870 SMILES Strings for Receptor-interacting serine/threonine-protein kinase 3

Compound Name
SMILES String
Cc1n[nH]cc1-c1c(c2c(CCNC2=O)n1Cc1ccc(F)cc1C#N)-c1ccc(F)cc1 |(-2.24,2.53,;-3.01,1.19,;-4.47,.72,;-4.47,-.82,;-3.01,-1.3,;-2.1,-.05,;-.56,-.05,;.34,1.19,;1.81,.72,;1.81,-.82,;3.14,-1.59,;4.47,-.82,;4.47,.72,;3.14,1.49,;3.14,3.03,;.34,-1.3,;-.06,-2.79,;1.03,-3.88,;2.52,-3.48,;3.61,-4.57,;3.21,-6.05,;4.3,-7.14,;1.72,-6.45,;.58,-5.38,;-.91,-5.78,;-2.4,-6.17,;-.06,2.68,;1.03,3.77,;.63,5.26,;-.85,5.66,;-1.25,7.14,;-1.94,4.57,;-1.54,3.08,)|
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2cccc(c2)C#N)c1-c1ccncc1
CC(=O)Nc1cc(ccn1)-c1c(c2c(CCNC2=O)n1CC1CCOCC1)-c1ccc(F)cc1
CC(=O)Nc1cc(ccn1)-c1c(c2c(CCNC2=O)n1Cc1ccc(C)cc1)-c1ccc(F)cc1
O=C1NCCc2c1c(c(-c1ccncc1)n2CC1CCOCC1)-c1cccc(c1)-c1ccccc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2ccc(cc2F)C(F)(F)F)c1-c1ccnc(Cl)c1
CC(C)C(=O)Nc1cc(ccn1)-c1c(c2c(CCNC2=O)n1Cc1ccc(cc1F)C(F)(F)F)-c1ccc(F)cc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2ccc(cc2F)C(F)(F)F)c1-c1ccnc(NC(=O)C2CC2)c1
Fc1ccc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2ccc(cc2)C(F)(F)F)c(c1)C#N
CNc1cc(ccn1)-c1c(c2c(CCNC2=O)n1Cc1ccc(cc1F)C(F)(F)F)-c1ccc(F)cc1
Fc1ccc(Cn2c3CCNC(=O)c3c(c2-c2ccnc(Cl)c2)-c2cccnc2)c(c1)C#N
Nc1cc(ccn1)-c1c(c2c(CCNC2=O)n1Cc1ccc(cc1F)C(F)(F)F)-c1ccc(F)cc1
Cc1noc(n1)-c1ccc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2ccc(F)cc2)cc1
Fc1ccc(Cn2c3CCNC(=O)c3c(-c3cccs3)c2-c2ccncc2)c(c1)C#N
COc1cnccc1-c1c(c2c(CCNC2=O)n1Cc1ccc(F)cc1C#N)-c1ccc(F)cc1 |(-2.87,3.95,;-2.1,2.61,;-2.87,1.28,;-4.41,1.28,;-5.18,-.05,;-4.41,-1.39,;-2.87,-1.39,;-2.1,-.05,;-.56,-.05,;.34,1.19,;1.81,.72,;1.81,-.82,;3.14,-1.59,;4.47,-.82,;4.47,.72,;3.14,1.49,;3.14,3.03,;.34,-1.3,;-.06,-2.79,;1.03,-3.88,;2.52,-3.48,;3.61,-4.57,;3.21,-6.05,;4.3,-7.14,;1.72,-6.45,;.58,-5.38,;-.91,-5.78,;-2.4,-6.17,;-.06,2.68,;1.03,3.77,;.63,5.26,;-.85,5.66,;-1.25,7.14,;-1.94,4.57,;-1.54,3.08,)|
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2ccc(F)cc2C#N)c1-c1ccnc(c1)C(F)(F)F
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2ccc(F)cc2C#N)c1-c1cncnc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2ccc(F)cc2C#N)c1-c1ccnc(F)c1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2ccc(F)cc2C#N)c1-c1ccc2[nH]ccc2c1
Cc1cc(ccn1)-c1c(c2c(CCNC2=O)n1Cc1ccc(F)cc1C#N)-c1ccc(F)cc1
CC(=O)Nc1cccc(c1)-c1c(c2c(CCNC2=O)n1Cc1ccc(F)cc1C#N)-c1ccc(F)cc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2ccc(F)cc2C#N)c1-c1ccnc(Cl)c1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2ccc(F)cc2C#N)c1-c1ccoc1
Cn1cc(cn1)-c1c(c2c(CCNC2=O)n1Cc1ccc(F)cc1C#N)-c1ccc(F)cc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2ccc(F)cc2C#N)c1-c1ccsc1
COc1ncc(cn1)-c1c(c2c(CCNC2=O)n1Cc1ccc(F)cc1C#N)-c1ccc(F)cc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2ccc(F)cc2C#N)c1-c1ccncc1F |(-1.25,7.14,;-.85,5.66,;.63,5.26,;1.03,3.77,;-.06,2.68,;-1.54,3.08,;-1.94,4.57,;.34,1.19,;1.81,.72,;1.81,-.82,;3.14,-1.59,;4.47,-.82,;4.47,.72,;3.14,1.49,;3.14,3.03,;.34,-1.3,;-.06,-2.79,;1.03,-3.88,;2.52,-3.48,;3.61,-4.57,;3.21,-6.05,;4.3,-7.14,;1.72,-6.45,;.58,-5.38,;-.91,-5.78,;-2.4,-6.17,;-.56,-.05,;-2.1,-.05,;-2.87,1.28,;-4.41,1.28,;-5.18,-.05,;-4.41,-1.39,;-2.87,-1.39,;-2.1,-2.72,)|
