3.9,;-8.05,-2.36,;-9.39,-1.59,;-9.39,-.05,;-8.05,.72,;-6.72,-.05,;-5.25,.42,;-4.35,-.82,;-5.25,-2.07,;-4.78,-3.53,;-3.27,-3.86,;-2.24,-2.71,;-.73,-3.03,;-.26,-4.5,;-1.29,-5.64,;-2.8,-5.32,;1.25,-4.82,;1.72,-6.28,;2.75,-5.14,;2.34,-3.73,;-6.72,-1.59,;-4.78,1.89,;-5.81,3.03,;-5.33,4.5,;-3.83,4.82,;-3.35,6.28,;-2.8,3.67,;-3.27,2.21,;-1.29,3.99,;-.81,5.46,;-.26,2.85,;1.25,3.17,;2.39,2.14,;3.73,2.91,;3.41,4.41,;1.87,4.57,;1.1,5.91,;5.13,2.28,;5.29,.75,;6.38,3.19,;6.62,4.71,;8.14,4.47,;9.39,5.37,;7.9,2.94,)|
CC(C)(F)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1Cl)-c1cc(CN2CCC(CC2)C(F)(F)F)c2c(N)ncnn12
CC(O)(CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1Cl)-c1cc(CN2CCC(CC2)C(F)(F)F)c2c(N)ncnn12)C(F)(F)F
CC(C)CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1Cl)-c1cc(CN2CCC(CC2)C(F)(F)F)c2c(N)ncnn12
Nc1ncnn2c(cc(CN3CCC(CC3)C(F)(F)F)c12)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(F)(F)F
Nc1ncnn2c(cc(CN3CCC(CC3)C(F)(F)F)c12)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(O)(C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(CN3CCC(CC3)C(F)(F)F)c12)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1
Nc1ncnn2c(cc(CN3CCC(CC3)C(F)(F)F)c12)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccccc1F
C[C@@](O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1Cl)-c1cc(CN2CCC(CC2)C(F)(F)F)c2c(N)ncnn12)C(F)(F)F
Nc1ncnn2c(cc(CN3CCC(CC3)C(F)(F)F)c12)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)CC1
Nc1ncnn2c(cc(CN3CCC(CC3)C(F)(F)F)c12)-c1ccc(Cl)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)C1
CC(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1Cl)-c1cc(CN2CCC(CC2)C(F)(F)F)c2c(N)ncnn12)C(F)(F)F
CCC(O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(ccc1Cl)-c1cc(CN2CCC(CC2)C(F)(F)F)c2c(N)ncnn12)C(F)(F)F
Nc1ncnn2c(cc(CN3CC(F)(F)C3)c12)-c1cccc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@H](O)C(F)(F)F
CC(C)CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cccc(c1)-c1cc(CN2CC(F)(F)C2)c2c(N)ncnn12
CC(C)(O)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cccc(c1)-c1cc(CN2CC(F)(F)C2)c2c(N)ncnn12
CC(C)(F)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cccc(c1)-c1cc(CN2CC(F)(F)C2)c2c(N)ncnn12
Nc1ncnn2c(cc(CN3CC(F)(F)C3)c12)-c1cccc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC1
Nc1ncnn2c(cc(CN3CC(F)(F)C3)c12)-c1cccc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(F)(F)F
CC(C)(C)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cccc(c1)-c1cc(CN2CC(F)(F)C2)c2c(N)ncnn12
Nc1ncnn2c(cc(CN3CC(F)(F)C3)c12)-c1cccc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccccc1F
CC(C)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cccc(c1)-c1cc(CN2CC(F)(F)C2)c2c(N)ncnn12
Nc1ncnn2c(cc(CN3CC(F)(F)C3)c12)-c1cccc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccc(F)cc1
Nc1ncnn2c(cc(CN3CC(F)(F)C3)c12)-c1cccc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)C1 |wU:30.35,26.29,(-8.05,-4.19,;-8.05,-2.65,;-9.39,-1.88,;-9.39,-.34,;-8.05,.43,;-6.72,-.34,;-5.25,.14,;-4.35,-1.11,;-5.25,-2.35,;-4.78,-3.82,;-3.27,-4.14,;-1.98,-3.3,;-1.14,-4.59,;0,-5.62,;.32,-4.12,;-2.43,-5.43,;-6.72,-1.88,;-4.78,1.6,;-5.81,2.75,;-5.33,4.21,;-3.83,4.53,;-2.8,3.39,;-3.27,1.92,;-1.29,3.71,;-.81,5.17,;-.26,2.56,;1.25,2.88,;2.39,1.85,;3.73,2.62,;3.41,4.13,;1.87,4.29,;1.1,5.62,;5.13,2,;5.29,.46,;6.38,2.9,;6.62,4.42,;8.14,4.18,;9.39,5.09,;7.9,2.66,)|
CC(C)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cccc(c1)-c1cc(CN2CC(F)(F)C2)c2c(N)ncnn12)C(F)(F)F
Nc1ncnn2c(cc(CN3CC(F)(F)C3)c12)-c1cccc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC1(F)F
Nc1ncnn2c(cc(CN3CC(F)(F)C3)c12)-c1cccc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)C1
Nc1ncnn2c(cc(CN3CC(F)(F)C3)c12)-c1cccc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)CC1
C[C@@](O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cccc(c1)-c1cc(CN2CC(F)(F)C2)c2c(N)ncnn12)C(F)(F)F
Nc1ncnn2c(cc(CN3CC(F)(F)C3)c12)-c1cccc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1
Cc1nc(C)c(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1(F)CC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1nc(C)c(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1nc(C)c(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccc(F)cc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1nc(C)c(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1nc(C)c(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccccc1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F
CC(CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(-c2cc(c3c(N)ncnn23)C(F)(F)F)c(C)nc1C)C(F)(F)F
Cc1nc(C)c(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1c(F)cncc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1nc(C)c(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccccc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1nc(C)c(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccccc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1nc(C)c(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1cccc(F)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1nc(C)c(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccncc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1nc(C)c(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C(F)(F)F)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1nc(C)c(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C)(O)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CC(C)CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(-c2cc(c3c(N)ncnn23)C(F)(F)F)c(C)nc1C
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COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC1CC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC1CCCC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC1CCC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC1CC1(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC1CC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC1(C)CC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC1(O)CCCCC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ccnc(n1)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cnc1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1cccnn1)-c1cc(c2c(N)ncnn12)C(F)(F)F
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COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC1CCCCC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
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COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C(F)(F)F)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
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COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C)(O)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
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COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccncc1)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccc(Cl)cc1)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1cccc(F)c1)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccccc1Cl)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1cc(F)ccc1F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1c(F)cccc1F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1c(F)cncc1F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ncccc1Cl)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1(F)CC1)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C)(O)C(F)(F)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C)C)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccnc(C)c1)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C(F)(F)F)C(F)(F)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccncc1F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1c(F)cc(F)cc1F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1cnccc1Cl)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccc(F)cc1Cl)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccccn1)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1cnccc1C(F)(F)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1cscn1)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccc(Cl)cn1)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C)C(F)(F)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1cc(C)ncc1F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)O)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(F)(F)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccc(F)c(F)c1)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ncc(F)cc1F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccc(F)cn1)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1cccc(F)c1Cl)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)C(F)(F)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1cc(F)cc(F)c1)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccncc1Cl)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
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COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)C(F)(F)F)-c1cc(CN2CC(F)(F)C2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)C)-c1cc(CN2CC(F)(F)C2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)CC(F)(F)F)-c1cc(CN2CC(F)(F)C2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)CCC(F)(F)F)-c1cc(CN2CC(F)(F)C2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)c1ccc(F)cc1)-c1cc(CN2CC(F)(F)C2)c2c(N)ncnn12
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COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)c1cn(C)nc1C(F)(F)F)-c1cc(CN2CC(F)(F)C2)c2c(N)ncnn12
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COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)C1CC1)-c1cc(CN2CC(F)(F)C2)c2c(N)ncnn12
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COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(C)(=O)=O)-c1cc(CN2CC(F)(F)C2)c2c(N)ncnn12
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COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)CCc1ccccc1)-c1cc(CN2CC(F)(F)C2)c2c(N)ncnn12
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COc1ncc(cc1C(=O)Nc1nc(co1)C(=O)NCC1CC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)Nc1nc(co1)C(=O)NC(C)C)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)Nc1nc(co1)C(=O)NC1CCCC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCCN(CC1CC1)C(=O)c1coc(NC(=O)c2cc(cnc2OC)-c2cc(c3c(N)ncnn23)C(F)(F)F)n1
COc1ncc(cc1C(=O)Nc1ncc(s1)C(=O)NCc1cc(OC(F)(F)F)ccc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CC(C)(F)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(-c2cc(CN3CC(F)(F)C3)c3c(N)ncnn23)c(F)cc1Cl
Nc1ncnn2c(cc(CN3CC(F)(F)C3)c12)-c1cc(C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)CC(F)(F)F)c(Cl)cc1F
CC(C)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(-c2cc(CN3CC(F)(F)C3)c3c(N)ncnn23)c(F)cc1Cl)C(F)(F)F
Nc1ncnn2c(cc(CN3CC(F)(F)C3)c12)-c1cc(C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)C2CC(F)(F)C2)c(Cl)cc1F
Nc1ncnn2c(cc(CN3CC(F)(F)C3)c12)-c1cc(C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)C2CCC(F)(F)C2)c(Cl)cc1F
Nc1ncnn2c(cc(CN3CC(F)(F)C3)c12)-c1cc(C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)C2CC(F)C2)c(Cl)cc1F |wU:27.31,23.25,(-8.05,-4.38,;-8.05,-2.84,;-9.39,-2.07,;-9.39,-.53,;-8.05,.24,;-6.72,-.53,;-5.25,-.05,;-4.35,-1.3,;-5.25,-2.54,;-4.78,-4.01,;-3.27,-4.33,;-1.98,-3.49,;-1.14,-4.78,;0,-5.81,;.32,-4.3,;-2.43,-5.62,;-6.72,-2.07,;-4.78,1.42,;-3.27,1.74,;-2.8,3.2,;-1.29,3.52,;-.81,4.98,;-.26,2.38,;1.25,2.7,;2.39,1.67,;3.73,2.44,;3.41,3.94,;1.87,4.1,;1.1,5.44,;5.13,1.81,;5.29,.28,;6.38,2.71,;6.62,4.24,;8.14,3.99,;9.39,4.9,;7.9,2.47,;-3.83,4.34,;-3.35,5.81,;-5.33,4.02,;-5.81,2.56,;-7.31,2.24,)|
C[C@@](O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(-c2cc(CN3CC(F)(F)C3)c3c(N)ncnn23)c(F)cc1Cl)C(F)(F)F
C[C@@](O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(F)cc(c1)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(F)cc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1
CCC(O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(F)cc(c1)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(F)cc(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC11CC1
Cc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(C(F)(F)F)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1cccnc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccncc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1cncc(F)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1c(F)cncc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCC(O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cc(F)c1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
C[C@@](O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cc(F)c1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
C[C@@](O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cc(F)c1F)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(F)c(F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)C1
CC(O)(CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cc(F)c1F)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
CC(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cc(F)c1F)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
Nc1ncnn2c(cc(c12)C(F)(F)F)-c1cc(F)c(F)c(c1)C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1
CCC(O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cc(F)c1F)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
CCc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(c2c(NC(=O)C(C)(C)F)ncnn12)C(F)(F)F |r|
COc1ncc(cc1C(=O)Nc1ncn(Cc2ccccc2)n1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N(C)[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1ncc(cc1C(=O)N(C)[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(OC)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1ncc(cc1C(=O)N[C@H](C)c1cc(OC(F)(F)F)ccc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(C(=O)N2CC(F)(F)C2)c2c(N)ncnn12 |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(C(=O)N2CC(F)(F)C2)c2c(N)ncnn12 |r|
COc1ccc(cc1C(=O)N[C@H](C)c1cc(ccc1F)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1ccc(cc1C(=O)NCc1ccccc1Oc1ccccc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(C[C@@H]1F)C1CC(C)c2ccccc12)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C1CCc2ccccc12)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C1CCc2c1cccc2F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C1CCc2cc(F)ccc12)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C1CCCCc2ccccc12)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C1CCC(C)c2ccccc12)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C1CCCc2c(Br)cccc12)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C1CCc2cccc(Cl)c12)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C1CCCc2ccccc12)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(Cc2cccc(=O)[nH]2)C[C@@H]1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(C)CC(O)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)[C@@H](C)C1CCC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)[C@H](C)CC(O)(c1ccccc1)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(C)CC(O)(C(F)(F)F)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)[C@H](C)C1CCC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)[C@@H](C)CC(O)(c1ccccc1)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C1CCCC1O)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(C)C(C)(C)O)-c1cc(c2c(N)ncnn12)C(F)(F)F
COC(=O)N1C[C@H](F)C(C1)NC(=O)c1cc(cnc1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COCCOC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cnc1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCCOC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cnc1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)Oc1ccccc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCOC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cnc1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCCCOC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cnc1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCC(C)OC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cnc1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)OCC(C)C)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)OCC=C)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)OCC(C)(C)C)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)OC(C)C(C)C)-c1cc(c2c(N)ncnn12)C(F)(F)F
COCC(C)OC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cnc1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)OCC(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)OCC1CCC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCOCCOC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cnc1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)OC1(CC1)C1CC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)OC1CCCC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)OCC#C)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)OC1(C)CC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)O[C@H](C)CO)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)OC1CC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)OC(C(F)(F)F)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(C[C@@H]1F)S(=O)(=O)C(C)C)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)C1CC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)C1CCCCC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)C1CCCC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)C(C)C(C)C)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)C(C)CC(C)C)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)C(C)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)CC(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)\C=C/F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)c1ccc(C)c(C)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ccc(OC)c(c1)S(=O)(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cnc1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)c1cccc2ccccc12)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CCN(C1)S(=O)(=O)Cc1ccc(F)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)Cc1cccc(C)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ccccc1S(=O)(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cnc1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ccc(C)cc1S(=O)(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cnc1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)c1ccccc1C)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)c1cccc(C)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)c1ccc(C)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)C1CCOC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)C1CC2CCC1C2)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)C1CCS(=O)(=O)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCCCS(=O)(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cnc1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)C1CCCCC1O)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)CCC(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)C1CCOCC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)C1=CCCCC1)-c1cc(c2c(N)ncnn12)C(F)(F)F |t:22|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)Cc1cccc(c1)[N+]([O-])=O)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)Cc1ccc(F)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)c1cc(F)ccc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)Cc1cccc(F)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)Cc1cccc(Cl)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)Cc1c(Cl)cccc1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)Cc1ccccc1Cl)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)Cc1ccccn1)-c1cc(c2c(N)ncnn12)C(F)(F)F
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COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)OCCCF)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
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COC(=O)N1C[C@H](F)[C@H](NC(=O)c2cc(cnc2OC)-c2cc(CN3CCC(F)(F)CC3)c3c(N)ncnn23)C1C1CC1(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)OC(C(F)(F)F)C(F)(F)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)OC(C(C)C)C(F)(F)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)OCC(F)(F)C(F)C(F)(F)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)OC(C1CC1)C(F)(F)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)OC(C(C)(C)C)C(F)(F)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)OC(C)C(F)(F)C(F)(F)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)OC1CC(F)(F)C1(F)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)OCC(C)C(F)(F)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
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CCCOC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cnc1OC)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)CCC(F)(F)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
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COc1ncc(cc1C(=O)NC1CN(C[C@@H]1F)C(=O)OCC(F)(F)F)-c1cc(CC2CC(F)(F)C2)c2c(N)ncnn12 |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(CN2CCCC2)c2c(N)ncnn12 |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(CN2CC3(CCC3)C2)c2c(N)ncnn12 |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(CN2CCC(C2)C(F)(F)F)c2c(N)ncnn12 |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(CN2CC(C2)C(F)(F)F)c2c(N)ncnn12 |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)OCC(F)(F)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12 |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(CN2CCC2)c2c(N)ncnn12 |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)OCC(F)(F)F)-c1cc(CN2CCC2)c2c(N)ncnn12 |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(O)(C(F)(F)F)C(F)(F)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12 |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@H]1CC1(F)F)-c1cc(CN2CC(F)(F)C2)c2c(N)ncnn12 |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@H]1CC1(F)F)-c1cc(CN2CC(F)(F)C2)c2c(N)ncnn12 |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@H]1CC1(F)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12 |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@H]1CC1(F)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12 |r|
Cc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)OC(C)(C)C)-c1cc(CN2CC(F)(F)C2)c2c(N)ncnn12 |r|
Cc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(CN2CC(F)(F)C2)c2c(N)ncnn12 |r|
Cc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(CN2CC(F)(F)C2)c2c(N)ncnn12 |r|
Cc1c(F)cc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC1(F)F)-c1cc(CN2CC(F)(F)C2)c2c(N)ncnn12 |r|
CO\N=C(/C)c1cc(-c2cnc(OC)c(c2)C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)[C@@](C)(O)C(F)(F)F)n2ncnc(N)c12 |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(C2CC2)c2c(N)ncnn12 |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(C2CC2)c2c(N)ncnn12 |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(-c2cncc(c2)C#N)c2c(N)ncnn12 |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(C#N)c2c(N)ncnn12 |r|
COc1cc(F)c(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12 |r|
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)OCC(F)(F)F)-c1cc(CN2CCC(CC2)C(F)(F)F)c2c(N)ncnn12 |r|
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)OCC(F)(F)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12 |r|
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)OCC(F)(F)F)-c1cc(CN2CCS(=O)(=O)CC2)c2c(N)ncnn12 |r|
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)OCC(F)(F)F)-c1cc(CN2CCOCC2)c2c(N)ncnn12 |r|
Cc1cc(F)c(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12 |r|
COc1ncc(cc1C(=O)NC1CN(CCC1F)C(=O)C1CC1(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@H]1CN(CC[C@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(CN2CCC(F)(F)C2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(CN2CC(F)C2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(CN2CCCCC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(CN2CC(C)(C)C2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(CN2CCC[C@H]2C(F)(F)F)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(CN2CCCC(C2)C(F)(F)F)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(CN2CCCC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(CN2CCC(F)(F)C2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(CN2CC(C2)C(F)(F)F)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(C(C)=O)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(C)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(Cl)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1ccc2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(CN2CCC(CC2)C(F)(F)F)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(CN2CCC(CC2)C(F)(F)F)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(-c2ccc(N)cc2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(CN2CCc3ccccc3C2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(OS(=O)(=O)c2ccc(C)cc2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(C(F)F)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1c(F)cc2c(N)ncnn12
COc1cc(-c2cnc(OC)c(c2)C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)[C@@](C)(O)C(F)(F)F)n2ncnc(N)c12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(F)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(OC(F)F)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(CN2CC3C(C2)C3(F)F)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(CN2[C@H]3CC[C@@H]2CC(F)(F)C3)c2c(N)ncnn12 |TLB:29:30:35.36.39:32.33|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(CN2CCC(C)(C)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(CN2CCC3(CC3(F)F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(CN2[C@H]3CC[C@@H]2CC(F)(F)C3)c2c(N)ncnn12 |TLB:28:29:34.35.38:31.32|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)OCC(F)(F)F)-c1cc(CN2CCC3(CC3(F)F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)OCC(F)(F)F)-c1cc(CN2CCC(CC2)C(F)(F)F)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccccc1F)-c1cc(CN2CCC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC1(F)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)C(F)(F)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CCC(F)(F)C1)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
CCC(O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cnc1OC)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1ccccc1F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1cc(F)c(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1cc(F)c(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC1(F)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1cc(F)c(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(O)(C(F)(F)F)C(F)(F)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1cc(F)c(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
CCC(O)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(-c2cc(CN3CCC(F)(F)CC3)c3c(N)ncnn23)c(F)cc1OC)C(F)(F)F
COc1cc(F)c(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)C(F)(F)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1cc(F)c(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(CN2CCC(CC2)C(F)(F)F)c2c(N)ncnn12
COc1cc(F)c(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(CN2CCC(CC2)C(F)(F)F)c2c(N)ncnn12
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(O)(C(F)(F)F)C(F)(F)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(CN2CCC(CC2)C(F)(F)F)c2c(N)ncnn12
Cc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(O)(C(F)(F)F)C(F)(F)F)-c1cc(CN2CCC(CC2)C(F)(F)F)c2c(N)ncnn12
Cc1cc(F)c(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC1(F)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
Cc1cc(F)c(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)CC(O)(C(F)(F)F)C(F)(F)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
Cc1cc(F)c(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)C(F)(F)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
Cc1cc(F)c(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
CC(C)CC(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(-c2cc(CN3CCC(F)(F)CC3)c3c(N)ncnn23)c(F)cc1C
Cc1cc(F)c(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)NC1CN(CCC1F)C(=O)CC(O)(C(F)(F)F)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CN(CCC1F)C(=O)C1CC(F)(F)C1)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)NC1CN(CCC1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)NC1CN(CCC1F)C(=O)c1ccccc1F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)NC1CN(CCC1F)C(=O)CC(O)(C(F)(F)F)C(F)(F)F)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1cncs1)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)c1cnc(Cl)s1)-c1cc(c2c(N)ncnn12)C(F)(F)F
CCCC(N)(C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cnc1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)N(C)C(=O)OC(C)(C)C)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(O)(O)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1(CC1)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1(CCN(C1)C(=O)OC(C)(C)C)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)(C)CNC(=O)OC(C)(C)C)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1(C)COC(C)(C)OC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(C)(C)C(C)=O)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1ncc(cc1C(=O)Nc1nnc(Cc2ccccc2)o1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)Nc1ncc(Cc2ccccc2)s1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@H]1CC[C@H](C1)c1ccc(Br)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1ncc(cc1C(=O)NC1CCC(C1)c1ccccc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CCCC(C1)c1ccccc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CCC(O)(C1)c1ccccc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NC1CCCCC(C1)c1ccccc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CCC[C@H](C1)c1ccccc1)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1ncc(cc1C(=O)N[C@H]1CCC[C@H](C1)c1ccccc1)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1ncc(cc1C(=O)NC1CCCN(C1)c1ccccc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@H]1CCC[C@H](C1)c1ccccc1)-c1cc(CN2CCC(F)(F)CC2)c2c(N)ncnn12 |r|
COc1ncc(cc1C(=O)N[C@H]1CCC[C@H](C1)c1ccc(F)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1ncc(cc1C(=O)N[C@H]1C[C@@H]1c1ccccc1)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1ncc(cc1C(=O)N[C@H]1CCC[C@H](C1)c1ccc(Cl)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COC[C@@H]1C[C@@H](CN1C(=O)OC(C)(C)C)NC(=O)c1cc(cnc1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COC[C@@H]1C[C@@H](CN1C(=O)C1CC(F)(F)C1)NC(=O)c1cc(cnc1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1ncc(cc1C(=O)N[C@H]1C[C@@H](COCc2ccccc2)N(C1)C(=O)C1CC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1ccc2c(N)nc(F)nn12 |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(Cn2ccnc2C)c2c(N)ncnn12 |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(Cn2cnc(C)c2)c2c(N)ncnn12 |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(Cn2cnc(Cl)c2)c2c(N)ncnn12 |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(Cn2cncn2)c2c(N)ncnn12 |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(Cn2cnc3ccccc23)c2c(N)ncnn12 |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(Cn2cccn2)c2c(N)ncnn12 |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(Cn2cnnn2)c2c(N)ncnn12 |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(Cn2cnc(c2)-c2ccccc2)c2c(N)ncnn12 |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(Cn2cncc2-c2ccccc2)c2c(N)ncnn12 |r|
CONCc1cc(-c2cnc(OC)c(c2)C(=O)N[C@@H]2CN(C[C@@H]2F)C(=O)C2CC(F)(F)C2)n2ncnc(N)c12 |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(CN2CCCC(=O)N2)c2c(N)ncnn12 |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C1CC(F)(F)C1)-c1cc(CN2CCCCN2)c2c(N)ncnn12 |r|
COc1ccc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)OCC(F)(F)F)-c1cc(CN2CCOCC2)c2c(N)ncnn12 |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)CCC(F)(F)F)-c1cc(CN2CCOCC2)c2c(N)ncnn12 |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)S(=O)(=O)CC(F)(F)F)-c1cc(CN2CCOCC2)c2c(N)ncnn12 |r|
Cc1ncc(cc1C(=O)NCCN1CCOC(C1)c1ccccc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)NCCN1CCOCC1c1ccccc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NCCN1CCCC(C1)c1ccccc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)Nc1ccn(Cc2ccccc2)n1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)Nc1ccn(Cc2ccccc2)n1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)NCC(C)(O)Cc1ccc(F)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)N1CCCC(C1)C(O)c1ccc(F)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NCC(C)(O)Cc1ccc(F)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N1CCCC(C1)C(O)c1ccc(F)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)N1CCCC(C)(C1)C(O)c1ccc(F)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N1CCCC(O)(Cc2ccc(F)cc2)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)N1CCCC(O)(Cc2ccc(F)cc2)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NCC(C)(O)C(O)c1ccc(F)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)NCC(C)(O)C(O)c1ccc(F)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)NCC(C)(O)CC(C)(C)C)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N1CCCC(O)(C1)C(O)c1ccc(F)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)N1CCCC(O)(C1)C(O)c1ccc(F)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)N1CC(O)CC(O)(Cc2ccc(F)cc2)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)NCC(O)CC(O)(C(F)(F)F)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COC(c1ccc(F)cc1)C(C)(O)CNC(=O)c1cc(cnc1C)-c1cc(c2c(N)ncnn12)C(F)(F)F
CO[C@H](c1ccc(F)cc1)C(C)(O)CNC(=O)c1cc(cnc1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