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2ccc(cc2)C#N)c1-c1ccncc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(c1-c1ccncc1)-c1ccccc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(CC2CCNCC2)c1-c1ccncc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(CC2CCOCC2)c1-c1ccncc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(CC2CCCNC2)c1-c1ccncc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2ccc(cc2)C(F)(F)F)c1-c1ccncc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2ccc(F)cc2C#N)c1-c1ccncc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2ccc(C#N)c(F)c2)c1-c1ccncc1
CC(c1ccccc1)n1c2CCNC(=O)c2c(c1-c1ccncc1)-c1ccc(F)cc1
COc1ccc(CCn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2ccc(F)cc2)cc1
COc1ccc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2ccc(F)cc2)cc1
CC(C)(C)c1ccc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2ccc(F)cc2)cc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2ccc(OC(F)(F)F)c(Cl)c2)c1-c1ccncc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2cc(F)cc(c2)C(F)(F)F)c1-c1ccncc1
CS(=O)(=O)c1ccc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2ccc(F)cc2)cc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2ccc(cc2F)C(F)(F)F)c1-c1ccncc1
Fc1ccc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2ccc(F)cc2)cc1
Cc1ccc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2ccc(F)cc2)cc1
Cc1cc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2ccc(F)cc2)ccc1F
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2nnc(s2)C2CC2)c1-c1ccncc1
Cc1nc(no1)-c1ccc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2ccc(F)cc2)c(F)c1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(CC#N)c1-c1ccncc1
Cc1noc(C)c1Cn1c2CCNC(=O)c2c(c1-c1ccncc1)-c1ccc(F)cc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2ccc(cc2F)C#N)c1-c1ccncc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2ccc(cc2)C2CC2)c1-c1ccncc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2ccc(cc2C(F)(F)F)C(F)(F)F)c1-c1ccncc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2ccc(cn2)C#N)c1-c1ccncc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2ccc(F)cc2C(F)(F)F)c1-c1ccncc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2nnc(o2)C2CC2)c1-c1ccncc1
CCCCCn1c2CCNC(=O)c2c(c1-c1ccncc1)-c1ccc(F)cc1
CC(C)Cn1c2CCNC(=O)c2c(c1-c1ccncc1)-c1ccc(F)cc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(CCCC#N)c1-c1ccncc1
Cc1nc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2ccc(F)cc2)cs1
CC(C)(C)Cn1c2CCNC(=O)c2c(c1-c1ccncc1)-c1ccc(F)cc1
CCn1c2CCNC(=O)c2c(c1-c1ccncc1)-c1ccc(F)cc1
CCC(C)n1c2CCNC(=O)c2c(c1-c1ccncc1)-c1ccc(F)cc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2ccc(F)cc2F)c1-c1ccncc1
Cc1cc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2ccc(F)cc2)n(C)n1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2ccncc2)c1-c1ccncc1
COc1cc(ccc1Cn1c2CCNC(=O)c2c(c1-c1ccncc1)-c1ccc(F)cc1)C(F)(F)F
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2ccccc2C#N)c1-c1ccncc1
OCCCn1c2CCNC(=O)c2c(c1-c1ccncc1)-c1ccc(F)cc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(CC(=O)N2CCCC2)c1-c1ccncc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2c(F)cc(F)cc2F)c1-c1ccncc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2ccncn2)c1-c1ccncc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2c(F)cccc2C(F)(F)F)c1-c1ccncc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2ccc(Cl)cc2F)c1-c1ccncc1
CC(C)(C)CCn1c2CCNC(=O)c2c(c1-c1ccncc1)-c1ccc(F)cc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2ccccn2)c1-c1ccncc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2c(F)cccc2C#N)c1-c1ccncc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(CC2CCCC2)c1-c1ccncc1
Cc1cc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2ccc(F)cc2)no1
Cn1ccnc1Cn1c2CCNC(=O)c2c(c1-c1ccncc1)-c1ccc(F)cc1
Cc1nc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2ccc(F)cc2)no1
OCCn1c2CCNC(=O)c2c(c1-c1ccncc1)-c1ccc(F)cc1
CC(C)NC(=O)Cn1c2CCNC(=O)c2c(c1-c1ccncc1)-c1ccc(F)cc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2c(F)cc(cc2F)C#N)c1-c1ccncc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(CC2CCOCC2)c1-c1ccnc(NC(=O)c2ccncc2)c1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(CC2CCOCC2)c1-c1ccnc(NC(=O)c2ccccc2)c1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(CC2CCOCC2)c1-c1ccnc(NC(=O)C2CC2)c1
CC(C)C(=O)Nc1cc(ccn1)-c1c(c2c(CCNC2=O)n1CC1CCOCC1)-c1ccc(F)cc1
COc1ccc(cc1)C(=O)Nc1cc(ccn1)-c1c(c2c(CCNC2=O)n1CC1CCOCC1)-c1ccc(F)cc1
CCC(=O)Nc1cc(ccn1)-c1c(c2c(CCNC2=O)n1CC1CCOCC1)-c1ccc(F)cc1
CC(C)OC(=O)Nc1cc(ccn1)-c1c(c2c(CCNC2=O)n1CC1CCOCC1)-c1ccc(F)cc1
CS(=O)(=O)Nc1cc(ccn1)-c1c(c2c(CCNC2=O)n1CC1CCOCC1)-c1ccc(F)cc1
CC(C)CC(=O)Nc1cc(ccn1)-c1c(c2c(CCNC2=O)n1CC1CCOCC1)-c1ccc(F)cc1
CCCC(=O)Nc1cc(ccn1)-c1c(c2c(CCNC2=O)n1CC1CCOCC1)-c1ccc(F)cc1
CCOC(=O)Nc1cc(ccn1)-c1c(c2c(CCNC2=O)n1CC1CCOCC1)-c1ccc(F)cc1
CNC(=O)Nc1cc(ccn1)-c1c(c2c(CCNC2=O)n1CC1CCOCC1)-c1ccc(F)cc1
CCNC(=O)Nc1cc(ccn1)-c1c(c2c(CCNC2=O)n1CC1CCOCC1)-c1ccc(F)cc1
CC(=O)Nc1cc(ccn1)-c1c(c2c(CCNC2=O)n1Cc1ccc(F)c(c1)C#N)-c1ccc(F)cc1
CC(=O)Nc1cc(ccn1)-c1c(c2c(CCNC2=O)n1Cc1ccc(F)cc1C#N)-c1ccc(F)cc1
CC(=O)Nc1cc(ccn1)-c1c(c2c(CCNC2=O)n1Cc1ccc(cc1F)C(F)(F)F)-c1ccc(F)cc1
CC(=O)Nc1cc(ccn1)-c1c(c2c(CCNC2=O)n1Cc1ccc(cc1)C(F)(F)F)-c1ccc(F)cc1
Cc1ccc(-c2c3c(CCNC3=O)n(CC3CCOCC3)c2-c2ccncc2)c(C)c1 |(-1.25,7.14,;-.85,5.66,;-1.94,4.57,;-1.54,3.08,;-.06,2.68,;.34,1.19,;1.81,.72,;1.81,-.82,;3.14,-1.59,;4.47,-.82,;4.47,.72,;3.14,1.49,;3.14,3.03,;.34,-1.3,;-.06,-2.79,;1.03,-3.88,;.58,-5.38,;1.72,-6.45,;3.21,-6.05,;3.61,-4.57,;2.52,-3.48,;-.56,-.05,;-2.1,-.05,;-2.87,1.28,;-4.41,1.28,;-5.18,-.05,;-4.41,-1.39,;-2.87,-1.39,;1.03,3.77,;2.52,3.37,;.63,5.26,)|
COc1ccc(cc1)-c1c2c(CCNC2=O)n(CC2CCOCC2)c1-c1ccncc1
FC(F)(F)c1cccc(c1)-c1c2c(CCNC2=O)n(CC2CCOCC2)c1-c1ccncc1
CC(=O)Nc1cccc(c1)-c1c2c(CCNC2=O)n(CC2CCOCC2)c1-c1ccncc1
COc1ccc(cn1)-c1c2c(CCNC2=O)n(CC2CCOCC2)c1-c1ccncc1
O=C1NCCc2c1c(c(-c1ccncc1)n2CC1CCOCC1)-c1cccnc1
CN(C)c1cccc(c1)-c1c2c(CCNC2=O)n(CC2CCOCC2)c1-c1ccncc1