CO[C@@H](c1ccc(F)cc1)C(C)(O)CNC(=O)c1cc(cnc1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COC(C(C)C(F)(F)F)C(C)(O)CNC(=O)c1cc(cnc1C)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)NCC(C)(O)C(=O)c1ccc(F)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)NCC(C)(O)C(O)c1ccccc1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)NCC(C)(O)C(O)c1cccc(F)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)NCC(C)(O)C(O)c1ccc(F)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COC(c1ccc(F)cc1)C(C)(O)CNC(=O)c1cc(ccc1C)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)NCC(C)(O)C(OC(F)F)c1ccc(F)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NCC(C)(O)C(OC(F)F)c1ccc(F)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1NC(=O)CCC(O)c1ccc(Cl)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NCC(O)C(O)c1ccccc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)NCC(O)C(O)c1ccccc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)NCCC(O)C1CC1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)NCC(Cc1ccccc1)NC(=O)OC(C)(C)C)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1NC(=O)c1cn(Cc2ccccc2)cn1)-c1cc(c2c(N)ncnn12)C(F)(F)F
CC(c1ccc(F)cc1)n1cnc(NC(=O)c2cc(cnc2C)-c2cc(c3c(N)ncnn23)C(F)(F)F)c1
COc1ncc(cc1C(=O)Nc1cn(cn1)C(C)c1ccc(F)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)Nc1cnn(Cc2cc(OC(F)(F)F)ccc2F)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)Nc1cnn(c1)C(C)c1ccc(F)cc1)-c1cc(c2c(N)ncnn12)C(F)(F)F
CC(c1ccc(F)cc1)n1cc(NC(=O)c2cc(cnc2C)-c2cc(c3c(N)ncnn23)C(F)(F)F)cn1
Cc1ncc(cc1C(=O)Nc1cn(Cc2cc(OC(F)(F)F)ccc2F)cn1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)Nc1cn(CC(C)(O)C(F)(F)F)cn1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)Nc1cn(CC(C)(O)C(F)(F)F)cn1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)Nc1cn(CCC(C)(O)C(F)(F)F)cn1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)NCCC(O)(C(F)(F)F)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)NCCC(O)(C(F)(F)F)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)Nc1cn(CCc2ccccc2)cn1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)Nc1cn(CCc2ccccc2)cn1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)Nc1cnn(CCc2ccccc2)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)Nc1cnn(CCc2ccccc2)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)Nc1cnn(CC(C)(O)C(F)(F)F)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)Nc1cnn(CC(C)(O)C(F)(F)F)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)Nc1cnn(CCC(C)(O)C(F)(F)F)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)Nc1cnn(CCC(C)(O)C(F)(F)F)c1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)Nc1cn(Cc2ccccc2)cn1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)Nc1ccn(Cc2ccccc2)n1)-c1cc(c2c(N)ncnn12)C(F)(F)F
CC(c1ccc(F)cc1)n1cc(NC(=O)c2cc(ccc2C)-c2cc(c3c(N)ncnn23)C(F)(F)F)cn1
Cc1c(NC(=O)c2cc(ccc2C)-c2cc(c3c(N)ncnn23)C(F)(F)F)ncn1Cc1ccccc1
COc1ncc(cc1C(=O)Nc1cn(cn1)C(c1ccccc1)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)Nc1cn(cn1)C(c1ccccc1)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)Nc1cn(cn1)C(c1ccccc1)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)Nc1cn(Cc2ccc(F)cc2)cn1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)Nc1cn(Cc2ccc(F)cc2)cn1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)Nc1cn(Cc2ccc(F)cc2)cn1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)Nc1cn(Cc2ccc(cc2)C(F)(F)F)cn1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)Nc1cn(Cc2ccc(cc2)C(F)(F)F)cn1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)Nc1cn(Cc2ccc(cc2)C(F)(F)F)cn1)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)Nc1cn(Cc2ccc(Cl)cc2)cn1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)Nc1cn(Cc2ccc(Cl)cc2)cn1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)Nc1cn(Cc2ccc(Cl)cc2)cn1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)Nc1ccn(Cc2ccc(F)cc2)n1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)Nc1ccn(Cc2ccc(F)cc2)n1)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1cc(NC(=O)c2cc(cnc2C)-c2cc(c3c(N)ncnn23)C(F)(F)F)nn1Cc1ccc(F)cc1
Cc1cc(NC(=O)c2cc(ccc2C)-c2cc(c3c(N)ncnn23)C(F)(F)F)nn1Cc1ccc(F)cc1
Cc1ncc(cc1C(=O)Nc1cnn(c1)C(c1ccccc1)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)Nc1cnn(c1)C(c1ccccc1)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)Nc1ccn(n1)C(c1ccccc1)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)Nc1ccn(n1)C(c1ccccc1)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ccc(cc1C(=O)Nc1cn(cn1)C(c1ccc(F)cc1)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
Cc1ncc(cc1C(=O)Nc1cn(cn1)C(c1ccc(F)cc1)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(CC(C)(O)C(F)(F)F)C[C@@H]1F)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(CC(O)CC(F)(F)F)C[C@@H]1F)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
CCC(O)(CN1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cnc1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(CC(O)(c2ccccc2)C(F)(F)F)C[C@@H]1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(CC(O)(C2CC2)C(F)(F)F)C[C@@H]1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(CC(O)(c2nccs2)C(F)(F)F)C[C@@H]1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(CC(O)(C(F)(F)F)C(F)(F)F)C[C@@H]1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(CC(O)CF)C[C@@H]1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(CC(O)COC(F)(F)C(F)F)C[C@@H]1F)-c1cc(c2c(N)ncnn12)C(F)(F)F
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)C(C)(N)C(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)[C@@](C)(O)C(F)(F)F)-c1ccc2c(N)ncnn12 |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)N1CCC(F)(F)C1)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)NC1CCCCC1)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)NCC(F)(F)F)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1ncc(cc1C(=O)N[C@@H]1CN(C[C@@H]1F)C(=O)N1CCCCC1)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
CCN(C)C(=O)N1C[C@H](F)[C@@H](C1)NC(=O)c1cc(cnc1OC)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1ncc(cc1C(=O)N[C@@H]1CC2(C[C@@H]1F)OCC(C)(C)CO2)-c1cc(c2c(N)ncnn12)C(F)(F)F |r|
COc1ncc(cc1C(=O)Nc1cc(Cl)n(Cc2ccccc2)n1)-c1cc(c2c(N)ncnn12)C(F)(F)F
O=C(NC1CCc2ccccc2-n2ccnc12)c1n[nH]c(Cc2ccccc2)n1 |w:3.2|
O=C(NC1CCc2ccccc2-n2ccnc12)c1nccc(n1)-c1ccccc1 |w:3.2|
O=C(N[C@H]1COc2ccccc2-n2nnnc12)c1n[nH]c(Cc2ccccc2)n1 |r|
O=C(NC1CCc2ccccc2-n2ccnc12)c1n[nH]c(Cc2ccccc2)n1
Clc1cccc(Cl)c1Cn1cnc(n1)C(=O)NC1CCc2ccccc2-n2ccnc12 |w:17.18|
O=C(N[C@H]1COc2ccccc2-n2nnnc12)c1cc(Cc2ccccc2)on1 |r|
O=C(NC1CCc2ccccc2-n2ccnc12)c1cc(Cc2ccccc2)on1 |w:3.2|
Clc1cccc(Cl)c1Cn1cnc(n1)C(=O)N[C@H]1COc2ccccc2-n2nnnc12 |r|
Clc1cccc(Cl)c1Cn1cnc(n1)C(=O)NC1CCc2ccccc2-n2ccnc12
Fc1ccccc1Cn1cnc(n1)C(=O)NC1CCc2ccccc2-n2ccnc12 |w:16.17|
Clc1cccc(Cl)c1Cc1nc(n[nH]1)C(=O)NC1CCc2ccccc2-n2ccnc12
Cc1cccc(C)c1Cn1cnc(n1)C(=O)N[C@H]1COc2ccccc2-n2nnnc12 |r|
Fc1ccccc1Cn1cnc(n1)C(=O)N[C@H]1COc2ccccc2-n2nnnc12 |r|
Fc1ccc(Cn2cnc(n2)C(=O)N[C@H]2CSc3ccccc3-n3nnnc23)cc1 |r|
O=C(N[C@H]1CSc2ccccc2-n2nnnc12)c1cc(Cc2ccccc2)on1 |r|
O=C(N[C@H]1CSc2ccccc2-n2nnnc12)c1n[nH]c(Cc2ccccc2)n1 |r|
O=C(N[C@H]1CS(=O)(=O)c2ccccc2-n2nnnc12)c1cc(Cc2ccccc2)on1 |r|
O=C(N[C@H]1CS(=O)c2ccccc2-n2nnnc12)c1cc(Cc2ccccc2)on1 |r|
Clc1cccc(Cl)c1Cn1cnc(n1)C(=O)NC1COc2ccccc2-n2cccc12 |w:17.18|
O=C(N[C@H]1CSc2ccccc2-n2c1noc2=O)c1cc(Cc2ccccc2)on1 |r|
Clc1cccc(Cl)c1Cn1cnc(n1)C(=O)NC1CSc2cccn2-n2ccnc12 |w:17.18|
Fc1ccc(Cc2nc(n[nH]2)C(=O)N[C@H]2CSc3ccccc3-n3nnnc23)cc1 |r|
Fc1ccc(Cc2nc(n[nH]2)C(=O)N[C@H]2CSc3ccccc3-n3c2noc3=O)cc1 |r|
Fc1ccc(Cn2cnc(n2)C(=O)N[C@H]2CSc3ccccc3-n3c2noc3=O)cc1 |r|
O=C(N[C@H]1CSc2ccccc2-n2c1noc2=O)c1n[nH]c(Cc2ccccc2)n1 |r|
O=C(NC1COc2ccccc2-n2cccc12)c1n[nH]c(Cc2ccccc2)n1 |w:3.2|
Cc1cn-2c(n1)C(CCc1ccccc-21)NC(=O)c1ncn(Cc2c(Cl)cccc2Cl)n1 |w:6.17|
Clc1cccc(Cl)c1Cn1cnc(n1)C(=O)NC1CCc2ccccc2-n2c1n[nH]c2=O
Fc1ccc(Cc2nc(n[nH]2)C(=O)NC2COc3ccccc3-n3cccc23)cc1 |w:14.14|
Fc1ccccc1Cn1cnc(n1)C(=O)NC1COc2ccccc2-n2cccc12
O=C(NC1CCc2ccc(CN3CCN(CC3)c3ccncc3)cc2-n2ccnc12)c1n[nH]c(Cc2ccccc2)n1
O=C(N[C@H]1COc2ccccc2-n2c1noc2=O)c1n[nH]c(Cc2ccccc2)n1 |r|
Clc1cccc(Cl)c1Cn1cnc(n1)C(=O)N[C@H]1COc2ccccc2-n2c1noc2=O |r|
O=C(N[C@H]1COc2ccccc2-n2c1noc2=O)c1cc(Cc2ccccc2)on1 |r|
Cc1cnc2C(CCc3ccccc3-n12)NC(=O)c1ncn(Cc2c(Cl)cccc2Cl)n1
O=C(NC1CSc2cccn2-n2ccnc12)c1n[nH]c(Cc2ccccc2)n1
O=C(N[C@H]1COc2ncccc2-n2c1noc2=O)c1cc(Cc2ccccc2)on1 |r|
Clc1cccc(Cl)c1Cn1cnc(n1)C(=O)NC1CCc2ccc(CN3CCN(CC3)c3ccncc3)cc2-n2ccnc12
O=C(NC1CCc2ccccc2-n2c1noc2=O)c1n[nH]c(Cc2ccccc2)n1
Fc1ccc(Cc2nc(n[nH]2)C(=O)N[C@H]2COc3ccccc3-n3c2noc3=O)c(F)c1 |r|
Fc1ccc(Cc2nc(n[nH]2)C(=O)N[C@H]2COc3ccccc3-n3c2noc3=O)cc1 |r|
O=C(NC1CCc2ccccc2-n2ccnc12)c1cc(Oc2ccccc2)ccn1
O=C(NC1CCc2ccccc2-n2c1noc2=O)c1cc(Oc2ccccc2)ccn1
O=C(N[C@H]1COc2ccccc2-n2c1noc2=O)c1cc(Oc2ccccc2)ccn1 |r|
O=C(NC1COc2ccccc2-n2cccc12)c1cc(Oc2ccccc2)ccn1
CC(C)(O)C#Cc1ccc2CCC(NC(=O)c3n[nH]c(Cc4ccccc4)n3)c3nccn3-c2c1
CC(C)(O)C#Cc1ccc2CCC(NC(=O)c3cc(Oc4ccccc4)ccn3)c3nccn3-c2c1
O=C(NC1CCc2ccccc2-n2cnnc12)c1n[nH]c(Cc2ccccc2)n1
Clc1cccc(Cl)c1Cn1cnc(n1)C(=O)NC1CCc2ccccc2-n2cnnc12
O=C(NC1CCc2ccccc2-n2cnnc12)c1cc(Oc2ccccc2)ccn1
Cn1nc2C(CCc3ccccc3-n2c1=O)NC(=O)c1ncn(Cc2c(Cl)cccc2Cl)n1
Clc1cccc(Cl)c1Cn1cnc(n1)C(=O)NC1CCc2ccc(cc2-n2ccnc12)N1CCC2(CCOCC2)CC1
O=C(NC1CCc2ccc(cc2-n2ccnc12)N1CCC2(CCOCC2)CC1)c1cc(Oc2ccccc2)ccn1
O=C(NC1CCc2ccccc2-n2cnnc12)c1ncn(Cc2ccccc2)n1
O=C(NC1CCc2ccc(cc2-n2ccnc12)N1CCC2(CCOCC2)CC1)c1n[nH]c(Cc2ccccc2)n1
O=C(NC1CCc2ccc(cc2-n2c1noc2=O)N1CCC2(CCOCC2)CC1)c1n[nH]c(Cc2ccccc2)n1
O=C(NC1Cc2ccccc2-n2ccnc12)c1n[nH]c(Cc2ccccc2)n1
O=C(NC1Cc2ccccc2-n2ccnc12)c1cc(Oc2ccccc2)ccn1
CC(C)(O)CCc1ccc2CCC(NC(=O)c3n[nH]c(Cc4ccccc4)n3)c3nccn3-c2c1
CC(C)(O)C#Cc1ccc2OC[C@H](NC(=O)c3n[nH]c(Cc4ccccc4)n3)c3nnnn3-c2c1 |r|
Clc1cnc2C(CCc3ccccc3-n12)NC(=O)c1cc(Cc2ccccc2)on1
CC(C)(O)C#Cc1ccc2CCC(NC(=O)c3n[nH]c(Cc4ccccc4)n3)c3nncn3-c2c1
Clc1nc2C(CCc3ccccc3-n2c1Cl)NC(=O)c1ncn(Cc2c(Cl)cccc2Cl)n1
Clc1cnc2C(CCc3ccccc3-n12)NC(=O)c1ncn(Cc2c(Cl)cccc2Cl)n1
Oc1cc(nn1Cc1ccccc1)C(=O)N[C@H]1COc2ccccc2-n2c1noc2=O |r|
O=C(NC1CCc2ccc(cc2-n2ccnc12)N1CCC2(CCOCC2)CC1)c1ccn(Cc2ccccc2)n1
CN1c2ccc(cc2OC[C@H](N2CCc3c(Cl)n(Cc4ccccc4)nc3C2=O)C1=O)C#CC(C)(C)O |r|
Clc1c2CN([C@H]3COc4ccccc4-n4nnnc34)C(=O)c2nn1Cc1ccccc1 |r|
Clc1nc2C(CCc3ccccc3-n2c1Cl)NC(=O)c1n[nH]c(Cc2ccccc2)n1
Clc1cnc2C(CCc3ccccc3-n12)NC(=O)c1n[nH]c(Cc2ccccc2)n1
CC(C)(O)C#Cc1ccc2CC[C@H](NC(=O)c3n[nH]c(Cc4ccccc4)n3)c3nccn3-c2c1 |r|
O=C(N[C@H]1CCc2ccc(cc2-n2ccnc12)N1CCC2(CCOCC2)CC1)c1n[nH]c(Cc2ccccc2)n1 |r|
O=C(NC1CCc2ccc(cc2-n2ccnc12)N1CC2(C1)CCOCC2)c1n[nH]c(Cc2ccccc2)n1
O=C(NC1CCc2ccc(cc2-n2ccnc12)N1CC2(C1)CCOCC2)c1ccn(Cc2ccccc2)n1
O=C(N[C@H]1CCc2ccc(cc2-n2ccnc12)N1CC2(C1)CCOCC2)c1n[nH]c(Cc2ccccc2)n1 |r|
O=C(NC1COc2ccc(cc2-n2ccnc12)N1CC2(C1)CCOCC2)c1n[nH]c(Cc2ccccc2)n1
O=C(N[C@H]1COc2ccc(cc2-n2ccnc12)N1CC2(C1)CCOCC2)c1cc(Oc2ccccc2)ccn1 |r|
O=C(N[C@H]1COc2ccc(cc2-n2ccnc12)C#Cc1ccccn1)c1n[nH]c(Cc2ccccc2)n1 |r|
CC(C)(O)C#Cc1ccc2OCC(NC(=O)c3n[nH]c(Cc4ccccc4)n3)c3nccn3-c2c1
CC(C)(O)C#Cc1ccc2CCC(NC(=O)n3cc(Cc4ccc(F)cc4)cn3)c3nccn3-c2c1
Cc1cc(=O)c(nn1-c1ccccc1)C(=O)Nc1cccc(Cl)c1F
Cc1cc(=O)c(nn1Cc1ccccc1)C(=O)Nc1cccc(Cl)c1F
Cc1cc(=O)c(nn1-c1ccccc1)C(=O)NCc1cc(F)cc(F)c1
Cc1cc(=O)c(nn1-c1ccccc1)C(=O)Nc1cccc(Cl)c1
Cc1cc(=O)c(nn1-c1ccccc1)C(=O)Nc1cc(Cl)cc(c1)C#N
Cc1cc(=O)c(nn1-c1cccc(Cl)c1F)C(=O)Nc1ccccc1
Cc1cc(=O)c(nn1-c1ccccc1F)C(=O)Nc1cccc(Cl)c1F
Cc1cc(=O)c(nn1-c1cc(F)ccc1F)C(=O)Nc1cccc(Cl)c1F
Cc1cc(=O)c(nn1-c1ccccc1)C(=O)Nc1cncc(Cl)c1
Cc1cc(=O)c(nn1-c1ccccc1)C(=O)Nc1ccn2nccc2c1
Cc1cc(=O)c(nn1-c1ccccc1)C(=O)Nc1cc(Cl)c2ncsc2c1
Cc1cc(=O)c(nn1-c1ccccc1)C(=O)Nc1ccc(N=N)c(N)c1
Cc1nn(C)c(C)c1NC(=O)c1nn(c(C)cc1=O)-c1ccccc1
Cc1cc(NC(=O)c2nn(c(C)cc2=O)-c2ccccc2)ncn1
Cc1noc(C)c1NC(=O)c1nn(c(C)cc1=O)-c1ccccc1
Cc1cc(=O)c(nn1-c1cccc(Cl)c1)C(=O)Nc1cccc(Cl)c1F
Cc1cc(=O)c(nn1-c1ccccc1)C(=O)Nc1cc(N)c(C=N)c(Cl)c1
Cc1n[nH]c(C)c1NC(=O)c1nn(c(C)cc1=O)-c1ccccc1
Cc1nccc(NC(=O)c2nn(c(C)cc2=O)-c2ccccc2)n1
Cc1cc(=O)c(nn1-c1ccccc1)C(=O)Nc1ccc(s1)C#N
Cc1cccc(C)c1NC(=O)c1nn(c(C)cc1=O)-c1ccccc1
Cc1cc(=O)c(nn1-c1ccccc1)C(=O)Nc1c2CCCCc2nc2ccccc12
CC(C)c1cccc(Br)c1NC(=O)c1nn(c(C)cc1=O)-c1ccccc1
Cc1cc(=O)c(nn1-c1ccccc1)C(=O)Nc1c(C)ncnc1C
Cc1cccc(C2CC2)c1NC(=O)c1nn(c(C)cc1=O)-c1ccccc1
CC(C)c1cccc(F)c1NC(=O)c1nn(c(C)cc1=O)-c1ccccc1
Cc1cccc(c1NC(=O)c1nn(c(C)cc1=O)-c1ccccc1)C(C)(C)C
Cc1cccc(c1NC(=O)c1nn(c(C)cc1=O)-c1ccccc1)C(F)(F)F
Cc1cc(=O)c(nn1-c1ccccc1)C(=O)Nc1ccccc1C1CC1
Cc1cnc2ccccc2c1NC(=O)c1nn(c(C)cc1=O)-c1ccccc1
Cc1cc(=O)c(nn1-c1ccccc1)C(=O)Nc1cc2NC(=O)Cc2c(Cl)c1
Cc1cc(=O)c(nn1-c1ccccc1)C(=O)Nc1c2ccccc2nc2ccccc12
CC(C)c1ncnc(C(C)C)c1NC(=O)c1nn(c(C)cc1=O)-c1ccccc1
COCc1cc(=O)c(nn1-c1ccccc1)C(=O)Nc1cccc(Cl)c1F
Cc1cc(=O)c(nn1-c1ccccc1)C(=O)NC1CCc2ccccc2NC1=O
Cc1c(Cl)c(=O)c(nn1-c1ccccc1)C(=O)NC1CCc2ccccc2NC1=O
Cc1c(Cl)c(=O)c(nn1-c1ccccc1)C(=O)NC1CCc2cc(Cl)ccc2NC1=O
CN1c2ccccc2CCC(NC(=O)c2nn(c(C)cc2=O)-c2ccccc2)C1=O
Cc1c(Br)c(=O)c(nn1-c1ccccc1)C(=O)NC1CCc2ccccc2NC1=O
Cc1c(Br)c(=O)c(nn1-c1ccccc1)C(=O)NC1CCc2cc(Br)ccc2NC1=O
Cc1c(Br)c(=O)c(nn1-c1ccccc1)C(=O)NC1CCc2cc(ccc2NC1=O)C#N
CN1c2ccc(Cl)cc2CCC(NC(=O)c2nn(-c3ccccc3)c(C)c(Cl)c2=O)C1=O
CN1c2ccc(Cl)cc2CCC(NC(=O)c2nn(-c3ccccc3)c(CCl)c(Cl)c2=O)C1=O
CN1c2ccccc2CCC(NC(=O)c2nn(-c3ccccc3)c(C)c(C#N)c2=O)C1=O
Cc1cc(=O)c(nn1-c1ccccc1)C(=O)NC1CCc2cc(F)cc(F)c2NC1=O
CN1c2c(F)cc(F)cc2CCC(NC(=O)c2nn(c(C)cc2=O)-c2ccccc2)C1=O
CN1c2ncccc2OC[C@H](NC(=O)c2nn(c(C)cc2=O)-c2ccccc2)C1=O |r|
Cc1ccc(cn1)-n1nc(C(=O)NC2CCc3ccccc3NC2=O)c(=O)cc1C
Cc1ccc(cc1F)-n1nc(C(=O)NC2CCc3ccccc3NC2=O)c(=O)cc1C
Cc1cc(=O)c(nn1-c1cccc(c1)C#N)C(=O)NC1CCc2ccccc2NC1=O
Cc1cc(=O)c(nn1-c1cccc(F)c1)C(=O)NC1CCc2ccccc2NC1=O
CN1c2ccc(cc2OC[C@H](NC(=O)c2nn(c(C)cc2=O)-c2ccccc2)C1=O)C#N |r|
Cc1cc(=O)c(nn1-c1ccc(cc1)C#N)C(=O)NC1CCc2ccccc2NC1=O
Cc1cc(=O)c(nn1-c1ccc(F)cc1)C(=O)NC1CCc2ccccc2NC1=O
Cc1cc(=O)c(nn1-c1ccccc1F)C(=O)NC1CCc2ccccc2NC1=O
CN1c2ccc(cc2OC[C@H](NC(=O)c2nn(c(C)cc2=O)-c2ccc(cc2)C#N)C1=O)C#N |r|
CN1c2ccc(cc2OC[C@H](NC(=O)c2nn(c(C)cc2=O)-c2cccc(F)c2)C1=O)C#N |r|
CN1c2ccc(cc2OC[C@H](NC(=O)c2nn(c(C)cc2=O)-c2ccc(C)c(F)c2)C1=O)C#N |r|
Cc1cccc(c1)-n1nc(C(=O)NC2CCc3ccccc3NC2=O)c(=O)cc1C
COc1ccc(cc1)-n1nc(C(=O)NC2CCc3ccccc3NC2=O)c(=O)cc1C
Cc1cc(=O)c(nn1-c1ccc(Cl)cc1)C(=O)NC1CCc2ccccc2NC1=O
COc1cccc(c1)-n1nc(C(=O)NC2CCc3ccccc3NC2=O)c(=O)cc1C
Cc1cc(=O)c(nn1-c1cccc(Cl)c1)C(=O)NC1CCc2ccccc2NC1=O
Cc1cc(=O)c(nn1-c1ccccc1)C(=O)NC1CCc2cc(F)cc(F)c2NC1
O=C(NC1CCc2ccccc2NC1=O)c1nn(-c2ccccc2)c2ccccc2c1=O
Cc1ccc(cc1)-n1nc(C(=O)NC2CCc3ccccc3NC2=O)c(=O)cc1C
CN1c2ccnn2CCC(NC(=O)c2nn(c(C)cc2=O)-c2ccccc2)C1=O
Cc1cc(=O)c(nn1-c1ccccc1)C(=O)Nc1nc(c(Br)s1)C(F)(F)F
Cc1cc(=O)c(nn1-c1ccccc1)C(=O)NC(C)(C)C
Cc1nocc1NC(=O)c1nn(c(C)cc1=O)-c1ccccc1
Cc1cc(C)c2nc(NC(=O)c3nn(c(C)cc3=O)-c3ccccc3)sc2c1
COCc1cc(=O)c(nn1C)C(=O)Nc1cccc(Cl)c1F
CC(C)c1nn(C)c(C(C)C)c1NC(=O)c1nn(c(C)cc1=O)-c1ccccc1
CC(C)c1n[nH]c(C(C)C)c1NC(=O)c1nn(c(C)cc1=O)-c1ccccc1
Cc1cc(=O)c(nn1-c1ccccc1)C(=O)NC1CC1
Cc1cc(=O)c(nn1-c1ccccc1)C(=O)Nc1cc(F)cc(F)c1
Cc1cc(=O)c(nn1-c1ccccc1)C(=O)Nc1cccc(F)c1
Cc1ccnc(NC(=O)c2nn(c(C)cc2=O)-c2ccccc2F)c1
Cc1cccc(NC(=O)c2nn(c(C)cc2=O)-c2ccccc2F)n1
CC(NC(=O)c1nn(c(C)cc1=O)-c1ccccc1)C1CC1
Cc1ccc(NC(=O)c2nn(c(C)cc2=O)-c2ccccc2)cc1
Cc1cc(=O)c(nn1-c1ccccc1)C(=O)NC(C1CC1)c1ccccc1
Cc1cccc(NC(=O)c2nn(c(C)cc2=O)-c2ccccc2)n1
Cc1cc(=O)c(nn1-c1ccccc1F)C(=O)Nc1ccc(Cl)cn1
CCn1c(NC(=O)c2nn(c(C)cc2=O)-c2ccccc2)nc2ccccc12
Cc1cc(=O)c(nn1-c1ccccc1Cl)C(=O)Nc1ccccn1
Cc1cc(=O)c(nn1-c1ccc(Cl)cc1)C(=O)Nc1ccccn1
Cc1cc(=O)c(nn1-c1ccccc1)C(=O)NCC1CCC1
CC(NC(=O)c1nn(c(C)cc1=O)-c1ccccc1)c1nc(C)no1
Cc1cc(=O)c(nn1-c1ccccc1)C(=O)Nc1ccccn1
Cc1cccc(NC(=O)c2nn(c(C)cc2=O)-c2ccccc2F)c1
Cc1cc(=O)c(nn1-c1ccccc1)C(=O)Nc1ccccc1F
Cc1cc(=O)c(nn1-c1ccccc1)C(=O)Nc1ccc(F)cc1
Cc1cc(=O)c(nn1-c1ccccc1)C(=O)NCC#C
Cc1cc(NC(=O)c2nn(c(C)cc2=O)-c2ccccc2)sn1
Cc1noc(C2CC2)c1NC(=O)c1nn(c(C)cc1=O)-c1ccccc1
Cc1cc(=O)c(nn1-c1ccccc1)C(=O)N1CCC(C1)Oc1ccccn1
Cc1ccnc(NC(=O)c2nn(c(C)cc2=O)-c2ccccc2)c1
Cc1cc(=O)c(nn1-c1ccccc1)C(=O)Nc1ccncc1
Cc1cc(=O)c(nn1-c1ccccc1)C(=O)Nc1cnns1
CC(C)c1cccc(C(C)C)c1NC(=O)c1nn(c(C)cc1=O)-c1ccccc1
Fc1cccc(Cn2nc3c(CCN(C3=O)c3cccc(Cl)c3F)c2Cl)c1F
Fc1c(Cl)cccc1N1CCc2c(Cl)n(Cc3ccccc3)nc2C1=O
Fc1cc(F)cc(Cn2nc3c(CCN(C3=O)c3cccc(Cl)c3F)c2Cl)c1
Cc1nc(nn1Cc1cnccn1)C(=O)Nc1cccc(Cl)c1F
Cc1cc(nn1Cc1ccccc1)C(=O)Nc1cccc(Cl)c1F
Cc1c(F)c(nn1Cc1ccccc1)C(=O)Nc1cccc(Cl)c1F
Fc1c(Cl)cccc1NC(=O)c1ccn(Cc2ccccc2)n1
Oc1cc(nn1Cc1cnccn1)C(=O)Nc1cccc(Cl)c1F
Fc1c(Cl)cccc1NC(=O)c1n[nH]c(Cc2ccccc2)n1
Cn1nc(nc1Cc1ccccc1)C(=O)Nc1cccc(Cl)c1F
Cn1cc(cn1)-c1cc(F)c(F)c(NC(=O)c2n[nH]c(Cc3ccccc3)n2)c1
Fc1ccccc1Cn1cnc(n1)C(=O)Nc1cccc(Cl)c1F
Cc1nc(nn1Cc1ccccc1)C(=O)Nc1cccc(Cl)c1F
Fc1c(Cl)cccc1NC(=O)c1nc(Cc2ccccc2)c[nH]1
Fc1c(Cl)cccc1N1CCn2cc(Cc3ccccc3)nc2C1=O
Fc1c(Cl)cccc1N1CCn2c(Cl)c(Cc3ccccc3)nc2C1=O
CC1CN(c2cccc(Cl)c2)C(=O)c2nc(Cc3ccccc3)cn2C1
Fc1c(Cl)cccc1NC(=O)c1nc(Cc2ccccc2)c(Cl)[nH]1
Fc1c(Cl)cccc1NC(=O)c1nnc(Cc2ccccc2)o1
Fc1ccccc1NC(=O)c1n[nH]c(Cc2ccccc2)n1
Clc1cccc(NC(=O)c2n[nH]c(Cc3ccccc3)n2)c1
Fc1cccc(NC(=O)c2n[nH]c(Cc3ccccc3)n2)c1F
Fc1cc(F)c(F)c(NC(=O)c2n[nH]c(Cc3ccccc3)n2)c1
Clc1cc(Cl)cc(NC(=O)c2n[nH]c(Cc3ccccc3)n2)c1
Cn1cc(cn1)-c1cc(Cl)c(F)c(NC(=O)c2n[nH]c(Cc3ccccc3)n2)c1
CC(C)(C#N)c1cc(Cl)cc(NC(=O)c2n[nH]c(Cc3ccccc3)n2)c1F
Fc1c(Cl)cccc1NC(=O)c1ncn(Cc2ccccc2)n1
Fc1ccc(NC(=O)c2ncn(Cc3ccccc3)n2)c(F)c1Cl
Fc1c(Cl)cccc1NC(=O)c1ncn(Cc2cccc(c2)C#N)n1
COc1ccc(NC(=O)c2ncn(Cc3ccccc3)n2)c(F)c1Cl
Oc1ccc(NC(=O)c2ncn(Cc3ccccc3)n2)c(F)c1Cl
Fc1c(Cl)cccc1NC(=O)c1ncn(Cc2cnccn2)n1
Fc1c(Cl)cccc1NC(=O)c1ncn(Cc2ccc(cc2)C#N)n1
Cc1nc(nn1Cc1cccc(c1)C#N)C(=O)Nc1cccc(Cl)c1F
Fc1c(Cl)cc(cc1NC(=O)c1ncn(Cc2ccccc2)n1)C#N
Cn1cc(cn1)-c1cc(Cl)c(F)c(NC(=O)c2ncn(Cc3ccccc3)n2)c1
Fc1c(NC(=O)c2ncn(Cc3ccccc3)n2)ccc(Cl)c1Cl
Fc1c(Cl)cc(cc1NC(=O)c1ncn(Cc2ccccc2)n1)C(F)(F)F
Fc1c(NC(=O)c2ncn(Cc3ccccc3)n2)ccc(C#N)c1Cl
Fc1c(NC(=O)c2ncn(Cc3ccccc3)n2)ccc(Br)c1Cl
CN(C(=O)c1ncn(Cc2ccccc2)n1)c1ccc(CO)c(Cl)c1F
Clc1c(Cc2ccccc2)nc2C(=O)N(CCn12)c1cccc(Cl)c1
Clc1cccc(c1)N1CCn2cc(Cc3ccccc3)nc2C1=O
Cn1cc(nc1Cc1ccccc1)C(=O)Nc1cccc(Cl)c1F
Fc1c(Cl)cccc1NC(=O)c1c[nH]c(Cc2ccccc2)n1
F[C@H]1C[C@@H](c2ccccc2)n2nc(nc12)C(=O)Nc1cccc(Cl)c1F |r|
Fc1ccccc1N1Cc2ccc(Cc3ccccc3)cc2C1=O
Fc1ccccc1N1Cc2ccc(Cc3ccccc3)nc2C1=O
Fc1ccc(F)c(Cn2nc3c(CCN(C3=O)c3cccc(Cl)c3F)c2Cl)c1
Fc1cc(OC(F)(F)F)ccc1NC(=O)c1ncn(Cc2ccccc2)n1
Cc1nc(nn1Cc1ccccc1)C(=O)Nc1ccc(OC(F)(F)F)cc1
Cc1cc(NC(=O)c2ncn(Cc3ccccc3)n2)ccc1OC(F)(F)F
Fc1cncc(Cn2nc3c(CCN(C3=O)c3cccc(Cl)c3F)c2Cl)c1
CC(c1cccc(F)c1F)n1nc2c(CCN(C2=O)c2cccc(Cl)c2F)c1Cl
C[C@H](c1cccc(F)c1F)n1nc2c(CCN(C2=O)c2cccc(Cl)c2F)c1Cl |r|
C[C@@H](c1cccc(F)c1F)n1nc2c(CCN(C2=O)c2cccc(Cl)c2F)c1Cl |r|
CC(c1cccc(c1)C#N)n1cnc(n1)C(=O)Nc1cccc(Cl)c1F
C[C@H](c1cccc(c1)C#N)n1cnc(n1)C(=O)Nc1cccc(Cl)c1F |r|
C[C@@H](c1cccc(c1)C#N)n1cnc(n1)C(=O)Nc1cccc(Cl)c1F |r|
COc1c2CCN(C(=O)c2nn1Cc1cc(F)ccc1F)c1cccc(Cl)c1F
NC(=O)c1cccc(Cn2nc3c(CCN(C3=O)c3cccc(Cl)c3F)c2Cl)c1
Cc1ccc(Cn2cnc(n2)C(=O)Nc2cccc(Cl)c2F)cc1
Cc1ccc(Cn2cnc(n2)C(=O)Nc2cccc(Cl)c2F)cc1F
Fc1cccc(Cn2cnc(n2)C(=O)Nc2cccc(Cl)c2F)c1
Fc1ccc(Cn2cnc(n2)C(=O)Nc2cccc(Cl)c2F)nc1
Cc1ccc(Cn2cnc(n2)C(=O)Nc2cccc(Cl)c2F)cn1
O=C(Nc1cccc2nn[nH]c12)c1ncn(Cc2ccccc2)n1
Fc1ccc(F)c(Cn2nc3c(CCN(C3=O)c3cccc(Cl)c3F)c2Br)c1
Fc1cccnc1Cn1cnc(n1)C(=O)Nc1cccc(Cl)c1F
Fc1cncc(Cn2cnc(n2)C(=O)Nc2cccc(Cl)c2F)c1
CN(C[C@@H](O)Cc1ccccc1)C(=O)c1cncc(c1)C#Cc1cnn(C)c1 |r|
CN(C[C@@H](O)Cc1ccccc1)C(=O)c1cncc(c1)C#Cc1cnn(c1)C(F)F |r|
CN(C[C@@H](O)Cc1ccccc1)C(=O)c1cncc(c1)C#Cc1cnn(C)n1 |r|
CN(C[C@@H](O)Cc1ccccc1)C(=O)c1cncc(c1)C#Cc1cnn(c1)C(F)(F)F |r|
CN(C[C@@H](O)Cc1ccccc1)C(=O)c1cncc(c1)C#Cc1cnn(c1)C1CC1 |r|
CN(C[C@@H](O)Cc1ccccc1)C(=O)c1cncc(c1)C#Cc1cnn(c1)C1CCC1 |r|
CN(C[C@@H](O)[C@@H](F)c1ccccc1)C(=O)c1cncc(c1)C#Cc1cnn(C)c1 |r|
CN(C[C@@H](O)Cc1ccccc1)C(=O)c1cncc(c1)C#Cc1cnn2CCOCc12 |r|
CN(C[C@H](O)Cc1ccccc1)C(=O)c1cnc(C(F)F)c(c1)C#Cc1cnn(C)c1 |r|
CN(C[C@@H](O)Cc1ccccc1)C(=O)c1cncc(c1)C#Cc1cnn(n1)C1COC1 |r|
CN(C[C@@H](O)Cc1ccccc1)C(=O)c1cncc(c1)C#Cc1cnn(C)c1C1CC1 |r|
CN(C[C@@H](O)Cc1cccc(F)c1)C(=O)c1cncc(c1)C#Cc1cnn(C)c1 |r|
COc1ncc(cc1C#Cc1cnn(C)c1)C(=O)N(C)C[C@@H](O)Cc1ccccc1 |r|
CN(C[C@@H](O)Cc1ccccc1)C(=O)c1cnc(C)c(c1)C#Cc1cnn(C)c1 |r|
CN(C[C@@H](O)Cc1ccccc1)C(=O)c1cncc(c1)C#Cc1cnc(C)s1 |r|
CN(C[C@@H](O)Cc1ccccc1)C(=O)c1cnc(C)c(c1)C#Cc1cncs1 |r|
CN(C[C@@H](O)Cc1ccccc1)C(=O)c1cncc(c1)C#Cc1cnc(C)o1 |r|
CN(C[C@@H](O)Cc1ccccc1)C(=O)c1cncc(c1)C#Cc1cnn(C(F)F)c1C
COc1ccc(CNC(=O)c2c[nH]c3ccc(cc23)-c2ccc3nc(NC(=O)C4CC4)sc3c2)cc1
Fc1ccc(CNC(=O)c2c[nH]c3ccc(cc23)-c2ccc3nc(NC(=O)C4CC4)sc3c2)cc1F
Fc1cc(F)cc(CNC(=O)c2c[nH]c3ccc(cc23)-c2ccc3nc(NC(=O)C4CC4)sc3c2)c1
Fc1cccc(CNC(=O)c2c[nH]c3ccc(cc23)-c2ccc3nc(NC(=O)C4CC4)sc3c2)c1
FC(F)(F)c1cc(CNC(=O)c2c[nH]c3ccc(cc23)-c2ccc3nc(NC(=O)C4CC4)sc3c2)cc(c1)C(F)(F)F
Fc1ccc(CNC(=O)c2c[nH]c3ccc(cc23)-c2ccc3nc(NC(=O)C4CC4)sc3c2)cc1
O=C(Nc1nc2ccc(cc2s1)-c1ccc2[nH]cc(C(=O)NCc3ccc(cc3)C#N)c2c1)C1CC1
FC(F)(F)c1cccc(CNC(=O)c2c[nH]c3ccc(cc23)-c2ccc3nc(NC(=O)C4CC4)sc3c2)c1
Fc1ccc(CNC(=O)c2c[nH]c3ccc(cc23)-c2ccc3nc(NC(=O)C4CC4)sc3c2)c(F)c1
[O-][N+](=O)c1cccc(CNC(=O)c2c[nH]c3ccc(cc23)-c2ccc3nc(NC(=O)C4CC4)sc3c2)c1
COc1cc(CNC(=O)c2c[nH]c3ccc(cc23)-c2ccc3nc(NC(=O)C4CC4)sc3c2)cc(OC)c1
COc1cccc(CNC(=O)c2c[nH]c3ccc(cc23)-c2ccc3nc(NC(=O)C4CC4)sc3c2)c1
Cc1ccc(CNC(=O)c2c[nH]c3ccc(cc23)-c2ccc3nc(NC(=O)C4CC4)sc3c2)cc1
O=C(Nc1nc2ccc(cc2s1)-c1ccc2[nH]cc(C(=O)NCc3cccc4ccccc34)c2c1)C1CC1
Cc1cccc(CNC(=O)c2c[nH]c3ccc(cc23)-c2ccc3nc(NC(=O)C4CC4)sc3c2)c1
FC(F)(F)c1ccc(CNC(=O)c2c[nH]c3ccc(cc23)-c2ccc3nc(NC(=O)C4CC4)sc3c2)cc1
O=C(Nc1nc2ccc(cc2s1)-c1ccc2[nH]cc(C(=O)NCc3ccco3)c2c1)C1CC1
O=C(Nc1nc2ccc(cc2s1)-c1ccc2[nH]cc(C(=O)NCc3cccs3)c2c1)C1CC1
FC(F)(F)Oc1cccc(CNC(=O)c2c[nH]c3ccc(cc23)-c2ccc3nc(NC(=O)C4CC4)sc3c2)c1
O=C(Nc1nc2ccc(cc2s1)-c1ccc2[nH]cc(C(=O)NCc3ccncc3)c2c1)C1CC1
Fc1ccccc1CNC(=O)c1c[nH]c2ccc(cc12)-c1ccc2nc(NC(=O)C3CC3)sc2c1
Clc1cccc(CNC(=O)c2c[nH]c3ccc(cc23)-c2ccc3nc(NC(=O)C4CC4)sc3c2)c1
Brc1cccc(CNC(=O)c2c[nH]c3ccc(cc23)-c2ccc3nc(NC(=O)C4CC4)sc3c2)c1
FC(F)(F)c1ccccc1CNC(=O)c1c[nH]c2ccc(cc12)-c1ccc2nc(NC(=O)C3CC3)sc2c1
Fc1ccc(F)c(CNC(=O)c2c[nH]c3ccc(cc23)-c2ccc3nc(NC(=O)C4CC4)sc3c2)c1
COc1ccc(CNC(=O)c2c[nH]c3ccc(cc23)-c2ccc3nc(NC(=O)C4CC4)sc3c2)cc1OC
O=C(Nc1nc2ccc(cc2s1)-c1ccc2[nH]cc(C(=O)NCc3ccccc3)c2c1)C1CC1
CC(C)c1ccc(CNC(=O)c2c[nH]c3ccc(cc23)-c2ccc3nc(NC(=O)C4CC4)sc3c2)cc1
CC(C)(C)c1ccc(CNC(=O)c2c[nH]c3ccc(cc23)-c2ccc3nc(NC(=O)C4CC4)sc3c2)cc1
C[C@H](NC(=O)c1c[nH]c2ccc(cc12)-c1ccc2nc(NC(=O)C3CC3)sc2c1)c1ccc(F)cc1 |r|
C[C@@H](NC(=O)c1c[nH]c2ccc(cc12)-c1ccc2nc(NC(=O)C3CC3)sc2c1)c1ccc(F)cc1 |r|
COc1ccc(cc1)[C@@H](C)NC(=O)c1c[nH]c2ccc(cc12)-c1ccc2nc(NC(=O)C3CC3)sc2c1 |r|
COc1ccc(cc1)[C@H](C)NC(=O)c1c[nH]c2ccc(cc12)-c1ccc2nc(NC(=O)C3CC3)sc2c1 |r|
C[C@H](NC(=O)c1c[nH]c2ccc(cc12)-c1ccc2nc(NC(=O)C3CC3)sc2c1)c1cccc(F)c1 |r|
C[C@@H](NC(=O)c1c[nH]c2ccc(cc12)-c1ccc2nc(NC(=O)C3CC3)sc2c1)c1cccc(F)c1 |r|
C[C@@H](NC(=O)c1c[nH]c2ccc(cc12)-c1ccc2nc(NC(=O)C3CC3)sc2c1)c1cccc(Cl)c1 |r|
C[C@H](NC(=O)c1c[nH]c2ccc(cc12)-c1ccc2nc(NC(=O)C3CC3)sc2c1)c1cccc(Cl)c1 |r|
COc1cccc(c1)[C@H](C)NC(=O)c1c[nH]c2ccc(cc12)-c1ccc2nc(NC(=O)C3CC3)sc2c1 |r|
COc1cccc(c1)[C@@H](C)NC(=O)c1c[nH]c2ccc(cc12)-c1ccc2nc(NC(=O)C3CC3)sc2c1 |r|
C[C@H](NC(=O)c1c[nH]c2ccc(cc12)-c1ccc2sc(NC(=O)C3CC3)nc2c1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1c[nH]c2ccc(cc12)-c1ccc(NC(=O)C2CC2)nc1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1c[nH]c2ccc(cc12)-c1ccc(NC(=O)C2CC2)cc1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1c[nH]c2ccc(cc12)-c1cnc(NC(=O)C2CC2)nc1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1c[nH]c2ccc(cc12)-c1ccc2nc(NC(=O)C3CC3)ncc2c1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1c[nH]c2ccc(cc12)-c1ccc2nc(NC(=O)C3CC3)nn2c1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccc2nc(NC(=O)C3CC3)sc2c1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1c[nH]c2ccc(cc12)-c1ccc2nc(NC(=O)C3CCC3)sc2c1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1c[nH]c2ccc(cc12)-c1ccc2nc(NC(=O)C3CCCC3)sc2c1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1c[nH]c2ccc(cc12)-c1ccc2nc(NC(=O)C3CCCCC3)sc2c1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1c[nH]c2ccc(cc12)-c1ccc2nc(NC(=O)C(C)(C)C)sc2c1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1c[nH]c2ccc(cc12)-c1ccc2nc(NC(=O)C3CCOCC3)sc2c1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1c[nH]c2ccc(cc12)-c1ccc2nc(NC(=O)C(F)(F)F)sc2c1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1c[nH]c2ccc(cc12)-c1ccc2nc(NC(=O)C3CCN(C)CC3)sc2c1)c1cccc(F)c1 |r|
Cn1cc(C(=O)NCc2cc(F)ccc2F)c2cc(ccc12)-c1ccc2nc(NC(=O)C3CC3)sc2c1
CC(C)C(=O)Nc1nc2ccc(cc2s1)-c1ccc2[nH]cc(C(=O)N[C@@H](C)c3cccc(F)c3)c2c1 |r|
CC(C)n1cc(C(=O)NCc2cc(F)ccc2F)c2cc(ccc12)-c1ccc2nc(NC(=O)C3CC3)sc2c1
CCCn1cc(C(=O)NCc2cc(F)ccc2F)c2cc(ccc12)-c1ccc2nc(NC(=O)C3CC3)sc2c1
CCCCn1cc(C(=O)NCc2cc(F)ccc2F)c2cc(ccc12)-c1ccc2nc(NC(=O)C3CC3)sc2c1
C[C@H](NC(=O)c1n[nH]c2ccc(cc12)-c1ccc2nc(NC(=O)C3CC3)sc2c1)c1cccc(F)c1 |r|
COc1cc(F)ccc1NC(=O)c1c[nH]c2ncc(cc12)-c1ccc2nc(NC(=O)C3CC3)sc2c1
COc1cc(F)ccc1NC(=O)c1n[nH]c2ccc(cc12)-c1ccc2nc(NC(=O)C3CC3)sc2c1
C[C@H](NC(=O)c1c[nH]c2ncc(cc12)-c1ccc2nc(NC(=O)C3CC3)sc2c1)c1cccc(F)c1 |r|
COc1ccc(NC(=O)c2c[nH]c3ncc(cc23)-c2ccc3nc(NC(=O)C4CC4)sc3c2)cc1OC
COc1ccc(CNC(=O)c2c[nH]c3ncc(cc23)-c2ccc3nc(NC(=O)C4CC4)sc3c2)cc1OC
COc1ccc(CNC(=O)c2cn(C)c3ccc(cc23)-c2ccc3nc(NC(=O)C4CC4)sc3c2)cc1OC
Cn1cc(C(=O)N2CCN(Cc3ccc4OCOc4c3)CC2)c2cc(ccc12)-c1ccc2nc(NC(=O)C3CC3)sc2c1
COc1cc(CN2CCN(CC2)C(=O)c2cn(C)c3ccc(cc23)-c2ccc3nc(NC(=O)C4CC4)sc3c2)cc(OC)c1OC
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccc(CN2CCN(C)CC2)cc1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1c[nH]c2ncc(cc12)-c1c(C)noc1C)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccc(cc1)C(=O)N1CCOCC1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccnn1C1CCCCO1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccc(cc1)N1CCOCC1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccc(nc1)N1CCOCC1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1c[nH]c2ncc(cc12)-c1ccc(cc1)C(=O)N1CCOCC1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1c[nH]c2ncc(cc12)-c1ccnn1C1CCCCO1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1c[nH]c2ncc(cc12)-c1ccc(cc1)N1CCOCC1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1c[nH]c2ncc(cc12)-c1ccc(nc1)N1CCOCC1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1cc[nH]n1)c1cccc(F)c1 |r|
Cn1cc(C(=O)NCc2ccc(F)cc2)c2cc(ccc12)-c1ccc2nc(NC(=O)C3CC3)sc2c1
Fc1ccc(CNC(=O)c2c[nH]c3ncc(cc23)-c2ccc3nc(NC(=O)C4CC4)sc3c2)c(F)c1
C[C@H](NC(=O)c1c[nH]c2ccc(cc12)-c1ccc2nc(NC(=O)C3CC3)[nH]c2c1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1c[nH]c2ccc(cc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1c[nH]c2ccc(cc12)-c1ccc2c(N)ncnn12)c1cccc(F)c1 |r|
Cc1noc(C)c1CNC(=O)c1c[nH]c2ccc(cc12)-c1ccc2nc(NC(=O)C3CC3)sc2c1
O=C(Nc1nc2ccc(cc2s1)-c1ccc2[nH]cc(C(=O)NCc3ccn[nH]3)c2c1)C1CC1
Cn1cc(CNC(=O)c2c[nH]c3ccc(cc23)-c2ccc3nc(NC(=O)C4CC4)sc3c2)cn1
O=C(Nc1nc2ccc(cc2s1)-c1ccc2[nH]cc(C(=O)NCc3ccc4[nH]ccc4c3)c2c1)C1CC1
C[C@H](NC(=O)c1c[nH]c2ccc(cc12)-c1ccc2nc(NC(=O)C3CC3)sc2n1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccc2nc(NC(=O)C3CC3)sc2n1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccc2nc(NC(=O)C3CC3)nn2c1)c1cccc(F)c1 |r|
COCC(=O)Nc1nc2ccc(nc2s1)-c1ccc2n(C)cc(C(=O)N[C@@H](C)c3cccc(F)c3)c2c1 |r|
COCC(=O)Nc1nc2ccc(cn2n1)-c1ccc2[nH]cc(C(=O)N[C@@H](C)c3cccc(F)c3)c2c1 |r|
O=C(Nc1nc2ccc(cc2s1)-c1ccc2[nH]cc(C(=O)NCc3ccc(cc3)N3CCOCC3)c2c1)C1CC1
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1)c1cccc(F)c1 |r|
COCC(=O)Nc1nc2ccc(cn2n1)-c1ccc2[nH]cc(C(=O)NCc3cccc(F)c3)c2c1
COCC(=O)Nc1nc2ccc(cn2n1)-c1ccc2n(C)cc(C(=O)N[C@@H](C)c3cccc(F)c3)c2c1 |r|
O=C(Nc1nc2cc(ccn2n1)-c1ccc2[nH]cc(C(=O)NCc3ccc(cc3)N3CCOCC3)c2c1)C1CC1
Cn1cc(C(=O)NCc2ccc(cc2)N2CCOCC2)c2cc(ccc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1
O=C(Nc1nc2ccc(nc2s1)-c1ccc2[nH]cc(C(=O)NCc3ccc(cc3)N3CCOCC3)c2c1)C1CC1
Cn1cc(C(=O)NCc2ccc(cc2)N2CCOCC2)c2cc(ccc12)-c1ccc2nc(NC(=O)C3CC3)sc2n1
Cc1ccc(CCNC(=O)c2n[nH]c3ccc(cc23)-c2ccc3c(N)ncnn23)cc1
Nc1ncnn2c(ccc12)-c1ccc2[nH]nc(C(=O)NCCc3cccc(F)c3)c2c1
Nc1ncnn2c(ccc12)-c1ccc2[nH]nc(C(=O)NCCc3ccc(F)cc3)c2c1
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccc2c(NC(=O)C3CC3)n[nH]c2c1)c1cccc(F)c1 |r|
CC(C)C(=O)Nc1nc2cc(ccn2n1)-c1ccc2n(C)cc(C(=O)NC(C)c3ccccc3)c2c1
CC(C)C(=O)Nc1nc2cc(ccn2n1)-c1ccc2n(C)cc(C(=O)N[C@@H](C)c3cccc(F)c3)c2c1 |r|
CC(C)C(=O)Nc1nc2ccc(cn2n1)-c1ccc2n(C)cc(C(=O)N[C@@H](C)c3cccc(F)c3)c2c1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)C3CC3)cc2n1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccc2nc(NC(=O)C3CC3)cn2n1)c1cccc(F)c1 |r|
CCn1cc(C(=O)N[C@@H](C)c2cccc(F)c2)c2cc(ccc12)-c1ccc2c(NC(=O)C3CC3)n[nH]c2c1 |r|
CC(C)n1cc(C(=O)N[C@@H](C)c2cccc(F)c2)c2cc(ccc12)-c1ccc2c(NC(=O)C3CC3)n[nH]c2c1 |r|
CCCn1cc(C(=O)N[C@@H](C)c2cccc(F)c2)c2cc(ccc12)-c1ccc2c(NC(=O)C3CC3)n[nH]c2c1 |r|
CCCCn1cc(C(=O)N[C@@H](C)c2cccc(F)c2)c2cc(ccc12)-c1ccc2c(NC(=O)C3CC3)n[nH]c2c1 |r|
CC(C)Cn1cc(C(=O)N[C@@H](C)c2cccc(F)c2)c2cc(ccc12)-c1ccc2c(NC(=O)C3CC3)n[nH]c2c1 |r|
COCCn1cc(C(=O)N[C@@H](C)c2cccc(F)c2)c2cc(ccc12)-c1ccc2c(NC(=O)C3CC3)n[nH]c2c1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccc2c(NC(=O)C3CC3)c[nH]c2c1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccc2c(c[nH]c2c1)C(=O)NC1CC1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccc2c(c[nH]c2c1)C(=O)NCC(C)(C)C)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1)c1ccc(C)cc1 |r|
CC(C)C(=O)Nc1nc2cc(ccn2n1)-c1ccc2n(C)cc(C(=O)N[C@H](C)c3ccccc3)c2c1 |r|
CC(C)C(=O)Nc1nc2cc(ccn2n1)-c1ccc2n(C)cc(C(=O)N[C@@H](C)c3ccccc3)c2c1 |r|
CC(C)C(=O)Nc1nc2cc(ccn2n1)-c1ccc2n(C)cc(C(=O)NC(C)(C)c3ccccc3)c2c1
CC(C)C(=O)Nc1nc2cc(ccn2n1)-c1ccc2n(C)cc(C(=O)NC(C)c3cccc(F)c3)c2c1
CC(C)C(=O)Nc1nc2cc(ccn2n1)-c1ccc2n(C)cc(C(=O)N[C@H](C)c3cccc(F)c3)c2c1 |r|
CC(C)C(=O)Nc1nc2cc(ccn2n1)-c1ccc2n(C)cc(C(=O)N[C@H](C)c3cccc(Cl)c3)c2c1 |r|
CC(C)C(=O)Nc1nc2cc(ccn2n1)-c1ccc2n(C)cc(C(=O)N[C@@H](C)c3cccc(Cl)c3)c2c1 |r|
COc1cccc(c1)[C@@H](C)NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)C(C)C)nc2c1 |r|
COc1cccc(c1)[C@H](C)NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)C(C)C)nc2c1 |r|
CC(C)C(=O)Nc1nc2cc(ccn2n1)-c1ccc2n(C)cc(C(=O)NC(C)c3ccc(F)cc3)c2c1
CC(C)C(=O)Nc1nc2cc(ccn2n1)-c1ccc2n(C)cc(C(=O)N[C@@H](C)c3ccc(F)cc3)c2c1 |r|
CC(C)C(=O)Nc1nc2cc(ccn2n1)-c1ccc2n(C)cc(C(=O)N[C@H](C)c3ccc(F)cc3)c2c1 |r|
COc1ccc(cc1)[C@H](C)NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)C(C)C)nc2c1 |r|
COc1ccc(cc1)[C@@H](C)NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)C(C)C)nc2c1 |r|
CC(C)C(=O)Nc1nc2cc(ccn2n1)-c1ccc2n(C)cc(C(=O)NC(C)c3ccccn3)c2c1
CC(C)C(=O)Nc1nc2cc(ccn2n1)-c1ccc2n(C)cc(C(=O)N[C@H](C)c3ccccn3)c2c1 |r|
CC(C)C(=O)Nc1nc2cc(ccn2n1)-c1ccc2n(C)cc(C(=O)N[C@@H](C)c3ccccn3)c2c1 |r|
CC(C)C(=O)Nc1nc2cc(ccn2n1)-c1ccc2n(C)cc(C(=O)NC(C)c3cccnc3)c2c1
CC(C)C(=O)Nc1nc2cc(ccn2n1)-c1ccc2n(C)cc(C(=O)NC(C)c3ccncc3)c2c1
CC(C)C(=O)Nc1nc2cc(ccn2n1)-c1ccc2n(C)cc(C(=O)N[C@H]3CCCc4ccccc34)c2c1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(N)nc2c1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)C3CC3(F)F)nc2c1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)[C@H]3C[C@H]3F)nc2c1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)nc2c1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)C3(F)CC3)nc2c1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)C3CC(F)(F)C3)nc2c1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)C3CCC(F)(F)CC3)nc2c1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)C(C)(C)CCl)nc2c1)c1cccc(F)c1 |r|
CCn1cc(C(=O)N[C@@H](C)c2cccc(F)c2)c2cc(ccc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1 |r|
CC(C)n1cc(C(=O)N[C@@H](C)c2cccc(F)c2)c2cc(ccc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1 |r|
CCCn1cc(C(=O)N[C@@H](C)c2cccc(F)c2)c2cc(ccc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1 |r|
CCCCn1cc(C(=O)N[C@@H](C)c2cccc(F)c2)c2cc(ccc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1 |r|
CC(C)Cn1cc(C(=O)N[C@@H](C)c2cccc(F)c2)c2cc(ccc12)-c1ccn2nc(NC(=O)C(C)C)nc2c1 |r|
COCCn1cc(C(=O)N[C@@H](C)c2cccc(F)c2)c2cc(ccc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1 |r|
C[C@@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1)c1cccc(F)c1 |r|
CC(C)C(=O)Nc1nc2cc(ccn2n1)-c1cnc2[nH]cc(C(=O)N[C@@H](C)c3cccc(F)c3)c2c1 |r|
CC(C)C(=O)Nc1nc2cc(ccn2n1)-c1cnc2n(C)cc(C(=O)N[C@@H](C)c3cccc(F)c3)c2c1 |r|
CC(C)C(=O)Nc1nc2cc(ccn2n1)-c1cn(C)c2ncc(cc12)C(=O)N[C@@H](C)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1ccc2ncc(cc2c1)-c1ccn2nc(NC(=O)C3CC3)nc2c1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)C3CCCO3)nc2c1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)N3CC[C@@H](O)C3)nc2c1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)N3CC[C@H](O)C3)nc2c1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)N3CCC[C@H]3CO)nc2c1)c1cccc(F)c1 |r|
C[C@@H](CO)NC(=O)Nc1nc2cc(ccn2n1)-c1ccc2n(C)cc(C(=O)N[C@@H](C)c3cccc(F)c3)c2c1 |r|
COC(=O)Nc1nc2cc(ccn2n1)-c1ccc2n(C)cc(C(=O)N[C@@H](C)c3ccc(F)cc3)c2c1 |r|
CC(NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1)c1ccc(F)c(F)c1
Cn1cc(C(=O)N2CCCC2c2cccc(F)c2)c2cc(ccc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)N3CCCC(O)C3)nc2c1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)N3CCC(O)CC3)nc2c1)c1cccc(F)c1 |r|
CC(C)CNc1nc2cc(ccn2n1)-c1ccc2n(C)cc(C(=O)N[C@@H](C)c3cccc(F)c3)c2c1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)N3CC(O)C3)nc2c1)c1cccc(F)c1 |r|
Cn1cc(C(=O)N2CCC[C@H]2c2cccc(F)c2)c2cc(ccc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1 |r|
Cn1cc(C(=O)N2CCC[C@H]2c2ccc(F)cc2)c2cc(ccc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1 |r|
CC(C)C(=O)Nc1nc2cc(ccn2n1)-c1ccc2n(C)cc(C(=O)N[C@@H](C)c3ccncc3)c2c1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1)c1ccncc1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)N3CCC[C@@H]3CO)nc2c1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)N3CCNCC3)nc2c1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)[C@H]3CCCN3)nc2c1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)[C@@H]3CCCN3)nc2c1)c1cccc(F)c1 |r|
COc1ccc(cc1F)[C@H](C)NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1)c1ccc(F)c(F)c1 |r|
Cn1cc(C(=O)N[C@H]2CCc3ccc(F)cc23)c2cc(ccc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1 |r|
Cn1cc(C(=O)N[C@H]2CCCc3ccc(F)cc23)c2cc(ccc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1 |r|
Cn1cc(C(=O)N2CCCC2c2cccc(F)c2)c2cc(ccc12)-c1ccn2nc(NC(=O)C3CC3)cc2n1
C[C@H](NC(=O)c1cn(C)c2ncc(cc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1)c1cccc(F)c1 |r|
Cn1cc(C(=O)N2CCCC2c2cccc(F)c2)c2cc(ccc12)-c1ccc2nc(NC(=O)C3CC3)cn2n1
Cn1cc(C(=O)N[C@H]2CCCc3ccccc23)c2cc(ccc12)-c1ccc2nc(NC(=O)C3CC3)cn2n1 |r|
Cc1cccc(c1)C1CCCN1C(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1
Cn1cc(C(=O)N2CCCC2c2cc(F)ccc2F)c2cc(ccc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1
Cn1cc(C(=O)N2CCC[C@H]2c2ccc(F)c(F)c2)c2cc(ccc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1 |r|
Cn1cc(C(=O)N2CCC[C@H]2c2cc(F)cc(F)c2)c2cc(ccc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1 |r|
Cn1cc(C(=O)N2CCC[C@H]2c2cccc(Cl)c2)c2cc(ccc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1 |r|
Cn1cc(C(=O)N2CCC[C@H]2c2ccc(Cl)cc2)c2cc(ccc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1 |r|
CNC(=O)Nc1nc2cc(ccn2n1)-c1ccc2n(C)cc(C(=O)N[C@@H](C)c3cccc(F)c3)c2c1 |r|
C[C@@H](CO)Nc1nc2cc(ccn2n1)-c1ccc2n(C)cc(C(=O)N[C@@H](C)c3cccc(F)c3)c2c1 |r|
CCn1cc(C(=O)N2CCC[C@H]2c2ccc(F)cc2)c2cc(cnc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1 |r|
CCn1cc(C(=O)N2CCC[C@H]2c2ccc(F)cc2)c2cc(ccc12)-c1ccn2nc(NC(=O)[C@H](C)OC(C)=O)nc2c1 |r|
CC[C@H](NC(=O)c1cn(CC)c2ccc(cc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1)c1ccc(F)cc1 |r|
CCn1cc(C(=O)N[C@@H](C2CC2)c2ccc(F)cc2)c2cc(ccc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1 |r|
CCn1cc(C(=O)N2CCC[C@H]2c2ccc(F)cc2)c2cc(ccc12)-c1ccn2nc(NC(=O)CN(C)C)nc2c1 |r|
Cn1cc(C(=O)N2C(CO)CC[C@H]2c2ccc(F)cc2)c2cc(ccc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1 |r|
Cn1cc(C(=O)N[C@@H](CO)c2ccc(F)cc2)c2cc(ccc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1 |r|
CCn1cc(C(=O)N2CCC[C@H]2c2ccc(F)cc2)c2cc(ccc12)-c1ccn2nc(NC(=O)[C@@H](C)O)nc2c1 |r|
CCn1cc(C(=O)N2CCC[C@H]2c2ccc(F)cc2)c2cc(ccc12)-c1ccn2nc(NC(=O)[C@H](C)O)nc2c1 |r|
Cn1cc(C(=O)N[C@@H](C2CC2)c2ccc(F)cc2)c2cc(ccc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1 |r|
CN(C)CC(=O)Nc1nc2cc(ccn2n1)-c1ccc2n(C)cc(C(=O)N[C@@H](C3CC3)c3ccc(F)cc3)c2c1 |r|
CC[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1)c1ccc(F)cc1 |r|
CCN(CC)CC(=O)Nc1nc2cc(ccn2n1)-c1ccc2n(C)cc(C(=O)N3CCC[C@H]3c3ccc(F)cc3)c2c1 |r|
CCn1cc(C(=O)N[C@@H](C2CC2)c2ccc(F)cc2)c2cc(ccc12)-c1ccn2nc(NC(=O)CN(C)C)nc2c1 |r|
CC[C@H](NC(=O)c1cn(CC)c2ccc(cc12)-c1ccn2nc(NC(=O)CN(C)C)nc2c1)c1ccc(F)cc1 |r|
CCn1cc(C(=O)N[C@@H](CF)c2ccc(F)cc2)c2cc(ccc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1 |r|
C[C@H]1CC[C@H](N1C(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1)c1ccc(F)cc1 |r|
CCn1cc(C(=O)N[C@@H](C2CC2)c2ccc(F)cc2)c2cc(ccc12)-c1ccn2nc(NC3CC3)nc2c1 |r|
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(cc1)-c1cncn(C)c1=O
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(c(F)c1)-c1cncn(C)c1=O
CC[C@H](C)n1cncc(-c2ccc(cc2)C2(CC2)NC(=O)c2ncc3cnn(C(C)C)c3n2)c1=O |r|
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(cc1)-c1cncn([C@H]2C[C@@H]2F)c1=O |r|
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(cn1)-c1cncn(C)c1=O
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(-c2cncn(C)c2=O)c(c1)C(F)(F)F
CC[C@@H](C)n1cncc(-c2ccc(cc2)C2(CC2)NC(=O)c2ncc3cnn(C(C)C)c3n2)c1=O |r|
C[C@H](n1cncc(-c2ccc(cc2)C2(CC2)NC(=O)c2ncc3cnn(CC4CC4)c3n2)c1=O)C(F)(F)F |r|
Cn1cncc(-c2ccc(cc2)C2(CC2)NC(=O)c2nnc(Cc3ccccc3)[nH]2)c1=O
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(c(Cl)c1)-c1cncn(C)c1=O
CC(C)Cn1cncc(-c2ccc(cc2)C2(CC2)NC(=O)c2ncc3cnn(C(C)C)c3n2)c1=O
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(cc1)-c1cncn([C@@H]2C[C@@H]2F)c1=O |r|
Cn1cncc(-c2ccc(cc2)C2(CC2)NC(=O)c2ncc3cnn(-c4ccccc4)c3n2)c1=O
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(cc1F)-c1cncn(C)c1=O
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(cc1F)-c1cncn([C@H](C)C(F)(F)F)c1=O |r|
C[C@@H](n1cncc(-c2ccc(cc2)C2(CC2)NC(=O)c2ncc3cnn(CC4CC4)c3n2)c1=O)C(F)(F)F |r|
Cn1cncc(-c2ccc(cc2)C2(CC2)NC(=O)c2cc(Cc3ccccc3)on2)c1=O
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(c(C)c1)-c1cncn(C)c1=O
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(cc1F)-c1cncn([C@@H](C)C(F)(F)F)c1=O |r|
C[C@H](n1cncc(-c2ccc(c(F)c2)C2(CC2)NC(=O)c2ncc3cnn(CC4CC4)c3n2)c1=O)C(F)(F)F |r|
CC(C)Cc1nc(ncc1Cl)C(=O)NC1(CC1)c1ccc(cc1)-c1cncn(C)c1=O
Cn1cncc(-c2ccc(c(F)c2)C2(CC2)NC(=O)c2n[nH]c(Cc3ccccc3)n2)c1=O
CC(C)n1cncc(-c2ccc(c(F)c2)C2(CC2)NC(=O)c2ncc3cnn(CC4CC4)c3n2)c1=O
Cn1c(N)ncc(-c2ccc(cc2)C2(CC2)NC(=O)c2nnc(Cc3ccccc3)[nH]2)c1=O
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(cc1)-c1cncn(C(C)C)c1=O
Cn1cncc(-c2ccc(cc2)C2(CC2)NC(=O)c2nc3CC[C@@H](c4ccccc4)n3n2)c1=O |r|
CC(C)n1cncc(-c2ccc(cc2F)C2(CC2)NC(=O)c2ncc3cnn(CC4CC4)c3n2)c1=O
Cn1cncc(-c2ccc(cc2)C2(CC2)NC(=O)c2ncn(Cc3ccccc3)n2)c1=O
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(cc1)-c1cnc(N)n(C)c1=O
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(cc1F)-c1cncn(CC2CC2)c1=O
Cn1cncc(-c2ccc(cc2)C2(CC2)NC(=O)c2noc(Cc3ccccc3)n2)c1=O
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(cc1)-c1cnc(C)n(C)c1=O
C[C@H](c1ccccc1)n1cnc(n1)C(=O)NC1(CC1)c1ccc(cc1)-c1cncn(C)c1=O |r|
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(c(F)c1)-c1cncn(CC2CC2)c1=O
Cn1cncc(-c2ccc(cc2)C2(CC2)NC(=O)c2ncc(Cc3ccccc3)o2)c1=O
C[C@@H](n1cncc(-c2ccc(c(F)c2)C2(CC2)NC(=O)c2ncc3cnn(CC4CC4)c3n2)c1=O)C(F)(F)F |r|
Cn1cncc(-c2ccc(cc2)C2(CC2)NC(=O)c2nnc(Cc3ccccc3)o2)c1=O
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(c(Cl)c1)-c1cncn(C(C)C)c1=O
C[C@@H](c1nnc([nH]1)C(=O)NC1(CC1)c1ccc(cc1)-c1cncn(C)c1=O)c1ccccc1 |r|
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(cc1)-c1cncn(C2CCOCC2)c1=O
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(cc1)-c1cncn(C2CC2)c1=O
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(cc1F)-c1cncn(C(C)C)c1=O
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(cc1)-c1cncn(c1=O)C1(C)CC1
CC(C)n1cncc(-c2ccc(cc2)C2(CC2)NC(=O)c2nnc(Cc3ccccc3)o2)c1=O
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(c(F)c1)-c1cncn(C(C)C)c1=O
CC(C)n1cncc(-c2ccc(cc2)C2(CC2)NC(=O)c2ncc3cnn(C(C)C4CC4)c3n2)c1=O
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(cc1)-c1cncn([C@H]2CCOC2)c1=O |r|
CC(C)n1cncc(-c2ccc(cc2)C2(CC2)NC(=O)c2nnc(Cc3ccccc3)[nH]2)c1=O
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(cc1)-c1cncn(CC2CC2)c1=O
CC(C)n1cncc(-c2ccc(cc2)C2(CC2)NC(=O)c2ncc3cnn(C4COC4)c3n2)c1=O
CC(C)n1cncc(-c2ccc(cc2)C2(CC2)NC(=O)c2nc3CC[C@H](c4ccccc4)n3n2)c1=O |r|
CCn1cncc(-c2ccc(cc2)C2(CC2)NC(=O)c2ncc3cnn(C(C)C)c3n2)c1=O
CC(C)n1cncc(-c2ccc(cc2)C2(CC2)NC(=O)c2ncc3cnn(CC4CC4)c3n2)c1=O
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(cc1)-c1cncn([C@@H](C)C#N)c1=O |r|
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(cc1)-c1cncn(CC(F)(F)F)c1=O
CC(C)n1cncc(-c2ccc(cc2)C2(CC2)NC(=O)c2ncc3cnn(CC4CCC4)c3n2)c1=O
CC(C)n1cncc(-c2ccc(cc2)C2(CC2)NC(=O)c2ncn(Cc3ccccc3)n2)c1=O
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(cc1)-c1cncn([C@H](C)C(F)(F)F)c1=O |r|
CC(C)n1cncc(-c2ccc(cc2)C2(CC2)NC(=O)c2ncc3cnn(-c4ccccn4)c3n2)c1=O
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(cc1)-c1cncn([C@H](C)C2CC2)c1=O |r|
Cn1cncc(-c2ccc(cc2)C2(CC2)NC(=O)c2nnc(Cc3c(F)cccc3F)[nH]2)c1=O
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(cc1)-c1cncn([C@@H](C)C(F)(F)F)c1=O |r|
O=C(NC1(CC1)c1ccc(cc1)-c1cncn(CC2CC2)c1=O)c1ncc2cnn(CC3CC3)c2n1
CC(C)n1cncc(-c2ccc(cc2)C2(CC2)NC(=O)c2ncc3cnn(-c4ccccc4)c3n2)c1=O
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(cc1)-c1cncn(C2COC2)c1=O
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(cc1)-c1cncn(C2CC(F)(F)C2)c1=O
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(cc1)-c1cncn(c1=O)C1(C)CCC1
CC(C)Cc1nc(ncc1Cl)C(=O)NC1(CC1)c1ccc(cc1)-c1cncn(C(C)C)c1=O
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(cc1)-c1cncn(C2CCC2)c1=O
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(cc1)-c1cncn(CC2CCC2)c1=O
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(cc1)-c1cncn(CC2(C)CC2)c1=O
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(cc1)-c1cncn(C2C[C@H](F)C2)c1=O |r,wU:31.35,(5.19,2.62,;4.72,1.16,;3.21,.84,;5.75,.02,;7.28,.18,;7.91,-1.23,;6.76,-2.26,;6.76,-3.8,;5.43,-4.57,;4.1,-3.8,;4.1,-2.26,;5.43,-1.49,;2.76,-4.57,;2.76,-6.11,;1.43,-3.8,;.08,-4.55,;-.69,-5.88,;.85,-5.88,;-1.23,-3.75,;-1.23,-2.21,;-2.57,-1.44,;-3.9,-2.21,;-3.9,-3.75,;-2.57,-4.52,;-5.24,-1.46,;-6.57,-2.23,;-7.91,-1.46,;-7.91,.08,;-6.57,.85,;-6.57,2.39,;-5.53,3.52,;-6.65,4.57,;-6.63,6.11,;-7.7,3.44,;-5.24,.08,;-3.89,.82,)|
CC(C)n1cncc(-c2ccc(cc2)C2(CC2)NC(=O)c2ncc3cnn([C@H](C)C4CC4)c3n2)c1=O |r|
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(c(F)c1F)-c1cncn(C(C)C)c1=O
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(c(Cl)c1F)-c1cncn(C(C)C)c1=O
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1cc(F)c(cc1F)-c1cncn(CC2CC2)c1=O
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1c(F)cc(cc1F)-c1cncn(C(C)C)c1=O
CC(C)n1ncc2cnc(nc12)C(=O)NC1(CC1)c1ccc(c(F)c1F)-c1cncn(CC2CC2)c1=O
O=c1n2[C@@H](CCc2nn1C12CCC(CC1)C2)c1ccccc1 |r|
O=c1n2[C@@H](CCc2nn1C12CC(C1)CC2)c1cnccn1 |r,wU:3.18,(.66,.94,;.34,-.57,;-1.06,-1.19,;-2.57,-.87,;-3.34,-2.2,;-2.31,-3.35,;-.9,-2.72,;.6,-3.04,;1.37,-1.71,;2.9,-1.55,;3.64,-.19,;5.15,-.47,;4.44,-1.55,;5.36,-2,;3.97,-2.66,;-3.2,.54,;-4.73,.7,;-5.36,2.1,;-4.45,3.35,;-2.92,3.19,;-2.29,1.78,)|
Fc1cc(F)cc(c1)[C@@H]1CCc2nn(c(=O)n12)C12CC(F)(C1)C2 |r|
Clc1cccc(c1)[C@@H]1CCc2nn(c(=O)n12)C12CC(C1)(C2)C#N |r|
Fc1cc(F)cc(c1)[C@@H]1CCc2nn(c(=O)n12)C12CCC(F)(CC1)C2 |r|
FC12CC(C1)(C2)n1nc2CC[C@@H](c3cccc(Cl)c3)n2c1=O |r|
Fc1cc(F)cc(c1)[C@@H]1CCc2nn(c(=O)n12)C12CC(C1)CC2 |r,wU:8.8,(-1.69,3.89,;-2.46,2.55,;-4,2.55,;-4.77,1.22,;-6.31,1.22,;-4,-.11,;-2.46,-.11,;-1.69,1.22,;-1.69,-1.45,;-2.31,-2.86,;-1.17,-3.89,;.16,-3.12,;1.7,-3.28,;2.32,-1.87,;1.18,-.84,;1.34,.69,;-.16,-1.61,;3.83,-1.55,;4.46,-.14,;5.99,-.3,;5.37,-1.55,;6.31,-1.81,;4.97,-2.58,)|
Fc1cc(F)cc(c1)[C@H]1CSc2nn(c(=O)n12)C12CC(C1)(C2)C#N |r|
Fc1cc(F)cc(c1)[C@@H]1CCc2nn(c(=O)n12)C12CC(C1)(C2)C#N |r|
Fc1cc(F)cc(c1)[C@@H]1CSc2nn(c(=O)n12)C12CC(C1)(C2)C#N |r|
FC12CC(C1)(C2)n1nc2CC[C@@H](c3ccccc3)n2c1=O |r|
COc1ccc(cc1)[C@@H]1CCc2nn(c(=O)n12)C12CC(F)(C1)C2 |r|
Fc1cc(F)cc(c1)[C@@H]1CCc2nn(c(=O)n12)C12CC(C1)C2 |r|
FC12CC(C1)(C2)n1nc2CC[C@@H](c3ccc(cc3)C#N)n2c1=O |r|
Fc1cc(F)cc(c1)[C@@H]1CCc2nn(c(=O)n12)C12CC(Cl)(C1)C2 |r|
Cc1cncc(n1)[C@@H]1CCc2nn(c(=O)n12)C12CC(Cl)(C1)C2 |r|
Fc1ccccc1[C@@H]1CCc2nn(c(=O)n12)C12CC(F)(C1)C2 |r|
C[C@@H]1C[C@@H](c2cc(F)cc(F)c2)n2c1nn(c2=O)C12CC(C1)(C2)C#N |r|
Fc1cncc(c1)[C@@H]1CCc2nn(c(=O)n12)C12CC(F)(C1)C2 |r|
C[C@H]1C[C@@H](c2cc(F)cc(F)c2)n2c1nn(c2=O)C12CC(C1)(C2)C#N |r|
Fc1cncc(c1)[C@@H]1CCc2nn(c(=O)n12)C12CC(C1)(C2)C#N |r|
Fc1ccc(nc1)[C@@H]1CCc2nn(c(=O)n12)C12CC(Cl)(C1)C2 |r|
Fc1cc(F)cc(c1)[C@@H]1CCc2nn(c(=O)n12)C12CC(C1)(C2)c1ccccc1 |r|
Cc1c(F)cc(cc1Cl)[C@@H]1CCc2nn(c(=O)n12)C12CC(F)(C1)C2 |r|
Fc1cncc(c1)[C@@H]1CCc2nn(c(=O)n12)C12CC(C1)(C2)c1ccccc1 |r|
Oc1c(F)cc(cc1F)[C@@H]1CCc2nn(c(=O)n12)C12CC(F)(C1)C2 |r|
CC12CC(C1)(CO2)n1nc2CC[C@@H](c3cc(F)cc(F)c3)n2c1=O |r,wU:12.14,(6.48,-.93,;5.23,-1.84,;3.77,-1.36,;2.86,-2.61,;4.4,-2.61,;3.77,-3.86,;5.23,-3.38,;1.32,-2.61,;.42,-3.86,;-1.05,-3.38,;-2.51,-3.86,;-3.42,-2.61,;-2.51,-1.36,;-2.99,.1,;-1.96,1.25,;-2.43,2.71,;-1.4,3.86,;-3.94,3.03,;-4.97,1.89,;-6.48,2.21,;-4.5,.42,;-1.05,-1.84,;.42,-1.36,;.89,.1,)|
Cc1cc(F)c([C@@H]2CCc3nn(c(=O)n23)C23CC(F)(C2)C3)c(F)c1 |r|
Fc1cncc(c1)[C@@H]1CCc2nn(c(=O)n12)C12CC(Cl)(C1)C2 |r|
Fc1cc(ccc1Cl)[C@@H]1CCc2nn(c(=O)n12)C12CC(F)(C1)C2 |r|
Fc1cccc(c1)[C@@H]1CCc2nn(c(=O)n12)C12CC(F)(C1)C2 |r|
Fc1cc(cc(F)c1F)[C@@H]1CCc2nn(c(=O)n12)C12CC(F)(C1)C2 |r|
O=c1n2[C@@H](CCc2nn1C12CC(C1)(C2)C#N)c1ccccc1 |r|
Fc1cc(cc(F)c1Cl)[C@@H]1CCc2nn(c(=O)n12)C12CC(F)(C1)C2 |r|
COC(=O)C12CC(C1)(C2)n1nc2CC[C@@H](c3cc(F)cc(F)c3)n2c1=O |r|
FC12CC(C1)(C2)n1nc2COC[C@@H](c3ccccc3)n2c1=O |r|
COC(=O)C12CC(C1)(C2)n1nc2CC[C@@H](c3ccccc3)n2c1=O |r|
Fc1cc(F)cc(c1)[C@@H]1COCc2nn(c(=O)n12)C12CC(C1)(C2)C#N |r|
Fc1cc(F)cc(c1)[C@@H]1CCc2nn(c(=O)n12)C12C3C4C1C1C2C3C41F |r,wU:8.8,(-1.69,3.98,;-2.72,2.83,;-4.23,3.15,;-5.26,2.01,;-6.77,2.33,;-4.79,.54,;-3.28,.22,;-2.25,1.37,;-2.8,-1.24,;-3.71,-2.49,;-2.8,-3.73,;-1.34,-3.26,;.13,-3.73,;1.03,-2.49,;.13,-1.24,;.6,.22,;-1.34,-1.72,;2.57,-2.49,;3.34,-1.16,;4.83,-.76,;4.06,-2.09,;4.46,-3.58,;2.97,-3.98,;3.74,-2.65,;5.23,-2.25,;6.77,-2.25,)|
FC12CC(C1)(C2)n1nc2CCC[C@@H](c3ccccc3)n2c1=O |r|
Fc1cc(F)cc(c1)[C@@H]1CCc2nn(c(=O)n12)C12C3C4C1C1C2C3C41C#N |r,wU:8.8,(-2.46,3.98,;-3.49,2.83,;-5,3.15,;-6.03,2.01,;-7.54,2.33,;-5.56,.54,;-4.05,.22,;-3.02,1.37,;-3.57,-1.24,;-4.48,-2.49,;-3.57,-3.73,;-2.11,-3.26,;-.64,-3.73,;.26,-2.49,;-.64,-1.24,;-.17,.22,;-2.11,-1.72,;1.8,-2.49,;2.57,-1.16,;4.06,-.76,;3.29,-2.09,;3.69,-3.58,;2.2,-3.98,;2.97,-2.65,;4.46,-2.25,;6,-2.25,;7.54,-2.25,)|
Fc1cc(F)cc(c1)[C@@H]1CCc2nn(c(=O)n12)C12CC(C1)(C#N)C2(F)F |r|
Clc1cncc(c1)[C@@H]1CCc2nn(c(=O)n12)C12CC(C1)(C2)C#N |r|
COC(=O)C12CC(C1)(n1nc3CC[C@@H](c4ccccc4)n3c1=O)C2(F)F |r|
Fc1ccccc1[C@@H]1CCc2nn(c(=O)n12)C12CC(C1)(C2)C#N |r|
FC1(F)C2(CC1(C2)n1nc2CC[C@@H](c3ccccc3)n2c1=O)C#N |r|
Fc1cccc(c1)[C@@H]1CCc2nn(c(=O)n12)C12CC(C1)(C2)C#N |r|
O=c1n(nc2CCC(c3cnccn3)n12)C12CC(C1)(C2)C#N
Fc1cc(F)cc(c1)[C@@H]1CCc2nn(c(=O)n12)C12CCC(CC1)CC2 |r|
COc1cc(F)cc(c1)C1CCc2nn(c(=O)n12)C12CC(F)(C1)C2
COC12CCC(CC1)(C2)n1nc2CC[C@@H](c3cc(F)cc(F)c3)n2c1=O |r|
FC12CC(C1)(C2)n1nc2CCC(c3cccc(c3)C#N)n2c1=O
FC(F)C12CCC(CC1)(C2)n1nc2CC[C@@H](c3cc(F)cc(F)c3)n2c1=O |r|
FC12CC(C1)(C2)n1nc2CCC(c3cccc(c3)C#C)n2c1=O
FC(F)C12CC(C1)(C2)n1nc2CC[C@@H](c3cc(F)cc(F)c3)n2c1=O |r|
Fc1cccc(C2CCc3nn(c(=O)n23)C23CC(F)(C2)C3)c1F
Fc1cc(F)cc(c1)[C@@H]1CCc2nn(c(=O)n12)C12CCC(CC1)(C2)C#N |r|
Cc1cc(F)cc(c1)C1CCc2nn(c(=O)n12)C12CC(F)(C1)C2
O=c1n2[C@@H](CCc2nn1C12CCC(CC1)(C2)C#N)c1ccccc1 |r|
Cc1ccc(cc1)[C@@H]1CCc2nn(c(=O)n12)C12CC(C1)(C2)C#N |r|
FC(F)C12CC(C1)(C2)n1nc2CC[C@@H](c3ccccc3)n2c1=O |r|
O=c1n(nc2CC[C@@H](c3cnccn3)n12)C12CC(C1)(C2)C#N |r|
CC(F)(F)C12CC(C1)(C2)n1nc2CC[C@@H](c3ccccc3)n2c1=O |r|
Cc1cc(F)cc(c1)[C@@H]1CCc2nn(c(=O)n12)C12CC(F)(C1)C2 |r|
FC(F)C12CC(C1)(C2)n1nc2CC[C@@H](c3cccc(F)c3)n2c1=O |r|
FC(F)c1ccc(cc1)[C@@H]1CCc2nn(c(=O)n12)C12CC(F)(C1)C2 |r|
CC(F)(F)C12CC(C1)(C2)n1nc2CC[C@@H](c3cccc(F)c3)n2c1=O |r|
FC12CC(C1)(C2)n1nc2CC[C@@H](c3ccc(cc3)C3CC3)n2c1=O |r|
Fc1cc(F)cc(c1)[C@@H]1CCc2nn(c(=O)n12)C12CC(C1)(CC2)C#N |r,wU:8.8,(-7.1,2.21,;-5.59,1.89,;-4.56,3.03,;-3.05,2.71,;-2.02,3.86,;-2.58,1.25,;-3.61,.1,;-5.12,.42,;-3.13,-1.36,;-4.04,-2.61,;-3.13,-3.86,;-1.67,-3.38,;-.2,-3.86,;.7,-2.61,;-.2,-1.36,;.27,.1,;-1.67,-1.84,;2.24,-2.61,;3.15,-1.36,;4.61,-1.84,;3.73,-2.74,;4.61,-3.38,;3.15,-3.86,;5.86,-.93,;7.1,-.03,)|
FC12CC(C1)(C2)n1nc2CC[C@@H](c3cnccn3)n2c1=O |r|
COC(=O)C12CC(C1)(n1nc3CC[C@@H](c4cc(F)cc(F)c4)n3c1=O)C2(F)F |r|
Cc1cncc(n1)[C@@H]1CCc2nn(c(=O)n12)C12CC(F)(C1)C2 |r|
Fc1ccc(cc1)[C@@H]1CCc2nn(c(=O)n12)C12CC(F)(C1)C2 |r|
Cc1cnc(cn1)[C@@H]1CCc2nn(c(=O)n12)C12CC(F)(C1)C2 |r|
Fc1ccc(cc1)[C@@H]1CCc2nn(c(=O)n12)C12CC(C1)(C2)C#N |r|
Cc1ccccc1[C@@H]1CCc2nn(c(=O)n12)C12CC(F)(C1)C2 |r|
O=c1n2[C@@H](CCc2nn1C12CC(C1)(CC2)C#N)c1ccccc1 |r,wU:3.20,(-.48,.51,;-.96,-.95,;-2.42,-1.43,;-3.89,-.95,;-4.79,-2.2,;-3.89,-3.44,;-2.42,-2.97,;-.96,-3.44,;-.05,-2.2,;1.49,-2.2,;2.39,-.95,;3.86,-1.43,;2.89,-2.43,;3.86,-2.97,;2.39,-3.44,;5.1,-.52,;6.34,.38,;-4.36,.51,;-3.33,1.66,;-3.81,3.12,;-5.31,3.44,;-6.34,2.3,;-5.87,.83,)|
FC(F)(F)c1cnc(cn1)[C@@H]1CCc2nn(c(=O)n12)C12CC(F)(C1)C2 |r|
Fc1cccc(F)c1[C@@H]1CCc2nn(c(=O)n12)C12CC(F)(C1)C2 |r|
F[C@H]1C[C@@H](c2cnccn2)n2c1nn(c2=O)C12CC(F)(C1)C2 |r|
ClC12CC(C1)(C2)n1nc2CC[C@@H](c3ccccc3)n2c1=O |r|
O[C@@H]1C[C@@H](c2cc(F)cc(F)c2)n2c1nn(c2=O)C12CC(F)(C1)C2 |r|
Fc1cccc(c1)[C@@H]1CCc2nn(c(=O)n12)C12CC(Cl)(C1)C2 |r|
O[C@H]1C[C@@H](c2cc(F)cc(F)c2)n2c1nn(c2=O)C12CC(F)(C1)C2 |r|
Fc1cccc(F)c1[C@@H]1CCc2nn(c(=O)n12)C12CC(C1)(C2)C#N |r|
FC1C[C@@H](c2cc(F)cc(F)c2)n2c1nn(c2=O)C12CC(F)(C1)C2 |r|
Fc1ccc(cc1F)[C@@H]1CCc2nn(c(=O)n12)C12CC(C1)(C2)C#N |r|
FC12CC(C1)(C2)n1nc2CC[C@@H](c3ccc(Cl)cc3)n2c1=O |r|
FC1C[C@@H](c2ccccc2)n2c1nn(c2=O)C12CC(F)(C1)C2 |r|
Clc1ccc(cc1)[C@@H]1CCc2nn(c(=O)n12)C12CC(C1)(C2)C#N |r|
Fc1ccc([C@@H]2CCc3nn(c(=O)n23)C23CC(C2)(C3)C#N)c(F)c1 |r|
FC1C[C@@H](c2cc(F)cc(F)c2)n2c1nn(c2=O)C12CC(C1)(C2)C#N |r|
Fc1ccc([C@@H]2CCc3nn(c(=O)n23)C23CC(F)(C2)C3)c(F)c1 |r|
FC(F)(F)c1cccc(c1)[C@@H]1CCc2nn(c(=O)n12)C12CC(C1)(C2)C#N |r|
FC1C[C@@H](c2ccccc2)n2c1nn(c2=O)C12CC(C1)(C2)C#N |r|
FC(F)(F)c1ccc(cc1)[C@@H]1CCc2nn(c(=O)n12)C12CC(C1)(C2)C#N |r|
Cc1c(F)cc(cc1F)[C@@H]1CCc2nn(c(=O)n12)C12CC(C1)(C2)C#N |r|
FC1C[C@@H](c2ccccc2F)n2c1nn(c2=O)C12CC(C1)(C2)C#N |r|
CC1Cc2nn(c(=O)n2C1c1cc(F)cc(F)c1)C12CC(C1)(C2)C#N
Fc1cc(F)cc(c1)[C@@H]1CCCc2nn(c(=O)n12)C12CC(C1)(C2)C#N |r|
FC(F)c1ccc(cc1)[C@@H]1CCc2nn(c(=O)n12)C12CC(C1)(C2)C#N |r|
O=c1n2C(CCc2nn1C12CC(C1)(C2)C#N)C1CCCC1
O=c1n(nc2CCC(C3CCCCC3)n12)C12CC(C1)(C2)C#N
Cc1c(F)cc(cc1F)[C@@H]1CCc2nn(c(=O)n12)C12CC(F)(C1)C2 |r|
FC(F)C12CC(C1)(C2)n1nc2CC[C@@H](c3cncc(F)c3)n2c1=O |r|
Fc1cc(F)cc(c1)[C@@H]1CCCc2nn(c(=O)n12)C12CC(F)(C1)C2 |r|
ClC12CC(C1)(C2)n1nc2CC[C@@H](c3cnccn3)n2c1=O |r|
O=c1n(nc2CC[C@@H](c3cnccn3)n12)C12CC(C1)(CC2)C#N |r,wU:7.7,(-.35,.94,;-.67,-.57,;.36,-1.71,;-.41,-3.04,;-1.92,-2.72,;-3.32,-3.35,;-4.35,-2.2,;-3.58,-.87,;-4.21,.54,;-5.74,.7,;-6.37,2.1,;-5.46,3.35,;-3.93,3.19,;-3.3,1.78,;-2.08,-1.19,;1.89,-1.55,;2.62,-.19,;4.23,-.34,;3.43,-1.55,;4.34,-2,;2.95,-2.66,;5.33,.73,;6.43,1.81,)|
CC(C)(C)C(=O)N1C[C@@H]2C[C@H]1c3ccccc3O2
CC(C)(C(F)F)C(=O)N1C[C@@H]2C[C@H]1c3ccccc3O2
CC1(CCC1)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
O=C(N1C[C@@H]2C[C@H]1c1ccccc1O2)C12CCC(CC1)C2 |r|
CC1(CCCCC1)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
CC1(CCCC1)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
CC(C)(COC(F)(F)F)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
O=C(C1CCCCC1)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
FC1(CCCCC1)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
O=C(N1C[C@@H]2C[C@H]1c1ccccc1O2)C12CC(C1)CCC2 |r,wD:6.5,4.4,(.32,2.88,;.88,1.44,;-.08,.24,;.59,-1.15,;-.08,-2.53,;-1.58,-1.23,;-1.58,.58,;-2.78,-.38,;-4.12,.39,;-5.45,-.38,;-5.45,-1.92,;-4.12,-2.69,;-2.78,-1.92,;-1.58,-2.88,;2.41,1.21,;3.37,2.42,;4.89,2.19,;3.89,.82,;5.45,.76,;4.49,-.45,;2.97,-.22,)|
CC(C)(C1CCC1)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
CC(F)(F)C1(CCC1)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
FC(F)C1(CCCC1)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
CC1(CC1(F)F)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
CC1(C)C(C(=O)N2C[C@@H]3C[C@H]2c2ccccc2O3)C1(C)C |r|
FC(F)(F)C1(CCC1)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
CC(F)(F)C(C)(C)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
CC(C)(C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2)C(F)(F)F |r|
FC1(CCCC1)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
CC1(CC1(Cl)Cl)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
CC(C)(C)CC(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
CCC(C)(C)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
O=C(N1C[C@@H]2C[C@H]1c1ccccc1O2)C12CC3CC(CC(C3)C1)C2 |r,TLB:17:18:22:16.21.15,21:16:23:22.20.19,21:20:23:17.16.15,THB:17:16:22:23.18.19|
CC(C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2)(C(F)(F)F)C(F)(F)F |r|
CN(C)C1(CCC1)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
FC(F)(F)C1(CCCC1)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
CC1(C)CCC1C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
CC(C)(C1CC1)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
FC(F)C1(CCC1)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
O=C(N1C[C@@H]2C[C@H]1c1ccccc1O2)C1(CCC1)C#N |r|
CC1(CC(F)(F)C1)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
C[C@H]1CC[C@@](C)(C(=O)N2C[C@@H]3C[C@H]2c2ccccc2O3)C1(C)C |r|
CC(CF)(CF)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
O=C(N1C[C@@H]2C[C@H]1c1ccccc1O2)C12CC3CC(C1)C23 |r|
O=C(C1CCCCC11CC1)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
O=C(C1CCN(CC1)c1cc(ncn1)C#N)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
O=C(C1CCN(CC1)c1ncnc2scnc12)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
O=C(N1C[C@@H]2C[C@H]1c1ccccc1O2)C12CC(C1)C2 |r|
O=C(C1CCN(CC1)c1nccn2ncnc12)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
FC12CCC(CC1)(C2)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
FC(F)C12CCC(CC1)(C2)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
CC12CC(C1)(CO2)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r,wD:13.14,11.13,(5.84,2.33,;4.47,1.62,;3.1,2.31,;2.02,1.21,;3.35,.44,;2.72,-.15,;4.24,.1,;.49,1.44,;-.07,2.88,;-.47,.24,;.2,-1.15,;-.47,-2.53,;-1.97,-1.27,;-1.97,.58,;-3.17,-.38,;-4.51,.39,;-5.84,-.38,;-5.84,-1.92,;-4.51,-2.69,;-3.17,-1.92,;-1.97,-2.88,)|
O=C(N1C[C@@H]2C[C@H]1c1ccccc1O2)C12CCC(CC1)CC2 |r|
FC(F)(F)C12CCC(CC1)(C2)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
CC1(C)C2CCC1(CC2)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
COC12CCC(CC1)(C2)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
O=C(N1C[C@@H]2C[C@H]1c1ccccc1O2)C12CCC(CC1)(CC2)C#N |r|
CC1(CCN(CC1)c1cc(ncn1)C#N)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
FC1(CCN(CC1)c1cc(ncn1)C#N)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
CC1(CCOC1)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
O=C(N1C[C@@H]2C[C@H]1c1ccccc1O2)C12CCC(CC1)(CC2)c1ccccc1 |r|
FC(F)(F)C12CC(C1)(C2)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
FC(F)(F)C12CCC(CC1)(CC2)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
FC(F)C12CCC(CC1)(CC2)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
COC(=O)C12CCC(CC1)(C2)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
Clc1ccc(CNC(=O)C(=O)N2C[C@@H]3C[C@H]2c2ccccc2O3)cc1 |r|
CC(C)(CC#N)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
COc1ccc(CC(C)(C)C(=O)N2C[C@@H]3C[C@H]2c2ccccc2O3)cc1 |r|
CC(C)(C#N)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
FC(F)C12CC(C1)(C2)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1O2 |r|
CC(C)(C(F)F)C(=O)N1C[C@@H]2C[C@H]1c1cc(Cl)ccc1O2 |r|
CC(C)(C(F)F)C(=O)N1C[C@@H]2C[C@H]1c1cc(ccc1O2)C#N |r|
Cc1ccc2O[C@H]3C[C@H](N(C3)C(=O)C(C)(C)C(F)F)c2c1 |r|
CC(C)(C)C(=O)N1C[C@@H]2C[C@H]1c1cc(F)cc(F)c1O2 |r|
CC(C)(C)C(=O)N1C[C@@H]2C[C@H]1c1cc(F)ccc1O2 |r|
CC(C)(C)C(=O)N1C[C@@H]2C[C@H]1c1cccc(F)c1O2 |r|
CC(C)(C(F)F)C(=O)N1C[C@@H]2C[C@H]1c1cc(F)ccc1O2 |r|
CC(C)(C(F)F)C(=O)N1C[C@@H]2C[C@H]1c1cccc(F)c1O2 |r|
CC1(CCC1)C(=O)N1C[C@@H]2C[C@H]1c1cc(F)ccc1O2 |r|
CC1(CCC1)C(=O)N1C[C@@H]2C[C@H]1c1cccc(F)c1O2 |r|
CC(C)(C(F)F)C(=O)N1C[C@@H]2C[C@H]1c1cc(F)cc(C#N)c1O2 |r|
CC(F)(F)C(C)(C)C(=O)N1C[C@@H]2C[C@H]1c1cccc(F)c1O2 |r|
CC(F)(F)C(C)(C)C(=O)N1C[C@@H]2C[C@H]1c1cc(F)ccc1O2 |r|
Fc1ccc2O[C@H]3C[C@H](N(C3)C(=O)C34CCC(CC3)C4)c2c1 |r|
Fc1cccc2[C@@H]3C[C@@H](CN3C(=O)C34CCC(CC3)C4)Oc12 |r|
CC(F)(F)C(C)(C)C(=O)N1C[C@@H]2C[C@H]1c1ccc(Cl)cc1O2 |r|
CC(C)(CC#N)C(=O)N1C[C@@H]2C[C@H]1c1cccc(F)c1O2 |r|
CC(C)(CC#N)C(=O)N1C[C@@H]2C[C@H]1c1cc(F)ccc1O2 |r|
CC(C)(C(F)F)C(=O)N1C[C@@H]2C[C@H]1c1cccc(C#N)c1O2 |r|
CC(C)(C(F)F)C(=O)N1C[C@@H]2C[C@H]1c1cccc(Cl)c1O2 |r|
CC(C)(C(F)F)C(=O)N1C[C@@H]2C[C@H]1c1ccc(Cl)cc1O2 |r|
CC(C)(C(F)F)C(=O)N1C[C@@H]2C[C@H]1c1ccc(cc1O2)C#N |r|
CC(C)(CC#N)C(=O)N1C[C@@H]2C[C@H]1c1ccc(Cl)cc1O2 |r|
CC(C)(C(F)F)C(=O)N1C[C@@H]2C[C@H]1c1cc(F)cc(Cl)c1O2 |r|
Fc1cc(C#N)c2O[C@H]3C[C@H](N(C3)C(=O)C34CCC(F)(CC3)C4)c2c1 |r|
CC(C)(C(F)F)C(=O)N1C[C@@H]2C[C@H]1c1cc(F)cc(F)c1O2 |r|
CC(C)(CC#N)C(=O)N1C[C@@H]2C[C@H]1c1cc(F)cc(F)c1O2 |r|
Fc1cccc2[C@@H]3C[C@@H](CN3C(=O)C3(CC#N)CCC3)Oc12 |r|
CC1(CC(C1)C#N)C(=O)N1C[C@@H]2C[C@H]1c1cc(F)ccc1O2 |r,wD:13.13,11.12,(1.6,2.7,;2,1.21,;2.91,-.02,;4.15,.89,;3.23,2.13,;5.67,.66,;7.19,.43,;.47,1.44,;-.09,2.88,;-.49,.24,;.18,-1.15,;-.49,-2.53,;-1.99,-1.27,;-1.99,.58,;-3.19,-.38,;-4.53,.39,;-5.86,-.38,;-7.19,.39,;-5.86,-1.92,;-4.53,-2.69,;-3.19,-1.92,;-1.99,-2.88,)|
CC1(CC(C1)C#N)C(=O)N1C[C@@H]2C[C@H]1c1cccc(F)c1O2 |r,wD:13.13,11.12,(.93,3.38,;1.33,1.89,;2.24,.65,;3.48,1.56,;2.57,2.8,;5,1.34,;6.53,1.11,;-.19,2.12,;-.76,3.55,;-1.15,.92,;-.49,-.47,;-1.15,-1.86,;-2.66,-.59,;-2.66,1.26,;-3.86,.3,;-5.19,1.07,;-6.53,.3,;-6.53,-1.24,;-5.19,-2.01,;-5.19,-3.55,;-3.86,-1.24,;-2.66,-2.2,)|
C[C@@H]1[C@@H]2C[C@H](N1C(=O)C(C)(C)C)c1ccccc1O2 |r|
FC12CCC(CC1)(C2)C(=O)N1C[C@@H]2C[C@H]1c1cc(Cl)ccc1O2 |r|
FC12CCC(CC1)(C2)C(=O)N1C[C@@H]2C[C@H]1c1ccc(Cl)cc1O2 |r|
Fc1cc(F)c2O[C@H]3C[C@H](N(C3)C(=O)C3(F)CCN(CC3)c3nccc(n3)C#N)c2c1 |r|
Fc1cc(F)c2O[C@H]3C[C@H](N(C3)C(=O)C34CCC(F)(CC3)C4)c2c1 |r|
Fc1cc(F)c2O[C@H]3C[C@H](N(C3)C(=O)C34CC(C3)(CC4)C#N)c2c1 |r,wD:9.8,7.7,(-6.88,1.07,;-5.54,.3,;-5.54,-1.24,;-4.21,-2.01,;-4.21,-3.55,;-2.88,-1.24,;-1.67,-2.2,;-.17,-1.86,;-1.67,-.59,;-1.67,1.26,;-.17,.92,;.5,-.47,;.79,2.12,;.23,3.55,;2.31,1.89,;3.08,.56,;4.7,.76,;3.7,1.89,;4.75,2.41,;3.34,3.03,;5.83,-.28,;6.97,-1.32,;-2.88,.3,;-4.21,1.07,)|
CC(C)(C)C(=O)N1[C@@H]2CC[C@H]1c1ccccc1OC2 |THB:4:6:8.9:11.16.17.18|
CC(C)(C)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1C2
CC(C)(CC#N)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1C2
FC(F)(F)C12CCC(CC1)(C2)C(=O)N1C[C@@H]2C[C@H]1c1ccccc1C2
CC(C)(C)C(=O)N1C[C@]2(C)C[C@H]1c1ccccc1C2
CC(C)(C(F)F)C(=O)N1C[C@]2(C)C[C@H]1c1ccccc1C2
C[C@]12C[C@H](N(C1)C(=O)C13CCC(CC1)C3)c1ccccc1C2
C[C@]12C[C@H](N(O1)C(=O)C13CCC(F)(CC1)C3)c1ccccc1C2
CC12CC(N(C1)C(=O)C13CCC(CC1)(C3)C(F)(F)F)c1ccccc1O2
CN1c2ccccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O |r|
CN1c2sc(C#Cc3cnn(C)c3)c(C)c2SC[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2sc(C#Cc3cccnc3)c(C)c2SC[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2sc(C#CC3CCOCC3)c(C)c2SC[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2sc(C#CC3CC3)c(C)c2SC[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2sc(C#Cc3ccccn3)c(C)c2SC[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2sc(C#Cc3ccncc3)c(C)c2SC[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#Cc1ccccn1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#Cc1cccnc1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#Cc1ccncc1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#Cc1cnn(C)c1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CC1CCOCC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CC1CC1 |r|
COCC#Cc1ccc2OC[C@H](NC(=O)c3nnc(Cc4ccccc4)[nH]3)C(=O)N(C)c2c1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O)C#CC(C)(C)O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O)C#CC1(O)COC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O)C#C[C@@](C)(O)c1cc(C)on1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O)C#C[C@](C)(O)c1cc(C)on1 |r|
CN1c2sc(C#Cc3cncn3C)c(C)c2SC[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
COCC#Cc1sc2N(C)C(=O)[C@H](CSc2c1C)NC(=O)c1nnc(Cc2ccccc2)[nH]1 |r|
CN1c2sc(C#CC(C)(C)O)c(C)c2SC[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2sc(C#CC3(O)COC3)c(C)c2SC[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2sc(C#C[C@@](C)(O)c3cc(C)on3)c(C)c2SC[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2ncc(Cc3ccccc3)o2)C1=O)C#Cc1cccnc1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O)C#Cc1cccnc1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Cc3ccccc3)ccn2)C1=O)C#Cc1cccnc1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1n[nH]c(Cc2ccccc2)n1)C#CCN1CCN(CC#C)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1n[nH]c(Cc2ccccc2)n1)C#CCN1CCN(CC#Cc2ccc3O[C@H](C)[C@H](NC(=O)c4n[nH]c(Cc5ccccc5)n4)C(=O)N(C)c3c2)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1n[nH]c(Cc2ccccc2)n1)C#CCN1CCN(CC#Cc2ccc3OC[C@H](NC(=O)c4n[nH]c(Cc5ccccc5)n4)C(=O)N(C)c3c2)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1ncn(Cc2ccccc2)n1)C#CCN1CCN(CC#Cc2ccc3O[C@H](C)[C@H](NC(=O)c4n[nH]c(Cc5ccccc5)n4)C(=O)N(C)c3c2)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1n[nH]c(Cc2ccccc2)n1)C#CCN1CCN(CC#Cc2ccc3OC[C@H](NC(=O)c4ncn(Cc5ccccc5)n4)C(=O)N(C)c3c2)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1n[nH]c(Cc2ccccc2)n1)C#CCN1CCN(CC#Cc2ccc3O[C@H](C)[C@H](NC(=O)c4nnn(Cc5ccccc5)n4)C(=O)N(C)c3c2)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1n[nH]c(Cc2ccccc2)n1)C#CCN1CCN(CC#Cc2ccc3OC[C@H](NC(=O)c4nnn(Cc5ccccc5)n4)C(=O)N(C)c3c2)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1cn(Cc2ccccc2)cn1)C#CCN1CCN(CC#Cc2ccc3O[C@H](C)[C@H](NC(=O)c4n[nH]c(Cc5ccccc5)n4)C(=O)N(C)c3c2)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1n[nH]c(Cc2ccccc2)n1)C#CCN1CCN(CC#Cc2ccc3OC[C@H](NC(=O)c4cn(Cc5ccccc5)cn4)C(=O)N(C)c3c2)CC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CCN1CCN(CC#C)CC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CCN1CCN(CC#Cc2ccc3OC[C@H](NC(=O)c4n[nH]c(Cc5ccccc5)n4)C(=O)N(C)c3c2)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1ncn(Cc2ccccc2)n1)C#CCN1CCN(CC#Cc2ccc3OC[C@H](NC(=O)c4n[nH]c(Cc5ccccc5)n4)C(=O)N(C)c3c2)CC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O)C#CCN1CCN(CC#Cc2ccc3OC[C@H](NC(=O)c4n[nH]c(Cc5ccccc5)n4)C(=O)N(C)c3c2)CC1 |r|
C[C@H]1Oc2ccc(cc2NC(=O)[C@H]1NC(=O)c1n[nH]c(Cc2ccccc2)n1)C#CCN1CCN(CC#C)CC1 |r|
C[C@H]1Oc2ccc(cc2NC(=O)[C@H]1NC(=O)c1n[nH]c(Cc2ccccc2)n1)C#CCN1CCN(CC#Cc2ccc3O[C@H](C)[C@H](NC(=O)c4n[nH]c(Cc5ccccc5)n4)C(=O)Nc3c2)CC1 |r|
C[C@@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1n[nH]c(Cc2ccccc2)n1)C#CCN1CCN(CC#C)CC1 |r|
C[C@@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1n[nH]c(Cc2ccccc2)n1)C#CCN1CCN(CC#Cc2ccc3O[C@@H](C)[C@H](NC(=O)c4n[nH]c(Cc5ccccc5)n4)C(=O)N(C)c3c2)CC1 |r|
O=C(N[C@H]1COc2ccc(cc2NC1=O)C#CCN1CCN(CC#C)CC1)c1n[nH]c(Cc2ccccc2)n1 |r|
O=C(N[C@H]1COc2ccc(cc2NC1=O)C#CCN1CCN(CC#Cc2ccc3OC[C@H](NC(=O)c4n[nH]c(Cc5ccccc5)n4)C(=O)Nc3c2)CC1)c1n[nH]c(Cc2ccccc2)n1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1ncn(Cc2ccccc2)n1)C#CCN1CCN(CC#C)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1ncn(Cc2ccccc2)n1)C#CCN1CCN(CC#Cc2ccc3O[C@H](C)[C@H](NC(=O)c4ncn(Cc5ccccc5)n4)C(=O)N(C)c3c2)CC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O)C#CCN1CCN(CC#Cc2ccc3OC[C@H](NC(=O)c4ncn(Cc5ccccc5)n4)C(=O)N(C)c3c2)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1ncn(Cc2ccccc2)n1)C#CCN1CCN(CC#Cc2ccc3O[C@H](C)[C@H](NC(=O)c4nnn(Cc5ccccc5)n4)C(=O)N(C)c3c2)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1ncn(Cc2ccccc2)n1)C#CCN1CCN(CC#Cc2ccc3OC[C@H](NC(=O)c4nnn(Cc5ccccc5)n4)C(=O)N(C)c3c2)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1cn(Cc2ccccc2)cn1)C#CCN1CCN(CC#Cc2ccc3O[C@H](C)[C@H](NC(=O)c4ncn(Cc5ccccc5)n4)C(=O)N(C)c3c2)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1ncn(Cc2ccccc2)n1)C#CCN1CCN(CC#Cc2ccc3OC[C@H](NC(=O)c4cn(Cc5ccccc5)cn4)C(=O)N(C)c3c2)CC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O)C#CCN1CCN(CC#C)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1ncn(Cc2ccccc2)n1)C#CCN1CCN(CC#Cc2ccc3OC[C@H](NC(=O)c4ncn(Cc5ccccc5)n4)C(=O)N(C)c3c2)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1cn(Cc2ccccc2)cn1)C#CCN1CCN(CC#Cc2ccc3OC[C@H](NC(=O)c4ncn(Cc5ccccc5)n4)C(=O)N(C)c3c2)CC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cn(Cc3ccccc3)cn2)C1=O)C#CCN1CCN(CC#Cc2ccc3OC[C@H](NC(=O)c4ncn(Cc5ccccc5)n4)C(=O)N(C)c3c2)CC1 |r|
C[C@H]1Oc2ccc(cc2NC(=O)[C@H]1NC(=O)c1ncn(Cc2ccccc2)n1)C#CCN1CCN(CC#Cc2ccc3O[C@H](C)[C@H](NC(=O)c4ncn(Cc5ccccc5)n4)C(=O)Nc3c2)CC1 |r|
C[C@@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1ncn(Cc2ccccc2)n1)C#CCN1CCN(CC#C)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1ncn(Cc2ccccc2)n1)C#CCN1CCN(CC#Cc2ccc3O[C@@H](C)[C@H](NC(=O)c4ncn(Cc5ccccc5)n4)C(=O)N(C)c3c2)CC1 |r|
C[C@@H]1Oc2ccc(cc2NC(=O)[C@H]1NC(=O)c1ncn(Cc2ccccc2)n1)C#CCN1CCN(CC#C)CC1 |r|
O=C(N[C@H]1COc2ccc(cc2NC1=O)C#CCN1CCN(CC#Cc2ccc3OC[C@H](NC(=O)c4ncn(Cc5ccccc5)n4)C(=O)Nc3c2)CC1)c1ncn(Cc2ccccc2)n1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1ncc(Cc2ccccc2)o1)C#CCN1CCN(CC#C)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1ncc(Cc2ccccc2)o1)C#CCN1CCN(CC#Cc2ccc3O[C@H](C)[C@H](NC(=O)c4ncc(Cc5ccccc5)o4)C(=O)N(C)c3c2)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1cc(Cc2ccccc2)on1)C#CCN1CCN(CC#C)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1cc(Cc2ccccc2)on1)C#CCN1CCN(CC#Cc2ccc3O[C@H](C)[C@H](NC(=O)c4cc(Cc5ccccc5)on4)C(=O)N(C)c3c2)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1cnn(Cc2ccccc2)c1)C#CCN1CCN(CC#C)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1cnn(Cc2ccccc2)c1)C#CCN1CCN(CC#Cc2ccc3O[C@H](C)[C@H](NC(=O)c4cnn(Cc5ccccc5)c4)C(=O)N(C)c3c2)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1nnc(Cc2ccccc2)o1)C#CCN1CCN(CC#C)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1nnc(Cc2ccccc2)o1)C#CCN1CCN(CC#Cc2ccc3O[C@H](C)[C@H](NC(=O)c4nnc(Cc5ccccc5)o4)C(=O)N(C)c3c2)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1noc(Cc2ccccc2)n1)C#CCN1CCN(CC#C)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1noc(Cc2ccccc2)n1)C#CCN1CCN(CC#Cc2ccc3O[C@H](C)[C@H](NC(=O)c4noc(Cc5ccccc5)n4)C(=O)N(C)c3c2)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1cn(Cc2ccccc2)nn1)C#CCN1CCN(CC#C)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1cn(Cc2ccccc2)nn1)C#CCN1CCN(CC#Cc2ccc3O[C@H](C)[C@H](NC(=O)c4cn(Cc5ccccc5)nn4)C(=O)N(C)c3c2)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1nnn(Cc2ccccc2)n1)C#CCN1CCN(CC#C)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1nnn(Cc2ccccc2)n1)C#CCN1CCN(CC#Cc2ccc3O[C@H](C)[C@H](NC(=O)c4nnn(Cc5ccccc5)n4)C(=O)N(C)c3c2)CC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2nnn(Cc3ccccc3)n2)C1=O)C#CCN1CCN(CC#C)CC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2nnn(Cc3ccccc3)n2)C1=O)C#CCN1CCN(CC#Cc2ccc3OC[C@H](NC(=O)c4nnn(Cc5ccccc5)n4)C(=O)N(C)c3c2)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1cn(Cc2ccccc2)cn1)C#CCN1CCN(CC#C)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1cn(Cc2ccccc2)cn1)C#CCN1CCN(CC#Cc2ccc3O[C@H](C)[C@H](NC(=O)c4cn(Cc5ccccc5)cn4)C(=O)N(C)c3c2)CC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cn(Cc3ccccc3)cn2)C1=O)C#CCN1CCN(CC#C)CC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cn(Cc3ccccc3)cn2)C1=O)C#CCN1CCN(CC#Cc2ccc3OC[C@H](NC(=O)c4cn(Cc5ccccc5)cn4)C(=O)N(C)c3c2)CC1 |r|
C[C@@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1cn(Cc2ccccc2)cn1)C#CCN1CCN(CC#C)CC1 |r|