FC(F)(F)Oc1cccc(c1)-c1c2c(CCNC2=O)n(CC2CCOCC2)c1-c1ccncc1
O=C1NCCc2c1c(c(-c1ccncc1)n2CC1CCOCC1)-c1cnc2ccccc2c1
O=C1NCCc2c1c(c(-c1ccncc1)n2CC1CCOCC1)-c1cccc2ccncc12 |(3.14,3.03,;3.14,1.49,;4.47,.72,;4.47,-.82,;3.14,-1.59,;1.81,-.82,;1.81,.72,;.34,1.19,;-.56,-.05,;-2.1,-.05,;-2.87,1.28,;-4.41,1.28,;-5.18,-.05,;-4.41,-1.39,;-2.87,-1.39,;.34,-1.3,;-.06,-2.79,;1.03,-3.88,;.58,-5.38,;1.72,-6.45,;3.21,-6.05,;3.61,-4.57,;2.52,-3.48,;-.06,2.68,;1.03,3.77,;.63,5.26,;-.85,5.66,;-1.94,4.57,;-3.43,4.96,;-4.52,3.88,;-4.12,2.39,;-2.63,1.99,;-1.54,3.08,)|
COc1ccc(cc1OC)-c1c2c(CCNC2=O)n(Cc2ccc(F)cc2C#N)c1-c1ccncc1
Fc1ccc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2cccc(OC(F)(F)F)c2)c(c1)C#N
Fc1ccc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2ccc(F)c(F)c2)c(c1)C#N
Fc1ccc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2ccc3ncccc3c2)c(c1)C#N
COc1cc(F)cc(c1)-c1c2c(CCNC2=O)n(Cc2ccc(F)cc2C#N)c1-c1ccncc1
Cn1ccc2cc(ccc12)-c1c2c(CCNC2=O)n(Cc2ccc(F)cc2C#N)c1-c1ccncc1
Fc1ccc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2cccnc2)c(c1)C#N
Fc1ccc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2cccc(c2)-c2ccccc2)c(c1)C#N
COc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2ccc(F)cc2C#N)c1-c1ccncc1
Fc1ccc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2ccc(OC(F)(F)F)cc2)c(c1)C#N
Fc1ccc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2cccc(c2)C(F)(F)F)c(c1)C#N
COc1ccc(cn1)-c1c2c(CCNC2=O)n(Cc2ccc(F)cc2C#N)c1-c1ccncc1
Fc1ccc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2ccccc2-c2ccccc2)c(c1)C#N |(4.3,-7.14,;3.21,-6.05,;3.61,-4.57,;2.52,-3.48,;1.03,-3.88,;-.06,-2.79,;.34,-1.3,;1.81,-.82,;3.14,-1.59,;4.47,-.82,;4.47,.72,;3.14,1.49,;3.14,3.03,;1.81,.72,;.34,1.19,;-.56,-.05,;-2.1,-.05,;-2.87,1.28,;-4.41,1.28,;-5.18,-.05,;-4.41,-1.39,;-2.87,-1.39,;-.06,2.68,;-1.54,3.08,;-1.94,4.57,;-.85,5.66,;.63,5.26,;1.03,3.77,;2.5,4.24,;3.64,3.21,;5.11,3.69,;5.43,5.2,;4.28,6.23,;2.82,5.75,;.58,-5.38,;1.72,-6.45,;-.91,-5.78,;-2.41,-6.1,)|
CS(=O)(=O)c1cccc(c1)-c1c2c(CCNC2=O)n(Cc2ccc(F)cc2C#N)c1-c1ccncc1
Oc1cccc(c1)-c1c2c(CCNC2=O)n(Cc2ccc(F)cc2C#N)c1-c1ccncc1
Fc1ccc(Cn2c3CCNC(=O)c3c(-c3ccsc3)c2-c2ccncc2)c(c1)C#N
Fc1ccc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2cccc(Cl)c2Cl)c(c1)C#N |(4.3,-7.14,;3.21,-6.05,;3.61,-4.57,;2.52,-3.48,;1.03,-3.88,;-.06,-2.79,;.34,-1.3,;1.81,-.82,;3.14,-1.59,;4.47,-.82,;4.47,.72,;3.14,1.49,;3.14,3.03,;1.81,.72,;.34,1.19,;-.56,-.05,;-2.1,-.05,;-2.87,1.28,;-4.41,1.28,;-5.18,-.05,;-4.41,-1.39,;-2.87,-1.39,;-.06,2.68,;1.03,3.77,;.63,5.26,;-.85,5.66,;-1.94,4.57,;-3.43,4.96,;-1.54,3.08,;-2.63,1.99,;.58,-5.38,;1.72,-6.45,;-.91,-5.78,;-2.41,-6.1,)|
Fc1ccc(Cn2c3CCNC(=O)c3c(-c3ccc(Cl)s3)c2-c2ccncc2)c(c1)C#N
COc1ccncc1-c1c2c(CCNC2=O)n(Cc2ccc(F)cc2C#N)c1-c1ccncc1 |(-4.12,2.39,;-2.63,1.99,;-1.54,3.08,;-1.94,4.57,;-.85,5.66,;.63,5.26,;1.03,3.77,;-.06,2.68,;.34,1.19,;1.81,.72,;1.81,-.82,;3.14,-1.59,;4.47,-.82,;4.47,.72,;3.14,1.49,;3.14,3.03,;.34,-1.3,;-.06,-2.79,;1.03,-3.88,;2.52,-3.48,;3.61,-4.57,;3.21,-6.05,;4.3,-7.14,;1.72,-6.45,;.58,-5.38,;-.91,-5.78,;-2.41,-6.1,;-.56,-.05,;-2.1,-.05,;-2.87,1.28,;-4.41,1.28,;-5.18,-.05,;-4.41,-1.39,;-2.87,-1.39,)|