C[C@@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1cn(Cc2ccccc2)cn1)C#CCN1CCN(CC#Cc2ccc3O[C@@H](C)[C@H](NC(=O)c4cn(Cc5ccccc5)cn4)C(=O)N(C)c3c2)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1n[nH]c(Cc2ccncc2)n1)C#CCN1CCN(CC#C)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1n[nH]c(Cc2ccncc2)n1)C#CCN1CCN(CC#Cc2ccc3O[C@H](C)[C@H](NC(=O)c4n[nH]c(Cc5ccncc5)n4)C(=O)N(C)c3c2)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1n[nH]c(Cc2cccnc2)n1)C#CCN1CCN(CC#C)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1n[nH]c(Cc2cccnc2)n1)C#CCN1CCN(CC#Cc2ccc3O[C@H](C)[C@H](NC(=O)c4n[nH]c(Cc5cccnc5)n4)C(=O)N(C)c3c2)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1n[nH]c(Cc2cccc(O)c2)n1)C#CCN1CCN(CC#C)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1n[nH]c(Cc2cccc(O)c2)n1)C#CCN1CCN(CC#Cc2ccc3O[C@H](C)[C@H](NC(=O)c4n[nH]c(Cc5cccc(O)c5)n4)C(=O)N(C)c3c2)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1n[nH]c(Cc2cccc(N)c2)n1)C#CCN1CCN(CC#C)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1n[nH]c(Cc2cccc(N)c2)n1)C#CCN1CCN(CC#Cc2ccc3O[C@H](C)[C@H](NC(=O)c4n[nH]c(Cc5cccc(N)c5)n4)C(=O)N(C)c3c2)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1ncn(Cc2cccnc2)n1)C#CCN1CCN(CC#C)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1ncn(Cc2cccnc2)n1)C#CCN1CCN(CC#Cc2ccc3O[C@H](C)[C@H](NC(=O)c4ncn(Cc5cccnc5)n4)C(=O)N(C)c3c2)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1ncn(Cc2cccc(O)c2)n1)C#CCN1CCN(CC#C)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1ncn(Cc2cccc(O)c2)n1)C#CCN1CCN(CC#Cc2ccc3O[C@H](C)[C@H](NC(=O)c4ncn(Cc5cccc(O)c5)n4)C(=O)N(C)c3c2)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1ncn(Cc2cccc(N)c2)n1)C#CCN1CCN(CC#C)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1ncn(Cc2cccc(N)c2)n1)C#CCN1CCN(CC#Cc2ccc3O[C@H](C)[C@H](NC(=O)c4ncn(Cc5cccc(N)c5)n4)C(=O)N(C)c3c2)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1n[nH]c(Cc2ccccc2)n1)C#CCCCCC#Cc1ccc2O[C@H](C)[C@H](NC(=O)c3n[nH]c(Cc4ccccc4)n3)C(=O)N(C)c2c1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CCCCCC#Cc1ccc2OC[C@H](NC(=O)c3n[nH]c(Cc4ccccc4)n3)C(=O)N(C)c2c1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1n[nH]c(Cc2ccccc2)n1)C#CCOCCOCCOCCOCCOCC#Cc1ccc2O[C@H](C)[C@H](NC(=O)c3n[nH]c(Cc4ccccc4)n3)C(=O)N(C)c2c1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1n[nH]c(Cc2ccccc2)n1)C#CCOCCOCCOCCOCCOCC#C |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CCOCCOCCOCCOCCOCC#Cc1ccc2OC[C@H](NC(=O)c3n[nH]c(Cc4ccccc4)n3)C(=O)N(C)c2c1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CCOCCOCCOCCOCCOCC#C |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1n[nH]c(Cc2ccccc2)n1)C#CCOCCOCCOCCOCCOCC#Cc1ccc2OC[C@H](NC(=O)c3n[nH]c(Cc4ccccc4)n3)C(=O)N(C)c2c1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1ncn(Cc2ccccc2)n1)C#CCOCCOCCOCCOCCOCC#Cc1ccc2O[C@H](C)[C@H](NC(=O)c3ncn(Cc4ccccc4)n3)C(=O)N(C)c2c1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1ncn(Cc2ccccc2)n1)C#CCOCCOCCOCCOCCOCC#C |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O)C#CCOCCOCCOCCOCCOCC#Cc1ccc2OC[C@H](NC(=O)c3ncn(Cc4ccccc4)n3)C(=O)N(C)c2c1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O)C#CCOCCOCCOCCOCCOCC#C |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1ncn(Cc2ccccc2)n1)C#CCOCCOCCOCCOCCOCC#Cc1ccc2OC[C@H](NC(=O)c3ncn(Cc4ccccc4)n3)C(=O)N(C)c2c1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1n[nH]c(Cc2ccccc2)n1)C#CCOCCOCCOCCOCCOCC#CC#CCOCCOCCOCCOCCOCC#Cc1ccc2O[C@H](C)[C@H](NC(=O)c3n[nH]c(Cc4ccccc4)n3)C(=O)N(C)c2c1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CCOCCOCCOCCOCCOCC#CC#CCOCCOCCOCCOCCOCC#Cc1ccc2OC[C@H](NC(=O)c3n[nH]c(Cc4ccccc4)n3)C(=O)N(C)c2c1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@@H]1NC(=O)c1ncn(Cc2ccccc2)n1)C#CCOCCOCCOCCOCCOCC#CC#CCOCCOCCOCCOCCOCC#Cc1ccc2O[C@H](C)[C@@H](NC(=O)c3ncn(Cc4ccccc4)n3)C(=O)N(C)c2c1 |r|
CN1c2cc(ccc2OC[C@@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O)C#CCOCCOCCOCCOCCOCC#CC#CCOCCOCCOCCOCCOCC#Cc1ccc2OC[C@@H](NC(=O)c3ncn(Cc4ccccc4)n3)C(=O)N(C)c2c1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1n[nH]c(Cc2ccccc2)n1)C#CCN1CCN(CC#CC#CCN2CCN(CC#Cc3ccc4O[C@H](C)[C@H](NC(=O)c5n[nH]c(Cc6ccccc6)n5)C(=O)N(C)c4c3)CC2)CC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O)C#CCN1CCN(CC#CC#CCN2CCN(CC#Cc3ccc4OC[C@H](NC(=O)c5n[nH]c(Cc6ccccc6)n5)C(=O)N(C)c4c3)CC2)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1ncn(Cc2ccccc2)n1)C#CCN1CCN(CC#CC#CCN2CCN(CC#Cc3ccc4O[C@H](C)[C@H](NC(=O)c5ncn(Cc6ccccc6)n5)C(=O)N(C)c4c3)CC2)CC1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O)C#CCN1CCN(CC#CC#CCN2CCN(CC#Cc3ccc4OC[C@H](NC(=O)c5ncn(Cc6ccccc6)n5)C(=O)N(C)c4c3)CC2)CC1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1n[nH]c(Cc2ccccc2)n1)C#CCCCN(C)CCCC#Cc1ccc2O[C@H](C)[C@H](NC(=O)c3n[nH]c(Cc4ccccc4)n3)C(=O)N(C)c2c1 |r|
CN(CCCC#Cc1ccc2OC[C@H](NC(=O)c3n[nH]c(Cc4ccccc4)n3)C(=O)N(C)c2c1)CCCC#Cc1ccc2OC[C@H](NC(=O)c3n[nH]c(Cc4ccccc4)n3)C(=O)N(C)c2c1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1ncn(Cc2ccccc2)n1)C#CCCCN(C)CCCC#Cc1ccc2O[C@H](C)[C@H](NC(=O)c3ncn(Cc4ccccc4)n3)C(=O)N(C)c2c1 |r|
CN(CCCC#Cc1ccc2OC[C@H](NC(=O)c3ncn(Cc4ccccc4)n3)C(=O)N(C)c2c1)CCCC#Cc1ccc2OC[C@H](NC(=O)c3ncn(Cc4ccccc4)n3)C(=O)N(C)c2c1 |r|
COCCOCCOCCOCCOCC#Cc1ccc2O[C@H](C)[C@H](NC(=O)c3n[nH]c(Cc4ccccc4)n3)C(=O)N(C)c2c1 |r|
COCCOCCOCCOCCOCC#Cc1ccc2OC[C@H](NC(=O)c3n[nH]c(Cc4ccccc4)n3)C(=O)N(C)c2c1 |r|
COCCOCCOCCOCCOCC#Cc1ccc2O[C@H](C)[C@H](NC(=O)c3ncn(Cc4ccccc4)n3)C(=O)N(C)c2c1 |r|
COCCOCCOCCOCCOCC#Cc1ccc2OC[C@H](NC(=O)c3ncn(Cc4ccccc4)n3)C(=O)N(C)c2c1 |r|
CC(O)C#Cc1ccc2O[C@H](C)[C@H](NC(=O)c3n[nH]c(Cc4ccccc4)n3)C(=O)N(C)c2c1 |r|
CC(O)C#Cc1ccc2O[C@H](C)[C@H](NC(=O)c3ncn(Cc4ccccc4)n3)C(=O)N(C)c2c1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1n[nH]c(Cc2ccccc2)n1)C#CCCO |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1ncn(Cc2ccccc2)n1)C#CCCO |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1n[nH]c(Cc2ccccc2)n1)C#CCCCCC(O)=O |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1ncn(Cc2ccccc2)n1)C#CCCCCC(O)=O |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1n[nH]c(Cc2ccccc2)n1)C#Cc1ccncc1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1ncn(Cc2ccccc2)n1)C#Cc1ccncc1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1n[nH]c(Cc2ccccc2)n1)C#Cc1cccnc1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1ncn(Cc2ccccc2)n1)C#Cc1cccnc1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1n[nH]c(Cc2ccccc2)n1)C#Cc1cccc(c1)S(O)(=O)=O |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1ncn(Cc2ccccc2)n1)C#Cc1cccc(c1)S(O)(=O)=O |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1n[nH]c(Cc2ccccc2)n1)C#Cc1cccc(c1)[N+]([O-])=O |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1ncn(Cc2ccccc2)n1)C#Cc1cccc(c1)[N+]([O-])=O |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1ncn(Cc2ccccc2)n1)C#Cc1cccc(N)c1 |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1nc(Cc2ccccc2)n[nH]1)C#C |r|
C[C@H]1Oc2ccc(cc2N(C)C(=O)[C@H]1NC(=O)c1ncn(Cc2ccccc2)n1)C#C |r|
CN1c2cc(CCCN3CCN(CCCc4ccc5OC[C@H](NC(=O)c6ncn(Cc7ccccc7)n6)C(=O)N(C)c5c4)CC3)ccc2OC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O |r|
C[C@H]1Oc2ccc(CCCN3CCN(CCCc4ccc5O[C@H](C)[C@H](NC(=O)c6ncn(Cc7ccccc7)n6)C(=O)N(C)c5c4)CC3)cc2N(C)C(=O)[C@H]1NC(=O)c1ncn(Cc2ccccc2)n1 |r|
CN1c2cc(CCCN3CCN(CCCc4ccc5OC[C@H](NC(=O)c6n[nH]c(Cc7ccccc7)n6)C(=O)N(C)c5c4)CC3)ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O |r|
C[C@H]1Oc2ccc(CCCN3CCN(CCCc4ccc5O[C@H](C)[C@H](NC(=O)c6n[nH]c(Cc7ccccc7)n6)C(=O)N(C)c5c4)CC3)cc2N(C)C(=O)[C@H]1NC(=O)c1n[nH]c(Cc2ccccc2)n1 |r|
CN1c2c(F)cc(F)cc2CC[C@H](NC(=O)c2nnc(Cc3ccccc3)[nH]2)C1=O |r|
Fc1cc(F)c2NC(=O)[C@H](CCc2c1)NC(=O)c1n[nH]c(Cc2ccccc2)n1 |r|
FC(F)CN1CCc2c(Cl)n(Cc3ccccc3)nc2C1=O
FC(F)CN1CCc2c(Cl)n(Cc3ccccc3F)nc2C1=O
FC(F)CN1CCc2c(Cl)n(Cc3c(F)cccc3F)nc2C1=O
C[C@H](C(F)F)N1CCc2c(Cl)n(Cc3c(F)cccc3F)nc2C1=O |r|
FC(F)CN1CCCc2c(Cl)n(Cc3ccccc3)nc2C1=O
CNC(=O)c1n[nH]c2cc(ccc12)N1CCCC(C1)C(=O)NCc1ccccc1OC(F)(F)F
CNC(=O)c1n[nH]c2cc(ccc12)N1CCN(C)C(C1)C(=O)NCc1ccccc1OC
CNC(=O)c1n[nH]c2cc(ccc12)N1CCOC(C1)C(=O)NCCC(O)c1ccc(F)c(F)c1
CNC(=O)c1n[nH]c2cc(ccc12)N1CCNC(C1)C(=O)NCCC(C)c1ccccc1
CNC(=O)c1n[nH]c2cc(ccc12)C1CCCN(C1)C(=O)NCCC(C)c1ccccc1
CNC(=O)c1n[nH]c2cc(ccc12)N1CCCC(C1)C(=O)NC[C@H](O)COc1ccccc1 |r|
CNC(=O)c1n[nH]c2cc(ccc12)N1CCCC(C1)C(=O)NC[C@@H](O)COc1ccccc1 |r|
CNC(=O)c1n[nH]c2cc(ccc12)N1CCCC(C1)C(=O)NCc1ccccc1Oc1ccccc1
CNC(=O)c1n[nH]c2cc(ccc12)N1CCCC(C1)C(=O)NCCCOc1ccccc1
CNC(=O)c1n[nH]c2cc(ccc12)N1CCCC(C1)C(=O)NCCC(O)c1ccccc1
CNC(=O)c1n[nH]c2cc(ccc12)N1CCCC(C1)C(=O)Nc1cnn(Cc2ccccc2)c1
CNC(=O)c1n[nH]c2cc(ccc12)N1CCCC(C1)C(=O)NCc1ccccc1OCC1CC1
CNC(=O)c1n[nH]c2cc(ccc12)N1CCCC(C1)C(=O)NCCCOc1ccc(F)cc1
CNC(=O)c1n[nH]c2cc(ccc12)N1CCCC(C1)C(=O)NCCC(O)c1ccc(F)c(F)c1
CNC(=O)c1n[nH]c2cc(ccc12)N1CCCC(C1)C(=O)NC1CCC[C@@H](C1)c1ccccc1 |r|
CNC(=O)c1n[nH]c2cc(ccc12)N1CCCC(C1)C(=O)NC1CCC[C@H](C1)c1ccccc1 |r|
CNC(=O)c1n[nH]c2cc(ccc12)N1CCCC(C1)C(=O)NCCC(C)c1ccccc1
CNC(=O)c1n[nH]c2cc(ccc12)N1CCN(C)C(C1)C(=O)NCCC(O)c1ccccc1
CNC(=O)c1n[nH]c2cc(ccc12)N1CCN(C)C(C1)C(=O)NCCC(C)c1ccc(F)cc1
CNC(=O)c1n[nH]c2cc(ccc12)N1CCN(C)C(C1)C(=O)NCCC(C)c1ccccc1
CNC(=O)c1n[nH]c2cc(ccc12)N1CCOC(C1)C(=O)Nc1cnn(Cc2ccccc2)c1
CNC(=O)c1n[nH]c2cc(ccc12)N1CCOC(C1)C(=O)NCCC(C)c1ccccc1
CNC(=O)c1n[nH]c2cc(ccc12)N1CCOC(C1)C(=O)NCC1CC1c1cccc(F)c1
CNC(=O)c1n[nH]c2cc(ccc12)N1CCOC(C1)C(=O)NCCC(C)c1ccc(F)cc1
CNC(=O)c1n[nH]c2cc(ccc12)N1CCOC(C1)C(=O)NCCC(O)c1ccc(Cl)cc1
CNC(=O)c1n[nH]c2cc(ccc12)N1CCOC(C1)C(=O)NC1CCCC(C1)c1ccccc1
CCC(C)(C)C(=O)N(O)Cc1cc(F)cc(F)c1
O=C(N(O)Cc1ccccc1)C1(C(F)(F)F)CCC1
CCC(C)(C)C(=O)N(O)Cc1ccc2c(c1)CCC2
CCC1(C(=O)N(O)Cc2ccccc2)CC1
O=C(C1CCN(c2ncc(F)cn2)CC1)N(O)Cc1ccccc1
O=C(C1CCN(c2ncc(F)cn2)CC1)N(O)Cc1cc(F)cc(F)c1
CCC(C)(C)C(=O)N(O)Cc1cnc(C)s1
Cc1ccsc1CN(O)C(=O)C(C)(C)C(F)(F)F
CCC(C)(C)C(=O)N(O)Cc1ccsc1
CCC(C)(C)C(=O)N(O)Cc1ccc(Cl)c(F)c1
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC([2H])([2H])C([2H])([2H])[2H])n[nH]c3c2)cc1C(=O)NC(C)c1cc(OC(F)(F)F)ccc1F
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC([2H])([2H])C([2H])([2H])[2H])n[nH]c3c2)cc1C(=O)N[C@H](C)c1ccccc1OC(F)(F)F
[2H]C([2H])([2H])NC(=O)c1n[nH]c2cc(-c3cnc(OC([2H])([2H])[2H])c(C(=O)N[C@H](C)c4cccc(C(F)(F)F)c4)c3)ccc12
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC)n[nH]c3c2)cc1C(=O)N[C@@H](c1cc(C(F)(F)F)ccc1F)C([2H])([2H])[2H]
[2H]C([2H])([2H])NC(=O)c1n[nH]c2cc(-c3cnc(OC([2H])([2H])[2H])c(C(=O)N[C@@H](C)c4cc(OC(F)(F)F)ccc4F)c3)ccc12
[2H]C([2H])([2H])NC(=O)c1n[nH]c2cc(-c3cnc(OC([2H])([2H])[2H])c(C(=O)N[C@H](C)c4cc(C(F)(F)F)ccc4F)c3)ccc12
[2H]C([2H])([2H])NC(=O)c1n[nH]c2cc(-c3cnc(OC([2H])([2H])[2H])c(C(=O)N[C@H](C)c4ccccc4OC(F)(F)F)c3)ccc12
[2H]C([2H])([2H])NC(=O)c1n[nH]c2cc(-c3cnc(OC([2H])([2H])[2H])c(C(=O)N[C@H](C)c4cccc(OC(F)(F)F)c4)c3)ccc12
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC)n[nH]c3c2)cc1C(=O)N[C@@H](c1cc(OC(F)(F)F)ccc1F)C([2H])([2H])[2H]
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC)n[nH]c3c2)cc1C(=O)N[C@H](c1cc(OC(F)(F)F)ccc1F)C([2H])([2H])[2H]
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC)n[nH]c3c2)cc1C(=O)N[C@@H](c1cccc(OC(F)(F)F)c1)C([2H])([2H])[2H]
[2H]C([2H])([2H])NC(=O)c1n[nH]c2cc(-c3cnc(OC([2H])([2H])[2H])c(C(=O)N[C@@H]4CN(C(=O)C5CC(F)(F)C5)C[C@@H]4F)c3)ccc12
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC4CC4)n[nH]c3c2)cc1C(=O)N[C@H](C)c1ccccc1OC(F)(F)F
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC)n[nH]c3c2)cc1C(=O)N[C@H](C)c1cccc(OC(F)(F)F)c1
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC)n[nH]c3c2)cc1C(=O)NC(C)c1ccccc1OC(F)(F)F
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC)n[nH]c3c2)cc1C(=O)NC([2H])([2H])c1ccccc1OC(F)(F)F
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NC4CCCC(NC(=O)C(C)(C)C)C4)c3)ccc12
CC[C@@H](c1ccccc1)n1nnc(-c2cc(-c3ccc4c(C(=O)NC)n[nH]c4c3)cnc2OC)n1
CC[C@H](c1ccccc1)n1nnc(-c2cc(-c3ccc4c(C(=O)NC)n[nH]c4c3)cnc2OC)n1
[2H]C([2H])([2H])NC(=O)c1n[nH]c2cc(-c3cnc(OC)c(-c4nnn([C@@H](C)c5ccc(F)cc5)n4)c3)ccc12
[2H]C([2H])([2H])NC(=O)c1n[nH]c2cc(-c3cnc(OC)c(-c4nnn([C@H](C)c5ccc(F)cc5)n4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(-c4nnn(Cc5ccccc5)n4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)N[C@H]4CCC[C@@H](c5ccccc5)C4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)N[C@@H]4CCC[C@@H](c5ccccc5)C4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)N[C@H]4CCC[C@H](c5ccccc5)C4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)N[C@@H]4CCC[C@H](c5ccccc5)C4)c3)ccc12
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC(C)C)n[nH]c3c2)cc1C(=O)NC(C)c1ccccc1OC(F)(F)F
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC4CCC(N(C([2H])([2H])[2H])C([2H])([2H])[2H])CC4)n[nH]c3c2)cc1C(=O)NC(C)c1cccc(OC(F)(F)F)c1
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NC(C)c4ccccc4C)c3)cc(F)c12
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1cc(O)ncn1)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1cc(F)ccn1)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1cccc(CO)n1)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1cccc(Cl)n1)CC2
Cc1cnc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)nc1
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1cc(C(F)F)ncn1)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1ccnc(C(F)F)n1)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1cc(F)ncc1F)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1cc(Cl)c(F)cn1)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1cc(Cl)ccn1)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1cccc(F)n1)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1ncnc3ccsc13)CC2
CSc1cc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)ncn1
Cc1csc2ncnc(N3CCC4(CC3)CN3CC[C@@H](c5cc(F)cc(F)c5)N3C4=O)c12
Cc1cc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)nc(C#N)n1
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1cc(-n3cccn3)ncn1)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1cc(-n3ccnc3)ncn1)CC2
Cc1cn(-c2cc(N3CCC4(CC3)CN3CC[C@@H](c5cc(F)cc(F)c5)N3C4=O)ncn2)cn1
CCc1nccc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)n1
Cn1nccc1-c1cc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)ncn1
CSc1cnc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)nc1
COc1nc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)ncc1C
NC(=O)c1ccnc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)n1
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1ncc(OC(F)F)cn1)CC2
Cc1nc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)ncc1OC(F)F
Cc1ccnc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)n1
CCc1cnc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)nc1
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1ncc(F)cn1)CC2
CN(C)c1nc(Cl)cc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)n1
COc1nc(OC)nc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)n1
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1ncc3c(n1)CCCC3)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1ncc3c(n1)CCCC3)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1ccc(Cl)nn1)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1cc(-c3ccccc3)ncn1)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1cnnc(Cl)c1)CC2
N#Cc1ccc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)nn1
Cc1c(Cl)ncnc1N1CCC2(CC1)CN1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1ccc(C(F)(F)F)cn1)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1cncc(Cl)n1)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1cnccn1)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1cnc(Cl)cn1)CC2
Cc1ncc(Cl)nc1N1CCC2(CC1)CN1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
Cc1cc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)nc(C(F)(F)F)n1
Cc1nccc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)n1
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1ccnc(C3CC3)n1)CC2
CC(C)c1nc(Cl)cc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)n1
Cc1cc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)nc(Cl)n1
CC(C)c1nccc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)n1
N#Cc1ccc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)nc1
N#Cc1c(F)c(F)nc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)c1F
N#Cc1cc(Cl)nc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)c1
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1nc(Cl)nc3[nH]ncc13)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1ncc(Br)cn1)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1ncccn1)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1ncc(C3CC3)cn1)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1ncc(F)c(C(F)F)n1)CC2
N#Cc1cccc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)n1
CC(C)Oc1cc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)ncc1C#N
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1cc(Br)cc(F)n1)CC2
CN(C)c1cc(Cl)nc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)n1
CC(=O)c1cnc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)cc1Cl
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1cccc(C(F)(F)F)n1)CC2
CC(=O)c1cccc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)n1
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1nc(Cl)nc3c1CCC3)CC2
CSc1ncc(C)c(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)n1
Cc1cc2c(N3CCC4(CC3)CN3CC[C@@H](c5cc(F)cc(F)c5)N3C4=O)ncnc2s1
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1ncnc3sccc13)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1cc(N3CCCC3)ncn1)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1cncc(-n3cccn3)n1)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1cccc(F)n1)CC2
CCc1nccc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)n1
Cc1csc2ncnc(N3CCC4(CC3)CN3CC[C@@H](c5cc(F)cc(F)c5)N3C4=O)c12
N#Cc1cc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)ncn1
N#Cc1ccnc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)n1
N#Cc1cnc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)nc1
CC(F)(F)c1ccnc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)n1
N#Cc1nccc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)n1
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1nccn3ncnc13)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1nc3ccccc3o1)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1noc3ccccc13)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1nnc(-c3ccccc3)o1)CC2
COc1cc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)ncn1
COc1nccc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)n1
COc1nc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)ncc1F
CNC(=O)c1cc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)ncn1
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1cc(-c3cnn(C(F)F)c3)ncn1)CC2
CN(C)C(=O)c1ccnc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)n1
COc1cc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)ccn1
CNC(=O)c1ccnc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)n1
Cn1cnc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)cc1=O
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1nccc(C(F)(F)F)n1)CC2
Cn1cc(-c2cc(N3CCC4(CC3)CN3CC[C@@H](c5cc(F)cc(F)c5)N3C4=O)ncn2)cn1
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1cc(C(F)(F)F)ncn1)CC2
COc1ccnc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)n1
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1cnnc(Cl)c1)CC2
N#Cc1ccc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)c2ccnn12
Cc1cc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)ccn1
N#Cc1cc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)ccn1
Cc1ccn(-c2ccnc(N3CCC4(CC3)CN3CC[C@@H](c5cc(F)cc(F)c5)N3C4=O)c2)n1
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1noc3ccccc13)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1ccnc3ccccc13)CC2
Cc1ccc2c(N3CCC4(CC3)CN3CC[C@@H](c5cc(F)cc(F)c5)N3C4=O)ccnc2c1
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1ncc(F)cc1C(F)F)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1ccnc3ccnn13)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1nccn3nccc13)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1cccc(-n3nccc3C(F)(F)F)n1)CC2
Cc1ccn(-c2cccc(N3CCC4(CC3)CN3CC[C@@H](c5cc(F)cc(F)c5)N3C4=O)n2)n1
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1cccc(-n3cccn3)n1)CC2
Cc1cnn(-c2cnc(N3CCC4(CC3)CN3CC[C@@H](c5cc(F)cc(F)c5)N3C4=O)cn2)c1
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1cnc(-c3ccccc3Cl)cn1)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1cnc(-c3cccc(Cl)c3)cn1)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1cnc(-c3ccc(Cl)cc3)cn1)CC2
N#Cc1cnc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)cn1
CSc1cnc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)cn1
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1ccc(OC(F)F)cn1)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1cc(-c3ccco3)ccn1)CC2
Cc1cc(-c2cncs2)nc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)c1
CCCOc1ccnc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)c1
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1cc(-n3ccnc3)ccn1)CC2
Cc1cnn(-c2ccnc(N3CCC4(CC3)CN3CC[C@@H](c5cc(F)cc(F)c5)N3C4=O)c2)c1
CCn6cnc5c(N1CCC4(CC1)CN3CC[C@@H](c2cc(F)cc(F)c2)N3C4=O)ncnc56
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1ncnc3scnc13)CC2
O=C(c1ncccn1)N1CCC2(CC1)CN1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
Cc1ccc(C(=O)N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)cc1
O=C(c1cccnc1)N1CCC2(CC1)CN1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
O=C(c1ccncc1)N1CCC2(CC1)CN1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
Cn1ccc(C(=O)N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)n1
N#Cc1cc(F)cc(C(=O)N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)c1
Cc1c(F)cccc1C(=O)N1CCC2(CC1)CN1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
O=C(c1c(F)ccc(F)c1F)N1CCC2(CC1)CN1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
O=C(c1cc(F)c(F)c(F)c1)N1CCC2(CC1)CN1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
O=C(c1cc(F)c(F)cc1F)N1CCC2(CC1)CN1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
O=C(c1cc(F)cc(F)c1F)N1CCC2(CC1)CN1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
Cc1ccc(F)cc1C(=O)N1CCC2(CC1)CN1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
Cc1ccc(F)cc1C(=O)N1CCC2(CC1)CN1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
N#Cc1ccc(C(=O)N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)cc1F
COc1ccc(C(=O)N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)cc1F
O=C(c1cncc(F)c1)N1CCC2(CC1)CN1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
Cc1cc(F)cc(C(=O)N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)c1
O=C(c1cc(F)cc(Cl)c1)N1CCC2(CC1)CN1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
O=C(c1cc(F)ccc1Cl)N1CCC2(CC1)CN1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
O=C(c1cc(F)ccc1F)N1CCC2(CC1)CN1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
Cc1ccc(C(=O)N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)cc1F
O=C(c1ccc(Cl)c(F)c1)N1CCC2(CC1)CN1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
O=C(c1ccc(F)c(F)c1)N1CCC2(CC1)CN1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
O=C(c1cccc(F)c1)N1CCC2(CC1)CN1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
Cc1cc(F)c(C(=O)N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)cc1F
COc1cc(F)cc(C(=O)N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)c1
O=C(c1cccc(F)c1Cl)N1CCC2(CC1)CN1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
O=C(c1cccc(F)c1F)N1CCC2(CC1)CN1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
COC(=O)N1CCC2(CC1)CN1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(S(=O)(=O)c1ccccc1)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1cncc(F)c1)CC2
O=C1N2[C@H](c3cc(F)cc(F)c3)CCN2CC12CCN(c1ccc(F)cc1)CC2
Cc1nc(N2CCC3(CC2)CN2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)ccc1F
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC)n[nH]c3c2)cc1C(=O)N[C@@H](C)c1cccc(OC(F)(F)F)c1
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC)n[nH]c3c2)cc1C(=O)NCCC(=O)OC(C)(C)C
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC)n[nH]c3c2)cc1C(=O)NCC[C@H](O)c1ccc(Cl)cc1
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC)n[nH]c3c2)cc1C(=O)NCC(C)(C)C(=O)OC(C)(C)C
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC)n[nH]c3c2)c(OC)c1C(=O)N[C@H](C)CC(=O)OC(C)(C)C
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC)n[nH]c3c2)cc1C(=O)N[C@H](C)c1cc(OC(F)(F)F)ccc1F
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC)n[nH]c3c2)cc1C(=O)N[C@H](C)c1cc(C(F)(F)F)ccc1F
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC)n[nH]c3c2)cc1C(=O)N[C@@H](C)c1cc(C(F)(F)F)ccc1F
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC)n[nH]c3c2)cc1C(=O)N[C@H](C)c1ccccc1C(F)(F)F
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC)n[nH]c3c2)cc1C(=O)N[C@H](C)c1cccc(C(F)(F)F)c1
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC)n[nH]c3c2)cc1C(=O)N[C@@H](C)c1cccc(C(F)(F)F)c1
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC)n[nH]c3c2)cc1C(=O)NC(C)c1cc(F)ccc1C(F)(F)F
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCCC(C)c4ccccc4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NC[C@H]4C[C@@H]4c4ccc(F)cc4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4ccc(F)cc4OC4CCOCC4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NC[C@H]4C[C@H]4c4ccccc4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NC[C@@H]4C[C@@H]4c4ccccc4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4ccccc4N4CCOCC4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4ccccc4CN(C)C)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCCCOc4ccccc4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCC(O)COc4ccccc4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4ccccc4N4CCC(CO)CC4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4ccccc4OC)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4ccccc4OCC(C)C)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCCCOC(C)(C)C)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCCCOC4CCCCO4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCCCOC4CCCCC4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCCCOc4ccc(F)cc4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCCCOCC(C)C)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCCC(O)c4ccc(Cl)cn4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4ccccc4S(C)(=O)=O)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)N[C@H]4CC[C@@H](c5ccccc5)C4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCC4(COc5ccccc5)CC4)c3)ccc12
CCCS(=O)(=O)c1ccccc1CNC(=O)c1cc(-c2ccc3c(C(=O)NC)n[nH]c3c2)cnc1OC
CNC(=O)c1[nH]nc2cc(-c3cnc(OC)c(C(=O)NC[C@@H]4C[C@H]4c4ccc(F)cc4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCC4(c5ccc(F)cc5)CC4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCC4(c5ccccc5OC(F)(F)F)CC4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4ccccc4NC(=O)OC(C)(C)C)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCCC(=O)OC(C)(C)C)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4ccccc4OCC(F)(F)F)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4cc(C(F)(F)F)ccc4OC)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NC[C@@H]4CCCC[C@H]4NC(=O)OC(C)(C)C)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4ccccc4OC(F)F)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCC4CCCOC4c4ccccc4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4ccccc4S(=O)(=O)C(C)C)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCC4CCCCC4(C)C)c3)ccc12
CCc1ccccc1CNC(=O)c1cc(-c2ccc3c(C(=O)NC)n[nH]c3c2)cnc1OC
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCC4CCCOC4C(C)(C)C)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4ccccc4C#N)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4ccccc4S(=O)(=O)NC4CC4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4ccccc4OCC4CCC4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NC4CCCC(OCC(F)(F)F)C4)c3)ccc12
CCOC(=O)C(C)(C)CNC(=O)c1cc(-c2ccc3c(C(=O)NC)n[nH]c3c2)cnc1OC
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCC/C(OC)=C(F)C=C(/C)F)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCC(C)(C)C(=O)OC(C)(C)C)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCC(C)(C)C(=O)NCc4ccc(F)cc4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4cccc(OC(F)(F)F)c4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4ccccc4OC(C)C)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4cccnc4OC)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NC45CC6CC(C4)CC(c4ccccc4)(C6)C5)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCC4CCCN4C(=O)C(C)(C)C(F)(F)F)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NC(C)c4cccc(OC(F)(F)F)c4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NC4CCCC(C(=O)N5CCOCC5)C4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NC4CCCC(C(=O)N5CCCC5)C4)c3)ccc12
CCCN(C)C(=O)C1CCCC(NC(=O)c2cc(-c3ccc4c(C(=O)NC)n[nH]c4c3)cnc2OC)C1
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NC(C)c4cccc(C(F)(F)F)c4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4cccc(C(F)(F)F)c4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCC(F)(F)COC(C)C)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4ccc(F)c(C(F)(F)F)c4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NC(C)c4ccc(F)c(C(F)(F)F)c4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4cccc(OCC5CC5)c4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4cccc(OC5CCCC5)c4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4ccccc4C(F)(F)F)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NC(C)c4ccccc4C(F)(F)F)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4ccccc4OCC4CCCC4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4cccc(OC(C)C)c4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4cccnc4OCC4CCC4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4ccccc4OC4CCCCC4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4cccc(C(F)(F)F)c4F)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4cccc(OCC5CCC5)c4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCC4CCCC4(C)C)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4ncccc4OCC4CCC4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NC4CCCC(Oc5ccccc5)C4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4cccc(OC(F)(F)F)c4F)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NC4CCCC(C(=O)N(C)C)C4)c3)ccc12
CCN(CC)C(=O)C1CCCC(NC(=O)c2cc(-c3ccc4c(C(=O)NC)n[nH]c4c3)cnc2OC)C1
CCN(C)C(=O)C1CCCC(NC(=O)c2cc(-c3ccc4c(C(=O)NC)n[nH]c4c3)cnc2OC)C1
CCCN(CC1CC1)C(=O)C1CCCC(NC(=O)c2cc(-c3ccc4c(C(=O)NC)n[nH]c4c3)cnc2OC)C1
CCN(CC1CCC1)C(=O)C1CCCC(NC(=O)c2cc(-c3ccc4c(C(=O)NC)n[nH]c4c3)cnc2OC)C1
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NC4CCCC(C(=O)N(C)C5CC5)C4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4cc(F)cc(F)c4OC(C)C)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4c(F)cccc4OC(C)C)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4cc(F)cc(F)c4OCC4CC4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NC(C)c4ccccc4C(F)(F)F)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4cc(F)ccc4OC(C)C)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4ccccc4OC4CCC(C)C4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NC4CCCC(C(=O)N5CC(F)(F)C5)C4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCC4(C(=O)OC5CCCCC5)CC4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)N4CCC[C@@H](Cc5ccc(F)cc5)C4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCCCC(=O)OC(C)(C)C)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)N[C@H]4CCN(C(=O)OC(C)(C)C)C4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4cc(OC(F)(F)F)ccc4F)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCC4CCCCC4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)N[C@@H](C)CC(=O)OC(C)(C)C)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCC4(C(=O)OC5CCCC5)CC4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)N[C@H](C)CC(=O)OC(C)(C)C)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCCCC(=O)N(CC4CC4)C4CC4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4cc(C(F)(F)F)ccn4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCC(C)(C)C(=O)OC(C)(C)C)c3)cc(F)c12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCC[C@H](O)c4ccc(Cl)cc4)c3)cc(F)c12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)N[C@@H](C)CC(=O)OC(C)(C)C)c3)cc(F)c12
CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NC(C)c4cccc(OC(F)(F)F)c4)c3)cc(F)c12
[2H]C([2H])([2H])NC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCC(C)(C)C(=O)OC4CCOCC4)c3)ccc12
[2H]C([2H])([2H])NC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCC(C)(C)C(=O)OC(C)(C)C)c3)ccc12
[2H]C([2H])([2H])NC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCCC(=O)OC(C)(C)C)c3)ccc12
[2H]C([2H])([2H])NC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NC(C)c4cccc(OC(F)(F)F)c4)c3)ccc12
[2H]C([2H])([2H])NC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NC(C)c4ccccc4OC(F)(F)F)c3)ccc12
[2H]C([2H])([2H])NC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4ccccc4OC(F)(F)F)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(C)c(C(=O)N[C@H]4CC[C@@H](c5ccccc5)C4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(C)c(C(=O)NC(C)c4cccc(OC(F)(F)F)c4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(C)c(C(=O)NC(C)c4cccc(OC(F)(F)F)c4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cnc(C)c(C(=O)NCc4cc(F)ccc4OC4CCCC4)c3)ccc12
CNC(=O)c1n[nH]c2cc(-c3cc(C(=O)NC(C)c4ccccc4OC(F)(F)F)c(OC)nc3C)ccc12
CNC(=O)c1n[nH]c2cc(-c3cc(C(=O)NCC4CCCC4(C)C)c(OC)nc3C)ccc12
CNC(=O)c1n[nH]c2cc(-c3cc(C(=O)NCc4cccc(OC(F)(F)F)c4)c(OC)nc3C)ccc12
CNC(=O)c1n[nH]c2cc(-c3cc(C(=O)NCc4cc(OC(F)(F)F)ccc4F)c(OC)nc3C)ccc12
CNC(=O)c1n[nH]c2cc(-c3cc(C(=O)NC(C)c4ccccc4OC(F)(F)F)c(C)nc3C)ccc12
CNC(=O)c1n[nH]c2cc(-c3cc(C(=O)NC(C)c4cccc(OC(F)(F)F)c4)c(C)nc3C)ccc12
CNC(=O)c1n[nH]c2cc(-c3cc(C(=O)NC(C)c4cccc(OC(F)(F)F)c4)c(C)nc3C)ccc12
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NCC4CC4)n[nH]c3c2)cc1C(=O)NCCC(=O)OC(C)(C)C
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NCC4CC4)n[nH]c3c2)cc1C(=O)NC(C)c1cccc(OC(F)(F)F)c1
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NCC4CC4)n[nH]c3c2)cc1C(=O)NCC[C@H](O)c1ccc(Cl)cc1
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NCC4CC4)n[nH]c3c2)cc1C(=O)NC(C)c1ccccc1OC(F)(F)F
COc1ncc(-c2ccc3c(C(=O)NC4CCN(S(C)(=O)=O)CC4)n[nH]c3c2)cc1C(=O)NCc1ccccc1OC(F)(F)F
CCNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4ccccc4OC(F)(F)F)c3)ccc12
COc1ncc(-c2ccc3c(C(=O)N[C@H](C)C4CC4)n[nH]c3c2)cc1C(=O)NCc1ccccc1OC(F)(F)F
COc1ncc(-c2ccc3c(C(=O)NCC4CC4)n[nH]c3c2)cc1C(=O)NCc1ccccc1OC(F)(F)F
COc1ncc(-c2ccc3c(C(=O)N[C@@H](C)C4CC4)n[nH]c3c2)cc1C(=O)NCc1ccccc1OC(F)(F)F
COc1ncc(-c2ccc3c(C(=O)NC4CC4)n[nH]c3c2)cc1C(=O)NCc1ccccc1OC(F)(F)F
CCCCNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4ccccc4OC(F)(F)F)c3)ccc12
CCCNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4ccccc4OC(F)(F)F)c3)ccc12
COc1ncc(-c2ccc3c(C(=O)NCCCN4CCCC4=O)n[nH]c3c2)cc1C(=O)NCc1ccccc1OC(F)(F)F
COc1ncc(-c2ccc3c(C(=O)NCC(F)(F)F)n[nH]c3c2)cc1C(=O)NCc1ccccc1OC(F)(F)F
COc1ncc(-c2ccc3c(C(=O)NC(C)C)n[nH]c3c2)cc1C(=O)NCc1ccccc1OC(F)(F)F
COc1ncc(-c2ccc3c(C(=O)NC4CCN(C(C)=O)CC4)n[nH]c3c2)cc1C(=O)NCc1ccccc1OC(F)(F)F
COc1ncc(-c2ccc3c(C(=O)NC4CC(=O)N(C(C)C)C4)n[nH]c3c2)cc1C(=O)NCc1ccccc1OC(F)(F)F
COc1ncc(-c2ccc3c(C(=O)NCCO)n[nH]c3c2)cc1C(=O)NCc1ccccc1OC(F)(F)F