Fc1ccc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2cncc3ccccc23)c(c1)C#N |(4.3,-7.14,;3.21,-6.05,;3.61,-4.57,;2.52,-3.48,;1.03,-3.88,;-.06,-2.79,;.34,-1.3,;1.81,-.82,;3.14,-1.59,;4.47,-.82,;4.47,.72,;3.14,1.49,;3.14,3.03,;1.81,.72,;.34,1.19,;-.56,-.05,;-2.1,-.05,;-2.87,1.28,;-4.41,1.28,;-5.18,-.05,;-4.41,-1.39,;-2.87,-1.39,;-.06,2.68,;-1.54,3.08,;-1.94,4.57,;-.85,5.66,;.63,5.26,;1.72,6.35,;3.21,5.95,;3.61,4.46,;2.52,3.37,;1.03,3.77,;.58,-5.38,;1.72,-6.45,;-.91,-5.78,;-2.41,-6.1,)|
NS(=O)(=O)c1cccc(c1)-c1c2c(CCNC2=O)n(Cc2ccc(F)cc2C#N)c1-c1ccncc1
OCc1cccc(c1)-c1c2c(CCNC2=O)n(Cc2ccc(F)cc2C#N)c1-c1ccncc1
Fc1ccc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2ccc(OCc3ccccc3)cc2)c(c1)C#N
Fc1ccc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2ccc(Cl)c(Cl)c2)c(c1)C#N
Oc1ccccc1-c1c2c(CCNC2=O)n(Cc2ccc(F)cc2C#N)c1-c1ccncc1 |(-2.63,1.99,;-1.54,3.08,;-1.94,4.57,;-.85,5.66,;.63,5.26,;1.03,3.77,;-.06,2.68,;.34,1.19,;1.81,.72,;1.81,-.82,;3.14,-1.59,;4.47,-.82,;4.47,.72,;3.14,1.49,;3.14,3.03,;.34,-1.3,;-.06,-2.79,;1.03,-3.88,;2.52,-3.48,;3.61,-4.57,;3.21,-6.05,;4.3,-7.14,;1.72,-6.45,;.58,-5.38,;-.91,-5.78,;-2.41,-6.1,;-.56,-.05,;-2.1,-.05,;-2.87,1.28,;-4.41,1.28,;-5.18,-.05,;-4.41,-1.39,;-2.87,-1.39,)|
Fc1ccc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2cc(Cl)cc(Cl)c2)c(c1)C#N
Fc1ccc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2cccc(c2)C#N)c(c1)C#N
COc1cc(ccn1)-c1c2c(CCNC2=O)n(Cc2ccc(F)cc2C#N)c1-c1ccncc1
Fc1ccc(Cn2c3CCNC(=O)c3c(-c3ccoc3)c2-c2ccncc2)c(c1)C#N
Cc1csc(c1)-c1c2c(CCNC2=O)n(Cc2ccc(F)cc2C#N)c1-c1ccncc1
Cc1cscc1-c1c2c(CCNC2=O)n(Cc2ccc(F)cc2C#N)c1-c1ccncc1 |(2.39,3.93,;.85,3.93,;-.06,5.17,;-1.52,4.7,;-1.52,3.16,;-.06,2.68,;.34,1.19,;1.81,.72,;1.81,-.82,;3.14,-1.59,;4.47,-.82,;4.47,.72,;3.14,1.49,;3.14,3.03,;.34,-1.3,;-.06,-2.79,;1.03,-3.88,;2.52,-3.48,;3.61,-4.57,;3.21,-6.05,;4.3,-7.14,;1.72,-6.45,;.58,-5.38,;-.91,-5.78,;-2.41,-6.1,;-.56,-.05,;-2.1,-.05,;-2.87,1.28,;-4.41,1.28,;-5.18,-.05,;-4.41,-1.39,;-2.87,-1.39,)|
Fc1ccc(Cn2c3CCNC(=O)c3c(\C=C\c3ccccc3)c2-c2ccncc2)c(c1)C#N
OCCNc1cc(ccn1)-c1c(c2c(CCNC2=O)n1Cc1ccc(cc1F)C(F)(F)F)-c1ccc(F)cc1
COCCNc1cc(ccn1)-c1c(c2c(CCNC2=O)n1Cc1ccc(cc1F)C(F)(F)F)-c1ccc(F)cc1
CCC(=O)Nc1cc(ccn1)-c1c(c2c(CCNC2=O)n1Cc1ccc(cc1F)C(F)(F)F)-c1ccc(F)cc1
COCC(=O)Nc1cc(ccn1)-c1c(c2c(CCNC2=O)n1Cc1ccc(cc1F)C(F)(F)F)-c1ccc(F)cc1
CC(C)Nc1cc(ccn1)-c1c(c2c(CCNC2=O)n1Cc1ccc(cc1F)C(F)(F)F)-c1ccc(F)cc1
CC1(C)CNC(=O)c2c(c(-c3ccncc3)n(CC3CCOCC3)c12)-c1ccc(F)cc1
CC1(C)CNC(=O)c2c1[nH]c(c2-c1ccc(F)cc1)-c1ccncc1
Cn1c(c(c2c1C(C)(C)CNC2=O)-c1ccc(F)cc1)-c1ccncc1
CCC(=O)Nc1cc(ccn1)-c1c(-c2ccc(F)cc2)c2c(cc[nH]c2=O)n1Cc1ccc(cc1F)C(F)(F)F
Fc1ccc(cc1)-c1c(-c2ccncc2)n(Cc2ccc(cc2F)C(F)(F)F)c2cc[nH]c(=O)c12
CC(C)(C)OC(=O)Nc1cc(ccn1)-c1c(c2c(CCNC2=O)n1Cc1ccc(F)cc1C#N)-c1ccc(F)cc1
Nc1cc(ccn1)-c1c(c2c(CCNC2=O)n1Cc1ccc(F)cc1C#N)-c1ccc(F)cc1
Fc1ccc(cc1)-c1c2c(CCNC2=O)n(Cc2ccc(F)cc2C#N)c1-c1ccnc(NC(=O)C2CC2)c1
Cc1ccc(cc1)S(=O)(=O)n1c2CCNC(=O)c2c(c1-c1ccncc1)-c1ccc(F)cc1
CC(C)(C)OC(=O)Nc1cccc(c1)-c1c2c(CCNC2=O)n(Cc2ccc(Cl)cc2F)c1-c1ccncc1
Cc1ccc(s1)-c1c2c(CCNC2=O)n(Cc2ccc(Cl)cc2F)c1-c1ccncc1
Cn1cc(cn1)-c1c2c(CCNC2=O)n(Cc2ccc(Cl)cc2F)c1-c1ccncc1
Fc1cc(Cl)ccc1Cn1c2CCNC(=O)c2c(c1-c1ccncc1)-c1ccncc1F |(-.91,-5.78,;.58,-5.38,;1.72,-6.45,;3.21,-6.05,;4.3,-7.14,;3.61,-4.57,;2.52,-3.48,;1.03,-3.88,;-.06,-2.79,;.34,-1.3,;1.81,-.82,;3.14,-1.59,;4.47,-.82,;4.47,.72,;3.14,1.49,;3.14,3.03,;1.81,.72,;.34,1.19,;-.56,-.05,;-2.1,-.05,;-2.87,1.28,;-4.41,1.28,;-5.18,-.05,;-4.41,-1.39,;-2.87,-1.39,;-.06,2.68,;1.03,3.77,;.63,5.26,;-.85,5.66,;-1.94,4.57,;-1.54,3.08,;-2.63,1.99,)|
COC(=O)c1cccc(c1)-c1c2c(CCNC2=O)n(Cc2ccc(Cl)cc2F)c1-c1ccncc1
Cc1cc(ccn1)-c1c2c(CCNC2=O)n(Cc2ccc(Cl)cc2F)c1-c1ccncc1
Nc1cccc(c1)-c1c2c(CCNC2=O)n(Cc2ccc(Cl)cc2F)c1-c1ccncc1
CCCC(=O)Nc1cccc(c1)-c1c2c(CCNC2=O)n(Cc2ccc(Cl)cc2F)c1-c1ccncc1
Cc1cc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2cccc(NC(=O)OC(C)(C)C)c2)n(C)n1
COC(=O)c1cccc(c1)-c1c2c(CCNC2=O)n(Cc2cc(C)nn2C)c1-c1ccncc1
Cc1cc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2cccc(c2)-c2c(C)noc2C)n(C)n1
Cc1cc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2cccc(N)c2)n(C)n1
Cc1cc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2cccc(NC(=O)Cc3ccccc3)c2)n(C)n1
Cc1cc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2cccc(NC(=O)c3ccccc3)c2)n(C)n1
Cc1cc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2cccc(NC(=O)C3CC3)c2)n(C)n1
Cc1cc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2cccc(NC=O)c2)n(C)n1
CCC(=O)Nc1cccc(c1)-c1c2c(CCNC2=O)n(Cc2cc(C)nn2C)c1-c1ccncc1
Cc1cc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2cccc(CCc3ccccc3)c2)n(C)n1
Cc1cc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2)-c2cccc(CCC3CCCCC3)c2)n(C)n1
Cc1cc(Cn2c3CCNC(=O)c3c(c2-c2ccncc2F)-c2ccc(F)cc2)n(C)n1 |(4.7,-5.44,;3.19,-5.12,;2.56,-3.71,;1.03,-3.88,;-.06,-2.79,;.34,-1.3,;1.81,-.82,;3.14,-1.59,;4.47,-.82,;4.47,.72,;3.14,1.49,;3.14,3.03,;1.81,.72,;.34,1.19,;-.56,-.05,;-2.1,-.05,;-2.87,1.28,;-4.41,1.28,;-5.18,-.05,;-4.41,-1.39,;-2.87,-1.39,;-2.1,-2.72,;-.06,2.68,;1.03,3.77,;.63,5.26,;-.85,5.66,;-1.25,7.14,;-1.94,4.57,;-1.54,3.08,;.71,-5.38,;-.69,-6.01,;2.05,-6.15,)|
COc1cnccc1-c1c(c2c(CCNC2=O)n1Cc1cc(C)nn1C)-c1ccc(F)cc1 |(-2.87,-4.05,;-2.1,-2.72,;-2.87,-1.39,;-4.41,-1.39,;-5.18,-.05,;-4.41,1.28,;-2.87,1.28,;-2.1,-.05,;-.56,-.05,;.34,1.19,;1.81,.72,;1.81,-.82,;3.14,-1.59,;4.47,-.82,;4.47,.72,;3.14,1.49,;3.14,3.03,;.34,-1.3,;-.06,-2.79,;1.03,-3.88,;2.56,-3.71,;3.19,-5.12,;4.7,-5.44,;2.05,-6.15,;.71,-5.38,;-.69,-6.01,;-.06,2.68,;1.03,3.77,;.63,5.26,;-.85,5.66,;-1.25,7.14,;-1.94,4.57,;-1.54,3.08,)|
Cc1cc(Cn2c3CCNC(=O)c3c(c2-c2cn[nH]c2)-c2ccc(F)cc2)n(C)n1
Cc1cc(Cn2c3CCNC(=O)c3c(c2-c2ccnc(NC(=O)C3CC3)c2)-c2cccc(NC(=O)OC(C)(C)C)c2)n(C)n1
CCS(=O)(=O)Nc1ccc(-c2nn(C)c3c(-c4cccnc4)cnc(N)c23)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2nn(C)c3c(NC(C)=O)cnc(N)c23)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2coc3c(-c4cnn(C5CCOCC5)c4)cnc(N)c23)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2coc3c(-c4cnn(CCO)c4)cnc(N)c23)cc1OCc1ccc(F)cc1