[2H]C([2H])([2H])C([2H])([2H])NC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4ccccc4OC(F)(F)F)c3)ccc12
CCN(CC)C1CCC(NC(=O)c2n[nH]c3cc(-c4cnc(OC)c(C(=O)NCc5ccccc5OC(F)(F)F)c4)ccc23)CC1
COc1ncc(-c2ccc3c(C(=O)NC4CCC(N(C)C)CC4)n[nH]c3c2)cc1C(=O)NCc1ccccc1OC(F)(F)F
COc1ccccc1N1CC(NC(=O)c2n[nH]c3cc(-c4cnc(OC)c(C(=O)NCc5ccccc5OC(F)(F)F)c4)ccc23)CC1=O
COc1ncc(-c2ccc3c(C(=O)NC4CC(=O)N(C)C4)n[nH]c3c2)cc1C(=O)NCc1ccccc1OC(F)(F)F
[2H]C([2H])([2H])C(NC1CCC(NC(=O)c2n[nH]c3cc(-c4cnc(OC)c(C(=O)NCc5ccccc5OC(F)(F)F)c4)ccc23)CC1)C([2H])([2H])[2H]
COc1ncc(-c2ccc3c(C(=O)NC4CCC(O)CC4)n[nH]c3c2)cc1C(=O)NCc1ccccc1OC(F)(F)F
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC4CC4)n[nH]c3c2)cc1C(=O)N[C@@H]1CN(C(=O)C2CC(F)(F)C2)C[C@@H]1F
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC4CC(F)(F)C4)n[nH]c3c2)cc1C(=O)N[C@@H]1CN(C(=O)C2CC(F)(F)C2)C[C@@H]1F
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NCC([2H])([2H])C([2H])([2H])[2H])n[nH]c3c2)cc1C(=O)N[C@@H]1CN(C(=O)C2CC(F)(F)C2)C[C@@H]1F
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NCC(C)(C)F)n[nH]c3c2)cc1C(=O)N[C@@H]1CN(C(=O)C2CC(F)(F)C2)C[C@@H]1F
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC4CC4)n[nH]c3c2)cc1C(=O)N[C@@H](C)c1cc(C(F)(F)F)ccc1F
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC4CC4)n[nH]c3c2)cc1C(=O)N[C@@H](C)CC(=O)OC(C)(C)C
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC4CC4)n[nH]c3c2)cc1C(=O)N[C@H](C)CC(=O)OC(C)(C)C
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC4CC4)n[nH]c3c2)cc1C(=O)NC(C)c1cccc(OC(F)(F)F)c1
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC4CC4)n[nH]c3c2)cc1C(=O)NCC[C@H](O)c1ccc(Cl)cc1
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC4CC4)n[nH]c3c2)cc1C(=O)N[C@@H]1CN(C(=O)C2CCC(F)(F)C2)C[C@@H]1F
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC4CC4)n[nH]c3c2)cc1C(=O)NCC(C)(C)C(=O)OC(C)(C)C
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC4CC4)n[nH]c3c2)cc1C(=O)N[C@H](C)c1cc(OC(F)(F)F)ccc1F
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC4CC4)n[nH]c3c2)cc1C(=O)N[C@H](C)c1cccc(OC(F)(F)F)c1
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC4CC4)n[nH]c3c2)cc1C(=O)NC1CCCC(C(=O)N2CCC(F)(F)C2)C1
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC4CC4)n[nH]c3c2)cc1C(=O)NC1CCCC(C(=O)N2CCCC2)C1
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC4CC4)n[nH]c3c2)cc1C(=O)N[C@@H](c1cccc(OC(F)(F)F)c1)C([2H])([2H])[2H]
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC4CC4)n[nH]c3c2)cc1C(=O)N[C@H](c1cc(OC(F)(F)F)ccc1F)C([2H])([2H])[2H]
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC4CC4)n[nH]c3c2)cc1C(=O)N[C@@H](c1cc(OC(F)(F)F)ccc1F)C([2H])([2H])[2H]
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC4CC4)n[nH]c3c2)cc1C(=O)N[C@H](c1cc(OC(F)(F)F)ccc1[3H])C([2H])([2H])[2H]
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC4CC4)n[nH]c3c2)cc1C(=O)N[C@@H](C)c1ccccc1C(F)(F)F
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC4CC4)n[nH]c3c2)cc1C(=O)N[C@H](C)c1cccc(C(F)(F)F)c1
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC4CC4)n[nH]c3c2)cc1C(=O)N[C@@H](C)c1cccc(C(F)(F)F)c1
[2H]C([2H])([2H])NC(=O)c1n[nH]c2cc(-c3cnc(OC([2H])([2H])[2H])c(C(=O)NC(C)c4cc(F)ccc4C(F)(F)F)c3)ccc12
[2H]C([2H])([2H])NC(=O)c1n[nH]c2cc(-c3cnc(OC([2H])([2H])[2H])c(C(=O)N[C@@H](C)c4cc(C(F)(F)F)ccc4F)c3)ccc12
[2H]C([2H])([2H])NC(=O)c1n[nH]c2cc(-c3cnc(OC([2H])([2H])[2H])c(C(=O)N[C@@H](C)c4cccc(C(F)(F)F)c4)c3)ccc12
[2H]C([2H])([2H])NC(=O)c1n[nH]c2cc(-c3cnc(OC([2H])([2H])[2H])c(C(=O)N[C@H](c4cc(C(F)(F)F)ccc4F)C([2H])([2H])[2H])c3)ccc12
[2H]C([2H])([2H])NC(=O)c1n[nH]c2cc(-c3cnc(OC([2H])([2H])[2H])c(C(=O)N[C@@H](c4cc(C(F)(F)F)ccc4F)C([2H])([2H])[2H])c3)ccc12
[2H]C([2H])([2H])NC(=O)c1n[nH]c2cc(-c3cnc(OC([2H])([2H])[2H])c(C(=O)N[C@H](c4cccc(OC(F)(F)F)c4)C([2H])([2H])[2H])c3)ccc12
[2H]C([2H])([2H])NC(=O)c1n[nH]c2cc(-c3cnc(OC([2H])([2H])[2H])c(C(=O)N[C@H](C)c4cc(OC(F)(F)F)ccc4F)c3)ccc12
[2H]C([2H])([2H])NC(=O)c1nn(C)c2cc(-c3cnc(OC([2H])([2H])[2H])c(C(=O)N[C@H](C)c4ccccc4C(F)(F)F)c3)ccc12
[2H]C([2H])([2H])NC(=O)c1nn(C)c2cc(-c3cnc(OC([2H])([2H])[2H])c(C(=O)N[C@@H](C)c4cccc(OC(F)(F)F)c4)c3)ccc12
[2H]C([2H])([2H])NC(=O)c1nn(C)c2cc(-c3cnc(OC([2H])([2H])[2H])c(C(=O)N[C@@H](c4cccc(OC(F)(F)F)c4)C([2H])([2H])[2H])c3)ccc12
[2H]C([2H])([2H])NC(=O)c1nn(C)c2cc(-c3cnc(OC([2H])([2H])[2H])c(C(=O)N[C@@H](c4cc(OC(F)(F)F)ccc4F)C([2H])([2H])[2H])c3)ccc12
[2H]C([2H])([2H])NC(=O)c1nn(C)c2cc(-c3cnc(OC([2H])([2H])[2H])c(C(=O)N[C@@H](c4cc(C(F)(F)F)ccc4F)C([2H])([2H])[2H])c3)ccc12
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC([2H])([2H])C([2H])([2H])[2H])n[nH]c3c2)cc1C(=O)N[C@H](C)c1cc(OC(F)(F)F)ccc1F
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC([2H])([2H])C([2H])([2H])[2H])n[nH]c3c2)cc1C(=O)N[C@@H](C)c1cc(OC(F)(F)F)ccc1F
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC([2H])([2H])C([2H])([2H])[2H])n[nH]c3c2)cc1C(=O)N[C@H](C)c1cc(C(F)(F)F)ccc1F
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC([2H])([2H])C([2H])([2H])[2H])n[nH]c3c2)cc1C(=O)N[C@@H](C)c1cc(C(F)(F)F)ccc1F
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC([2H])([2H])C([2H])([2H])[2H])n[nH]c3c2)cc1C(=O)NC(C)c1cc(F)ccc1C(F)(F)F
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC([2H])([2H])C([2H])([2H])[2H])n[nH]c3c2)cc1C(=O)NC(C)c1cccc(C(F)(F)F)c1
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC([2H])([2H])C([2H])([2H])[2H])n[nH]c3c2)cc1C(=O)N[C@H](C)c1cccc(C(F)(F)F)c1
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC([2H])([2H])C([2H])([2H])[2H])n[nH]c3c2)cc1C(=O)N[C@@H](C)c1cccc(OC(F)(F)F)c1
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC([2H])([2H])C([2H])([2H])[2H])n[nH]c3c2)cc1C(=O)N[C@H](c1cccc(OC(F)(F)F)c1)C([2H])([2H])[2H]
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC([2H])([2H])C([2H])([2H])[2H])n[nH]c3c2)cc1C(=O)N[C@H](c1cc(OC(F)(F)F)ccc1F)C([2H])([2H])[2H]
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC([2H])([2H])C([2H])([2H])[2H])n[nH]c3c2)cc1C(=O)N[C@H](c1cc(C(F)(F)F)ccc1F)C([2H])([2H])[2H]
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC([2H])([2H])C([2H])([2H])[2H])n[nH]c3c2)cc1C(=O)N[C@@H](C)c1ccccc1C(F)(F)F
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC([2H])([2H])C([2H])([2H])[2H])n[nH]c3c2)cc1C(=O)N[C@@H](c1cc(C(F)(F)F)ccc1F)C([2H])([2H])[2H]
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC([2H])([2H])C([2H])([2H])[2H])n[nH]c3c2)cc1C(=O)NCC[C@H](O)c1ccc(Cl)cc1
[2H]C([2H])([2H])Oc1ncc(-c2ccc3c(C(=O)NC([2H])([2H])C([2H])([2H])[2H])n[nH]c3c2)cc1C(=O)N[C@H](C)CC(=O)OC(C)(C)C
O=C(c1ccccc1)N1CCC2(CC1)O[C@@H]1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
COC(=O)N1CCC2(CC1)O[C@@H]1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
O=C(c1ccccc1)N1CCC2(CC1)O[C@@H]1CC[C@@H](c3ccccc3)N1C2=O
O=C(c1ccccc1)N1CCC2(CC1)O[C@@H]1CC[C@@H](c3cncc(F)c3)N1C2=O
O=C(c1ccccc1)N1CCC2(CC1)O[C@@H]1CC[C@@H](c3cccc(F)c3)N1C2=O
O=C(c1cc(F)ccc1F)N1CCC2(CC1)O[C@@H]1CC[C@@H](c3cccc(F)c3)N1C2=O
O=C(c1ccccc1F)N1CCC2(CC1)O[C@@H]1CC[C@@H](c3cccc(F)c3)N1C2=O
O=C(C1CC1)N1CCC2(CC1)O[C@@H]1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
O=C(c1ccccc1F)N1CCC2(CC1)O[C@@H]1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
O=C(c1ccccc1F)N1CCC2(CC1)O[C@@H]1CC[C@@H](c3ccccc3)N1C2=O
O=C(c1cc(F)ccc1F)N1CCC2(CC1)O[C@@H]1CC[C@@H](c3ccccc3)N1C2=O
O=C(c1cc(F)ccc1F)N1CCC2(CC1)O[C@@H]1CC[C@@H](c3ccccc3F)N1C2=O
O=C(c1ccccc1)N1CCC2(CC1)O[C@@H]1CC[C@@H](c3ccccc3F)N1C2=O
O=C(c1cc(Cl)ccc1F)N1CCC2(CC1)O[C@@H]1CC[C@@H](c3ccccc3F)N1C2=O
O=C(c1cc(F)ccc1Cl)N1CCC2(CC1)O[C@@H]1CC[C@@H](c3ccccc3F)N1C2=O
O=C(c1ccccc1F)N1CCC2(CC1)O[C@@H]1CC[C@@H](c3ccccc3F)N1C2=O
Cc1ccc(F)c(C(=O)N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4F)N2C3=O)c1
O=C(c1cc(F)ccc1F)N1CC2(C1)O[C@@H]1CC[C@@H](c3ccccc3F)N1C2=O
O=C(c1ccccc1)N1CC2(C1)O[C@@H]1CC[C@@H](c3ccccc3F)N1C2=O
O=C(c1cc(F)ccc1F)N1CC2(C1)O[C@@H]1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
O=C(c1ccccc1)N1CCC2(CC1)SC1CC[C@H](c3cc(F)cc(F)c3)N1C2=O
O=C(c1ccccc1)N1CCC2(CC1)SC1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
O=C(c1ccccc1)N1CCC2(CC1)S[C@@H]1CC[C@@H](c3ccccc3)N1C2=O
O=C(c1cc(F)ccc1F)N1CCC2(CC1)SC1CCC(c3ccccc3)N1C2=O
O=C(c1ccccc1)N1CC2(C1)S[C@@H]1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
Cc1ncc([C@@H]2CC[C@H]3OC4(CN(C(=O)c5ccccc5)C4)C(=O)N32)cc1F
O=C(c1ccccc1)N1CCC2(O[C@@H]3CC[C@@H](c4ccccc4)N3C2=O)C(F)C1
O=C(c1ccccc1)N1CCC2(O[C@@H]3CC[C@@H](c4ccccc4)N3C2=O)C(F)C1
CC1CN(C(=O)c2ccccc2)CCC12O[C@@H]1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
CC1CN(C(=O)c2ccccc2)CCC12O[C@@H]1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
CC1CN(C(=O)c2ccccc2)CCC12O[C@@H]1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
CC1CN(C(=O)c2ccccc2)CCC12O[C@@H]1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
O=C(c1ccccc1)N1CCC2(CC1)O[C@@H]1CC[C@@H](c3ccc(F)cc3)N1C2=O
Cc1ncc([C@@H]2CC[C@H]3OC4(CCN(C(=O)c5ccccc5)CC4F)C(=O)N32)cc1F
Cc1ncc([C@@H]2CC[C@H]3OC4(CCN(C(=O)c5ccccc5)CC4F)C(=O)N32)cc1F
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1ccnc3c(F)cnn13)CC2
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ccnc3c(F)cnn13)CC2
Cc1cc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)nc(C#N)n1
O=C1N2C(CCC2c2cc(F)cc(F)c2)OC12CCN(c1cc(F)ccn1)CC2
N#Cc1cc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)ncn1
N#Cc1nccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)n1
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1ccnc3ccnn13)CC2
N#Cc1cncc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)n1
N#Cc1ccnc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)c1
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1ccnc(C(F)F)n1)CC2
COc1ccnc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)n1
COc1cc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)ncn1
N#Cc1ccnc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)n1
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1cc(-c3ccccc3)ncn1)CC2
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1cc(F)ccn1)CC2
O=C1N2[C@H](CC[C@H]2c2cccc(F)c2)OC12CCN(c1ccnc3c(F)cnn13)CC2
Cc1cc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)cc(C#N)n1
COc1nccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)n1
N#Cc1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)cc1F
N#Cc1cnnc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)c1
N#Cc1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)cc1Cl
COc1nc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)ncc1F
Cc1nc(Cl)c(C)c(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)n1
CCOC(=O)c1cc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)ncn1
N#Cc1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)c(F)c1
Cc1nccn1-c1cc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)ncn1
Cc1cnn(-c2cc(N3CCC4(CC3)O[C@@H]3CC[C@@H](c5ccccc5)N3C4=O)ncn2)c1
CSc1cc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)ncn1
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ccnc3ccnn13)CC2
N#Cc1cccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)n1
Cc1c(Cl)ncnc1N1CCC2(CC1)O[C@@H]1CC[C@@H](c3ccccc3)N1C2=O
N#Cc1cc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)ccn1
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1cc(-c3ccccc3)ncn1)CC2
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1cc(C(F)(F)F)ncn1)CC2
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1cc(Cl)nc(C3CCCCC3)n1)CC2
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1cc(-n3cccn3)ncn1)CC2
CSc1nc(C)cc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)n1
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ncnc3ccsc13)CC2
COc1nc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)ncc1C#N
COc1cc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)ncn1
N#Cc1cc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)ncn1
CC(C)Oc1cc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)ncc1C#N
Cc1nc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)ccc1C#N
COc1cc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)ncc1C#N
N#Cc1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)nc1
N#Cc1ncc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)cn1
Cc1ncc([C@@H]2CC[C@H]3OC4(CCN(c5ccc(C#N)c(C)n5)CC4)C(=O)N32)cc1F
Cc1cc(C#N)cnc1N1CCC2(CC1)O[C@@H]1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
N#CN1CCC2(CC1)O[C@@H]1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
O=C1N2[C@@H](CC[C@H]2c2cncc(F)c2)OC12CCN(c1ccnc3c(F)cnn13)CC2
N#Cc1cnc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cccc(F)c4)N2C3=O)c(F)c1
COc1cc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cccc(F)c4)N2C3=O)ncn1
O=C1N2[C@@H](CC[C@H]2c2cccc(F)c2)OC12CCN(c1cc(C(F)F)ncn1)CC2
N#Cc1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cccc(F)c4)N2C3=O)c(F)c1
N#Cc1ccnc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cccc(F)c4)N2C3=O)c1
CSc1cnc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)nc1
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1ncc(C3CC3)cn1)CC2
CCOc1cnc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)nc1
Cc1nc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)ncc1OC(F)F
COc1nc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)ncc1C
CCc1cnc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)nc1
Cc1nc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)ncc1F
COc1nc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)ncc1Cl
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1ncc(Cl)cn1)CC2
COc1cnc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)nc1
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1ncc(F)c(C3CC3)n1)CC2
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1ncc(F)c(C(F)F)n1)CC2
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1ncc(F)cn1)CC2
N#Cc1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)cc1
COc1cc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)nc(C)c1C#N
N#Cc1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)cc1-n1ccnn1
CSc1cc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)ncc1C#N
N#Cc1cnc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)c(F)c1
N#Cc1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)c(F)c1
Cc1nc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)ccc1C#N
N#Cc1cnc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)cc1F
N#Cc1cnc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)nc1
Cc1nc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cccc(F)c4)N2C3=O)ccc1C#N
Cc1nc(N2CCC3(CC2)C[C@@H]2OC[C@@H](c4ccccc4)N2C3=O)ccc1C#N
O=C1N2C(=NC13CCN(c1ccnc4c(F)cnn14)CC3)CC[C@H]2c1cc(F)cc(F)c1
N#Cc1cc(N2CCC3(CC2)N=C2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)ncn1
C[C@@]12CC[C@@H](c3ccccc3)N1C(=O)C1(CCN(c3ccnc4c(F)cnn34)CC1)O2
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1nccc3nccn13)CC2
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1ccnc3ncnn13)CC2
O=C1N2[C@@H](CC[C@H]2c2cncc(F)c2)OC12CCN(c1ccnc3c(F)cnn13)CC2
Cc1cc2nccc(N3CCC4(CC3)O[C@@H]3CC[C@@H](c5cc(F)cc(F)c5)N3C4=O)n2n1
CSc1cc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)n2nccc2n1
O=C1N2[C@@H](CC[C@H]2C2CCCCC2)OC12CCN(c1ccnc3c(F)cnn13)CC2
O=C1N2[C@@H](CC[C@H]2C2CCCC2)OC12CCN(c1ccnc3c(F)cnn13)CC2
Cc1ncc([C@@H]2CC[C@H]3OC4(CCN(c5ccnc6ccnn56)CC4)C(=O)N32)cc1F
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1ncc(F)c3ncnn13)CC2
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ccnc3c(F)cnn13)CC2F
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ccnc3c(F)cnn13)CC2F
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ncnc3ccnn13)CC2
N#Cc1cc(N2CCC3(O[C@@H]4CC[C@@H](c5ccccc5)N4C3=O)C(F)C2)ncn1
N#Cc1cc(N2CCC3(O[C@@H]4CC[C@@H](c5ccccc5)N4C3=O)C(F)C2)ncn1
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CN(c1ccnc3c(F)cnn13)C2
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ncnc3ccnn13)CC2F
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ncnc3ccnn13)CC2F
O=C1N2[C@@H](CC[C@H]2c2ccccc2F)OC12CCN(c1cc(Cl)ncn1)CC2
N#Cc1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)nn1
N#Cc1cnc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)s1
O=C1N2[C@@H](CC[C@H]2c2ccccc2F)OC12CCN(c1ccnc3c(F)cnn13)CC2
O=C1N2[C@@H](CC[C@H]2c2ccccc2F)OC12CCN(c1ccnc3ccnn13)CC2
N#Cc1cc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4F)N2C3=O)ncn1
Cc1nc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4F)N2C3=O)ccc1C#N
N#Cc1cnc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4F)N2C3=O)nc1
O=C1N2[C@@H](CC[C@H]2c2ccccc2F)OC12CN(c1cc(Cl)ncn1)C2
O=C1N2[C@@H](CC[C@H]2c2ccccc2F)OC12CN(c1ccnc3ccnn13)C2
O=C1N2[C@@H](CC[C@H]2c2ccccc2F)OC12CN(c1ccnc(Cl)c1)C2
O=C1N2C(CCC2c2cc(F)cc(F)c2)SC12CCN(c1ccnc3c(F)cnn13)CC2
N#Cc1cc(N2CCC3(CC2)SC2CCC(c4cc(F)cc(F)c4)N2C3=O)ncn1
N#Cc1cncc([C@@H]2CC[C@H]3SC4(CCN(c5ccnc6c(F)cnn56)CC4)C(=O)N32)c1
N#Cc1cc(N2CCC3(CC2)C[C@@H]2OC[C@@H](c4ccccc4)N2C3=O)ncn1
O=C1N2[C@@H](CC[C@H]2c2cc(F)ccc2F)OC12CCN(c1ccnc3ccnn13)CC2
O=C1N2[C@H](CC[C@@H]2c2ccccc2)SC12CCN(c1ccnc3ccnn13)CC2
O=C1N2[C@@H](CC[C@H]2c2ccccc2)SC12CCN(c1ccnc3ccnn13)CC2
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CN(c1ccnc3c(F)cnn13)C2
N#Cc1cc(N2CC3(C2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)ncn1
N#Cc1cnc(N2CC3(C2)O[C@@H]2CC[C@@H](c4ccccc4F)N2C3=O)nc1
O=C1N2[C@H](CC13CCN(c1ccnc4c(F)cnn14)CC3)OC[C@H]2c1ccccc1
N#Cc1cc(F)cc([C@@H]2CC[C@H]3OC4(CCN(c5ccnc6c(F)cnn56)CC4)C(=O)N32)c1
N#Cc1cc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cccc(F)c4)N2C3=O)ncn1
O=C1N2[C@@H](CC[C@H]2c2cccc(F)c2)OC12CCN(c1ccnc3ccnn13)CC2
O=C1N2[C@@H](CC[C@H]2c2ccc(F)cc2)OC12CCN(c1ccnc3c(F)cnn13)CC2
O=C1N2[C@@H](CC[C@H]2c2cccc(F)c2)OC12CCN(c1cc(-c3ccccc3)ncn1)CC2
O=C1N2[C@@H](CC[C@H]2c2cccc(F)c2)OC12CCN(c1cc(F)ccn1)CC2
N#Cc1cncc([C@@H]2CC[C@H]3OC4(CCN(c5ccnc6c(F)cnn56)CC4)C(=O)N32)c1
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1ncnc3ccnn13)CC2
O=C1N2[C@@H](CC[C@H]2c2cccc(F)c2)OC12CCN(c1ccnc3c(F)cnn13)CC2
Cc1ncc([C@@H]2CC[C@H]3OC4(CCN(c5ccnc6c(F)cnn56)CC4F)C(=O)N32)cc1F
Cc1ncc([C@@H]2CC[C@H]3OC4(CCN(c5ccnc6c(F)cnn56)CC4F)C(=O)N32)cc1F
O=C1N2[C@@H](CC[C@H]2c2ccccc2)SC12CCN(c1ccnc3c(F)cnn13)CC2
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CN(c1cccc3ncnn13)C2
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CN(c1ccnc3ccnn13)C2
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CN(c1cccc3ncnn13)C2
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CN(c1ccnc3ccnn13)C2
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CN(c1ncnc3ccnn13)C2
O=C1N2[C@@H](CC[C@H]2c2ccccc2F)OC12CN(c1ccnc(-c3cnn(C(F)F)c3)c1)C2
O=C1N2[C@@H](CC[C@H]2c2ccccc2F)OC12CN(c1ccnc(-c3ccc(F)cc3)c1)C2
O=C1N2[C@@H](CC[C@H]2c2cnccn2)OC12CCN(c1ccnc3c(F)cnn13)CC2
N#Cc1ccc(N2CCC3(CC2)OC2CCC(c4cnccn4)N2C3=O)n2ncnc12
Cc1nc(N2CCC3(CC2)OC2CCC(c4cnccn4)N2C3=O)ccc1C#N
O=C1N2[C@@H](CC[C@H]2c2cnccn2)OC12CCN(c1ccnc3c(F)cnn13)CC2
Cc1nccnc1[C@@H]1CC[C@H]2OC3(CCN(c4ccnc5c(F)cnn45)CC3)C(=O)N21
N#Cc1ccc(N2CCC3(CC2)S[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)n2nccc12
N#Cc1cnc(N2CCC3(CC2)S[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)n2ncnc12
O=C1N2[C@@H](CO[C@H]2c2cc(F)cc(F)c2)CC12CCN(c1ccnc3ccnn13)CC2
O=C1N2[C@@H](CO[C@H]2c2cc(F)cc(F)c2)CC12CCN(c1ccnc3c(F)cnn13)CC2
O=C1N2[C@H](OC13CCN(c1ccnc4c(F)cnn14)CC3)[C@H](O)C[C@H]2c1ccccc1
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1cccn3nccc13)CC2
NC(=O)c1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4F)N2C3=O)n2ncnc12
NC(=O)c1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cccc(F)c4)N2C3=O)n2ncnc12
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ccc(Cl)c3ccnn13)CC2
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1nc3ccccc3o1)CC2
NC(=O)c1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)n2nccc12
N#Cc1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4F)N2C3=O)n2nccc12
N#Cc1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cccc(F)c4)N2C3=O)n2nccc12
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1nc3ccncc3o1)CC2
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1nc3cnccc3o1)CC2
COc1ccc2oc(N3CCC4(CC3)O[C@@H]3CC[C@@H](c5ccccc5)N3C4=O)nc2c1
O=C(c1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)nc1)C(F)F
CC(C)(C)OC(=O)/C=C/c1cnc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)cc1Cl
CC(C)(C)OC(=O)/C=C/c1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)nc1
COCOc1cc(-c2ccc(N3CCC4(CC3)O[C@@H]3CC[C@@H](c5ccccc5)N3C4=O)nc2)on1
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ccc(-c3nnc(C(F)(F)F)o3)cn1)CC2
O=C3N1[C@@H](CC[C@H]1c2ccccc2)OC37CCN(c6ccc(c5nc4ccccc4[nH]5)cn6)CC7
CN(C)C(=O)c1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)nc1
CC(C)(C)OC(=O)/C=C/c1cnc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)cc1Cl
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1cc(-c3ccco3)ccn1)CC2
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1cc(-c3ccsc3)ccn1)CC2
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1cc(-n3ccnc3)ncn1)CC2
Cc1cn(-c2cc(N3CCC4(CC3)O[C@@H]3CC[C@@H](c5ccccc5)N3C4=O)ncn2)cn1
CCOC(=O)c1coc(-c2ccnc(N3CCC4(CC3)O[C@@H]3CC[C@@H](c5ccccc5)N3C4=O)c2)n1
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1cc(-n3cccn3)ncn1)CC2
Cc1nccn1-c1cc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)ncn1
Cc1cnn(-c2cc(N3CCC4(CC3)O[C@@H]3CC[C@@H](c5ccccc5)N3C4=O)ncn2)c1
N#Cc1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)n2ncc(F)c12
N#Cc1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)n2ncc(C#N)c12
N#Cc1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)n2ncc(C(F)F)c12
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ccc(-c3ncco3)c3ncnn13)CC2
N#Cc1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)n2ncc(-c3ncco3)c12
N#Cc1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)n2ncc(Cl)c12
N#Cc1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)n2ncc(Br)c12
NC(=O)c1nc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)ncc1F
NC(=O)c1cc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)ncn1
CC(=O)c1cnc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)cc1Cl
Cc1cc2c(nc1N1CCC3(CC1)O[C@@H]1CC[C@@H](c4ccccc4)N1C3=O)CNC2=O
COC(=O)c1cc(C)c(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)nc1C#N
COC(=O)c1cnc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)nc1C
CC(C)OC(=O)c1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)nc1
COCCN1Cc2nc(N3CCC4(CC3)O[C@@H]3CC[C@@H](c5ccccc5)N3C4=O)ccc2C1=O
COC(=O)c1c(C)cc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)nc1C#N
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ccc(-c3cc(O)no3)cn1)CC2
COC(=O)c1cnc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)nc1
CC(C)N1Cc2nc(N3CCC4(CC3)O[C@@H]3CC[C@@H](c5ccccc5)N3C4=O)ccc2C1=O
O=C1CCc2nc(N3CCC4(CC3)O[C@@H]3CC[C@@H](c5ccccc5)N3C4=O)ccc21
COC(=O)c1cnc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)c(OC)c1
CC(C)(C)OC(=O)c1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)nc1
NC(=O)c1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)nc1
CCOC(=O)c1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)nc1
NC(=O)c1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)nc1Cl
COC(=O)c1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)nc1
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1cc(CF)ncn1)CC2
O=C1N2[C@@H](CC[C@H]2c2cccc(F)c2)OC12CCN(c1ncnc3ccnn13)CC2
CCOC(=O)c1nc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)ncc1F
N#Cc1cnc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)cc1OC(F)F
Cc1cc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)ncc1[N+](=O)[O-]
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1cc(-c3ccc(F)cc3)c([N+](=O)[O-])cn1)CC2
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1cc(F)c(O)cn1)CC2
COC(=O)c1cnc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)cc1OC
COC(=O)c1cnc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)cc1Cl
NC(=O)c1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)n2ncnc12
CC1CC2(CCN1c1ncnc3ccnn13)O[C@@H]1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
CC(F)c1cc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)ncn1
CC(F)c1cc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)ncn1
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ccc(Br)n3ncnc13)CC2
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ncnc3c1CCO3)CC2
N#Cc1cnn2c(N3CCC4(CC3)O[C@@H]3CC[C@@H](c5ccccc5)N3C4=O)ncnc12
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ncnc3c(I)cnn13)CC2
COc1cc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)ncc1C#N
CCc1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)n2ncnc12
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ncnc3c1COC3)CC2
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ccc(F)c3ncnn13)CC2
CC1CC2(CCN1c1ccnc3c(F)cnn13)O[C@@H]1CC[C@@H](c3ccccc3)N1C2=O
CC1CC2(CCN1c1ccnc3c(F)cnn13)O[C@@H]1CC[C@@H](c3ccccc3)N1C2=O
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ncnn3c(F)cnc13)CC2
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ncnn3ccnc13)CC2
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1ncnn3ccnc13)CC2
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ncnc3ccnn13)CC2
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1ncnc3ccnn13)CC2
CC1CC2(CCN1c1ccnc3ccnn13)O[C@@H]1CC[C@@H](c3ccccc3)N1C2=O
CC1CC2(CCN1c1ccnc3ccnn13)O[C@@H]1CC[C@@H](c3ccccc3)N1C2=O
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ncnc3c(F)cnn13)CC2
CC1CN(c2cc(C#N)ncn2)CCC12O[C@@H]1CC[C@@H](c3ccccc3)N1C2=O
CC1CN(c2ccnc3ccnn23)CCC12O[C@@H]1CC[C@@H](c3ccccc3)N1C2=O
CC1CN(c2cc(C#N)ncn2)CCC12O[C@@H]1CC[C@@H](c3ccccc3)N1C2=O
CC1CN(c2cc(C#N)ncn2)CCC12O[C@@H]1CC[C@@H](c3ccccc3)N1C2=O
CC1CN(c2ccnc3ccnn23)CCC12O[C@@H]1CC[C@@H](c3ccccc3)N1C2=O
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ncc(Br)c3ncnn13)CC2
O=C1N2[C@@H](CC[C@H]2c2ccccc2F)OC12CCN(c1ncc(Br)c3ncnn13)CC2
N#Cc1cnc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)n2ncnc12
N#Cc1cnc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4F)N2C3=O)n2ncnc12
CC1CN(c2cccc3ncnn23)CCC12O[C@@H]1CC[C@@H](c3ccccc3)N1C2=O
CC1CN(c2cccc3ncnn23)CCC12O[C@@H]1CC[C@@H](c3ccccc3)N1C2=O
CC1CN(c2cccc3ncnn23)CCC12O[C@@H]1CC[C@@H](c3ccccc3)N1C2=O
CC1CN(c2ccnc3ccnn23)CCC12O[C@@H]1CC[C@@H](c3ccccc3)N1C2=O
CC1CC2(CCN1c1ccnc3ccnn13)O[C@@H]1CC[C@@H](c3ccccc3)N1C2=O
O=C1N2[C@H](OC13CCN(c1ccnc4ccnn14)CC3)[C@H](O)C[C@H]2c1ccccc1
N#Cc1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4F)N2C3=O)n2ncnc12
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1ncnc3c(F)cnn13)CC2
O=C1N2[C@H](OC13CCN(c1ccnc4ccnn14)CC3)[C@@H](O)C[C@H]2c1ccccc1
O=C1N2[C@@H](CC[C@H]2c2ccccc2F)OC12CCN(c1ncnc3ccnn13)CC2
O=C1N2[C@@H](CC[C@H]2c2ccccc2F)OC12CCN(c1cccc3ncnn13)CC2
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CC1CCC(C2)N1c1ccnc2c(F)cnn12
Cc1ccccc1[C@@H]1CC[C@H]2OC3(CCN(c4ccnc5c(F)cnn45)CC3)C(=O)N21
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ncccc1Cl)CC2
N#Cc1ccc(N2CCC3(O[C@@H]4CC[C@@H](c5ccccc5)N4C3=O)C(F)C2)n2ncnc12
N#Cc1ccc(N2CCC3(O[C@@H]4CC[C@@H](c5ccccc5)N4C3=O)C(F)C2)n2ncnc12
N#Cc1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cccc(F)c4)N2C3=O)n2ncnc12
O=C1N2[C@@H](CC[C@H]2c2ccccc2F)OC12CCN(c1ccnc3ccnn13)CC2
N#Cc1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)n2ncnc12
CC(F)(F)c1ccnc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)c1
Cc1ccn(-c2cccc(N3CCC4(CC3)O[C@@H]3CC[C@@H](c5ccccc5)N3C4=O)n2)n1
CC1CN(c2ncnc3ccnn23)CCC12O[C@@H]1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
CC1CN(c2cccc3ncnn23)CCC12O[C@@H]1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
CC1CN(c2cccc3ncnn23)CCC12O[C@@H]1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
CC1CN(c2ncnc3ccnn23)CCC12O[C@@H]1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
O=C1N2[C@@H](CC[C@H]2c2ccccc2F)OC12CCN(c1ccnc(Cl)c1)CC2
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ccc(C(F)F)c3ncnn13)CC2
CC(=O)c1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)n2ncnc12
O=C1N2[C@H](OC13CCN(c1ccnc4c(F)cnn14)CC3)[C@@H](O)C[C@H]2c1ccccc1
O=C1N2[C@@H](CC[C@H]2c2ccccc2F)OC12CN(c1ncco1)C2
Cc1nnc(N2CC3(C2)O[C@@H]2CC[C@@H](c4ccccc4F)N2C3=O)o1
O=C(c1cc(F)ccc1F)N1CCC2(CC1)O[C@@H]1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
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CC1CN(C(=O)c2ccccc2)CCC12O[C@@H]1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
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Cc1ocnc1C(=O)N1CCC2(CC1)O[C@@H]1CC[C@@H](c3ccccc3)N1C2=O
N#Cc1ccccc1C(=O)N1CCC2(CC1)O[C@@H]1CC[C@@H](c3ccccc3)N1C2=O
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N#Cc1ccc(C(=O)N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)cc1
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COc1ncnc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)c1F
COc1nc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)ncc1F
COc1ccnc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)c1
COc1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)nc1OC
Cc1nc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)sc1C
Cc1nc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)ccc1F
Cc1ncc(C)c(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)n1
O=C1N2[C@@H](CC[C@H]2c2ccccc2F)OC12CN(c1cc(-c3ccccc3)no1)C2
O=C(Nc1ccccc1)N1CCC2(CC1)O[C@@H]1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1cccc3ncnn13)CC2
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1cccc3ncnn13)CC2
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1ccnn3ccnc13)CC2
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1cncc3ncnn13)CC2
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1cccc3nccn13)CC2
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1ccc(Br)c3ccnn13)CC2
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1ccc(Br)c3ncnn13)CC2
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1cncc3nccn13)CC2
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1nnc3cccnn13)CC2
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1nccn3cccc13)CC2
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1ncnn3cccc13)CC2
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1nccn3nccc13)CC2
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1ncc(F)c3nncn13)CC2
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1nccn3cncc13)CC2
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1nccn3ccnc13)CC2
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1ccc(Cl)c3nccn13)CC2
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1cccc3ncnn13)CC2F
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1cccc3ncnn13)CC2F
N#Cc1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)c2ccnn12
O=C1N2[C@@H](CC[C@H]2c2ccccc2F)OC12CN(c1cccc3ncnn13)C2
N#Cc1ccc(N2CC3(C2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)c2ccnn12
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CN(c1cccc3ncnn13)C2
N#Cc1ccc(N2CC3(C2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)n2ncnc12
N#Cc1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)n2ncnc12
N#Cc1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)n2nccc12
N#Cc1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)n2ncnc12
N#Cc1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cncc(F)c4)N2C3=O)n2nccc12
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1ccc(Cl)c3ccnn13)CC2
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1cccc3ccnn13)CC2
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ccc(Cl)c3ncnn13)CC2
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1ccc(Cl)c3ncnn13)CC2
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1ccc(Br)c3ccnn13)CC2
O=C(c1ccccc1)N1CCC2(CC1)O[C@@H]1CC[C@@H](c3cnccn3)N1C2=O
O=C(c1ccccc1)N1CCC2(CC1)O[C@@H]1CC[C@@H](c3ccc4sccc4c3)N1C2=O
Cc1ccc([C@@H]2CC[C@H]3OC4(CCN(C(=O)c5ccccc5)CC4)C(=O)N32)cc1
N#Cc1cc([C@@H]2CC[C@H]3OC4(CCN(C(=O)c5ccccc5)CC4)C(=O)N32)ccc1F
COc5cccc([C@@H]4CC[C@H]3OC2(CCN(C(=O)c1ccccc1)CC2)C(=O)N34)n5
O=C(c1ccccc1)N1CCC2(CC1)O[C@@H]1CC[C@@H](c3ccc(F)cn3)N1C2=O
O=C(c1ccccc1)N1CCC2(CC1)O[C@@H]1CC[C@@H](c3cnsc3)N1C2=O
COc5ccc([C@@H]4CC[C@H]3OC2(CCN(C(=O)c1ccccc1)CC2)C(=O)N34)cc5
COc5cc(F)cc([C@@H]4CC[C@H]3OC2(CCN(C(=O)c1ccccc1)CC2)C(=O)N34)c5
O=C(c1ccccc1)N1CCC2(CC1)O[C@@H]1CC[C@@H](c3cccc(F)c3F)N1C2=O
Cc1ccc([C@@H]2CC[C@H]3OC4(CCN(C(=O)c5ccccc5)CC4)C(=O)N32)c(F)c1
O=C(c1ccccc1)N1CCC2(CC1)O[C@@H]1CC[C@@H](c3cnc4c(c3)CCC4)N1C2=O
N#Cc1cscc1[C@@H]1CC[C@H]2OC3(CCN(C(=O)c4ccccc4)CC3)C(=O)N21
O=C(c1ccccc1)N1CCC2(CC1)O[C@@H]1CC[C@@H](c3ccc(F)cc3F)N1C2=O
Cc1ccc([C@@H]2CC[C@H]3OC4(CCN(C(=O)c5ccccc5)CC4)C(=O)N32)cc1F
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1ccc(C3CCC3)c3ccnn13)CC2
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ccc(C3COC3)c3ccnn13)CC2
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CN(c1ccc(C3CCC3)c3ccnn13)C2
COc1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)n2nccc12
CCOc1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)n2nccc12
COc1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)n2ncnc12
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1ccc(OCC(F)F)c3ccnn13)CC2
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1ccc(OCC3CCO3)c3ccnn13)CC2
COc1cnc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)n2ncnc12
CCOc1cnc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)n2ncnc12
COc1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)n2ncnc12
Cn1cc([C@@H]2CC[C@H]3OC4(CCN(c5ccc(C#N)c6ncnn56)CC4)C(=O)N32)cn1
COc1cccc([C@@H]2CC[C@H]3OC4(CCN(c5ccc(C#N)c6ncnn56)CC4)C(=O)N32)c1
COc1cccc([C@@H]2CC[C@H]3OC4(CCN(c5cc(C#N)ncn5)CC4)C(=O)N32)c1
N#Cc1ccc(F)c([C@@H]2CC[C@H]3OC4(CCN(c5ccnc6c(F)cnn56)CC4)C(=O)N32)c1
N#Cc1cccc([C@@H]2CC[C@H]3OC4(CCN(c5ccnc6c(F)cnn56)CC4)C(=O)N32)c1F
N#Cc1cc([C@@H]2CC[C@H]3OC4(CCN(c5ccnc6c(F)cnn56)CC4)C(=O)N32)ccc1F
O=C1N2C(CCC2c2cccc(F)c2F)OC12CCN(c1ccnc3ccnn13)CC2
O=C1N2C(CCC2c2c(F)cccc2F)OC12CCN(c1ccnc3ccnn13)CC2
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(c1ccc(-c3ncco3)c3ncnn13)CC2
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ncc(-c3ncco3)c(C(F)(F)F)n1)CC2
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ncc(-c3ncco3)c(C(F)F)n1)CC2
Cc1nc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)ncc1-c1ncn(C)n1
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ncc(-c3cnco3)cc1F)CC2
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ncc(-c3cocn3)cc1F)CC2
Cc1nc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)ncc1-c1ncnn1C
Cc1nc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)ncc1-c1ccnn1C