Nc1ncc(-c2cnn(C3CCOCC3)c2)c2occ(-c3ccc(NS(=O)(=O)C(F)F)c(OCc4ccc(F)cc4)c3)c12
Nc1ncc(-c2cnn(CCO)c2)c2occ(-c3ccc(NS(=O)(=O)C(F)F)c(OCc4ccc(F)cc4)c3)c12
C[C@H](Oc1cc(-c2coc3c(-c4cnn(C5CCOCC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2coc3c(-c4cnn(C)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2coc3c(-c4cnn(CCO)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3ccnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
Nc1ncc(-c2cnn(C3CCOCC3)c2)c2occ(-c3ccc(NS(=O)(=O)CC(F)(F)F)c(OCc4ccc(F)cc4)c3)c12
Cn1nc(-c2ccc(NS(=O)(=O)C(F)F)c(OCc3ccc(F)cc3)c2)c2c(N)ncc(-c3cnn(CCO)c3)c21
Cn1nc(-c2ccc(NS(=O)(=O)C(F)F)c(OCc3ccc(F)cc3)c2)c2c(N)ncc(-c3cnn(C4CCOCC4)c3)c21
Cn1nc(-c2ccc(NS(=O)(=O)C(F)F)c(OCc3ccc(F)cc3)c2)c2c(N)ncc(-c3ccncc3)c21
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(CCO)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
Cn1cc(-c2cnc(N)c3c(-c4ccc(NS(=O)(=O)C(F)F)c(OCc5ccc(F)cc5)c4)nn(C)c23)cn1
C[C@H](Oc3cc(c1nn(C)c2ccnc(N)c12)ccc3NS(=O)(=O)C(F)F)c4ccc(F)cc4
C[C@H](Oc1cc(-c2nn(C)c3c(-c4ccncc4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCOCC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(C4=CCN(C)CC4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc3cc(C1C=NN2C=CN=C(N)C12)ccc3NS(=O)(=O)C(F)F)c4ccc(F)cc4
C[C@H](Oc1cc(-c2nn(C)c3c(-c4ccnc(C(F)(F)F)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
Cc1cc(-c2cnc(N)c3c(-c4ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c5ccc(F)cc5)c4)nn(C)c23)ccn1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cccnc4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
Cc1ccc(-c2cnc(N)c3c(-c4ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c5ccc(F)cc5)c4)nn(C)c23)cn1
COc1cc(-c2cnc(N)c3c(-c4ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c5ccc(F)cc5)c4)nn(C)c23)ccn1
COc1ccc(-c2cnc(N)c3c(-c4ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c5ccc(F)cc5)c4)nn(C)c23)cn1
COCCn1cc(-c2cnc(N)c3c(-c4ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c5ccc(F)cc5)c4)nn(C)c23)cn1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCCC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CC(C)n1cc(-c2cnc(N)c3c(-c4ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c5ccc(F)cc5)c4)nn(C)c23)cn1
Cc1cnccc1-c1cnc(N)c2c(-c3ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c4ccc(F)cc4)c3)nn(C)c12
Cc1noc(C)c1-c1cnc(N)c2c(-c3ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c4ccc(F)cc4)c3)nn(C)c12
C[C@H](Oc1cc(-c2nn(C)c3c(Cc4ccccc4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2cnn3c(-c4cnn(C)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2cnn3c(-c4cnn(C5CCOCC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2cnn3c(-c4cnn(CCO)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5COC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2cnn3c(-c4ccncc4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc4cc(c2nn(C)c3c(c1ccncn1)cnc(N)c23)ccc4NS(=O)(=O)C(F)F)c5ccc(F)cc5
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCOC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc4cc(c2nn(C)c3c(C1CCN(C)CC1)cnc(N)c23)ccc4NS(=O)(=O)C(F)F)c5ccc(F)cc5