Cc1nc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)ncc1-c1cnoc1
COc1nc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)ncc1-c1ncco1
Cc1nc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)ncc1-c1ncco1
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ncc(-c3nccs3)cn1)CC2
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ncc(-c3cscn3)cn1)CC2
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1cnc(-c3ncco3)cn1)CC2
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ncc(-c3ncco3)cn1)CC2
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ccc(-c3ncco3)cn1)CC2
Cc1cnc(-c2ccc(N3CCC4(CC3)O[C@@H]3CC[C@@H](c5ccccc5)N3C4=O)n3nccc23)o1
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ccc(-c3cc4n(n3)CCC4)c3ncnn13)CC2
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ccc(-c3cscn3)c3ncnn13)CC2
Cn1nc(C(F)(F)F)cc1-c1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)n2ncnc12
Cn1cnc(-c2ccc(N3CCC4(CC3)O[C@@H]3CC[C@@H](c5ccccc5)N3C4=O)n3ncnc23)c1
O=C1N2[C@@H](CC[C@H]2c2ccccc2)OC12CCN(c1ccc(-c3ncco3)c3ccnn13)CC2
C#Cc1cnc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)n2ncnc12
C#Cc1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)n2ncnc12
O=C1N2[C@@H](CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(C(c1ccccc1)C(F)F)CC2
O=C1N2C(CC[C@H]2c2cc(F)cc(F)c2)OC12CCN(C(c1ccccc1)C(F)F)CC2
N#Cc1ccccc1CN1CCC(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)CC1
Cc1cccc(CN2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)c1
Cc1ccccc1CN1CCC2(CC1)O[C@@H]1CC[C@@H](c3cc(F)cc(F)c3)N1C2=O
N#Cc1cccc(CN2CCC3(CC2)O[C@@H]2CC[C@@H](c4cc(F)cc(F)c4)N2C3=O)c1
O=C1N2[C@@H](CC[C@H]2c2ccccc2F)OC12CN(Cc1ccccc1)C2
O=C1N2[C@@H](CC[C@H]2c2ccccc2F)OC12CN(CCc1ccccc1)C2
NC(=O)c1ccc(N2CCC3(CC2)O[C@@H]2CC[C@@H](c4ccccc4)N2C3=O)n2ncnc12
CCS(=O)(=O)Nc1ccc(-c2nn(C)c3c(-c4cccnc4)cnc(N)c23)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2nn(C)c3c(NC(C)=O)cnc(N)c23)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2coc3c(-c4cnn(C5CCOCC5)c4)cnc(N)c23)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2coc3c(-c4cnn(CCO)c4)cnc(N)c23)cc1OCc1ccc(F)cc1
Nc1ncc(-c2cnn(C3CCOCC3)c2)c2occ(-c3ccc(NS(=O)(=O)C(F)F)c(OCc4ccc(F)cc4)c3)c12
Nc1ncc(-c2cnn(CCO)c2)c2occ(-c3ccc(NS(=O)(=O)C(F)F)c(OCc4ccc(F)cc4)c3)c12
C[C@H](Oc1cc(-c2coc3c(-c4cnn(C5CCOCC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2coc3c(-c4cnn(C)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2coc3c(-c4cnn(CCO)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3ccnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
Nc1ncc(-c2cnn(C3CCOCC3)c2)c2occ(-c3ccc(NS(=O)(=O)CC(F)(F)F)c(OCc4ccc(F)cc4)c3)c12
Cn1nc(-c2ccc(NS(=O)(=O)C(F)F)c(OCc3ccc(F)cc3)c2)c2c(N)ncc(-c3cnn(CCO)c3)c21
Cn1nc(-c2ccc(NS(=O)(=O)C(F)F)c(OCc3ccc(F)cc3)c2)c2c(N)ncc(-c3cnn(C4CCOCC4)c3)c21
Cn1nc(-c2ccc(NS(=O)(=O)C(F)F)c(OCc3ccc(F)cc3)c2)c2c(N)ncc(-c3ccncc3)c21
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(CCO)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
Cn1cc(-c2cnc(N)c3c(-c4ccc(NS(=O)(=O)C(F)F)c(OCc5ccc(F)cc5)c4)nn(C)c23)cn1
C[C@H](Oc3cc(c1nn(C)c2ccnc(N)c12)ccc3NS(=O)(=O)C(F)F)c4ccc(F)cc4
C[C@H](Oc1cc(-c2nn(C)c3c(-c4ccncc4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCOCC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(C4=CCN(C)CC4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc3cc(C1C=NN2C=CN=C(N)C12)ccc3NS(=O)(=O)C(F)F)c4ccc(F)cc4
C[C@H](Oc1cc(-c2nn(C)c3c(-c4ccnc(C(F)(F)F)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
Cc1cc(-c2cnc(N)c3c(-c4ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c5ccc(F)cc5)c4)nn(C)c23)ccn1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cccnc4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
Cc1ccc(-c2cnc(N)c3c(-c4ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c5ccc(F)cc5)c4)nn(C)c23)cn1
COc1cc(-c2cnc(N)c3c(-c4ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c5ccc(F)cc5)c4)nn(C)c23)ccn1
COc1ccc(-c2cnc(N)c3c(-c4ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c5ccc(F)cc5)c4)nn(C)c23)cn1
COCCn1cc(-c2cnc(N)c3c(-c4ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c5ccc(F)cc5)c4)nn(C)c23)cn1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCCC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CC(C)n1cc(-c2cnc(N)c3c(-c4ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c5ccc(F)cc5)c4)nn(C)c23)cn1
Cc1cnccc1-c1cnc(N)c2c(-c3ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c4ccc(F)cc4)c3)nn(C)c12
Cc1noc(C)c1-c1cnc(N)c2c(-c3ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c4ccc(F)cc4)c3)nn(C)c12
C[C@H](Oc1cc(-c2nn(C)c3c(Cc4ccccc4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2cnn3c(-c4cnn(C)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2cnn3c(-c4cnn(C5CCOCC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2cnn3c(-c4cnn(CCO)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5COC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2cnn3c(-c4ccncc4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc4cc(c2nn(C)c3c(c1ccncn1)cnc(N)c23)ccc4NS(=O)(=O)C(F)F)c5ccc(F)cc5
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCOC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc4cc(c2nn(C)c3c(C1CCN(C)CC1)cnc(N)c23)ccc4NS(=O)(=O)C(F)F)c5ccc(F)cc5
C[C@H](Oc1cc(-c2nn(C)c3c(C4=CCOCC4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc5cc(c3nn(C)c4c(c2cnn(C1CCOCC1)c2)cnc(N)c34)ccc5NS(=O)(=O)CC(F)(F)F)c6ccc(F)cc6
CCS(=O)(=O)Nc1ccc(-c2nn(C)c3c(-c4cnn(C5CCOCC5)c4)cnc(N)c23)cc1O[C@@H](C)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCN(C)CC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
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C[C@H](Oc1cc(-c2nn(C)c3c(-c4ccnc(C(C)(C)C)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4ccnc(N(C)C)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
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CC(C)n1nc(-c2ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c3ccc(F)cc3)c2)c2c(N)ncc(-c3cnn(C4CCOCC4)c3)c21
CC(C)n1nc(-c2ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c3ccc(F)cc3)c2)c2c(N)ncc(-c3cnn(C)c3)c21
CC(C)n4nc(c2ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c1ccc(F)cc1)c2)c3c(N)nccc34
C[C@H](Oc4cc(c2nn(C)c3c(C1CCCNC1)cnc(N)c23)ccc4NS(=O)(=O)C(F)F)c5ccc(F)cc5
C[C@H](Oc4cc(c2nn(C)c3c(C1CCCN(C)C1)cnc(N)c23)ccc4NS(=O)(=O)C(F)F)c5ccc(F)cc5
CC#Cc1cnc(N)c2c(-c3ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c4ccc(F)cc4)c3)nn(C)c12
C[C@H](Oc1cc(-c2nn(C)c3c(-c4ccnc(C(F)F)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(C#CC4CCOCC4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCNCC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(CCN5CCN(C)CC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCN(CC(F)(F)F)CC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CCS(=O)(=O)Nc3ccc(c1cccc2[nH]nc(N)c12)cc3OCc4ccc(F)cc4
CCS(=O)(=O)Nc3ccc(c1ncn2ccnc(N)c12)cc3OCc4ccc(F)cc4
CCS(=O)(=O)Nc3ccc(c1cnn2ccnc(N)c12)cc3OCc4ccc(F)cc4
Nc3n[nH]c4ccnc(c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc1ccc(F)cc1)c2)c34
Nc3n[nH]c4nccc(c2ccc(NS(=O)(=O)C(F)F)c(OCc1ccc(F)cc1)c2)c34
Nc3n[nH]c4nccc(c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc1ccc(F)cc1)c2)c34
Nc3n[nH]c4ccnc(c2ccc(NS(=O)(=O)C(F)F)c(OCc1ccc(F)cc1)c2)c34
Nc3n[nH]c4ncnc(c2ccc(NS(=O)(=O)C(F)F)c(OCc1ccc(F)cc1)c2)c34
Cc4cc(c2ccc(NS(=O)(=O)C(F)F)c(OCc1ccc(F)cc1)c2)c3c(N)n[nH]c3n4
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C[C@H](Oc3cc(c1ccnc2[nH]nc(N)c12)ccc3NS(=O)(=O)C(F)F)c4ccc(F)cc4
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CC6CCC(C5)N6C)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CNc1c(-c2cnn(C3CCCNCC3)c2)cnc(N)c1C(=N)c1ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c2ccc(F)cc2)c1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(CCN5CC(C)(C)C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CC(C)N1CC(n2cc(-c3cnc(N)c4c(-c5ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c6ccc(F)cc6)c5)nn(C)c34)cn2)C1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CN(CC(F)(F)F)C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CC6(CNC6)C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc4cc(c2nn(C)c3c(C#CC1CCNCC1)cnc(N)c23)ccc4NS(=O)(=O)C(F)F)c5ccc(F)cc5
C[C@H](Oc4cc(c2nn(C)c3c(C#CC1CCN(C)CC1)cnc(N)c23)ccc4NS(=O)(=O)C(F)F)c5ccc(F)cc5
CC(C)N(C)C(=O)C(C)n1cc(-c2cnc(N)c3c(-c4ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c5ccc(F)cc5)c4)nn(C)c23)cn1
CNCCn1cc(-c2cnc(N)c3c(-c4ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c5ccc(F)cc5)c4)nn(C)c23)cn1
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C[C@H](Oc1cc(-c2nn(C)c3c(-c4cccc(Cl)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4ccccc4Cl)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4ccccc4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4ccc(Cl)cc4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CNc1c(-c2cnn(CC3CCCN3)c2)cnc(N)c1C(=N)c1ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c2ccc(F)cc2)c1
C[C@H](Oc5cc(c3nn(C)c4c(c2cnn(C1(CN)CC1)c2)cnc(N)c34)ccc5NS(=O)(=O)C(F)F)c6ccc(F)cc6
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn5c4CNCC5)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc5cc(c3nn(C)c4c(c1cnn2CCN(C)Cc12)cnc(N)c34)ccc5NS(=O)(=O)C(F)F)c6ccc(F)cc6
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CN(C)C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCN(C)C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CNC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CC1CNCC(n2cc(-c3cnc(N)c4c(-c5ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c6ccc(F)cc6)c5)nn(C)c34)cn2)C1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5(C#N)CC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C(C)(C)CO)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc5cc(c3nn(C)c4c(c2cnn(C1(CC#N)COC1)c2)cnc(N)c34)ccc5NS(=O)(=O)C(F)F)c6ccc(F)cc6
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C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(CCN(C)C)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CC(C)N(C)CC(C)n1cc(-c2cnc(N)c3c(-c4ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c5ccc(F)cc5)c4)nn(C)c23)cn1
COCC(Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCOCC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
[2H]C([2H])([2H])N6CCC(n5cc(c3cnc(N)c4c(c2ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c1ccc(F)cc1)c2)nn(C)c34)cn5)CC6
C[C@H](Oc5cc(c3nn(C)c4c(c2cnn(C1CCC(C)(C)N(C)C1)c2)cnc(N)c34)ccc5NS(=O)(=O)C(F)F)c6ccc(F)cc6
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnc(N5CCN(C)CC5)nc4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
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C[C@@H](Oc1cc(-c2nn(C)c3c(-c4ccc(N5CCN(C)CC5)nc4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4ccc(N5CCN(C)CC5)nc4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CC(=O)N6CCC(n5cc(c3cnc(N)c4c(c2ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c1ccc(F)cc1)c2)nn(C)c34)cn5)CC6
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnc(N5CCOCC5)nc4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
COC[C@H](Oc5cc(c3nn(C)c4c(c2cnn(C1CCOCC1)c2)cnc(N)c34)ccc5NS(=O)(=O)C(F)F)c6ccc(F)cc6
COC[C@@H](Oc5cc(c3nn(C)c4c(c2cnn(C1CCOCC1)c2)cnc(N)c34)ccc5NS(=O)(=O)C(F)F)c6ccc(F)cc6
C[C@H](Oc5cc(c3nn(C)c4c(c2cnn(C1CCN(C)C(C)(C)C1)c2)cnc(N)c34)ccc5NS(=O)(=O)C(F)F)c6ccc(F)cc6
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnc(N5CCCC5)nc4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4ccc(N5CCOCC5)nc4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(CC(F)(F)F)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
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C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCOCC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccccc1F
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCOCC5)c4)cnc(N)c23)ccc1NS(C)(=O)=O)c1ccc(F)cc1
C[C@H](Oc5cc(c3nn(C)c4c(c2cnn(C1CCC(F)(F)C1)c2)cnc(N)c34)ccc5NS(=O)(=O)C(F)F)c6ccc(F)cc6
C[C@@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCOCC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCOCC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1cccc(Cl)c1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C(F)F)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCOCC5)c4)cnc(N)c23)ccc1NS(=O)(=O)N(C)C)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCOCC5)c4)cnc(N)c23)ccc1NS(=O)(=O)Cc1ccccc1)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4ccn(C)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCOCC5)c4)cnc(N)c23)ccc1NS(=O)(=O)Cc1ccccc1)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(C#CC4CCN(CC(F)(F)F)CC4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
COc1ccc([C@H](C)Oc2cc(-c3nn(C)c4c(-c5cnn(C6CCOCC6)c5)cnc(N)c34)ccc2NS(=O)(=O)C(F)F)cc1
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C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(CCC(F)(F)F)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
Cn1nc(-c2ccc(NS(=O)(=O)C(F)F)c(OCc3ccc(Cl)c(F)c3)c2)c2c(N)ncc(-c3cnn(C4CCOCC4)c3)c21
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C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C(F)(F)F)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
Cn1nc(-c2ccc(NS(=O)(=O)C(F)F)cc2OCc2cccc(F)c2)c2c(N)ncc(-c3cnn(C4CCOCC4)c3)c21
CNc1ncc(-c2cnc(N)c3c(-c4ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c5ccc(F)cc5)c4)nn(C)c23)cn1
COCC(Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCN(C)CC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
Cn1nc(-c2ccc(NS(=O)(=O)C(F)F)c(OC3(c4ccc(F)cc4)CC3)c2)c2c(N)ncc(-c3cnn(C4CCOCC4)c3)c21
C[C@H](Oc4cc(c2nn(C)c3c(N1CCOCC1)cnc(N)c23)ccc4NS(=O)(=O)C(F)F)c5ccc(F)cc5
CC(n1cc(-c2cnc(N)c3c(-c4ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c5ccc(F)cc5)c4)nn(C)c23)cn1)C(F)(F)F
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C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCN(C)C6(CC6)C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCC(F)(F)CC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
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C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CC6CCC(C5)N6CC(F)(F)F)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCN(C)C(C)(C)C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
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C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCN(C)C(C)(C)C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(Cl)cc1
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C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5C[C@H]6CNC[C@H]6C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5C[C@@H]6CN(C)C[C@@H]6C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4ccc5c(c4)CC(=O)N5C)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4ccc5c(cnn5C)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCN(CC(F)(F)F)C(C)(C)C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCC(N(C)C)C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCN(C)C6(CC6)C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCN(C)C6(CC6)C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CC1CN(C)CC(C)C1n1cc(-c2cnc(N)c3c(-c4ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c5ccc(F)cc5)c4)nn(C)c23)cn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1ccc(F)c(F)c1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1ccccc1F
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)cc1OCc1cccc(Cl)c1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)cc1OCc1ccc(Cl)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc3ccc(F)cc3)c2)n[nH]c1Nc1cccc(C(F)(F)F)n1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccnc3)c2C(N)=O)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCC1CCN(C(C)=O)CC1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)cc1OCc1ccc(F)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)Cc3cccc(Cl)c3)cc2)n[nH]c1Nc1cccc(C(F)(F)F)n1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)cc1OCC1CCCC1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(OC)n3)c2C(N)=O)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)cc1OCC(C)C
CCS(=O)(=O)Cc1ccc(-c2nn(C(C)(C)C)c(Cc3ccccn3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnc(OC)cn3)c2C(N)=O)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cncc(OC)n3)c2C(N)=O)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)cc1OCc1ccncc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cncc(C(F)(F)F)n3)c2C(N)=O)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccnc(OC)c3)c2C(N)=O)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Cc1ccc(-c2nn(COCC[Si](C)(C)C)c(Nc3cnccn3)c2C(N)=O)cc1Oc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccccn3)c2C(N)=O)cc1OCc1ccccc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)c(OCc2ccc(F)cc2)c1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Cc3cnc(C)cn3)c2C(N)=O)cc1OCc1ccc(F)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CCC(F)F)cc2)n[nH]c1Nc1cnccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1ccccc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1cccc(F)c1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccccn3)c2C(N)=O)cc1OCc1ccncc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1ccncc1
N#CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccccn3)c2C(N)=O)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccccn3)c2C(N)=O)cc1OCc1cccnc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1cccnc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)cc1OCc1cccnc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnc(C(C)C)cn3)c2C(N)=O)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccccn3)c2C(N)=O)cc1OCC1CCCCC1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccccn3)c2C(N)=O)cc1OCC1CCCC1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccccn3)c2C(N)=O)cc1OCC(C)C
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccccn3)c2C(N)=O)cc1OCc1cccc(Cl)c1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccccn3)c2C(N)=O)cc1OCc1ccc(Cl)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCC1CCCC1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1cccc(Cl)c1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1ccc(Cl)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)cc2)n[nH]c1Nc1cccc(C(F)(F)F)n1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cncc(C(F)(F)F)n3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCC(C)C
CCS(=O)(=O)Nc1ccc(-c2nn(C(C)(C)C)c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)cc1OCc1ccccc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCC1CCCCC1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)F)cc2)n[nH]c1Nc1ccccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)F)cc2)n[nH]c1Nc1cccc(C(F)(F)F)n1
COCCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)cc1
CN(C)CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C3CC3)cc2)n[nH]c1Nc1cccc(C(F)(F)F)n1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)F)cc2)n[nH]c1Nc1cccc(C(F)(F)F)n1
CC(C)S(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)Cc3ccc(F)cc3)cc2)n[nH]c1Nc1cccc(C(F)(F)F)n1
NC(=O)c1c(-c2ccc(NS(=O)(=O)Cc3ccc(Cl)c(Cl)c3)cc2)n[nH]c1Nc1cccc(C(F)(F)F)n1
Cc1ccc(CS(=O)(=O)Nc2ccc(-c3n[nH]c(Nc4cccc(C(F)(F)F)n4)c3C(N)=O)cc2)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)Cc3ccccc3Cl)cc2)n[nH]c1Nc1cccc(C(F)(F)F)n1
Cc1cccc(CS(=O)(=O)Nc2ccc(-c3n[nH]c(Nc4cccc(C(F)(F)F)n4)c3C(N)=O)cc2)c1Cl
NC(=O)c1c(-c2ccc(NS(=O)(=O)Cc3ccc(Cl)cc3)cc2)n[nH]c1Nc1cccc(C(F)(F)F)n1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OC
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1ccc(F)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)F)cc2)n[nH]c1Nc1cnccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccnn3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnc4cc(Cl)ccc4n3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnc(C(C)C)cn3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnc4ccccc4n3)c2C(N)=O)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C3CC3)cc2)n[nH]c1Nc1cnccn1
CC(C)(C)S(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)Cc3ccc(Cl)cc3)cc2)n[nH]c1Nc1cnccn1
CC(C)S(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1
CCCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1
Cc1cccc(S(=O)(=O)Nc2ccc(-c3n[nH]c(Nc4cnccn4)c3C(N)=O)cc2)c1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C3CCCCC3)cc2)n[nH]c1Nc1cnccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnc(C(F)(F)F)cn3)c2C(N)=O)cc1
Cc1ccc(CS(=O)(=O)Nc2ccc(-c3n[nH]c(Nc4cnccn4)c3C(N)=O)cc2)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)Cc3ccccc3)cc2)n[nH]c1Nc1cnccn1
Cc1ccc(S(=O)(=O)Nc2ccc(-c3n[nH]c(Nc4cnccn4)c3C(N)=O)cc2)cc1
Cc1ccc(S(=O)(=O)Nc2ccc(-c3n[nH]c(Nc4cnccn4)c3C(N)=O)cc2)cc1
Cc1ccc(CS(=O)(=O)Nc2ccc(-c3n[nH]c(Nc4cnccn4)c3C(N)=O)cc2)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC3CCC3)cc2)n[nH]c1Nc1cnccn1
COc1ccc(S(=O)(=O)Nc2ccc(-c3n[nH]c(Nc4cnccn4)c3C(N)=O)cc2)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)Cc3cccc(C(F)(F)F)c3)cc2)n[nH]c1Nc1cnccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cncc(C)n3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cc(C(F)(F)F)ccn3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccc4ccccc4c3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cc4ccccc4cn3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccc(OC)cn3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccc4ccccc4n3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnc(OC)cn3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccn(C)n3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)F)n3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccc(C(F)(F)F)cn3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C)n3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cc(C)ccn3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccccn3)c2C(N)=O)cc1
CCCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1
CCOc1nccc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)CC)cc3)c2C(N)=O)n1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cncc(OC)n3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnn(C)c3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnc(C)cn3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccc(C#N)cc3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccnc(C(F)(F)F)c3)c2C(N)=O)cc1
CCOc1cc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)CC)cc3)c2C(N)=O)ccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccnc(OCC(F)F)c3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(OC)n3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1
C#CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccnc(OCCOC)c3)c2C(N)=O)cc1
N#CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccnc(OCCOC)c3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cc(C)ncc3F)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cc(C)nc(C)c3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccnc(C)c3)c2C(N)=O)cc1
COCCOc1cc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)C(F)(F)F)cc3)c2C(N)=O)ccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccc(OC)nc3)c2C#N)cc1
COCCOc1cc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)CCN(C)C)cc3)c2C(N)=O)ccn1
CCS(=O)(=O)N(C)c1ccc(-c2n[nH]c(Nc3ccnc(OCCOC)c3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2nn(C(C)(C)C)c(Nc3cc(OC)ncc3C)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(NC)c2C(N)=O)cc1
COCCOc1cc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)COC)cc3)c2C(N)=O)ccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccnc(OC)c3)c2C(N)=O)cc1
COCCOc1cc(Nc2[nH]nc(-c3ccc(NS(C)(=O)=O)cc3)c2C(N)=O)ccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccnc(OC)n3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccccc3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccnc(C)n3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(C2=NN=C(Nc3ccnc(OCCOC)c3)C2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(OCCOC)n3)c2C(N)=O)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)Cc3cccc(Cl)c3)cc2)n[nH]c1Nc1ccccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CCc3ccccc3)cc2)n[nH]c1Nc1ccccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccccn3)c2C(N)=O)cc1
Cc1ccc(CS(=O)(=O)Nc2ccc(-c3n[nH]c(Nc4ccccn4)c3C(N)=O)cc2)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)c3ccccc3)cc2)n[nH]c1Nc1ccccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC3CCC3)cc2)n[nH]c1Nc1ccccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)cc2)n[nH]c1Nc1cnccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccc4ccc(Cl)cc4n3)c2C(N)=O)cc1OCc1ccc(F)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)cc2OCc2ccc(F)cc2)n[nH]c1Nc1cnccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)cc2OCc2ccc(F)cc2)n[nH]c1Nc1cccc(C(F)(F)F)n1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)c(OCc2ccc(F)cc2)c1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1c(C)cc(F)cc1C
COc1cnc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)CC(F)(F)F)c(OCc4ccc(F)cc4)c3)c2C(N)=O)cn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OC3(c4ccc(F)cc4)CC3)c2)n[nH]c1Nc1cnccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)F)cc2)n[nH]c1Nc1ccc(C(F)(F)F)cn1
Cc1cnc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)CC(F)(F)F)c(OCc4ccc(Cl)c(F)c4)c3)c2C(N)=O)cn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)F)c(Oc3ccc(F)cc3)c2)n[nH]c1Nc1cccc(C(F)(F)F)n1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(Oc3ccc(F)cc3)c2)n[nH]c1Nc1cccc(C(F)(F)F)n1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)cc1Oc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnc(C)cn3)c2C(N)=O)cc1OCc1ccc(F)c(Cl)c1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)F)c(OCc3ccc(F)c(F)c3)c2)n[nH]c1Nc1cccc(C(F)(F)F)n1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OC1(c2ccccc2)CC1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)cc2)n[nH]c1Nc1ccc(C(F)(F)F)cn1
C[C@H](Oc1cc(-c2n[nH]c(Nc3ccccn3)c2C(N)=O)ccc1NS(=O)(=O)CC(F)(F)F)c1ccc(F)cc1
Cc1cnc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)CC(F)(F)F)c(OCc4ccc(F)c(Cl)c4)c3)c2C(N)=O)cn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1ccc(F)cn1
COc1cnc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)CC(F)(F)F)c(OCc4ccc(Cl)cc4)c3)c2C(N)=O)cn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnc(C4CC4)cn3)c2C(N)=O)cc1
COc1ccc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)CC(F)(F)F)c(OCc4ccc(F)cc4)c3)c2C(N)=O)cn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc3ccc(F)c(F)c3)c2)n[nH]c1Nc1ccccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OC3(c4ccccc4)CC3)c2)n[nH]c1Nc1cnccn1
Cc1cnc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)CC(F)(F)F)c(OCc4ccc(Cl)cc4)c3)c2C(N)=O)cn1
Cc1cnc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)CC(F)(F)F)c(OCc4ccc(F)cc4)c3)c2C(N)=O)cn1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)ccc1NS(=O)(=O)CC(F)(F)F)c1ccc(F)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc3ccc(Cl)c(F)c3)c2)n[nH]c1Nc1cnccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1ccc(Cl)c(F)c1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(Oc3cccc(F)c3)c2)n[nH]c1Nc1cnccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(Oc3ccc(Cl)cc3)c2)n[nH]c1Nc1cnccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C3CC3)c(OCc3ccc(F)cc3)c2)n[nH]c1Nc1cnccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc3ccc(F)cc3)c2)n[nH]c1Nc1cnccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1ccc(F)cc1C
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(CC(F)(F)F)n3)c2C(N)=O)cc1OCc1ccc(F)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc3ccc(F)cc3)c2)n[nH]c1Nc1cccc(C(F)F)n1
CCS(=O)(=O)Cc1ccc(-c2n[nH]c(Nc3cccc(OCCOC)n3)c2C(N)=O)cc1OCc1ccc(F)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc3ccc(F)c(F)c3)c2)n[nH]c1Nc1cnccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc3ccc(F)cc3)c2)n[nH]c1Nc1ccc(C(F)(F)F)nc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)F)c(Oc3ccc(F)cc3)c2)n[nH]c1Nc1cnccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)F)c(OCc3ccc(F)cc3)c2)n[nH]c1Nc1cccc(C(F)(F)F)n1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)F)n3)c2C(N)=O)cc1OCc1ccc(F)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)F)c(OCc3ccc(F)cc3)c2)n[nH]c1Nc1cnccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnc(C(C)(C)C)cn3)c2C(N)=O)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CCC(F)(F)F)c(OCc3ccc(F)cc3)c2)n[nH]c1Nc1cccc(C(F)(F)F)n1
Cc1cnc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)CCC(F)(F)F)c(OCc4ccc(F)cc4)c3)c2C(N)=O)cn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CCC(F)(F)F)c(OCc3ccc(F)cc3)c2)n[nH]c1Nc1cnccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1Oc1ccc(Cl)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc3ccc(F)cc3)c2)n[nH]c1Nc1ccnc(C(F)(F)F)n1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCC1CCCN(C)C1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)F)c(OCc3ccc(F)cc3)c2)n[nH]c1Nc1ccc(C(F)(F)F)nc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CCC(F)(F)F)cc2)n[nH]c1Nc1cccc(C(F)(F)F)n1
COc1cnc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)C(F)F)c(OCc4ccc(Cl)cc4)c3)c2C(N)=O)cn1
COc1cnc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)C(F)F)c(OCc4ccc(F)cc4)c3)c2C(N)=O)cn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccnc3C(F)(F)F)c2C(N)=O)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1O[C@H](C)c1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccc(C(F)(F)F)nc3)c2C(N)=O)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccnc(C(F)(F)F)n3)c2C(N)=O)cc1OCc1ccc(F)cc1
COc1ccc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)C(F)F)c(OCc4ccc(F)cc4)c3)c2C(N)=O)nc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccc(OC)nc3)c2C(N)=O)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)c(OCc2ccc(Cl)cc2)c1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1O[C@@H](C)c1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)cc1OCC1CCCCC1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccccn3)c2C(N)=O)c(OCc2ccc(F)cc2)c1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)F)c(OCc3ccc(F)cc3)c2)n[nH]c1Nc1cnccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCC1CCN(C)CC1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1Oc1cccc(F)c1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)(F)F)cc2)n[nH]c1Nc1cccc(C(F)(F)F)n1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCCc1ccccc1Cl
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccc(C(F)(F)F)cn3)c2C(N)=O)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)c(OCc2cccc(F)c2)c1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)c(OC)c1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCCc1ccccc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCCc1ccccc1F
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCCc1cccc(Cl)c1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cc(C(F)(F)F)ccn3)c2C(N)=O)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1cccc(OC(F)(F)F)c1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1ccc(OC(F)(F)F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1ccc(C(F)(F)F)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)F)c(OCc3ccc(F)cc3)c2)n[nH]c1Nc1cccc(C(F)(F)F)n1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1cccc(C(F)(F)F)c1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCCc1cccc(F)c1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccc4cc(Cl)ccc4n3)c2C(N)=O)cc1OCc1ccc(F)cc1
COCCOc1cc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)N(C)C)cc3)c2C(N)=O)ccn1
CCS(=O)(=O)Nc1ccc(-c2c(C(N)=O)c(Nc3cnccn3)nn2C)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OC1CCCc2cc(F)ccc21
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc3ccc(F)c(Cl)c3)c2)n[nH]c1Nc1cnccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)F)c(OCc3ccc(F)c(F)c3)c2)n[nH]c1Nc1ccccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc3ccccn3)c2)n[nH]c1Nc1cnccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OC(C)(C)c1ccc(F)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1O[C@@H](C)c1ccccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc3ccc(F)cn3)c2)n[nH]c1Nc1cnccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OC1CCCc2ccccc21
CCC(Oc1cc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc3ccc(Cl)cc3)c2)n[nH]c1Nc1cnc(C(F)(F)F)cn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)F)c(OCc3ccc(Cl)cc3)c2)n[nH]c1Nc1cnc(C(F)(F)F)cn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)F)c(OC(c3ccc(F)cc3)C3CCC3)c2)n[nH]c1Nc1cnccn1
N#Cc1cccc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)CC(F)(F)F)cc3)c2C(N)=O)n1
NC(=O)c1c(-c2ccc(CS(=O)(=O)CC(F)(F)F)c(OCc3ccc(F)cc3)c2)n[nH]c1Nc1cnc(C(F)(F)F)cn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc3ccc(F)cc3)c2)n[nH]c1Nc1ccccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc3ccc(F)cn3)c2)n[nH]c1Nc1ccccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccccn3)c2C(N)=O)cc1OCc1ccc(F)cn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1ccc(Cl)cn1
C[C@H](Oc1cc(NS(=O)(=O)C(F)F)ccc1-c1n[nH]c(Nc2cnccn2)c1C(N)=O)c1ccc(F)cc1
C[C@H](Oc1cc(NS(=O)(=O)CC(F)(F)F)ccc1-c1n[nH]c(Nc2cnccn2)c1C(N)=O)c1ccc(F)cc1
Cc1cnc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c4ccc(F)cc4)c3)c2C(N)=O)cn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)F)c(OCc3ccc(F)cc3)c2)n[nH]c1Nc1cnc(C(F)(F)F)cn1
CCS(=O)(=O)Nc3ccc(c2n[nH]c(Nc1cnccn1)c2C#N)cc3OC5(c4ccc(F)c(C)c4)CC5
CCS(=O)(=O)Nc3ccc(c2n[nH]c(Nc1cnccn1)c2C#N)cc3OC5(c4ccc(F)cc4)CC5
C[C@H](Oc1cc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)ccc1NS(=O)(=O)CC(F)(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(Cl)cc1
C[C@H](Oc1cc(-c2c(C(N)=O)c(Nc3cnccn3)nn2C)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@@H](Oc1cc(NS(=O)(=O)CC(F)(F)F)ccc1-c1n[nH]c(Nc2cnccn2)c1C(N)=O)c1ccc(F)cc1
C[C@@H](Oc1cc(NS(=O)(=O)C(F)F)ccc1-c1n[nH]c(Nc2cnccn2)c1C(N)=O)c1ccc(F)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)ccc1NS(=O)(=O)CC(F)(F)F)c1cccc(Cl)c1
NC(=O)c1cccc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)C(F)F)cc3)c2C(N)=O)n1
N#Cc1cccc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)C(F)F)cc3)c2C(N)=O)n1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)ccc1NS(=O)(=O)CC(F)(F)F)c1ccc(Cl)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3ccccn3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1ccccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc3ccc(Cl)cn3)c2)n[nH]c1Nc1cnccn1
CCC(Oc1cc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)ccc1NS(=O)(=O)CC)c1ccc(F)cc1
Cc1cnc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)CC(F)(F)F)c(O[C@@H](C)c4ccc(F)cc4)c3)c2C(N)=O)cn1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)ccc1NS(=O)(=O)CC(F)(F)F)c1cccc(F)c1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OC(c3ccc(F)cc3)C3CCC3)c2)n[nH]c1Nc1cnccn1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)ccc1NS(=O)(=O)CC(F)(F)F)c1ccccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)cc2)n[nH]c1Nc1ccccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc3ccc(Cl)cc3)c2)n[nH]c1Nc1ccccn1
Cc1nn(C)cc1Nc1[nH]nc(-c2ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c3ccc(F)cc3)c2)c1C(N)=O
C[C@@H](Oc1cc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1O[C@@H](COC)c1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1O[C@H](COC)c1ccc(F)cc1
CCc1cc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c4ccc(F)cc4)c3)c2C(N)=O)no1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)F)c(OCc3nccs3)c2)n[nH]c1Nc1cnccn1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cc(C4(C)CC4)on3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cc(C(F)(F)F)n(C)n3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3ccc(C4CCOCC4)cn3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@@H](Oc1cc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)ccc1CS(=O)(=O)C(F)F)c1ncco1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)ccc1CS(=O)(=O)C(F)F)c1ncco1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cc(C4CCC4)on3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cc(C(C)(C)C)on3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3ncn(C)n3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
Cc1nc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c4ccc(F)cc4)c3)c2C(N)=O)sc1C
Cc1cc(Nc2[nH]nc(-c3ccc(CS(=O)(=O)C(F)F)c(O[C@@H](C)c4ccc(F)cc4)c3)c2C(N)=O)nn1C
Cc1cn(C)nc1Nc1[nH]nc(-c2ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c3ccc(F)cc3)c2)c1C(N)=O
C[C@H](Oc1cc(-c2n[nH]c(Nc3cc(C4CCOCC4)ccn3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
COCC(C)(C)c1cc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c4ccc(F)cc4)c3)c2C(N)=O)no1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cc(C4(C(F)(F)F)CC4)on3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
Cc1cnc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)C(F)F)c(OC4(c5ccc(F)cc5)CC4)c3)c2C(N)=O)cn1
Cc1ccc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)C(F)F)c(OCc4ccc(F)c(F)c4)c3)c2C(N)=O)nc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cc(C4(C)COC4)on3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CC(Oc1cc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ncco1
COc1cc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c4ccc(F)cc4)c3)c2C(N)=O)nn1C
C[C@H](Oc1cc(-c2n[nH]c(Nc3cc(C(C)(C)C)no3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cnc(C4CCOCC4)cn3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cc(C(C)(C)F)on3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
COCC(Oc1cc(-c2n[nH]c(Nc3cc(C)on3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CCS(=O)(=O)Cc1ccc(-c2n[nH]c(Nc3cc(C)on3)c2C(N)=O)cc1O[C@@H](COC)c1ccc(F)cc1
CCS(=O)(=O)Cc1ccc(-c2n[nH]c(Nc3cc(C)on3)c2C(N)=O)cc1O[C@H](COC)c1ccc(F)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cc(C4(C)CCOCC4)on3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
Cc1cc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c4ccc(F)cc4)c3)c2C(N)=O)on1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cc(C4CCOCC4)on3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cc(C45CC6CC(CC(C6)C4)C5)on3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cc(C4CCOC4)on3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cnn(C4CCOCC4)c3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)F)c(OC3(c4ccc(F)cc4)CC3)c2)n[nH]c1Nc1cnccn1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cc4n(n3)CCOC4)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
Cc1nccc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c4ccc(F)cc4)c3)c2C(N)=O)n1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cc(C4CC4)on3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cc(C)on3)c2C(N)=O)cc1O[C@@H](C)c1ccc(F)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cnc(C(C)(C)C)cn3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)F)c(OCc3ncco3)c2)n[nH]c1Nc1cnccn1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cc(C(F)F)on3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccc(C(=O)O)cn3)c2C(N)=O)cc1O[C@@H](C)c1ccc(F)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cnc(C4CC4)cn3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cc(C)on3)c2C(N)=O)cc1O[C@@H](C)c1ccc(F)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cc4n(n3)CCCN(C)C4)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
COCC(Oc1cc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
Cc1cc(Nc2c(C(N)=O)c(-c3ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c4ccc(F)cc4)c3)nn2C)no1
Cn1nc(-c2ccc(NS(=O)(=O)C(F)F)c(OCc3ccc(F)cc3)c2)c2c(N)nccc21
C[C@H](Oc1cc(-c2cnn3ccnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4ccncn4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(C4CCN(C)CC4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(C4=CCOCC4)cnc(N)c23)ccc1NS(=O)(=O)CC(F)(F)F)c1ccc(F)cc1
CC(C)n1nc(-c2ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c3ccc(F)cc3)c2)c2c(N)nccc21
CC(C)n1nc(-c2ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c3ccc(F)cc3)c2)c2c(N)ncc(C3=CCCNC3)c21
C[C@H](Oc1cc(-c2nn(C)c3c(C4=CCCN(C)C4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2cccc3[nH]nc(N)c23)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2ncn3ccnc(N)c23)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2cnn3ccnc(N)c23)cc1OCc1ccc(F)cc1
Nc1n[nH]c2ccnc(-c3ccc(NS(=O)(=O)CC(F)(F)F)c(OCc4ccc(F)cc4)c3)c12
Nc1n[nH]c2nccc(-c3ccc(NS(=O)(=O)C(F)F)c(OCc4ccc(F)cc4)c3)c12
Nc1n[nH]c2nccc(-c3ccc(NS(=O)(=O)CC(F)(F)F)c(OCc4ccc(F)cc4)c3)c12
Nc1n[nH]c2ccnc(-c3ccc(NS(=O)(=O)C(F)F)c(OCc4ccc(F)cc4)c3)c12
Nc1n[nH]c2ncnc(-c3ccc(NS(=O)(=O)C(F)F)c(OCc4ccc(F)cc4)c3)c12
Cc1cc(-c2ccc(NS(=O)(=O)C(F)F)c(OCc3ccc(F)cc3)c2)c2c(N)n[nH]c2n1
Nc1n[nH]c2nc(-c3ccccc3)cc(-c3ccc(NS(=O)(=O)C(F)F)c(OCc4ccc(F)cc4)c3)c12
C[C@H](Oc1cc(-c2ccnc3[nH]nc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCCNCC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CN(CC(F)(F)F)C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(C#CC4CCNCC4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(C#CC4CCN(C)CC4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(CC5CCCN5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5(CN)CC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn5c4CN(C)CC5)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5(CC#N)COC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CC6(C5)CN(C)C6)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCC(C)(C)N(C)C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4ccc(N5CCNCC5)nc4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CC(=O)N1CCC(n2cc(-c3cnc(N)c4c(-c5ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c6ccc(F)cc6)c5)nn(C)c34)cn2)CC1
COC[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCOCC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
COC[C@@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCOCC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCC(F)(F)C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
Nc1ncc(-c2cnn(C3CCOCC3)c2)c2[nH]nc(-c3ccc(NS(=O)(=O)C(F)F)c(OCc4cccc(Cl)c4)c3)c12
C[C@H](Oc1cc(-c2nn(C)c3c(N4CCOCC4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCN(C)C(C(F)(F)F)C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn([C@@H]5CCN(C)C(C)(C)C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
Fc1ccccc1CN1CCC2(CCN(CC2)C(=O)c2ccccc2)C1=O
Fc1ccc(F)c(CN2CCC3(CCN(CC3)C(=O)c3ccccc3)C2=O)c1
O=C(c1cnco1)N1CCC2(CC1)CCN(Cc1cc(F)ccc1F)C2=O
O=C(c1ccc2cc[nH]c2c1)N1CCC2(CC1)CCN(Cc1ccccc1F)C2=O
Fc1ccc(F)c(CN2CCC3(CCN(CC3)C(=O)c3ccc4cc[nH]c4c3)C2=O)c1
Cn1ccc2ccc(cc12)C(=O)N1CCC2(CCN(Cc3cc(F)ccc3F)C2=O)CC1
O=C(c1ccc2cc[nH]c2c1)N1CCC2(CC1)CCN(Cc1ccccc1F)C2=O
Nc1nc2cc(-c3ccc4c(c3)C(=O)N(Cc3cc(OC(F)(F)F)ccc3F)CCO4)ccn2n1
Nc1nc2cc(-c3ccc4c(c3)C(=O)N(Cc3cc(OC(F)(F)F)ccc3F)CCC4)ccn2n1
O=C(c1nc2n(n1)[C@H](c1cncc(F)c1)C[C@@H]2F)C1CC1
O=C(c1nc2n(n1)[C@@H](c1cncc(F)c1)C[C@H]2F)C1CC1
CC1(C)OCC2CC21C(=O)c1nc2n(n1)C(c1ccccc1)CC2F
CC(C)(CO)C(=O)c1nc2n(n1)[C@H](c1ccccc1)C[C@@H]2F
CC(C)(COC(F)F)C(=O)c1nc2n(n1)[C@H](c1ccccc1)C[C@@H]2F
CCC(=O)c1nc2n(n1)[C@H](c1cnn(C)c1)C[C@@H]2F
CC(=O)N1CC(C(=O)c2nc3n(n2)[C@H](c2ccccc2)C[C@@H]3F)C1
N#Cc1cccc([C@@H]2C[C@H](F)c3nc(C(=O)C4CC4)nn32)c1
O=C(c1nc2n(n1)[C@H](c1cccc(Cl)c1)C[C@@H]2F)C1CC1
O=C(c1nc2n(n1)CC[C@H]2c1ccccc1)C1CC1
COC(=O)C12CC(C(=O)N3N=CCC3c3cc(F)cc(F)c3)(C1)C2
O=C(O)C12CC(C(=O)N3N=CCC3c3cc(F)cc(F)c3)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3cc4cc(F)ccc4n3)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3cc4cc(F)ccc4n3)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(CF)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(COc3cc(Br)ncn3)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(COc3cc(Cl)ncn3)(C1)C2
NC(=O)c1cc(OCC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)ncn1
N#Cc1cc(OCC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)ncn1
CN(C)C(=O)C12CC(C(=O)N3N=CCC3c3cc(F)cc(F)c3)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(CCl)(C1)C2
N#Cc1cc(NCC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)ncn1
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(CN3CCOCC3)(C1)C2
O=C(N1N=CCC1c1cncc(F)c1)C12CC(Cn3ncc4c(F)cccc43)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3ncc4c(F)cncc43)(C1)C2
Cc1cc(=O)n(CC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)[nH]1
CP(C)(=O)c1cc(OCC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)ncn1
N#CCC12CC(C(=O)NC(CC=N)c3cc(F)cc(F)c3)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cc3nnn[nH]3)(C1)C2
Cc1nnc(CC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)o1
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3cc4c(F)cccc4n3)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3cc4c(F)cccc4n3)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3cnc4ccccc43)(C1)C2
O=C(N1CC(F)CC1c1cccc(F)c1)C12CC(CO)(C1)C2
Cc1cccc(C2CCCN2C(=O)C23CC(N4C(=O)CCC4=O)(C2)C3)c1
N#Cc1ccnc(OCC23CC(C(=O)N4CC(F)CC4c4cccc(F)c4)(C2)C3)c1
O=C(N1CC(F)CC1c1cccc(F)c1)C12CC(Cn3ncc4cc(F)ccc43)(C1)C2
O=C(N1CC(F)CC1c1cccc(F)c1)C12CC(COc3cc(Br)ncn3)(C1)C2
Cn1cc(-c2cc(OCC34CC(C(=O)N5CC(F)CC5c5cccc(F)c5)(C3)C4)ncn2)cn1
Cn1cc(-c2cc(OCC34CC(C(=O)N5CC(F)CC5c5cccc(F)c5)(C3)C4)ncn2)cn1
O=C(N1CC(F)CC1c1cccc(F)c1)C12CC(COc3ccccc3)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(CN3C(=O)C(F)(F)c4ccccc43)(C1)C2
N#Cc1cnn(CC23CC(C(=O)N4CC(F)CC4c4cccc(F)c4)(C2)C3)c1
COC(=O)C12CC(C(=O)N3CC(F)CC3c3cccc(F)c3)(C1)C2
COCC12CC(C(=O)N3CC(F)CC3c3cccc(F)c3)(C1)C2
N#Cc1ccn(CC23CC(C(=O)N4CC(F)CC4c4cccc(F)c4)(C2)C3)c(=O)c1
COC(=O)C12CC(C(=O)N3CC[C@@H](Oc4cc(F)ccc4F)C3)(C1)C2
O=C(N1CC[C@@H](Oc2cc(F)ccc2F)C1)C12CC(CO)(C1)C2
N#Cc1cc(OCC23CC(C(=O)N4CC[C@@H](Oc5cc(F)ccc5F)C4)(C2)C3)ncn1
O=C(N1CC(F)CC1c1cccc(F)c1)C12CC(C(O)c3ccccc3)(C1)C2
O=C(N1CC(F)CC1c1cccc(F)c1)C12CC(C(F)c3ccccc3)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(C(F)c3cccc(Cl)c3)(C1)C2
CC(Oc1cc(Cl)ncn1)C12CC(C(=O)N3CC(F)CC3c3cccc(F)c3)(C1)C2
O=C(N1N=CCC1c1ccccc1)C12CC(C1)C2
O=C(N1N=CCC1c1ccccc1)C12CC(O)(C1)C2
CCOC12CC(C(=O)NC(CC=N)c3ccccc3)(C1)C2
CC(=N)CC(NC(=O)C12CC(Cn3cc(C#N)cn3)(C1)C2)c1cc(F)cc(F)c1
O=C(N1CC(F)CC1c1cccc(F)c1)C12CC(Cn3ncc4ncccc43)(C1)C2
Cc1cnc(C2CC=NN2C(=O)C23CC(Cn4ncc5cc(C#N)ccc54)(C2)C3)cn1
Cc1cncc(C2CC=NN2C(=O)C23CC(Cn4ncc5cc(C#N)ccc54)(C2)C3)n1
N#Cc1ccc2c(cnn2CC23CC(C(=O)N4N=CCC4c4cnccn4)(C2)C3)c1
N#Cc1ccc2c(cnn2CC23CC(C(=O)N4N=CCC4c4ccccc4)(C2)C3)c1
N#Cc1ccc2c(cnn2CC23CC(C(=O)N4N=CCC4c4cc(F)ccc4F)(C2)C3)c1
NC(=O)c1cn(CC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)nn1
NC(=O)c1cnnn1CC12CC(C(=O)N3N=CCC3c3cc(F)cc(F)c3)(C1)C2
N#Cc1ccc2cn(CC34CC(C(=O)N5N=CCC5c5cc(F)cc(F)c5)(C3)C4)nc2c1
COc1ccc2cn(CC34CC(C(=O)N5N=CCC5c5cc(F)cc(F)c5)(C3)C4)nc2c1
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3cc4cccc(Cl)c4n3)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3cc4ncccc4n3)(C1)C2
N#Cc1cccc2nn(CC34CC(C(=O)N5N=CCC5c5cc(F)cc(F)c5)(C3)C4)cc12
N#Cc1ccc2nn(CC34CC(C(=O)N5N=CCC5c5cc(F)cc(F)c5)(C3)C4)cc2c1
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3cc4ccc(F)cc4n3)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3cc4c(Cl)cncc4n3)(C1)C2
N#Cc1ccc2c(cnn2CC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)c1
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3ncc4ncccc43)(C1)C2
N#Cc1ccc2cnn(CC34CC(C(=O)N5N=CCC5c5cc(F)cc(F)c5)(C3)C4)c2c1
N#Cc1cccc2c1cnn2CC12CC(C(=O)N3N=CCC3c3cc(F)cc(F)c3)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3ncc4cncc(Cl)c43)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3ncc4cccc(Cl)c43)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3ncc4ccc(F)cc43)(C1)C2
N#Cc1cnn(CC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)c1
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3cc(C(F)(F)F)cn3)(C1)C2
COc1ccc2cnn(CC34CC(C(=O)N5N=CCC5c5cc(F)cc(F)c5)(C3)C4)c2c1
Cc1cnn(CC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)c1
Cc1cc(C)n(CC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)n1
O=C(Nc1cc(Cl)ncn1)C12CC(C(=O)N3N=CCC3c3cc(F)cc(F)c3)(C1)C2
N#Cc1cccc(NC(=O)C23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)c1
CNC(=O)C12CC(C(=O)N3N=CCC3c3cc(F)cc(F)c3)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(CN3CC(F)(F)C3)(C1)C2
CS(=O)(=O)C1CN(CC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)C1
O=C(N1N=CCC1c1ccccc1)C12CC(Cn3ncc4c(F)cccc43)(C1)C2
N#Cc1cccc(C2CC=NN2C(=O)C23CC(Cn4ncc5c(F)cccc54)(C2)C3)c1
O=C(N1CC(F)CC1c1cccc(F)c1)C12CC(Cn3ncc4c(F)cccc43)(C1)C2
O=C(N1N=CCC1c1cc(F)ccc1F)C12CC(Cn3ncc4c(F)cccc43)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3nc4ccc(F)cc4n3)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3nc4ccccc4n3)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3ncc4ccncc43)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3cc4ccncc4n3)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3ncc4cccnc43)(C1)C2
C[C@H](NC(=O)C12CC(CO)(C1)C2)c1cc(F)cc(F)c1
O=C(NCc1cc(F)cc(F)c1)C12CC(CO)(C1)C2
N#Cc1cc(OCC23CC(C(=O)N4CC(F)CC4c4cccc(F)c4)(C2)C3)ncn1
Cc1ncnc(OCC23CC(C(=O)N4CC(F)CC4c4cccc(F)c4)(C2)C3)c1F
N#Cc1cccc(OCC23CC(C(=O)N4CC(F)CC4c4cccc(F)c4)(C2)C3)n1
NC(=O)c1ccnc(OCC23CC(C(=O)N4CC(F)CC4c4cccc(F)c4)(C2)C3)n1
N#Cc1cncc(OCC23CC(C(=O)N4CC(F)CC4c4cccc(F)c4)(C2)C3)n1
O=C(N1CC(F)CC1c1cccc(F)c1)C12CC(COc3ncc(F)cn3)(C1)C2
NC(=O)c1cc(OCC23CC(C(=O)N4CC(F)CC4c4cccc(F)c4)(C2)C3)ncn1
N#Cc1cc(OCC23CC(C(=O)N4CC(F)CC4c4cccc(F)c4)(C2)C3)ccn1
N#Cc1cnc(OCC23CC(C(=O)N4CC(F)CC4c4cccc(F)c4)(C2)C3)nc1
O=C(N1CC(F)CC1c1cccc(F)c1)C12CC(COc3nccc(Cl)n3)(C1)C2
N#Cc1cc(OCC23CC(C(=O)N[C@@H](C)c4cc(F)cc(F)c4)(C2)C3)ncn1
O=C(N1CC(F)CC1c1cccc(F)c1)C12CC(COc3cccc4nncn34)(C1)C2
N#Cc1cc(OCC23CC(C(=O)NCc4cc(F)cc(F)c4)(C2)C3)ncn1
Cc1cccc(C2CCCN2C(=O)C23CC(Nc4nccc(C#N)n4)(C2)C3)c1
O=C(N1CC(F)CC1c1cccc(F)c1)C12CC(Cn3cc4cc(F)ccc4n3)(C1)C2
N#Cc1cccc(OCC23CC(C(=O)N4CC(F)CC4c4cccc(F)c4)(C2)C3)c1
Cc1cccc(OCC23CC(C(=O)N4CC(F)CC4c4cccc(F)c4)(C2)C3)c1
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3c(=O)[nH]c4ccccc43)(C1)C2
Cn1c(=O)n(CC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)c2ccccc21
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3cc(-c4ccccn4)cn3)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3cc(-c4cnccn4)cn3)(C1)C2
Cc1cccc(C2CCCN2C(=O)C23CC(C2)C3)c1
O=C(N1CCC(Oc2ccccc2)C1)C12CC(F)(C1)C2
COC(=O)C12CC(C(=O)N[C@@H](C)c3cc(F)cc(F)c3)(C1)C2
N#CC12CC(C(=O)N3CCC(Oc4ccccc4)C3)(C1)C2
Cc1cccc(C2CCCN2C(=O)C23CC(NC(=O)c4ccccc4)(C2)C3)c1
CCC(=O)NC12CC(C(=O)N3CCCC3c3cccc(C)c3)(C1)C2
CC(=O)NC12CC(C(=O)N3CCCC3c3cccc(C)c3)(C1)C2
Cc1cccc(C2CCCN2C(=O)C23CC(O)(C2)C3)c1
COC(=O)C12CC(C(=O)NCc3cc(F)cc(F)c3)(C1)C2
CCOC12CC(C(=O)N3CCCC3c3cccc(C)c3)(C1)C2
N#Cc1cncn1CC12CC(C(=O)N3N=CCC3c3cc(F)cc(F)c3)(C1)C2
N#Cc1cn(CC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)cn1
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(CN3C(=O)C4(CC4)c4ccccc43)(C1)C2
N#Cc1cc(OCC23CC(C(=O)N4N=CCC4c4cncc(F)c4)(C2)C3)ncn1
N#Cc1ccc2nn(CC34CC(C(=O)N5N=CCC5c5cncc(F)c5)(C3)C4)cc2c1
N#Cc1ccc2c(cnn2CC23CC(C(=O)N4N=CCC4c4cncc(F)c4)(C2)C3)c1
Cc1c2cc(C#N)ccc2nn1CC12CC(C(=O)N3N=CCC3c3cncc(F)c3)(C1)C2
Cc1nn(CC23CC(C(=O)N4N=CCC4c4cncc(F)c4)(C2)C3)c2ccc(C#N)cc12
Cc1cnc(C2CC=NN2C(=O)C23CC(Cn4cc(C#N)cn4)(C2)C3)cn1
Cc1ccc2c(cnn2CC23CC(C(=O)N4N=CCC4c4cncc(F)c4)(C2)C3)n1
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3ccc4cc(F)ccc43)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3ccc4ncc(F)cc43)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3ncc4nccnc43)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3ccc4cncnc43)(C1)C2
N#Cc1cccc(C2CC=NN2C(=O)C23CC(Cn4cc(C#N)cn4)(C2)C3)c1
N#Cc1cnn(CC23CC(C(=O)N4N=CCC4c4ccccc4)(C2)C3)c1
N#Cc1cccc(C2CC=NN2C(=O)C23CC(Cn4ncc5ncccc54)(C2)C3)c1
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3nc4ccccc4c3Cl)(C1)C2
N#Cc1cccc2cn(CC34CC(C(=O)N5N=CCC5c5cc(F)cc(F)c5)(C3)C4)nc12
N#Cc1cccc2cn(CC34CC(C(=O)N5N=CCC5c5cc(F)cc(F)c5)(C3)C4)nc12
N#Cc1cccc2cnn(CC34CC(C(=O)N5N=CCC5c5cc(F)cc(F)c5)(C3)C4)c12
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3cc4c(n3)CCC4)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3ncc4c3CCC4)(C1)C2
N#Cc1cnn2ccn(CC34CC(C(=O)N5N=CCC5c5cc(F)cc(F)c5)(C3)C4)c12
O=C(N1N=CCC1c1ccccc1)C12CC(Cn3ncc4ncccc43)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3ncc4ncccc43)(C1)C2
COCc1cn(CC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)nn1
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3cc(CO)nn3)(C1)C2
Cc1cnc(C2CC=NN2C(=O)C23CC(Cn4ncc5ncccc54)(C2)C3)cn1
Cc1c2ccccc2nn1CC12CC(C(=O)N3N=CCC3c3cc(F)cc(F)c3)(C1)C2
Cc1nn(CC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)c2ccccc12
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(CN3CC(c4ccccc4)C3)(C1)C2
N#CC1CCN(CC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)C1
N#Cc1c(C)cnn1CC12CC(C(=O)N3N=CCC3c3cc(F)cc(F)c3)(C1)C2
Cc1cn(CC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)nc1C#N
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3ccn4nccc34)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3cc(C4CC4)nn3)(C1)C2
COc1cnn(CC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)c1
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3cc(F)c4ncc(F)cc43)(C1)C2
N#Cc1cc(N(C)CC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)ncn1
N#Cc1cn(CC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)nn1
COc1ccn(CC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)n1
Cc1ccc2c(cnn2CC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)n1
N#Cc1cnn(CC23CC(C(=O)N4N=CCC4c4cncc(F)c4)(C2)C3)c1
N#Cc1cnn(CC23CC(C(=O)N4N=CCC4c4cnccn4)(C2)C3)c1
N#Cc1cncc(C2CC=NN2C(=O)C23CC(Cn4cc(C#N)cn4)(C2)C3)c1
Cc1cncc(C2CC=NN2C(=O)C23CC(Cn4cc(C#N)cn4)(C2)C3)n1
Cc1csc(C2CC=NN2C(=O)C23CC(Cn4cc(C#N)cn4)(C2)C3)n1
Cc1ccc(C2CC=NN2C(=O)C23CC(Cn4cc(C#N)cn4)(C2)C3)nc1
CC1CC(c2cccc(F)c2)N(C(=O)C23CC(Cn4cc(C#N)cn4)(C2)C3)C1
N#Cc1ccc2c(cnn2CC23CC(C(=O)N4N=CCC4c4cncc(F)c4)(C2)C3)c1
Cc1ccc(C2CC=NN2C(=O)C23CC(Cn4ncc5cc(C#N)ccc54)(C2)C3)nc1
N#Cc1cccc(C2CC=NN2C(=O)C23CC(Cn4ncc5cc(C#N)ccc54)(C2)C3)c1
N#Cc1ccc2c(cnn2CC23CC(C(=O)N4CC(F)CC4c4cccc(F)c4)(C2)C3)c1
N#Cc1ccc2c(cnn2CC23CC(C(=O)N4CCC4c4ccccc4)(C2)C3)c1
N#Cc1ncn(CC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)n1
N#Cc1ccc2c(cnn2CC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)n1
N#Cc1ccc2nn(CC34CC(C(=O)N5N=CCC5c5cc(F)cc(F)c5)(C3)C4)cc2n1
N#Cc1cnc2ncn(CC34CC(C(=O)N5N=CCC5c5cc(F)cc(F)c5)(C3)C4)c2c1
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3nnc4cc(F)ccc43)(C1)C2
N#Cc1ccc2ncn(CC34CC(C(=O)N5N=CCC5c5cc(F)cc(F)c5)(C3)C4)c2c1
COc1ccc2ncn(CC34CC(C(=O)N5N=CCC5c5cc(F)cc(F)c5)(C3)C4)c2c1
Cc1nc2ccc(F)cc2n1CC12CC(C(=O)N3N=CCC3c3cc(F)cc(F)c3)(C1)C2
N#Cc1ccn(CC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)n1
Cc1ccn(CC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)n1
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3ccc(C4CC4)n3)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3cnc4ccc(F)cc43)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(Cn3cnc4ncccc43)(C1)C2
Cc1c(C#N)cnn1CC12CC(C(=O)N3N=CCC3c3cc(F)cc(F)c3)(C1)C2
N#Cc1cnc(OCC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)cn1
N#Cc1ccc(OCC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)c(Cl)c1
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(CO)(C1)C2
N#Cc1ccc2c(ccn2CC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)n1
N#Cc1cnc2c(ccn2CC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)c1
N#Cc1cc2cnn(CC34CC(C(=O)N5N=CCC5c5cc(F)cc(F)c5)(C3)C4)c2cn1
N#Cc1cnc2cnn(CC34CC(C(=O)N5N=CCC5c5cc(F)cc(F)c5)(C3)C4)c2c1
N#Cc1cc2cn(CC34CC(C(=O)N5N=CCC5c5cc(F)cc(F)c5)(C3)C4)nc2cn1
N#Cc1cnc2cn(CC34CC(C(=O)N5N=CCC5c5cc(F)cc(F)c5)(C3)C4)nc2c1
COc1cccc(C(F)C23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)c1
COc1ccc(C(F)C23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)cc1
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(C(O)c3cccc(Cl)c3)(C1)C2
N#Cc1ccc2c(cnn2CC23CC(C(=O)N4CCC4c4ccc(Cl)cc4)(C2)C3)c1
N#Cc1ccc2c(cnn2CC23CC(C(=O)N4CCC4c4ccc(F)cc4)(C2)C3)c1
N#Cc1ccc2c(cnn2CC23CC(C(=O)N4CCC4c4ccccc4F)(C2)C3)c1
N#Cc1ccc2c(cnn2CC23CC(C(=O)N4CCC4c4cccc(F)c4)(C2)C3)c1
N#Cc1ccc2c(cnn2CC23CC(C(=O)N4N=CC[C@H]4c4cc(F)cc(F)c4)(C2)C3)c1
N#Cc1ccc2c(cnn2CC23CC(C(=O)N4CCC4c4cccs4)(C2)C3)c1
N#Cc1ccc2c(cnn2CC23CC(C(=O)N4N=CCC4c4ccc5nccn5c4)(C2)C3)c1
N#Cc1ccc2c(cnn2CC23CC(C(=O)N4CCC4c4cccc(Cl)c4Cl)(C2)C3)c1
N#Cc1ccc2c(cnn2CC23CC(C(=O)NCc4cc(F)cc(F)c4)(C2)C3)c1
N#Cc1ccc(OCC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)nc1
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(COc3ncc(F)cc3F)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(COc3ncc(F)cn3)(C1)C2
N#Cc1cncc(OCC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)n1
COc1ccnc(OCC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)n1
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(COc3cc(F)cnc3F)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(COc3ccc(Br)cc3Cl)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(COc3ccc(Br)cc3F)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(COc3cccc(F)c3Cl)(C1)C2
N#Cc1ccc(OCC23CC(C(=O)N4N=CCC4c4cc(F)cc(F)c4)(C2)C3)c(F)c1
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(COc3ccc(F)cc3Cl)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(COc3ccc(F)cc3F)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(COc3ccccc3Cl)(C1)C2
Cc1ccccc1OCC12CC(C(=O)N3N=CCC3c3cc(F)cc(F)c3)(C1)C2
O=C(N1N=CCC1c1cc(F)cc(F)c1)C12CC(COc3cc(F)ccc3F)(C1)C2
C[C@@]12[C@@H]([C@@H](C[C@@H](O1)n3c4ccccc4c5c3c6n2c7ccccc7c6c8c5C(=O)NC8)N(C)C(=O)c9ccccc9)OC
C[C@@]12[C@](C[C@@H](O1)n3c4ccccc4c5c3c6n2c7ccccc7c6c8c5C(=O)NC8)(CO)O
CN1CCN(CC1)CC(=O)N(C)c2ccc(cc2)N/C(=C\3/c4ccc(cc4NC3=O)C(=O)OC)/c5ccccc5
C[C@@]12[C@@H]([C@@H](C[C@@H](O1)n3c4ccccc4c5c3c6n2c7ccccc7c6c8c5C(=O)NC8)NC)OC
CC(C)(C)c1cc(NC(=O)Nc2ccc(cc2)-c2cccc3c(N)nccc23)no1
CN1c2ccccc2NC[C@H](NC(=O)c2cc(Cc3ccccc3)on2)C1=O |r|
CN1c2ccccc2OC[C@@H](C1=O)NC(=O)c3cc(on3)Cc4ccccc4
O=C(N[C@H]1CS(=O)(=O)c2ccccc2NC1=O)c1cc(Cc2ccccc2)on1 |r|
O=C(N[C@@H]1COc2ccccc2NC1=O)c1cc(Cc2ccccc2)on1 |r|
CN1c2ccccc2OC[C@H](NC(=O)c2cc(Cc3cccc(c3)C3(N=N3)C(F)(F)F)[nH]n2)C1=O |r,c:27|
CCCCCc1cc(n[nH]1)C(=O)N[C@H]1COc2ccccc2NC1=O |r|
O=C(N[C@H]1COc2ccccc2NC1=O)c1cccc(Oc2ccccc2)c1 |r|
O=C(N[C@H]1CNc2ccccc2NC1=O)c1cc(Cc2ccccc2)on1 |r|
O=C(N[C@H]1COc2ccccc2NC1=O)c1cc(Cc2ccccc2)on1 |r|
CN1c2ccccc2SC[C@H](NC(=O)c2cc(Cc3ccccc3)on2)C1=O |r|
CN1c2ccc(cc2CC[C@H](NC(=O)c2cc(Cc3ccccc3)on2)C1=O)C1(N=N1)C(F)(F)F |r,c:33|
CN1c2ccccc2OC[C@H](NC(=O)c2cc(Cc3ccccc3)[nH]n2)C1=O |r|
CN1c2ccccc2CC[C@H](NC(=O)c2cc(Cc3ccccc3)on2)C1=O |r|
CC(C)(C)c1cc(NC(=O)Nc2ccc(cc2)-c2cn3c(n2)sc2cc(OCCN4CCOCC4)ccc32)no1
COc1cc2c(ncnc2cc1OCCCN1CCCCC1)N1CCN(CC1)C(=O)Nc1ccc(OC(C)C)cc1
CNC(=O)c1cc(ccn1)Oc2ccc(cc2)NC(=O)Nc3ccc(c(c3)C(F)(F)F)Cl
CO[C@@H]1[C@@H](C[C@H]2O[C@]1(C)n1c3ccccc3c3c4[C@H](O)NC(=O)c4c4c5ccccc5n2c4c13)N(C)C(=O)c1ccccc1 |r|
CNC(=O)c1ccccc1Sc2ccc3c(c2)[nH]nc3/C=C/c4ccccn4
CN1CCN(CC1)CCCOc2cc3c(cc2OC)c(c(cn3)C#N)Nc4cc(c(cc4Cl)Cl)OC
COc1cc(Oc2ccnc3cc(OC)c(OC)cc23)ccc1NC(=O)NC(C)c1nccs1
Cc1n[nH]c2ccc(cc12)-c1cncc(OC[C@@H](N)Cc2ccccc2)c1 |r|
CC1(C(=O)Nc2c(ccc(n2)Nc3c(cnc(n3)Nc4cc(c(c(c4)OC)OC)OC)F)O1)C
COCCOc1cc2c(cc1OCCOC)ncnc2Nc3cccc(c3)C#C
CN(C)C[C@@H]1CCn2cc(C3=C(C(=O)NC3=O)c3cn(CCO1)c1ccccc31)c1ccccc21 |r,t:10|
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(OCCN2CCOCC2)c2ccccc12)C(C)(C)C
CC(C)S(=O)(=O)c1ccccc1Nc2c(cnc(n2)Nc3ccc(cc3OC)N4CCC(CC4)N5CCN(CC5)C)Cl
Cn1c(Nc2ccc(cc2)C(F)(F)F)nc2cc(Oc3ccnc(c3)-c3ncc([nH]3)C(F)(F)F)ccc12
Cc1cnc2c(NCCN)nc3ccc(C)cc3n12
Fc1ccc(C(=O)NOCC2CC2)c(Nc2ccc(I)cc2Cl)c1F
O=C(N1CCNCC1)c1ccc(\C=C\c2n[nH]c3ccccc23)cc1
Cn1cc(cn1)-c1ccc2nnc(Sc3ccc4ncccc4c3)n2n1
CC(C)(C)c1cnc(o1)CSc2cnc(s2)NC(=O)C3CCNCC3
COc1ccc(cc1)COc2ccc(cc2OC)Cc3cnc(nc3N)N
CS(=O)(=O)N1CCN(Cc2cc3nc(nc(N4CCOCC4)c3s2)-c2cccc3[nH]ncc23)CC1
Oc1cccc(c1)-c1nc(N2CCOCC2)c2oc3ncccc3c2n1
CCN(CCCOc1ccc2c(c1)ncnc2Nc3cc(n[nH]3)CC(=O)Nc4cccc(c4)F)CCO
CC(C)n1nc(-c2cc3cc(O)ccc3[nH]2)c2c(N)ncnc12
Cc1cccc(c1NC(=O)c2cnc(s2)Nc3cc(nc(n3)C)N4CCN(CC4)CCO)Cl
CCC(C)(C)C(=O)N(O)Cc1cc(F)c(F)c(F)c1
CCC(C)(C)C(=O)N(O)Cc1ccc(F)c(F)c1F
CCC(C)(C)C(=O)N(O)Cc1ccc(F)cc1F
CCC(C)(C)C(=O)N(O)Cc1ccc(F)cc1
CCC(C)(C)C(=O)N(O)Cc1ccccc1
CCC(C)(C)C(=O)NC1(CC1)c1ccccc1
CCC(C)(C)C(=O)N(C)C(CO)c1ccccc1
CCC(C)(C)C(=O)NC(CO)c1ccccc1
CCC(C)(C)C(=O)N(C)C(C)c1ccccc1
CCC(C)(C)C(=O)NC(C)c1ccccc1
CC1CCCCN1C(=O)N(C)Cc1cc(F)cc(F)c1F
CC(C)N(C(C)C)C(=O)N(C)Cc1cc(F)cc(F)c1F
CC(C)N(C)C(=O)N(C)Cc1cc(F)cc(F)c1F
CN(Cc1cc(F)cc(F)c1F)C(=O)C1(C)CCCCC1
CN(Cc1cc(F)cc(F)c1F)C(=O)C1(CCCC1)C(F)(F)F
CN(Cc1cc(F)cc(F)c1F)C(=O)C1(CCC1)C(F)(F)F
CN(Cc1cc(F)cc(F)c1F)C(=O)C1CCC1
CN(Cc1cc(F)cc(F)c1F)C(=O)C1(C)CC1
CN(Cc1cc(F)cc(F)c1F)C(=O)C(C)(C)CO
COC(C)(C)C(=O)N(C)Cc1cc(F)cc(F)c1F
CN(Cc1cc(F)cc(F)c1F)C(=O)C(C)(C)C
CCC(C)(C)C(=O)N(C)Cc1ccn(C)n1
CCC(C)(C)C(=O)N(C)Cc1cnc(C)s1
CCC(C)(C)C(=O)N(C)Cc1ccco1
CCC(C)(C)C(=O)N(C)Cc1ccc(C)s1
CCC(C)(C)C(=O)N(C)Cc1sccc1C
CCC(C)(C)C(=O)N(C)Cc1cccs1
CCC(C)(C)C(=O)N(C)Cc1cccnc1
CCC(C)(C)C(=O)N(C)Cc1ccncc1
CCC(C)(C)C(=O)N(C)Cc1c(F)cc(F)cc1F
CCC(C)(C)C(=O)N(C)Cc1cc(F)ccc1F
CCC(C)(C)C(=O)N(C)Cc1ccc(F)cc1F
CCC(C)(C)C(=O)N(C)Cc1ccc(F)cc1
CCC(C)(C)C(=O)N(C)Cc1cccc(O)c1
CCC(C)(C)C(=O)N(C)Cc1cccc(Br)c1
CCC(C)(C)C(=O)N(C)Cc1cccc(F)c1
CCC(C)(C)C(=O)N(C)Cc1ccccc1Cl
CCN(Cc1ccccc1F)C(=O)C(C)(C)CC
CCC(C)(C)C(=O)N(C)Cc1ccccc1
CCC(C)(C)C(=O)NCc1cccc(Br)c1
CCC(C)(C)C(=O)NCc1ccccc1F
CCC(C)(C)C(=O)NCc1ccccc1
CCC(C)(C)C(=O)N(O)Cc1cc(F)cc(F)c1F
CCC(C)(C)C(=O)N(O)Cc1ccc(F)c(F)c1
CCC(C)(C)C(=O)N(C)C(C)(C)c1ccccc1
CCC(C)(C)C(=O)NC(C)(C)c1ccccc1
CC1CCCC(C)N1C(=O)N(C)Cc1cc(F)cc(F)c1F
CCC(C)(C)C(=O)N(C)Cc1cc(C)c(C)s1
CCC(C)(C)C(=O)N(C)Cc1cc(F)cc(F)c1F
CCC(C)(C)C(=O)N(C)Cc1cccc(F)c1F
CCC(C)(C)C(=O)N(C)Cc1ccncc1F
CCC(C)(C)C(=O)N(C)Cc1ccccc1F
CCC(C)(C)C(=O)N(C)Cc1cccc(Cl)c1
CCC(C)(C)C(=O)NCc1ccccc1Br
COc1c(Cl)cc2c3ccncc3[nH]c2c1NC(=O)c1cccnc1C
Cn1cnc2c1cc(c(c2F)Nc3ccc(cc3Cl)Br)C(=O)NOCCO
c1cc(c(c(c1)Cl)C2=C3C=CC(=NN3C=NC2=O)Sc4ccc(cc4F)F)Cl
CS(=O)(=O)CCNCc1ccc(o1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1
Cc1ccc(cc1Nc2nc(cs2)c3cccnc3)NC(=O)c4ccc(cc4)CN5CCN(CC5)C
C[C@@H](Oc1cc(cnc1N)-c1cnn(c1)C1CCNCC1)c1c(Cl)ccc(F)c1Cl |r|
C[C@@H](Oc1cc(sc1C(N)=O)-n1cnc2ccc(CN3CCN(C)CC3)cc12)c1ccccc1C(F)(F)F |r|
COc1ccc(c(c1C(=O)c2cnc(nc2N)NC3CCN(CC3)S(=O)(=O)C)F)F
CN1CCN(Cc2ccc(cc2)C(=O)Nc2ccc(C)c(Nc3nccc(n3)-c3cccnc3)c2)CC1
CN(C)C/C=C/C(=O)Nc1cc2c(cc1O[C@H]3CCOC3)ncnc2Nc4ccc(c(c4)Cl)F
Cc1[nH]c(\C=C2/C(=O)Nc3ccc(cc23)S(=O)(=O)Cc2c(Cl)cccc2Cl)c(C)c1C(=O)N1CCC[C@@H]1CN1CCCC1 |r|
CCn1c(nc2c(ncc(OC[C@H]3CCCNC3)c12)C#CC(C)(C)O)-c1nonc1N |r|
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(Cl)cc23)c1F
Clc1cccc(Cl)c1C(=O)Nc1cn[nH]c1C(=O)NC1CCNCC1
CCOc1cc2ncc(C#N)c(Nc3ccc(OCc4ccccn4)c(Cl)c3)c2cc1NC(=O)\C=C\CN(C)C
Nc1nc(N)c2nc(-c3cccc(O)c3)c(nc2n1)-c1cccc(O)c1
OCCn1cc(c(n1)-c1ccncc1)-c1ccc2C(CCc2c1)N=O
OC(=O)c1ccc(Nc2ncc3CN=C(c4cc(Cl)ccc4-c3n2)c2c(F)cccc2F)cc1 |c:13|
CC1(CNc2c1ccc(c2)NC(=O)c3cccnc3NCc4ccncc4)C
c1c[nH]c2c1c(ncn2)c3cnn(c3)[C@H](CC#N)C4CCCC4
C=CC(=O)Nc1cc2c(cc1OCCCN3CCOCC3)ncnc2Nc4ccc(c(c4)Cl)F
Cn1cc(C2=C(C(=O)NC2=O)c2cn(C3CCN(Cc4ccccn4)CC3)c3ccccc23)c2ccccc12 |t:4|
Clc1ccc(Nc2nnc(Cc3ccncc3)c3ccccc23)cc1
COc1cc2c(Oc3ccc(NC(=O)C4(CC4)C(=O)NC4=CCC(F)C=C4)cc3F)ccnc2cc1OCCCN1CCOCC1 |c:26,t:21|
C[C@@H]1CCN(C[C@@H]1N(C)c1ncnc2[nH]ccc12)C(=O)CC#N |r|
C[C@@H](O)COc1cn2ncnc(Oc3ccc4[nH]c(C)cc4c3F)c2c1C
CN1CCC(CC1)COc2cc3c(cc2OC)c(ncn3)Nc4ccc(cc4F)Br
Cc1cnc(nc1Nc2cccc(c2)S(=O)(=O)NC(C)(C)C)Nc3ccc(cc3)OCCN4CCCC4
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Cc3ccccc3)on2)C1=O)-c1n[nH]c(=O)o1 |r|
CN1c2ccccc2OC[C@H](NC(=O)c2ncc(Cc3ccccc3)o2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2cc(Cc3ccccc3)n(C)n2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2nnc(Cc3ccccc3)o2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2noc(Cc3ccccc3)n2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2cnn(Cc3ccccc3)c2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2c[nH]c(Cc3ccccc3)n2)C1=O |r|
[H][C@@]12CCCC[C@@]1([H])OC[C@H](NC(=O)c1cc(Cc3ccccc3)on1)C(=O)N2 |r|
O=C(N[C@H]1COCCNC1=O)c1cc(Cc2ccccc2)on1 |r|
O=C(N[C@H]1CCOc2ccccc2NC1=O)c1cc(Cc2ccccc2)on1 |r|
O=C(N[C@@H]1CNc2ccccc2OC1)c1cc(Cc2ccccc2)on1 |r|
CN([C@H]1COc2ccccc2NC1=O)C(=O)c1cc(Cc2ccccc2)on1 |r|
O=C(N[C@H]1COc2ccccc2N(C2CC2)C1=O)c1cc(Cc2ccccc2)on1 |r|
CN1c2ccccc2OC[C@H](NC(=O)c2ncn(Cc3ccccc3)n2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2cc(Cc3ccccc3)ccn2)C1=O |r|
CN1C[C@H](NC(=O)c2cc(Cc3ccccc3)on2)C(=O)N(C)c2ccccc12 |r|
O=C(NC1Cc2ccccc2NC1=O)c1cc(Cc2ccccc2)on1
CN1c2cc(NC(C)=O)ccc2OC[C@H](NC(=O)c2cc(Cc3ccccc3)on2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2cc(CN3CCCCC3)on2)C1=O |r|
CC(C)Cc1cc(no1)C(=O)N[C@H]1COc2ccccc2N(C)C1=O |r|
CCCCCc1cc(no1)C(=O)N[C@H]1COc2ccccc2N(C)C1=O |r|
COC(=O)Nc1ccc2OC[C@H](NC(=O)c3cc(Cc4ccccc4)on3)C(=O)N(C)c2c1 |r|
CN1c2cc(NS(C)(=O)=O)ccc2OC[C@H](NC(=O)c2cc(Cc3ccccc3)on2)C1=O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2cc(Cc3ccccc3)on2)C1=O)-c1cc[nH]n1 |r|
CN1c2ccccc2OC[C@H](NC(=O)c2coc(Cc3ccccc3)n2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2cn(Cc3ccccc3)nn2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2cccc(Cc3ccccc3)c2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2cc(CC3CCCCC3)on2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2cn(Cc3ccccc3)cn2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2nnn(Cc3ccccc3)n2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2cc(C)on2)C1=O |r|
CN1CC[C@@H]([C@H](O)C1)c1c(O)cc(O)c2c1oc(cc2=O)-c1ccccc1Cl |r|
C[C@@]1(COc2ccccc2NC1=O)NC(=O)c1cc(Cc2ccccc2)on1 |r|
CNC(=O)c1c(F)cccc1Nc1nc(Nc2cc3N(CCc3cc2OC)C(=O)CN(C)C)nc2[nH]ccc12
COc1cc2c(cc1OCCCN3CCOCC3)c(ncn2)Nc4ccc(c(c4)Cl)F
CC[C@H]1N(C2CCCC2)c2nc(Nc3ccc(cc3OC)C(=O)NC3CCN(C)CC3)ncc2N(C)C1=O |r|
CS(=O)c1ccc(cc1)-c1nc(c([nH]1)-c1ccc(F)cc1)-c1ccncc1
CN1c2c(cnc(n2)Nc3cccc(c3)SC)C=C(C1=O)c4c(cccc4Cl)Cl
COc1cc2c(Oc3ccc4[nH]c(C)cc4c3F)ncnc2cc1OCCCN1CCCC1
CN(C)CC(=O)N1CCC(CC1)c1ccc(NC(=O)c2ncc([nH]2)C#N)c(c1)C1=CCCCC1 |t:31|
Cc1cn(cn1)-c1cc(NC(=O)c2ccc(C)c(Nc3nccc(n3)-c3cccnc3)c2)cc(c1)C(F)(F)F
c1ccc(cc1)Cc2[nH]c3ccc(cc3n2)[N+](=O)[O-]
CN1c2ccccc2OC[C@H](N2CCn3nc(Cc4ccccc4)nc3C2=O)C1=O |r|
CN1c2ccccc2OC[C@H](N2CCn3cc(Cc4ccccc4)nc3C2=O)C1=O |r|
CN1c2ccccc2OC[C@H](N2CCc3cn(Cc4ccccc4)nc3C2=O)C1=O |r|
CN1c2ccccc2OC[C@H](N2CCc3cn(Cc4ccccc4F)nc3C2=O)C1=O |r|
CN1c2ccccc2OC[C@H](N2CCc3cn(Cc4cccc(F)c4)nc3C2=O)C1=O |r|
CN1c2ccccc2OC[C@H](N2CCc3cn(Cc4ccc(F)cc4)nc3C2=O)C1=O |r|
CN1c2ccccc2OC[C@H](N2CCc3cn(CC4CCC4)nc3C2=O)C1=O |r|
CN1c2ccccc2OC[C@H](N2CCc3cn(Cc4cccnc4)nc3C2=O)C1=O |r|
CN1c2ccccc2OC[C@H](N2CCc3cn(Cc4ccccn4)nc3C2=O)C1=O |r|
CN1c2ccccc2OC[C@H](N2CCc3cn(CC4CCS(=O)(=O)C4)nc3C2=O)C1=O |r|
CN1c2ccccc2OC[C@H](N2CCc3c(C)n(Cc4ccccc4)nc3C2=O)C1=O |r|
CN1c2ccc(cc2OC[C@@H](C1=O)N3CCc4c(nn(c4Cl)Cc5ccccc5)C3=O)C#N
CN1c2ccccc2OC[C@H](N2CCc3c(Cl)n(Cc4ccccc4)nc3C2=O)C1=O |r|
CN1c2ccccc2OC[C@H](N2CCc3c(nn(Cc4ccccc4)c3C(N)=O)C2=O)C1=O |r|
CN1c2cc(ccc2OC[C@H](N2CCc3c(Cl)n(Cc4ccccc4)nc3C2=O)C1=O)C#N |r|
CNC(=O)c1ccc2N(C)C(=O)[C@H](COc2c1)N1CCc2c(Cl)n(Cc3ccccc3)nc2C1=O |r|
CN1c2ccc(cc2OC[C@H](N2CCc3cn(Cc4ccccc4F)nc3C2=O)C1=O)C#N |r|
CN1c2ccc(cc2OC[C@H](N2CCc3cn(Cc4c(F)cccc4F)nc3C2=O)C1=O)C#N |r|
Nc1ncnc2occ(-c3ccc(NC(=O)Nc4cc(ccc4F)C(F)(F)F)cc3)c12
CN1c2ccccc2OC[C@H](N2CCc3nn(Cc4ccccc4)cc3C2=O)C1=O |r|
CN1c2ccccc2OC[C@H](N2CCc3cn(Cc4c(F)cccc4F)nc3C2=O)C1=O |r|
CN1c2ccccc2OC[C@H](N2CCc3cn(CC4CCS(=O)(=O)CC4)nc3C2=O)C1=O |r|
CN1c2ccccc2OC[C@H](N2CCc3c(nn(Cc4ccccc4)c3C#N)C2=O)C1=O |r|
CN(C)C(=O)c1ccc2N(C)C(=O)[C@H](COc2c1)N1CCc2c(Cl)n(Cc3ccccc3)nc2C1=O |r|
CN1c2ccccc2OC[C@H](N2CCc3[nH]c(Cc4ccccc4)nc3C2=O)C1=O |r|
Cc1[nH]nc(Nc2nc(Nc3ccc(NC(=O)C4CC4)cc3)nc(n2)N2CCOCC2)c1C
CN1CCN(CC1)c1cc(Nc2n[nH]c(C)c2C)nc(Nc2ccc(NC(=O)C3CCCCC3)cc2)n1
CN1CCN(CC1)c1nc(Nc2n[nH]c(C)c2C)nc(Sc2ccc(NC(=O)C3CC3)cc2)n1
Cc1cc(Nc2cc(nc(Nc3ccc(NC(=O)C4CC4)cc3)n2)N2CCCCC2)n[nH]1
Cc1cc(Nc2cc(nc(Nc3ccc(NC(=O)C4CC4)cc3)n2)N2CCOCC2)n[nH]1
CN1CCN(CC1)c1cc(Nc2cc(C)[nH]n2)nc(Nc2ccc(NC(=O)C3CC3)cc2)n1
CN1CCN(CC1)c1nc(Nc2cc(C)[nH]n2)nc(Sc2ccc(NC(=O)C3CCCCC3)cc2)n1
CN1C(=O)NC(Cc2c[nH]c3c(Cl)cccc23)C1=O
CN1CCN(CC1)c1nc(Nc2n[nH]c(C)c2C)nc(Sc2ccc(NC(=O)C3CCCCC3)cc2)n1
Cc1cc(Nc2cc(nc(Sc3ccc(NC(=O)C4CCCCC4)cc3)n2)N2CCOCC2)n[nH]1
Cc1[nH]nc(Nc2cc(nc(Sc3ccc(NC(=O)C4CCCCC4)cc3)n2)N2CCCCC2)c1C
Cc1cc(Nc2nc(Sc3ccc(NC(=O)C4CC4)cc3)nc(n2)N2CCOCC2)n[nH]1
Cc1[nH]nc(Nc2nc(Nc3ccc(NC(=O)C4CC4)cc3)nc(n2)N2CCCCC2)c1C
Cc1[nH]nc(Nc2cc(nc(Sc3ccc(NC(=O)C4CCCCC4)cc3)n2)N2CCOCC2)c1C
Cc1[nH]nc(Nc2nc(Nc3ccc(NC(=O)C4CCCCC4)cc3)nc(n2)N2CCCCC2)c1C
Cc1cc(Nc2nc(Nc3ccc(NC(=O)C4CC4)cc3)nc(n2)N2CCOCC2)n[nH]1
Cc1[nH]nc(Nc2nc(Sc3ccc(NC(=O)C4CC4)cc3)nc(n2)N2CCOCC2)c1C
CN1CCN(CC1)c1cc(Nc2cc(C)[nH]n2)nc(Sc2ccc(NC(=O)C3CC3)cc2)n1
Cc1[nH]nc(Nc2cc(nc(Nc3ccc(NC(=O)C4CCCCC4)cc3)n2)N2CCOCC2)c1C
Cc1cc(Nc2cc(nc(Nc3ccc(NC(=O)C4CCCCC4)cc3)n2)N2CCCCC2)n[nH]1
Cc1[nH]nc(Nc2cc(nc(Nc3ccc(NC(=O)C4CCCCC4)cc3)n2)N2CCCCC2)c1C
Cc1cc(Nc2cc(nc(Sc3ccc(NC(=O)C4CCCCC4)cc3)n2)N2CCCCC2)n[nH]1
Cc1cc(Nc2nc(Nc3ccc(NC(=O)C4CC4)cc3)nc(n2)N2CCCCC2)n[nH]1
Cc1cc(Nc2nc(Sc3ccc(NC(=O)C4CCCCC4)cc3)nc(n2)N2CCOCC2)n[nH]1
Cc1[nH]nc(Nc2nc(Nc3ccc(NC(=O)C4CCCCC4)cc3)nc(n2)N2CCOCC2)c1C
Cc1cc(Nc2cc(nc(Sc3ccc(NC(=O)C4CC4)cc3)n2)N2CCCCC2)n[nH]1
CN1CCN(CC1)c1nc(Nc2n[nH]c(C)c2C)nc(Nc2ccc(NC(=O)C3CC3)cc2)n1
Cc1cc(Nc2nc(Nc3ccc(NC(=O)C4CCCCC4)cc3)nc(n2)N2CCOCC2)n[nH]1
CN1CCN(CC1)c1nc(Nc2cc(C)[nH]n2)nc(Nc2ccc(NC(=O)C3CCCCC3)cc2)n1
CN1CCN(CC1)c1nc(Nc2cc(C)[nH]n2)nc(Nc2ccc(NC(=O)C3CC3)cc2)n1
CN1CCN(CC1)c1nc(Nc2n[nH]c(C)c2C)nc(Nc2ccc(NC(=O)C3CCCCC3)cc2)n1
Cc1cc(Nc2cc(nc(Sc3ccc(NC(=O)C4CC4)cc3)n2)N2CCOCC2)n[nH]1
Cc1[nH]nc(Nc2cc(nc(Nc3ccc(NC(=O)C4CC4)cc3)n2)N2CCCCC2)c1C
CN1CCN(CC1)c1cc(Nc2cc(C)[nH]n2)nc(Sc2ccc(NC(=O)C3CCCCC3)cc2)n1
CN1CCN(CC1)c1cc(Nc2cc(C)[nH]n2)nc(Nc2ccc(NC(=O)C3CCCCC3)cc2)n1
CN1CCN(CC1)c1cc(Nc2n[nH]c(C)c2C)nc(Sc2ccc(NC(=O)C3CCCCC3)cc2)n1
CCN1CCN(CC1)c1cc(Nc2n[nH]c(C)c2C)nc(Sc2ccc(NC(=O)C3CC3)cc2)n1
CN1CCN(CC1)c1cc(Nc2n[nH]c(C)c2C)nc(Nc2ccc(NC(=O)C3CC3)cc2)n1
Cc1[nH]nc(Nc2nc(Sc3ccc(NC(=O)C4CCCCC4)cc3)nc(n2)N2CCOCC2)c1C
CN1CCN(CC1)c1nc(Nc2cc(C)[nH]n2)nc(Sc2ccc(NC(=O)C3CC3)cc2)n1
Cc1cc(Nc2nc(Sc3ccc(NC(=O)C4CC4)cc3)nc(n2)N2CCCCC2)n[nH]1
Cc1[nH]nc(Nc2nc(Sc3ccc(NC(=O)C4CC4)cc3)nc(n2)N2CCCCC2)c1C
Cc1cc(Nc2nc(Nc3ccc(NC(=O)C4CCCCC4)cc3)nc(n2)N2CCCCC2)n[nH]1
Cc1cc(Nc2cc(nc(Nc3ccc(NC(=O)C4CCCCC4)cc3)n2)N2CCOCC2)n[nH]1
Cc1[nH]nc(Nc2cc(nc(Nc3ccc(NC(=O)C4CC4)cc3)n2)N2CCOCC2)c1C
Cc1[nH]nc(Nc2nc(Sc3ccc(NC(=O)C4CCCCC4)cc3)nc(n2)N2CCCCC2)c1C
Cc1cc(Nc2nc(Sc3ccc(NC(=O)C4CCCCC4)cc3)nc(n2)N2CCCCC2)n[nH]1
CC[C@H](CO)Nc1nc(NCc2ccccc2)c2ncn(C(C)C)c2n1 |r|
Oc1ccc(cc1)-c1nc(c([nH]1)-c1ccc(F)cc1)-c1ccncc1
NC(=O)c1ccc(cc1)-c1nc(c([nH]1)-c1ccc2OCOc2c1)-c1ccccn1
COCC(=O)NC\C=C\c1ccc2ncnc(Nc3ccc(Oc4ccc(C)nc4)c(C)c3)c2c1
CCOc1cc2c(cc1NC(=O)/C=C/CN(C)C)c(c(cn2)C#N)Nc3ccc(c(c3)Cl)F
CCOC1=CS(=O)(=O)c2cc3c(Nc4ccc5scnc5c4)ncnc3cc12 |t:3|
Nc1nccc2c(cccc12)-c1ccc(NC(=O)Nc2cccc(c2)C(F)(F)F)cc1
Nc1nccc2c(cccc12)-c1ccc(NC(=O)Nc2ccc(F)c(c2)C(F)(F)F)cc1
Nc1nccc2c(cccc12)-c1ccc(NC(=O)Nc2cc(F)cc(c2)C(F)(F)F)cc1
Nc1nccc2c(cccc12)-c1ccc(NC(=O)Nc2cc(ccc2F)C(F)(F)F)cc1
CC(C)(C)c1cc(NC(=O)Nc2ccc(cc2)-c2coc3ncnc(N)c23)no1
Nc1ncnc2occ(-c3ccc(NC(=O)Nc4cc(cc(c4)C(F)(F)F)C(F)(F)F)cc3)c12
Nc1ncnc2occ(-c3ccc(NC(=O)Nc4ccc5ccccc5c4)cc3)c12
Nc1ncnc2occ(-c3ccc(NC(=O)Nc4cccc(Cl)c4)cc3)c12
CCc1cccc(NC(=O)Nc2ccc(cc2)-c2coc3ncnc(N)c23)c1
Nc1ncnc2occ(-c3ccc(NC(=O)Nc4cc(ccc4Cl)C(F)(F)F)cc3)c12
Nc1ncnc2occ(-c3ccc(NC(=O)Nc4ccc(Cl)c(c4)C(F)(F)F)cc3)c12
Nc1ncnc2occ(-c3ccc(NC(=O)Nc4cccc(c4F)C(F)(F)F)cc3)c12
Nc1ncnc2occ(-c3ccc(NC(=O)Nc4cc(F)cc(c4)C(F)(F)F)cc3)c12
Nc1ncnc2occ(-c3ccc(NC(=O)Nc4ccc(F)c(c4)C(F)(F)F)cc3)c12
Nc1ncnc2occ(-c3ccc(NC(=O)Nc4cccc(c4)C(F)(F)F)cc3)c12
Fc1ccc(cc1NC(=O)Nc1cccc(c1)-c1c[nH]c2ncc(cc12)-c1cn[nH]c1)C(F)(F)F
Nc1ccc(cc1)-c1cnc2[nH]cc(-c3cccc(NC(=O)Nc4cc(ccc4F)C(F)(F)F)c3)c2c1
Nc1cccc(c1)-c1cnc2[nH]cc(-c3cccc(NC(=O)Nc4cc(ccc4F)C(F)(F)F)c3)c2c1
CS(=O)(=O)c1cccc(c1)-c1cnc2[nH]cc(-c3cccc(NC(=O)Nc4cc(ccc4F)C(F)(F)F)c3)c2c1
NC(=O)c1cccc(c1)-c1cnc2[nH]cc(-c3cccc(NC(=O)Nc4cc(ccc4F)C(F)(F)F)c3)c2c1
Fc1ccc(cc1NC(=O)Nc1cccc(c1)-c1c[nH]c2ncc(cc12)-c1cccnc1)C(F)(F)F
CCS(=O)(=O)c1ccc(cc1)-c1cnc2[nH]cc(-c3cccc(NC(=O)Nc4cc(ccc4F)C(F)(F)F)c3)c2c1
O=C(NC1CCCC1)Nc1cccc(c1)-c1c[nH]c2ncc(cc12)-c1ccccc1
Fc1ccc(cc1NC(=O)Nc1cccc(c1)-c1c[nH]c2ncc(cc12)-c1ccccc1)C(F)(F)F
CC(=O)c1cccc(NC(=O)Nc2cccc(c2)-c2c[nH]c3ncc(cc23)-c2ccccc2)c1
COc1cccc(NC(=O)Nc2cccc(c2)-c2c[nH]c3ncc(cc23)-c2ccccc2)c1
FC(F)(F)c1cccc(NC(=O)Nc2cccc(c2)-c2c[nH]c3ncc(cc23)-c2ccccc2)c1
[O-][N+](=O)c1cccc(NC(=O)Nc2cccc(c2)-c2c[nH]c3ncc(cc23)-c2ccccc2)c1
Cc1cccc(NC(=O)Nc2cccc(c2)-c2c[nH]c3ncc(cc23)-c2ccccc2)c1
O=C(Nc1ccccc1)Nc1cccc(c1)-c1c[nH]c2ncc(cc12)-c1ccccc1
Nc1nccc2c(cccc12)-c1ccc(NC(=O)Nc2cc(ccc2Cl)C(F)(F)F)cc1
Nc1nccc2c(cccc12)-c1ccc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)cc1
Nc1nccc2c(cccc12)-c1ccc(NC(=O)Nc2cccc(c2F)C(F)(F)F)cc1
Cn1nc(-c2ccc3N(CCc3c2)C(=O)Cc2cccc(OC(F)(F)F)c2)c2cncnc12
Cn1nc(-c2ccc3N(CCc3c2)C(=O)Cc2cccc(Br)c2)c2c(N)ncnc12
Cc1cc(ccc1NC(=O)Cc1cccc(c1)C(F)(F)F)-c1nn(C)c2ncnc(N)c12
CCCn1cc(-c2ccc3N(CCc3c2)C(=O)Cc2cccc(OC(F)(F)F)c2)c2c(N)ncnc12
Cc1cccc(CC(=O)N2CCc3cc(ccc23)-c2nn(C)c3ncnc(N)c23)c1
Cn1nc(-c2ccc(NC(=O)Cc3cccc(c3)C(F)(F)F)c(F)c2)c2c(N)ncnc12
CCn1cc(-c2ccc3N(CCc3c2)C(=O)Cc2cccc(OC(F)(F)F)c2)c2c(N)ncnc12
Cn1cc(-c2ccc3N(CCc3c2)C(=O)Cc2cccc(OC(F)(F)F)c2)c2c(N)ncnc12
Cn1nc(-c2ccc3N(CCc3c2)C(=O)Cc2cc(F)cc(c2)C(F)(F)F)c2c(N)ncnc12
Cn1nc(-c2ccc3N(CCc3c2)C(=O)Cc2cccc(c2)C#N)c2c(N)ncnc12
Cn1nc(-c2ccc3N(CCc3c2)C(=O)Cc2cccc(F)c2)c2c(N)ncnc12
CC(C)c1cc(ccc1NC(=O)Cc1cccc(c1)C(F)(F)F)-c1nn(C)c2ncnc(N)c12
Cn1nc(-c2ccc(NC(=O)Cc3cccc(c3)C(F)(F)F)cc2)c2c(N)ncnc12
CCCCn1cc(-c2ccc3N(CCc3c2)C(=O)Cc2cccc(OC(F)(F)F)c2)c2c(N)ncnc12
CC(C)n1cc(-c2ccc3N(CCc3c2)C(=O)Cc2cccc(OC(F)(F)F)c2)c2c(N)ncnc12
Cn1cc(-c2ccc3N(CCc3c2)C(=O)Cc2cccc(OC(F)(F)F)c2)c2cncnc12
Cn1nc(-c2ccc3N(CCc3c2)C(=O)Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2c(N)ncnc12
Cn1nc(-c2ccc3N(CCc3c2)C(=O)Cc2ccc(Br)cc2)c2c(N)ncnc12
Cn1nc(-c2ccc3N(CCc3c2)C(=O)Cc2ccc(Cl)cc2)c2c(N)ncnc12
Cn1nc(-c2ccc3N(CCc3c2)C(=O)Cc2ccc(cc2)C(F)(F)F)c2c(N)ncnc12
Cn1nc(-c2ccc3N(CCc3c2)C(=O)Cc2cccc(OC(F)(F)F)c2)c2c(N)ncnc12
Cn1nc(-c2ccc3N(CCc3c2)C(=O)Cc2cccc(Cl)c2)c2c(N)ncnc12
Cn1nc(-c2ccc3N(CCc3c2)C(=O)Nc2cccc(c2)C(F)(F)F)c2c(N)ncnc12
C[C@@H](C(=O)N1CCc2cc(ccc12)-c1nn(C)c2ncnc(N)c12)c1ccccc1 |r|
Cn1nc(-c2ccc3N(CCc3c2)C(=O)Cc2cccc(c2)C(F)(F)F)c2c(N)ncnc12
CCc1cc(ccc1NC(=O)Cc1cccc(c1)C(F)(F)F)-c1nn(C)c2ncnc(N)c12
COc1cc(ccc1NC(=O)Cc1cccc(c1)C(F)(F)F)-c1nn(C)c2ncnc(N)c12
Cn1nc(-c2ccc(NC(=O)Cc3cccc(c3)C(F)(F)F)c(Cl)c2)c2c(N)ncnc12
COCCn1cc(-c2ccc3N(CCc3c2)C(=O)Cc2cccc(OC(F)(F)F)c2)c2c(N)ncnc12
Cn1nc(-c2ccc3N(CCc3c2)C(=O)Cc2ccc(Cl)c(c2)C(F)(F)F)c2c(N)ncnc12
COc1cccc(CC(=O)N2CCc3cc(ccc23)-c2nn(C)c3ncnc(N)c23)c1
Cn1nc(-c2ccc(NC(=O)Cc3cccc(c3)C(F)(F)F)cc2F)c2c(N)ncnc12
Cn1nc(-c2ccc3N(CCc3c2)C(=O)CCc2cccc(c2)C(F)(F)F)c2c(N)ncnc12
C[C@H](C(=O)N1CCc2cc(ccc12)-c1nn(C)c2ncnc(N)c12)c1ccccc1 |r|
CN1c2ccccc2CC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O |r|
O=C(N[C@H]1COc2ccccc2NC1=O)c1n[nH]c(Cc2ccccc2)n1 |r|
O=C(N[C@H]1CCc2ccccc2NC1=O)c1n[nH]c(Cc2ccccc2)n1 |r|
CN1c2c(F)cc(F)cc2CC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O |r|
CN1c2ccccc2NC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3F)n2)C1=O |r|
Clc1ccc2NC(=O)[C@H](CNc2c1)NC(=O)c1nnc(Cc2ccccc2)[nH]1 |r|
Fc1cc(F)cc(c1)[C@@H]1CC=NN1C(=O)C1CCN(CC1)c1cc(ncn1)C#N |r,c:11|
Fc1ccccc1Cc1nnc([nH]1)C(=O)N[C@H]1CNc2cccc(F)c2NC1=O |r|
CN1c2c(F)cc(F)cc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O |r|
Cc1cc(NC(=O)c2cccn(-c3ccc(F)cc3)c2=O)ccc1Oc1ccnc(NC(=O)C2CC2)c1
Cc1ccc(COC(=O)Nc2cc(ccn2)-c2cc3c(CCNC3=O)[nH]2)cc1
Fc1ccc(cc1)-n1cccc(C(=O)Nc2ccc(Oc3ccnc4[nH]ccc34)c(F)c2)c1=O
c1cc(ccc1N2C=CC=C(C2=O)C(=O)Nc3ccc(c(c3)F)Oc4ccnc(c4)NC(=O)C5CC5)F
Fc1ccc(cc1)-n1cccc(C(=O)Nc2ccc(Oc3ccncc3)c(F)c2)c1=O
Cc1cc(NC(=O)c2cccn(-c3ccc(F)cc3)c2=O)cc(C)c1Oc1ccncc1
Cc1cc(NC(=O)c2cccn(-c3ccc(F)cc3)c2=O)cc(C)c1Oc1ccnc(NC(=O)C2CC2)c1
CC#Cc1c(N)nccc1Oc1ccc(NC(=O)c2cccn(-c3ccc(F)cc3)c2=O)cc1F
Nc1ccc(nc1)C#Cc1c(N)nccc1Oc1ccc(NC(=O)c2cccn(-c3ccc(F)cc3)c2=O)cc1F
Fc1ccc(cc1)-n1cccc(C(=O)Nc2ccc(Oc3ccncc3)c3ccccc23)c1=O
Fc1ccc(cc1)-c1cccc(c1)C(=O)Nc1ccc(Oc2ccncc2)c(F)c1
Cc1c(c(ccc1NC(=O)C2=CC=CN(C2=O)c3ccc(cc3)F)Oc4ccnc(c4)NC(=O)C5CC5)C
Cc1c(C)c(Oc2ccncc2)ccc1NC(=O)c1cccn(-c2ccc(F)cc2)c1=O
CC(=O)N1CCC(CC1)C(=O)N1N=CC[C@H]1c1ccccc1 |r,c:13|
CC(C)(C)C(=O)N1N=CCC1c1c[nH]cn1 |c:7|
O=C(C1CCCC1)N1N=CCC1c1ccccc1 |c:9|
O=C(N1N=CCC1c1ccccc1)c1ccccn1 |c:3|
CN1CCN(C(C1)c1ccccc1)C(=O)C(C)(C)C
CC(C)(C)C(=O)N1N=CCC1c1ccc(cc1)C(C)(C)C |c:7|
O=C(C1CCN(CC1)C(=O)c1ccccc1)N1N=CCC1c1ccccc1 |c:19|
O=C(C1CCN(CC1)c1ccccn1)N1N=CC[C@H]1c1ccccc1 |r,c:17|
Cc1nnc(o1)N1CCC(CC1)C(=O)N1N=CC[C@H]1c1cc(F)cc(F)c1 |r,c:17|
O=C(C1CCN(CC1)C(=O)c1ccccn1)N1N=CCC1c1ccccc1 |c:19|
O=C(C1CCN(CC1)c1cccnn1)N1N=CC[C@H]1c1ccccc1 |r,c:17|
CC(C)(C)C(=O)N1N=CCC1c1ccccc1 |c:7|
CN1CCC(CC1)C1CC=NN1C(=O)C(C)(C)C |c:10|
O=C(N1N=CCC1c1ccccc1)c1ccccc1 |c:3|
O=C(C1CCN(CC1)C(=O)c1cccnc1)N1N=CCC1c1ccccc1 |c:19|
CC(C)(C)C(=O)N1N=CC[C@H]1c1ccccc1 |r,c:7|
CC(C)(C)C(=O)N1CCSC1c1ccccc1
O=C(C1CCN(CC1)c1ccccc1)N1N=CC[C@H]1c1ccccc1 |r,c:17|
Cc1ccc(cc1)C1CC=NN1C(=O)C(C)(C)C |c:10|
CC(C)(C)C(=O)N1N=CCC1c1ccccn1 |c:7|
CC(C)C(=O)N1N=CCC1c1ccccc1 |c:6|
O=C(N1N=CCC1c1ccccc1)c1cccnc1 |c:3|
O=C(C1CCN(CC1)c1ncccn1)N1N=CC[C@H]1c1ccccc1 |r,c:17|
Fc1cc(F)cc(c1)[C@@H]1CC=NN1C(=O)C1CCN(CC1)c1ccc(nn1)C#N |r,c:11|
Fc1cc(F)cc(c1)[C@@H]1CC=NN1C(=O)C1CCN(CC1)c1cnc(cn1)C#N |r,c:11|
CC(C)(C)C(=O)N1N=CC[C@@H]1c1ccccc1 |r,c:7|
CC(C)(C)C(=O)N1N=CCC1c1cccc(F)c1 |c:7|
Cc1ccc(cc1F)C1CC=NN1C(=O)C(C)(C)C |c:11|
CC(C)(C)C(=O)N1N=CCC1c1cccc(Cl)c1 |c:7|
CC(C)(C)C(=O)N1N=CCC1c1cccnc1 |c:7|
CC(C)(C)C(=O)N1N=CCC1c1ccncc1 |c:7|
CC(C)(C)C(=O)N1N=CCC1c1cocn1 |c:7|
CC(C)(C)C(=O)N1N=CCC1C1CCCCC1 |c:7|
CC(C)(C)C(=O)N1N=CCC1C1CCOCC1 |c:7|
CC(C)(CO)C(=O)N1N=CCC1c1ccccc1 |c:8|
O=C(C1CCCCC1)N1N=CCC1c1ccccc1 |c:10|
O=C(C1CCC1)N1N=CCC1c1ccccc1 |c:8|
O=C(N1N=CCC1c1ccccc1)c1ccncc1 |c:3|
O=C(C1CCN(CC1)c1ccccc1)N1N=CCC1c1ccccc1 |c:17|
CC(=O)N1CCC(CC1)C(=O)N1N=CCC1c1ccccc1 |c:13|
O=C(C1CCN(CC1)C(=O)C1CCCCC1)N1N=CCC1c1ccccc1 |c:19|
O=C(C1CCN(CC1)C(=O)c1cnco1)N1N=CC[C@H]1c1ccccc1 |r,c:18|
O=C(C1CCN(CC1)C(=O)c1cn[nH]c1)N1N=CCC1c1ccccc1 |c:18|
O=C(C1CCN(CC1)C(=O)c1c[nH]nn1)N1N=CCC1c1ccccc1 |c:18|
Cc1nnc(o1)N1CCC(CC1)C(=O)N1N=CC[C@H]1c1ccccc1 |r,c:17|
Fc1cc(F)cc(c1)[C@@H]1CC=NN1C(=O)C1CCN(CC1)c1ccnc(n1)C#N |r,c:11|
CC(C)(C)C(=O)N1CCCC1c1ccccc1
CC(C)(C)C(=O)N1CCCC1c1cccc(F)c1
CC1=NN([C@@H](C1)c1ccccc1)C(=O)C(C)(C)C |r,t:1|
CC(C)(C)C(=O)N1CCCCC1c1ccccc1
CC(C)(C)C(=O)N1CCNCC1c1ccccc1
CC(C)(C)C(=O)N1N=CCC1c1cc(F)cc(F)c1 |c:7|
CC(C)(C)C(=O)N1N=CCC1c1ccc(Cl)cc1 |c:7|
CC(C)(C)C(=O)N1N=CCC1c1cc[nH]n1 |c:7|
CC(C)(C)C(=O)N1N=CCC1C1CCCC1 |c:7|
CC(C)(CN)C(=O)N1N=CCC1c1ccccc1 |c:8|
O=C(C1CCOC1)N1N=CCC1c1ccccc1 |c:9|
FC(F)(F)C(=O)N1CCC(CC1)C(=O)N1N=CCC1c1ccccc1 |c:16|
O=C(C1CCN(CC1)C(=O)c1cc[nH]n1)N1N=CCC1c1ccccc1 |c:18|
Clc1cccc(NC(=O)N2N=CCC2c2ccccc2)c1 |c:10|
CC(C)(C)C(=O)n1nccc1-c1ccccc1
CC(C)(C)C(=O)N1CCOCC1c1ccccc1
CC(C)(C)C(=O)N1CCC1c1ccccc1
O=C(C1CCOCC1)N1N=CCC1c1ccccc1 |c:10|
CN1CCC(CC1)C(=O)N1N=CCC1c1ccccc1 |c:11|
O=C(C1CCN(CC1)C(=O)c1cocn1)N1N=CCC1c1ccccc1 |c:18|
O=C(C1CCN(CC1)c1ccncn1)N1N=CC[C@H]1c1ccccc1 |r,c:17|
C[C@@H]1C=NN([C@@H]1c1ccccc1)C(=O)C(C)(C)C |r,c:2|
CC(C)(C)C(=O)N1N=CCC1c1ccc(cc1)S(C)(=O)=O |c:7|
O=C(C1CCN(CC1)C(=O)c1cscn1)N1N=CC[C@H]1c1ccccc1 |r,c:18|
CCC(=O)N1CCC(CC1)C(=O)N1N=CCC1c1ccccc1 |c:14|
Oc1ccc(cc1)-c1cc2cccnc2[nH]1
CC(C)S(=O)(=O)c1ccc2nccc(Nc3ccc4ncsc4c3)c2c1
COc1ccc2N(C)C(=O)[C@H](CCc2c1)NC(=O)c1nc2CC[C@@H](c3ccccc3)n2n1 |r|
CC(=O)Nc1nc2ccc(cc2s1)-c1cnc(Cl)c(CC(=O)Cc2ccccc2)c1
CC(=O)Nc1nc2ccc(cc2s1)-c1cnc(C)c(CC(=O)OC2CCCCC2)c1
Cc1ccc(cc1C#Cc2cnc3n2nccc3)C(=O)Nc4ccc(c(c4)C(F)(F)F)CN5CCN(CC5)C
Cn1cc(-c2ccc3N(CCc3c2F)C(=O)Cc2cccc(n2)C(F)(F)F)c2c(N)ncnc12
c1ccc(cc1)[C@H](C(=O)Nc2ccc(cc2)F)OC(=O)c3c(nccn3)N
Cc1cc(-c2cnc(N)c3c(csc23)-c2ccc3scnc3c2)n(C)n1
CNC(=O)c1ccc2n(cnc2c1)-c1ccc(CC(=O)OC(C)(C)C)cc1
CC(C)(C)c1nc(c(s1)c2ccnc(n2)N)c3cccc(c3F)NS(=O)(=O)c4c(cccc4F)F
Cc1ccc(Oc2ccnc3cc(ccc23)-c2cnn(c2)C2CCCCC2)cc1
Cc1ccc(O)cc1Nc1ccnc2cc(ccc12)-c1ccccn1
Cc1ccc(CCCCN2C(=O)N[C@H](Cc3c[nH]c4c(Cl)cccc34)C2=O)cc1C#Cc1cnc2cccnn12 |r|
Cn1cc(-c2ccc3N(CCc3c2)C(=O)Cc2cccc(c2)C(F)(F)F)c2c(N)ncnc12
COc1cc(O)c2C(=O)CC(O)(Oc2c1)c1ccc(OCc2ccccc2)cc1
CN(C)c1ccc(cc1)C(=O)Nc1cccc(NC(=O)COc2ccc3c(c2)occc3=O)c1
Cc1cccc(NC(=O)Nc2cc(Oc3ccc4nc(NC(=O)C5CC5)sc4c3)ccc2F)c1
Fc1ccc(Oc2ccc3nc(NC(=O)C4CC4)sc3c2)cc1NC(=O)Cc1ccc(F)c(c1)C(F)(F)F
Fc1ccc(Oc2ccc3nc(NC(=O)C4CC4)sc3c2)cc1NC(=O)Cc1cccc(n1)C(F)(F)F
c1cc(cc(c1)C(F)(F)F)CC(=O)Nc2cc(ccc2F)Oc3ccc4c(c3C#N)sc(n4)NC(=O)C5CC5
Fc1ccc(Oc2ccc3nc(NC(=O)C4CC4)sc3c2)cc1NC(=O)Cc1cccc(c1F)C(F)(F)F
Cc1cccc(CC(=O)Nc2cc(Oc3ccc4nc(NC(=O)C5CC5)sc4c3)ccc2F)c1
COc1cccc(CC(=O)Nc2cc(Oc3ccc4nc(NC(=O)C5CC5)sc4c3)ccc2F)c1
Fc1ccc(Oc2ccc3nc(NC(=O)C4CC4)sc3c2)cc1NC(=O)Cc1cccc(c1)C#N
Fc1ccc(Oc2ccc3nc(NC(=O)C4CC4)sc3c2)cc1NC(=O)Cc1ccc2OCOc2c1
Cn1cc(CC(=O)Nc2cc(Oc3ccc4nc(NC(=O)C5CC5)sc4c3)ccc2F)c2ccccc12
CCOC(=O)c1cccc(NC(=O)Nc2cc(Oc3ccc4nc(NC(=O)C5CC5)sc4c3)ccc2F)c1
CC(=O)c1cccc(NC(=O)Nc2cc(Oc3ccc4nc(NC(=O)C5CC5)sc4c3)ccc2F)c1
COc1cccc(NC(=O)Nc2cc(Oc3ccc4nc(NC(=O)C5CC5)sc4c3)ccc2F)c1
Cc1ccc(CC(=O)Nc2cc(Oc3ccc4nc(NC(=O)C5CC5)sc4c3)ccc2F)cc1C
Fc1ccc(Oc2ccc3nc(NC(=O)C4CC4)sc3c2)cc1NC(=O)Cc1cccc(OC(F)(F)F)c1
Fc1ccc(Oc2ccc3nc(NC(=O)C4CC4)sc3c2)cc1NC(=O)CCc1cccc(c1)C(F)(F)F
Fc1ccc(Oc2ccc3nc(NC(=O)C4CC4)sc3c2)cc1NC(=O)Nc1cccc(Br)c1
Fc1ccc(Oc2ccc3nc(NC(=O)C4CC4)sc3c2)cc1NC(=O)Cc1cccc(c1)C(F)(F)F
[O-][N+](=O)c1cccc(CC(=O)Nc2cc(Oc3ccc4nc(NC(=O)C5CC5)sc4c3)ccc2F)c1
CN1c2ccccc2OC[C@H](NC(=O)c2nnn3CCC(Cc23)C(F)(F)C(F)(F)F)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2nnc3ccc(nn23)C(F)(F)F)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2n[nH]c3ncc(cc23)C(F)(F)F)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2n[nH]c3CCC(C)(C)Cc23)C1=O |r|
C[C@H]1CCc2[nH]nc(C(=O)N[C@H]3COc4ccccc4N(C)C3=O)c2C1 |r|
CN1c2ccccc2OC[C@H](NC(=O)c2n[nH]c3CCC4CC4c23)C1=O |r|
C[C@@H]1CCc2[nH]nc(C(=O)N[C@H]3COc4ccccc4N(C)C3=O)c2C1 |r|
CC(C)c1cnc2[nH]nc(C(=O)N[C@H]3COc4ccccc4N(C)C3=O)c2c1 |r|
CN1c2ccccc2OC[C@H](NC(=O)c2n[nH]c3CCC(Cc23)n2cccn2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2n[nH]c3CC[C@H](Cc23)C(F)(F)F)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2n[nH]c3CC4(CC4)CCc23)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2n[nH]c3ncc(cc23)C(F)(F)C(F)(F)F)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2n[nH]c3ccc(cc23)C(F)(F)F)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2n[nH]c3CCC(Cc23)c2ccccc2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2nnc3ccc(nn23)C(F)(F)C(F)(F)F)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2ncn3ccc(cc23)C(F)(F)F)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2n[nH]c3CC[C@H](Cc23)C(C)(C)C)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2n[nH]c3CC4CC4Cc23)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2nnc[nH]2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2nnn3CC[C@H](Cc23)C(F)(F)F)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2nn(C)c3CC[C@H](Cc23)C(F)(F)F)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2n[nH]c3CCCCc23)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2n[nH]c3CC(C)(C)CCc23)C1=O |r|
CCCCNc1nc2ccc(cc2[nH]1)[N+]([O-])=O
CCCNc1nc2ccc(cc2[nH]1)[N+]([O-])=O
CC(C)Nc1nc2ccc(cc2[nH]1)[N+]([O-])=O
CC(C)CNc1nc2ccc(cc2[nH]1)[N+]([O-])=O
[O-][N+](=O)c1ccc2nc(NC3CCCCC3)[nH]c2c1
[O-][N+](=O)c1ccc2nc(Nc3ccccc3)[nH]c2c1
CCCCNc1nc2cccc(C(=O)OC)c2[nH]1
COC(=O)c1cccc2nc(NC3CCCCC3)[nH]c12
Clc1ccc2nc(NC3CCCCC3)[nH]c2c1
CCCCNc1nc2cc(cc(Br)c2[nH]1)C(F)(F)F
CCCCNc1nc2ccc(cc2s1)[N+]([O-])=O
CCCCNc1nc2cc(ccc2s1)[N+]([O-])=O
O=S1(=O)CC2(OCCO2)c2cc3nccc(Nc4ccc5scnc5c4)c3cc12
CC1(C)CC1C(=O)Nc1nc2ccc(Oc3ccc(F)c(NC(=O)Cc4cccc(c4)C(F)(F)F)c3)cc2s1
CC1(C)C[C@H]1C(=O)Nc1nc2ccc(Oc3ccc(F)c(NC(=O)Cc4cccc(c4)C(F)(F)F)c3)cc2s1 |r|
CC1(C)C[C@@H]1C(=O)Nc1nc2ccc(Oc3ccc(F)c(NC(=O)Cc4cccc(c4)C(F)(F)F)c3)cc2s1 |r|
Fc1cc(F)cc(c1)[C@@H]1CC=NN1C(=O)N1CC(C1)C(=O)c1ccccc1 |r,c:11|
Fc1cc(F)cc(c1)[C@@H]1CC=NN1C(=O)N1CC(C1)Oc1ccccc1F |r,c:11|
Fc1cc(F)cc(c1)[C@@H]1CC=NN1C(=O)N1CC(C1)Oc1ccccc1 |r,c:11|
Fc1cc(F)cc(c1)[C@@H]1CC=NN1C(=O)N1CC(C1)Sc1ccc(Br)cc1 |r,c:11|
C[C@H]1[C@H](CN1C(=O)N1N=CC[C@H]1c1ccc(Cl)cc1)Oc1ccc(F)cc1 |r,c:9|
O=C(N1CC(C1)Oc1ccccc1)N1N=CC[C@H]1c1ccccc1 |r,c:16|
Cc1ncc(cc1NC(=O)OC1CCOCC1)-c1ccc2nc(NC(=O)C3CC3)sc2c1
Fc1ccc(Oc2cc3nc(NC(=O)C4CC4)sc3cc2F)cc1NC(=O)Cc1cccc(c1)C(F)(F)F
Fc1ccc(Oc2cc3nc(NC(=O)C4CC4)sc3cc2F)cc1NC(=O)Cc1cccc(OC(F)(F)F)c1
Fc1ccc(Oc2cc3nc(NC(=O)C4CCOC4)sc3cc2F)cc1NC(=O)Cc1cccc(OC(F)(F)F)c1
Fc1ccc(Oc2cc3nc(NC(=O)C4CC(=O)C4)sc3cc2F)cc1NC(=O)Cc1cccc(OC(F)(F)F)c1
Fc1ccc(Oc2cc3nc(NC(=O)C4CCC(=O)C4)sc3cc2F)cc1NC(=O)Cc1cccc(OC(F)(F)F)c1
Fc1ccc(Oc2cc3nc(NC(=O)C4CCC(=O)CC4)sc3cc2F)cc1NC(=O)Cc1cccc(OC(F)(F)F)c1
CC1(C)CC1C(=O)Nc1nc2cc(Oc3ccc(F)c(NC(=O)Cc4cccc(OC(F)(F)F)c4)c3)c(F)cc2s1
FC1CC1C(=O)Nc1nc2cc(Oc3ccc(F)c(NC(=O)Cc4cccc(OC(F)(F)F)c4)c3)c(F)cc2s1
Cc1ccc(-c2cn([C@@H]3CC[C@H](N)CC3)c3ncnc(N)c23)c(F)c1 |r,wU:8.7,11.11,(2.17,7.19,;1.77,5.71,;.28,5.31,;-.11,3.82,;.97,2.74,;.58,1.25,;1.48,0,;.58,-1.24,;.97,-2.73,;-.11,-3.82,;.28,-5.31,;1.77,-5.71,;2.17,-7.19,;2.86,-4.62,;2.46,-3.13,;-.89,-.77,;-2.22,-1.54,;-3.56,-.77,;-3.56,.77,;-2.22,1.54,;-2.22,3.08,;-.89,.77,;2.47,3.14,;3.56,2.05,;2.86,4.62,)|
O=C(N1CCC2(CN(Cc3ccccc3)C2=O)CC1)c1ccccc1
CN1c2ccccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=S |r|
CN1c2ccccc2OC[C@H](NC(=O)c2nc(Cc3ccccc3)n(C)n2)C1=S |r|
CCn1nc(nc1Cc1ccccc1)C(=O)N[C@H]1COc2ccccc2N(C)C1=S |r|
CN1c2ccccc2OC[C@H](NC(=O)c2nc(Cc3ccccc3)n(CCF)n2)C1=S |r|
CN1c2ccccc2OC[C@H](NC(=O)c2nc(Cc3ccccc3)n(CC(F)(F)F)n2)C1=S |r|
CN1c2ccccc2OC[C@H](NC(=O)c2nc(Cc3ccccc3)n(n2)C2CCC2)C1=S |r|
CN1c2ccccc2OC[C@H](NC(=O)c2nc(Cc3ccccc3)n(n2)C2CCOC2)C1=S |r|
CNC(=O)c1cc(Oc2ccc(NC(=O)Nc3cc(nn3-c3cccc4ncccc34)C(C)(C)C)c(F)c2)ccn1
CN1C(=O)N(Cc2cnc(Nc3ccc(C)nc3)nc12)c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C
CN(c1ccc(cc1)NC(=O)Nc2ccc(cc2)OC(F)(F)F)c3ccnc(n3)Nc4cccc(c4)S(=O)(=O)N
CN(c1ccc(cc1)NC(=O)Nc2cc(ccc2F)C(F)(F)F)c3ccnc(n3)Nc4cccc(c4)S(=O)(=O)N
Fc1ccc(Oc2ccc3nc(NC(=O)C4CC4)sc3c2)cc1NC(=O)Cc1cccc(Br)c1
Fc1ccc(Oc2cc3sc(NC(=O)C4CC4)nc3cc2F)cc1NC(=O)Cc1cccc(c1)C(F)(F)F
[O-][N+](=O)c1nn(Cc2cc(F)ccc2F)cc1Br
COc1cc2c(ccnc2cc1OCCCN3CCOCC3)Oc4ccc(cc4F)NC(=O)C5(CC5)C(=O)Nc6ccc(cc6)F
Cc1[nH]c(CC2C(=O)Nc3ccc(F)cc23)c(C)c1C(=O)NC[C@@H](O)CN1CCOCC1 |r|
CN(C)CC(=O)N1CCC(CC1)c1ccc(NC(=O)c2nc(c[nH]2)C#N)c(c1)C1=CCCCC1 |t:31|
Cc1cccc(CC(=O)N2CCc3c2ccc(-c2cn(C)c4ncnc(N)c24)c3F)n1
CN1c2cc(ccc2OC[C@H](NC(=O)c2nc(Cc3ccccc3)n[nH]2)C1=O)C#CC1CC1 |r|
O=C(N1CCOc2ccccc2C1)c1cnn(Cc2ccccc2)c1
[H][C@@]12CCc3ccc(OC)cc3C1=CN([C@@H]2c1ccc(OC)c(F)c1)C(=O)CO |r,c:14|
C[C@@H](c1c(cccc1Cl)F)NC(=O)c2ccc(n2C)C#N
CN1c2cnc(cc2CC[C@@H](C1=O)NC(=O)c3nc4n(n3)[C@@H](CC4)c5ccccc5)OC
COC(=O)c1cccc(c1)C#Cc1ccc2OC[C@H](NC(=O)c3n[nH]c(Cc4ccccc4)n3)C(=S)N(C)c2c1 |r|
COC(=O)c1ccc(cc1)C#Cc1ccc2OC[C@H](NC(=O)c3n[nH]c(Cc4ccccc4)n3)C(=S)N(C)c2c1 |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=S)C#Cc1ccccc1C#N |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=S)C#Cc1cccc(c1)C#N |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=S)C#Cc1ccc(cc1)C#N |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=S)C#Cc1cccc(c1)[N+]([O-])=O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=S)C#Cc1ccc(cc1)[N+]([O-])=O |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=S)C#C |r|
CN1c2cc(ccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=S)C#CC1CC1 |r|
CN1c2ccccc2OC[C@H](NC(=O)c2cc3cccc(-c4ccccc4)c3[nH]2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2cc3cccc(-c4ccccc4F)c3[nH]2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2cc3cccc(-c4ccccc4C)c3[nH]2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2cc3cccc(-c4cccc(F)c4F)c3[nH]2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2cc3cccc(-c4ccc(F)cc4F)c3[nH]2)C1=O |r|
CN1c2ccccc2OC[C@H](NC(=O)c2cc3cccc(-c4cc(F)ccc4F)c3[nH]2)C1=O |r|
Nc1cc(ncn1)N1CCC(CC1)C(=O)N1OCC[C@H]1c1cc(F)cc(F)c1 |r|
Cc1c(F)cc(cc1C#N)[C@@H]1CCON1C(=O)C1CCN(CC1)c1cc(N)ncn1 |r|
Nc1cc(ncn1)N1CCC(CC1)C(=O)N1OCC[C@H]1c1cc(F)cc(c1)C#N |r|
COc1ncnc(N2CCC(CC2)C(=O)N2OCC[C@H]2c2cc(F)cc(c2)C#N)c1F |r|
COc1cc(ncn1)N1CCC(CC1)C(=O)N1OCC[C@H]1c1cc(F)c(C)c(c1)C#N |r|
COc1cc(ncn1)N1CCC(CC1)C(=O)N1OCC[C@H]1c1cc(F)cc(Cl)c1 |r|
CNC(=O)c1n[nH]c2cc(ccc12)-c1ccc(nc1)C(=O)NCc1ccc(OCCC2CC2)cc1
CC(NCC(=O)Nc1cccc(n1)-c1cc(C(=O)NCc2cccc(F)c2)n(C)c1)c1ccccc1F
Cc1cc(Oc2ccc(F)c(n2)C(=O)NCc2ccc(F)cc2)cc(c1)C(=O)NCc1ccc(Br)s1
CC(=O)Nc1cn2cc(ccc2n1)-c1ccc(CNC(=O)c2cc(F)ccc2OCC2CCCC2)nc1
CCOc1ccccc1CNCC(=O)c1cn2ccc(cc2n1)-c1ccn2nc(NC(=O)C(C)C)nc2c1
CC(NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)C3CC3)cc2n1)c1ccc(F)cc1
CC(NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)C3CC3)cc2n1)c1ccccc1
Fc1ccc(cc1NC(=O)Cc1cccc(OC(F)(F)F)c1)-c1ccc2nc(NC(=O)C3CC3)sc2c1
Fc1c(NC(=O)Cc2cccc(OC(F)(F)F)c2)cccc1-c1ccc2nc(NC(=O)C3CC3)sc2c1
CC(C)C(=O)NC1CCC(CC1)C(=O)Nc1nc2cc(F)c(Oc3ccc(F)c(NC(=O)Cc4cccc(c4)C(F)(F)F)c3)cc2s1 |(-12.06,-2.87,;-13.6,-2.87,;-14.37,-4.21,;-14.37,-1.54,;-15.91,-1.54,;-13.6,-.21,;-12.06,-.21,;-11.29,1.13,;-9.75,1.13,;-8.98,-.21,;-9.75,-1.54,;-11.29,-1.54,;-7.44,-.21,;-6.67,-1.54,;-6.67,1.13,;-5.13,1.13,;-4.23,-.12,;-2.76,.36,;-1.43,-.41,;-.09,.36,;1.24,-.41,;-.09,1.9,;1.24,2.67,;2.57,1.9,;2.57,.36,;3.91,-.41,;5.24,.36,;6.57,-.41,;5.24,1.9,;6.57,2.67,;7.91,1.9,;7.91,.36,;9.24,2.67,;10.58,1.9,;10.58,.36,;11.91,-.41,;13.24,.36,;13.24,1.9,;11.91,2.67,;14.58,2.67,;15.91,3.44,;15.91,1.9,;14.58,4.21,;3.91,2.67,;-1.43,2.67,;-2.76,1.9,;-4.23,2.37,)|
CCCCC(=O)NC1CCC(CC1)C(=O)Nc1nc2cc(F)c(Oc3ccc(F)c(NC(=O)Cc4cccc(c4)C(F)(F)F)c3)cc2s1 |(-9.75,-4.21,;-11.29,-4.21,;-12.06,-2.87,;-13.6,-2.87,;-14.37,-1.54,;-15.91,-1.54,;-13.6,-.21,;-12.06,-.21,;-11.29,1.13,;-9.75,1.13,;-8.98,-.21,;-9.75,-1.54,;-11.29,-1.54,;-7.44,-.21,;-6.67,-1.54,;-6.67,1.13,;-5.13,1.13,;-4.23,-.12,;-2.76,.36,;-1.43,-.41,;-.09,.36,;1.24,-.41,;-.09,1.9,;1.24,2.67,;2.57,1.9,;2.57,.36,;3.91,-.41,;5.24,.36,;6.57,-.41,;5.24,1.9,;6.57,2.67,;7.91,1.9,;7.91,.36,;9.24,2.67,;10.58,1.9,;10.58,.36,;11.91,-.41,;13.24,.36,;13.24,1.9,;11.91,2.67,;14.58,2.67,;15.91,3.44,;15.91,1.9,;14.58,4.21,;3.91,2.67,;-1.43,2.67,;-2.76,1.9,;-4.23,2.37,)|
Fc1ccc(Oc2cc3sc(NC(=O)C4CCC(CC4)NC(=O)CCCl)nc3cc2F)cc1NC(=O)Cc1cccc(c1)C(F)(F)F |(6.57,-.41,;5.24,.36,;3.91,-.41,;2.57,.36,;2.57,1.9,;1.24,2.67,;-.09,1.9,;-1.43,2.67,;-2.76,1.9,;-4.23,2.37,;-5.13,1.13,;-6.67,1.13,;-7.44,-.21,;-6.67,-1.54,;-8.98,-.21,;-9.75,1.13,;-11.29,1.13,;-12.06,-.21,;-11.29,-1.54,;-9.75,-1.54,;-13.6,-.21,;-14.37,-1.54,;-15.91,-1.54,;-13.6,-2.87,;-12.06,-2.87,;-11.29,-4.21,;-4.23,-.12,;-2.76,.36,;-1.43,-.41,;-.09,.36,;1.24,-.41,;3.91,2.67,;5.24,1.9,;6.57,2.67,;7.91,1.9,;7.91,.36,;9.24,2.67,;10.58,1.9,;10.58,.36,;11.91,-.41,;13.24,.36,;13.24,1.9,;11.91,2.67,;14.58,2.67,;15.91,3.44,;15.91,1.9,;14.58,4.21,)|
COCC(=O)NC1CCC(CC1)C(=O)Nc1nc2cc(F)c(Oc3ccc(F)c(NC(=O)Cc4cccc(c4)C(F)(F)F)c3)cc2s1 |(-11.29,-4.21,;-12.06,-2.87,;-13.6,-2.87,;-14.37,-1.54,;-15.91,-1.54,;-13.6,-.21,;-12.06,-.21,;-11.29,1.13,;-9.75,1.13,;-8.98,-.21,;-9.75,-1.54,;-11.29,-1.54,;-7.44,-.21,;-6.67,-1.54,;-6.67,1.13,;-5.13,1.13,;-4.23,-.12,;-2.76,.36,;-1.43,-.41,;-.09,.36,;1.24,-.41,;-.09,1.9,;1.24,2.67,;2.57,1.9,;2.57,.36,;3.91,-.41,;5.24,.36,;6.57,-.41,;5.24,1.9,;6.57,2.67,;7.91,1.9,;7.91,.36,;9.24,2.67,;10.58,1.9,;10.58,.36,;11.91,-.41,;13.24,.36,;13.24,1.9,;11.91,2.67,;14.58,2.67,;15.91,3.44,;15.91,1.9,;14.58,4.21,;3.91,2.67,;-1.43,2.67,;-2.76,1.9,;-4.23,2.37,)|
CCOCC(=O)NC1CCC(CC1)C(=O)Nc1nc2cc(F)c(Oc3ccc(F)c(NC(=O)Cc4cccc(c4)C(F)(F)F)c3)cc2s1 |(-9.75,-4.21,;-11.29,-4.21,;-12.06,-2.87,;-13.6,-2.87,;-14.37,-1.54,;-15.91,-1.54,;-13.6,-.21,;-12.06,-.21,;-11.29,1.13,;-9.75,1.13,;-8.98,-.21,;-9.75,-1.54,;-11.29,-1.54,;-7.44,-.21,;-6.67,-1.54,;-6.67,1.13,;-5.13,1.13,;-4.23,-.12,;-2.76,.36,;-1.43,-.41,;-.09,.36,;1.24,-.41,;-.09,1.9,;1.24,2.67,;2.57,1.9,;2.57,.36,;3.91,-.41,;5.24,.36,;6.57,-.41,;5.24,1.9,;6.57,2.67,;7.91,1.9,;7.91,.36,;9.24,2.67,;10.58,1.9,;10.58,.36,;11.91,-.41,;13.24,.36,;13.24,1.9,;11.91,2.67,;14.58,2.67,;15.91,3.44,;15.91,1.9,;14.58,4.21,;3.91,2.67,;-1.43,2.67,;-2.76,1.9,;-4.23,2.37,)|
Fc1ccc(Oc2cc3sc(NC(=O)C4CCC(CC4)NC(=O)c4cccs4)nc3cc2F)cc1NC(=O)Cc1cccc(c1)C(F)(F)F |(6.57,.14,;5.24,.91,;3.91,.14,;2.57,.91,;2.57,2.45,;1.24,3.22,;-.09,2.45,;-1.43,3.22,;-2.76,2.45,;-4.23,2.92,;-5.13,1.68,;-6.67,1.68,;-7.44,.34,;-6.67,-.99,;-8.98,.34,;-9.75,1.68,;-11.29,1.68,;-12.06,.34,;-11.29,-.99,;-9.75,-.99,;-13.6,.34,;-14.37,-.99,;-15.91,-.99,;-13.6,-2.32,;-12.07,-2.48,;-11.75,-3.99,;-13.08,-4.76,;-14.23,-3.73,;-4.23,.43,;-2.76,.91,;-1.43,.14,;-.09,.91,;1.24,.14,;3.91,3.22,;5.24,2.45,;6.57,3.22,;7.91,2.45,;7.91,.91,;9.24,3.22,;10.58,2.45,;10.58,.91,;11.91,.14,;13.24,.91,;13.24,2.45,;11.91,3.22,;14.58,3.22,;15.91,3.99,;15.91,2.45,;14.58,4.76,)|
CCS(=O)(=O)NC1CCC(CC1)C(=O)Nc1nc2cc(F)c(Oc3ccc(F)c(NC(=O)Cc4cccc(c4)C(F)(F)F)c3)cc2s1 |(-14.4,-4.21,;-13.63,-2.87,;-14.4,-1.54,;-15.49,-.45,;-15.88,-1.94,;-13.63,-.21,;-12.09,-.21,;-11.32,1.13,;-9.78,1.13,;-9.01,-.21,;-9.78,-1.54,;-11.32,-1.54,;-7.47,-.21,;-6.7,-1.54,;-6.7,1.13,;-5.16,1.13,;-4.25,-.12,;-2.79,.36,;-1.45,-.41,;-.12,.36,;1.21,-.41,;-.12,1.9,;1.21,2.67,;2.55,1.9,;2.55,.36,;3.88,-.41,;5.21,.36,;6.55,-.41,;5.21,1.9,;6.55,2.67,;7.88,1.9,;7.88,.36,;9.22,2.67,;10.55,1.9,;10.55,.36,;11.88,-.41,;13.22,.36,;13.22,1.9,;11.88,2.67,;14.55,2.67,;15.88,3.44,;15.88,1.9,;14.55,4.21,;3.88,2.67,;-1.45,2.67,;-2.79,1.9,;-4.25,2.37,)|
Oc1ccc(cc1)-c1cnc2[nH]ccc2c1
Oc1ccc(cc1)-c1cnc2[nH]ccc2n1
N#Cc1ccc(cc1)-c1cnc2[nH]ccc2c1
NC(=O)c1ccc(cc1)-c1cnc2[nH]ccc2c1
O\N=C\c1ccc(cc1)-c1cnc2[nH]ccc2c1
OCc1ccc(cc1)-c1cc2cccnc2[nH]1
OCCc1ccc(cc1)-c1cc2cccnc2[nH]1
Oc1ccccc1-c1cc2cccnc2[nH]1
Oc1cccc(c1)-c1cc2cccnc2[nH]1
Nc1ccc(cc1)-c1cc2cccnc2[nH]1
COc1ccc(cc1)-c1cc2ccc[nH]c2n1
CC(C)(C)Oc1ccc(cc1)-c1cc2cccnc2[nH]1
NC(=O)c1ccc(cc1)-c1cc2cccnc2[nH]1
Oc1ccc(cc1F)-c1cc2cccnc2[nH]1
COc1cc(ccc1O)-c1cc2cccnc2[nH]1
Oc1ccc(cc1Cl)-c1cc2cccnc2[nH]1
Oc1ccc2ccc(cc2c1)-c1cc2cccnc2[nH]1
O(c1ccccc1)c1ccc(cc1)-c1cc2cccnc2[nH]1
Oc1ccc(cc1)-c1ccc(cc1)-c1cc2cccnc2[nH]1
c1nc2ccc(cc2s1)-c1cc2cccnc2[nH]1
O\N=C\c1ccc(cc1)-c1cc2cccnc2[nH]1
C1COc2ccc(cc2C1)-c1cc2cccnc2[nH]1
CNC(=O)c1ccc(cc1)-c1cc2cccnc2[nH]1
CCNC(=O)c1ccc(cc1)-c1cc2cccnc2[nH]1
CCCNC(=O)c1ccc(cc1)-c1cc2cccnc2[nH]1
CC(C)NC(=O)c1ccc(cc1)-c1cc2cccnc2[nH]1
CC(C)(C)NC(=O)c1ccc(cc1)-c1cc2cccnc2[nH]1
CC(C)N(C(C)C)C(=O)c1ccc(cc1)-c1cc2cccnc2[nH]1
O=C(N1CCCC1)c1ccc(cc1)-c1cc2cccnc2[nH]1
O=C(N1CCCCC1)c1ccc(cc1)-c1cc2cccnc2[nH]1
O=C(N1CCNCC1)c1ccc(cc1)-c1cc2cccnc2[nH]1
O=C(N1CCOCC1)c1ccc(cc1)-c1cc2cccnc2[nH]1
CN1CCN(CC1)C(=O)c1ccc(cc1)-c1cc2cccnc2[nH]1
O=C(NC1CC1)c1ccc(cc1)-c1cc2cccnc2[nH]1
CN1C(=O)[C@@H](NC(=O)c2ccc3[nH]cc(-c4ccccc4)c3c2)COc2ccccc21
CN1C(=O)[C@@H](NC(=O)c2ccc3[nH]cc(-c4ccccc4F)c3c2)COc2ccccc21
CN1C(=O)[C@@H](NC(=O)c2ccc3[nH]cc(-c4cccc(F)c4)c3c2)COc2ccccc21
Cc1ccccc1-c1c[nH]c2ccc(C(=O)N[C@H]3COc4ccccc4N(C)C3=O)cc12
Cc1ccc(-c2c[nH]c3ccc(C(=O)N[C@H]4COc5ccccc5N(C)C4=O)cc23)cc1
CN1C(=O)[C@@H](NC(=O)c2ccc3[nH]cc(-c4ccccc4C(F)(F)F)c3c2)COc2ccccc21
COc1cccc(-c2c[nH]c3ccc(C(=O)N[C@H]4COc5ccccc5N(C)C4=O)cc23)c1
CN1C(=O)[C@@H](NC(=O)c2ccc3[nH]cc(-c4ccc(-c5ccccc5)cc4)c3c2)COc2ccccc21
CN1C(=O)[C@@H](NC(=O)c2ccc3[nH]cc(-c4cccc(F)c4F)c3c2)COc2ccccc21
CN1C(=O)[C@@H](NC(=O)c2ccc3[nH]cc(-c4ccc(F)cc4F)c3c2)COc2ccccc21
CN1C(=O)[C@@H](NC(=O)c2ccc3[nH]cc(-c4cc(F)ccc4F)c3c2)COc2ccccc21
CN1C(=O)[C@@H](NC(=O)c2ccc3[nH]cc(-c4c(F)cccc4F)c3c2)COc2ccccc21
Cc1cccc(-c2c[nH]c3ccc(C(=O)N[C@H]4COc5ccccc5N(C)C4=O)cc23)c1C
Cc1ccc(-c2c[nH]c3ccc(C(=O)N[C@H]4COc5ccccc5N(C)C4=O)cc23)c(C)c1
Cc1ccc(C)c(-c2c[nH]c3ccc(C(=O)N[C@H]4COc5ccccc5N(C)C4=O)cc23)c1
Cc1ccc(-c2c[nH]c3ccc(C(=O)N[C@H]4COc5ccccc5N(C)C4=O)cc23)cc1C
COc1ccc(-c2c[nH]c3ccc(C(=O)N[C@H]4COc5ccccc5N(C)C4=O)cc23)c(OC)c1
COc1ccc(-c2c[nH]c3ccc(C(=O)N[C@H]4COc5ccccc5N(C)C4=O)cc23)cc1OC
CN1C(=O)[C@@H](NC(=O)c2ccc3[nH]cc(-c4cccc5ccccc45)c3c2)COc2ccccc21
CN1C(=O)N[C@@H](Cc2c[nH]c3c(Cl)cccc23)C1=O
O=C(NC1CCOCC1)c1nsc2ncc(-c3ccc4nc(NC(=O)C5CC5)sc4c3)cc12
Cc1ccc(F)c(NC(=O)Nc2ccc(cc2)-c2cccc3[nH]nc(N)c23)c1
O=C(NCCc1ccccc1Cl)c1cn(-c2ccccc2)nn1
Cc1ccc(CCCCN2C(=O)NC(Cc3c[nH]c4c(Cl)cccc34)C2=O)cc1C#Cc1cnc2cccnn12
CN1C(=O)[C@@H](Cc2c[nH]c3c(Cl)c(F)ccc23)N(C=O)C1=O
O=C(Nc1cn2cc(-c3cnc4c(c3)N(C(=O)OC3CCOCC3)CC4)ccc2n1)C1CC1
Cc1ccc(C(=O)Nc2ccccc2)cc1-c1ccc2nc(NCCN3CCOCC3)ncc2c1
Cc1cc(Nc2cc(N3CCNCC3)nc(Nc3ccc(NC(=O)C4CC4)cc3)n2)n[nH]1
CC(=O)Nc1nc2ccc(cc2s1)-c1cnc(Cl)c(NC(=O)Cc2ccccc2)c1
Cn1cc(-c2ccc3N(CCc3c2)C(=O)Cc2cccc(n2)C(F)(F)F)c2c(N)ncnc12
Cc1cccc(CC(=O)N2CCc3cc(ccc23)-c2cn(C)c3ncnc(N)c23)n1
Cn1cc(-c2ccc3c(c2)CCN3C(=O)Cc2ccc(C(F)(F)F)cn2)c2c(N)ncnc21
CNC(=O)c1cc(Oc2ccc(NC(=O)Nc3cc(nn3-c3ccc4ncccc4c3)C(C)(C)C)c(F)c2)ccn1
COc1cc(CCc2cc(NC(=O)c3ccc(cc3)N3C[C@H](C)N[C@H](C)C3)n[nH]2)cc(OC)c1
NC(=O)c1cccc(-c2ccc3c(c2)CCN3C(=O)Cc2cccc(OC(F)(F)F)c2)c1
NC(=O)c1cncc(-c2ccc3c(c2)CCN3C(=O)Cc2cccc(OC(F)(F)F)c2)c1
NC(=O)c1cc(-c2ccc3c(c2)CCN3C(=O)Cc2cccc(OC(F)(F)F)c2)ccc1N
CCn1cc(-c2ccc3c(c2)CCN3C(=O)Cc2cccc(OC(F)(F)F)c2)c2ncnc(N)c21
CCNc1ncnc(N)c1-c1ccc2c(c1)CCN2C(=O)Cc1cccc(OC(F)(F)F)c1
Nc1nc2cccc(-c3ccc4c(c3)CCN4C(=O)Cc3cccc(OC(F)(F)F)c3)n2n1
CCn1cc(-c2ccc3c(c2)CCN3C(=O)Cc2cccc(OC(F)(F)F)c2)c2c(=O)[nH]cnc21
CCc1nc(-c2ccc3c(c2)CCN3C(=O)Cc2cccc(OC(F)(F)F)c2)c2c(N)nccn12
CCn1cc(-c2ccc3c(c2)CCN3C(=O)Cc2cccc(OC(F)(F)F)c2)c2c(N)n[nH]c(=O)c21
CCn1nc(-c2ccc3c(c2)CCN3C(=O)Cc2cccc(OC(F)(F)F)c2)c2c(N)n[nH]c(=O)c21
CCn1nc(-c2ccc3c(c2)CCN3C(C)=O)c2c(N)n[nH]c(=O)c21
CCn1nc(-c2ccc3c(c2)CCN3C(=O)Cc2ccccc2)c2c(N)n[nH]c(=O)c21
CCn1nc(-c2ccc3c(c2)CCN3C(=O)CC2CCCCC2)c2c(N)n[nH]c(=O)c21
CCn1nc(-c2ccc3c(c2)CCN3C(=O)[C@H](C)c2ccccc2)c2c(N)n[nH]c(=O)c21
CCn1nc(-c2ccc3c(c2)CCN3C(=O)C2(c3ccccc3)CC2)c2c(N)n[nH]c(=O)c21
CCn1nc(-c2ccc3c(c2)CCN3C(=O)CCc2ccccc2)c2c(N)n[nH]c(=O)c21
CCn1nc(-c2ccc3c(c2)CCN3C(=O)Cc2ccc(Oc3ccccc3)cc2)c2c(N)n[nH]c(=O)c21
CCn1nc(-c2ccc3c(c2)CCN3C(=O)Cc2ccc3c(c2)OCO3)c2c(N)n[nH]c(=O)c21
CCn1nc(-c2ccc3c(c2)CCN3C(=O)Cc2ccc(OC(F)(F)F)cc2)c2c(N)n[nH]c(=O)c21
CCn1nc(-c2ccc3c(c2)CCN3C(=O)Cc2cccc(C(F)(F)F)c2)c2c(N)n[nH]c(=O)c21
CCn1nc(-c2ccc3c(c2)CCN3C(=O)Cc2cccc(OC)c2)c2c(N)n[nH]c(=O)c21
CCn1nc(-c2ccc3c(c2)CCN3C(=O)Cc2cccc(F)c2)c2c(N)n[nH]c(=O)c21
CCn1nc(-c2ccc3c(c2)CCN3C(=O)Cc2cc(F)cc(C(F)(F)F)c2)c2c(N)n[nH]c(=O)c21
CCn1nc(-c2ccc3c(c2)CCN3C(=O)Cc2cccc(F)c2F)c2c(N)n[nH]c(=O)c21
CCn1nc(-c2ccc3c(c2)CCN3C(=O)CCc2cccc(OC(F)(F)F)c2)c2c(N)n[nH]c(=O)c21
CCn1nc(-c2ccc3c(c2)CCN3C(=O)CCc2cccc(C(F)(F)F)c2)c2c(N)n[nH]c(=O)c21
CCn1nc(-c2ccc3c(c2)CCN3C(=O)c2cccc(OC(F)(F)F)c2)c2c(N)n[nH]c(=O)c21
CCn1nc(-c2ccc3c(c2)CCN3Cc2cccc(OC(F)(F)F)c2)c2c(N)n[nH]c(=O)c21
Cn1nc(-c2ccc3c(c2)CCN3C(=O)Cc2cccc(OC(F)(F)F)c2)c2c(N)n[nH]c(=O)c21
CC(C)n1nc(-c2ccc3c(c2)CCN3C(=O)Cc2cccc(OC(F)(F)F)c2)c2c(N)n[nH]c(=O)c21
CC(C)Cn1nc(-c2ccc3c(c2)CCN3C(=O)Cc2cccc(OC(F)(F)F)c2)c2c(N)n[nH]c(=O)c21
Nc1n[nH]c(=O)c2c1c(-c1ccc3c(c1)CCN3C(=O)Cc1cccc(OC(F)(F)F)c1)nn2CC(F)F
CCCn1nc(-c2ccc3c(c2)CCN3C(=O)Cc2cccc(OC(F)(F)F)c2)c2c(N)n[nH]c(=O)c21
CCCCn1nc(-c2ccc3c(c2)CCN3C(=O)Cc2cccc(OC(F)(F)F)c2)c2c(N)n[nH]c(=O)c21
CC(C)=CCn1nc(-c2ccc3c(c2)CCN3C(=O)Cc2cccc(OC(F)(F)F)c2)c2c(N)n[nH]c(=O)c21
CC(C)CCn1nc(-c2ccc3c(c2)CCN3C(=O)Cc2cccc(OC(F)(F)F)c2)c2c(N)n[nH]c(=O)c21
Nc1n[nH]c(=O)c2c1c(-c1ccc3c(c1)CCN3C(=O)Cc1cccc(OC(F)(F)F)c1)nn2CCC1CC1
Nc1n[nH]c(=O)c2c1c(-c1ccc3c(c1)CCN3C(=O)Cc1cccc(OC(F)(F)F)c1)nn2CC1CC1
CC1(Cn2nc(-c3ccc4c(c3)CCN4C(=O)Cc3cccc(OC(F)(F)F)c3)c3c(N)n[nH]c(=O)c32)CC1
Nc1n[nH]c(=O)c2c1c(-c1ccc3c(c1)CCN3C(=O)Cc1cccc(OC(F)(F)F)c1)nn2CC1CCC1
Nc1n[nH]c(=O)c2c1c(-c1ccc3c(c1)CCN3C(=O)Cc1cccc(OC(F)(F)F)c1)nn2CC1CCCC1
Nc1n[nH]c(=O)c2c1c(-c1ccc3c(c1)CCN3C(=O)Cc1cccc(OC(F)(F)F)c1)nn2CCC1CCCC1
Nc1n[nH]c(=O)c2c1c(-c1ccc3c(c1)CCN3C(=O)Cc1cccc(OC(F)(F)F)c1)nn2CCC1CCCCC1
Nc1n[nH]c(=O)c2c1c(-c1ccc3c(c1)CCN3C(=O)Cc1cccc(OC(F)(F)F)c1)nn2CC1COC1
CC1(Cn2nc(-c3ccc4c(c3)CCN4C(=O)Cc3cccc(OC(F)(F)F)c3)c3c(N)n[nH]c(=O)c32)COC1
CCC1(Cn2nc(-c3ccc4c(c3)CCN4C(=O)Cc3cccc(OC(F)(F)F)c3)c3c(N)n[nH]c(=O)c32)COC1
Nc1n[nH]c(=O)c2c1c(-c1ccc3c(c1)CCN3C(=O)Cc1cccc(OC(F)(F)F)c1)nn2CCC1CNC1
COCCn1nc(-c2ccc3c(c2)CCN3C(=O)Cc2cccc(OC(F)(F)F)c2)c2c(N)n[nH]c(=O)c21
Nc1n[nH]c(=O)c2c1c(-c1ccc3c(c1)CCN3C(=O)Cc1cccc(OC(F)(F)F)c1)nn2CCN1CCCC1
Nc1n[nH]c(=O)c2c1c(-c1ccc3c(c1)CCN3C(=O)Cc1cccc(OC(F)(F)F)c1)nn2Cc1ccccc1
CC(C)(C)c1ccc(Cn2nc(-c3ccc4c(c3)CCN4C(=O)Cc3cccc(OC(F)(F)F)c3)c3c(N)n[nH]c(=O)c32)cc1
Nc1n[nH]c(=O)c2c1c(-c1ccc3c(c1)CCN3C(=O)Cc1cccc(OC(F)(F)F)c1)nn2Cc1ccc(F)cc1
CC(C)Cn1cc(-c2ccc3c(c2)CCN3C(=O)Cc2cccc(OC(F)(F)F)c2)c2c(N)n[nH]c(=O)c21
Nc1n[nH]c(=O)c2c1c(-c1ccc3c(c1)CCN3C(=O)Cc1cccc(OC(F)(F)F)c1)cn2CC1CC1
CC1(Cn2cc(-c3ccc4c(c3)CCN4C(=O)Cc3cccc(OC(F)(F)F)c3)c3c(N)n[nH]c(=O)c32)COC1
Nc1n[nH]c(=O)c2c1c(-c1ccc3c(c1)CCN3C(=O)Cc1cccc(C(F)(F)F)c1)cn2CC1CC1
CC1(Cn2cc(-c3ccc4c(c3)CCN4C(=O)Cc3cccc(C(F)(F)F)c3)c3c(N)n[nH]c(=O)c32)COC1
COCC(=O)Nc1nc2cc(-c3ccc4c(c3)c(C(=O)N[C@@H](C)c3cccc(F)c3)cn4C)ccn2n1
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccc2c(NC(=O)C3CC3)n[nH]c2c1)c1cccc(F)c1 |r|
C[C@H](NC(=O)c1cn(C)c2ccc(-c3ccc4c(C(=O)NC5CC5)n[nH]c4c3)cc12)c1cccc(F)c1
CC(C)Cn1cc(C(=O)N[C@@H](C)c2cccc(F)c2)c2cc(-c3ccn4nc(NC(=O)C5CC5)nc4c3)ccc21
CN1C(=O)NC(Cc2c[nH]c3c(F)cccc23)C1=O
Cn1cc(-c2cccc(NC(=O)c3cc4c(nc3O[C@H]3C[C@@H](O)C3)OC(C)(C)C4)n2)cn1
CC(C)S(=O)(=O)c1ccc2c(c1)c(ccn2)Nc3ccc4c(c3)ncs4
C=Cc1cc2c(Nc3ccc4scnc4c3)ncnc2cn1
Clc1ccc(/C=C/c2cc3c(Nc4ccc5scnc5c4)ncnc3cn2)cc1
Cc1ccc(Nc2ncnc3cnc(/C=C/c4ccc(Cl)cc4)cc23)cn1
Clc1cc2ncnc(Nc3ccc4scnc4c3)c2cc1-c1cccs1
Cc1ncc(-c2cc3c(Nc4ccc5scnc5c4)ncnc3cc2Cl)s1
Cn1cccc1-c1cc2c(Nc3ccc4scnc4c3)ncnc2cc1Cl
Cn1ccnc1-c1cc2c(Nc3ccc4scnc4c3)ncnc2cc1Cl
Cn1cnc(-c2cc3c(Nc4ccc5scnc5c4)ncnc3cc2Cl)c1
Cc1csc(-c2cc3c(Nc4ccc5scnc5c4)ncnc3cc2Cl)n1
Cn1cc(-c2cc3c(Nc4ccc5scnc5c4)ncnc3cc2Cl)cn1
Cn1cncc1-c1cc2c(Nc3ccc4scnc4c3)ncnc2cc1Cl
Cc1ncc(-c2cc3c(Nc4ccc5scnc5c4)ncnc3cc2Cl)n1C
Cn1nccc1-c1cc2c(Nc3ccc4scnc4c3)ncnc2cc1Cl
Cc1nc(-c2cc3c(Nc4ccc5scnc5c4)ncnc3cc2Cl)sc1C
Cn1nc(C(F)(F)F)cc1-c1cc2c(Nc3ccc4scnc4c3)ncnc2cc1Cl
Cc1ccsc1-c1cc2c(Nc3ccc4scnc4c3)ncnc2cc1Cl
Clc1cc2ncnc(Nc3ccc4scnc4c3)c2cc1-c1cc[nH]n1
COc1cccc(-c2cc3c(Nc4ccc5scnc5c4)ncnc3cc2Cl)n1
Clc1cc2ncnc(Nc3ccc4scnc4c3)c2cc1-c1ccccc1
Cc1cscc1-c1cc2c(Nc3ccc4scnc4c3)ncnc2cc1Cl
c1csc(-c2ccc3ncnc(Nc4ccc5scnc5c4)c3c2)c1
Cc1ncc(-c2ccc3ncnc(Nc4ccc5scnc5c4)c3c2)s1
Cn1cccc1-c1ccc2ncnc(Nc3ccc4scnc4c3)c2c1
Cn1ccnc1-c1ccc2ncnc(Nc3ccc4scnc4c3)c2c1
Cn1cnc(-c2ccc3ncnc(Nc4ccc5scnc5c4)c3c2)c1
Cc1csc(-c2ccc3ncnc(Nc4ccc5scnc5c4)c3c2)n1
Cn1cc(-c2ccc3ncnc(Nc4ccc5scnc5c4)c3c2)cn1
Cn1cncc1-c1ccc2ncnc(Nc3ccc4scnc4c3)c2c1
Cc1ncc(-c2ccc3ncnc(Nc4ccc5scnc5c4)c3c2)n1C
Cc1nc(-c2ccc3ncnc(Nc4ccc5scnc5c4)c3c2)sc1C
Cc1ccsc1-c1ccc2ncnc(Nc3ccc4scnc4c3)c2c1
c1nc(Nc2ccc3scnc3c2)c2cc(-c3cc[nH]n3)ccc2n1
COc1cccc(-c2ccc3ncnc(Nc4ccc5scnc5c4)c3c2)n1
c1ccc(-c2ccc3ncnc(Nc4ccc5scnc5c4)c3c2)cc1
Cc1cscc1-c1ccc2ncnc(Nc3ccc4scnc4c3)c2c1
OCc1cccc(-c2cc3ncnc(Nc4ccc5scnc5c4)c3cc2-c2cccs2)c1
Cn1cccc1-c1cc2c(Nc3ccc4scnc4c3)ncnc2cc1-c1cccc(CO)c1
Cc1ccsc1-c1cc2c(Nc3ccc4scnc4c3)ncnc2cc1-c1cccc(CO)c1
OCc1ccc(-c2cc3ncnc(Nc4ccc5scnc5c4)c3cc2-c2cccs2)o1
C1=C(c2cc3ncnc(Nc4ccc5scnc5c4)c3cc2-c2cccs2)COC1
Cc1cn(CCN2CCN(CC2)c2ccccc2-c2cc(cc(c2)C(=O)NCCCN2CCCC2)C#N)c2ccccc12