C[C@H](Oc1cc(-c2nn(C)c3c(C4=CCOCC4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc5cc(c3nn(C)c4c(c2cnn(C1CCOCC1)c2)cnc(N)c34)ccc5NS(=O)(=O)CC(F)(F)F)c6ccc(F)cc6
CCS(=O)(=O)Nc1ccc(-c2nn(C)c3c(-c4cnn(C5CCOCC5)c4)cnc(N)c23)cc1O[C@@H](C)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCN(C)CC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CC(=O)Nc1cnc(N)c2c(-c3ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c4ccc(F)cc4)c3)nn(C)c12
C[C@H](Oc1cc(-c2nn(C)c3c(-c4ccnc(C(C)(C)C)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4ccnc(N(C)C)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CC(C)n1nc(-c2ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c3ccc(F)cc3)c2)c2c(N)ncc(-c3ccncc3)c21
CC(C)n1nc(-c2ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c3ccc(F)cc3)c2)c2c(N)ncc(-c3cnn(C4CCOCC4)c3)c21
CC(C)n1nc(-c2ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c3ccc(F)cc3)c2)c2c(N)ncc(-c3cnn(C)c3)c21
CC(C)n4nc(c2ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c1ccc(F)cc1)c2)c3c(N)nccc34
C[C@H](Oc4cc(c2nn(C)c3c(C1CCCNC1)cnc(N)c23)ccc4NS(=O)(=O)C(F)F)c5ccc(F)cc5
C[C@H](Oc4cc(c2nn(C)c3c(C1CCCN(C)C1)cnc(N)c23)ccc4NS(=O)(=O)C(F)F)c5ccc(F)cc5
CC#Cc1cnc(N)c2c(-c3ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c4ccc(F)cc4)c3)nn(C)c12
C[C@H](Oc1cc(-c2nn(C)c3c(-c4ccnc(C(F)F)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(C#CC4CCOCC4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCNCC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(CCN5CCN(C)CC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCN(CC(F)(F)F)CC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CCS(=O)(=O)Nc3ccc(c1cccc2[nH]nc(N)c12)cc3OCc4ccc(F)cc4
CCS(=O)(=O)Nc3ccc(c1ncn2ccnc(N)c12)cc3OCc4ccc(F)cc4
CCS(=O)(=O)Nc3ccc(c1cnn2ccnc(N)c12)cc3OCc4ccc(F)cc4
Nc3n[nH]c4ccnc(c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc1ccc(F)cc1)c2)c34
Nc3n[nH]c4nccc(c2ccc(NS(=O)(=O)C(F)F)c(OCc1ccc(F)cc1)c2)c34
Nc3n[nH]c4nccc(c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc1ccc(F)cc1)c2)c34
Nc3n[nH]c4ccnc(c2ccc(NS(=O)(=O)C(F)F)c(OCc1ccc(F)cc1)c2)c34
Nc3n[nH]c4ncnc(c2ccc(NS(=O)(=O)C(F)F)c(OCc1ccc(F)cc1)c2)c34
Cc4cc(c2ccc(NS(=O)(=O)C(F)F)c(OCc1ccc(F)cc1)c2)c3c(N)n[nH]c3n4
Nc4n[nH]c5nc(c1ccccc1)cc(c3ccc(NS(=O)(=O)C(F)F)c(OCc2ccc(F)cc2)c3)c45
C[C@H](Oc3cc(c1ccnc2[nH]nc(N)c12)ccc3NS(=O)(=O)C(F)F)c4ccc(F)cc4
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CC6CCC(C5)N6C)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CNc1c(-c2cnn(C3CCCNCC3)c2)cnc(N)c1C(=N)c1ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c2ccc(F)cc2)c1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(CCN5CC(C)(C)C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CC(C)N1CC(n2cc(-c3cnc(N)c4c(-c5ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c6ccc(F)cc6)c5)nn(C)c34)cn2)C1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CN(CC(F)(F)F)C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CC6(CNC6)C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc4cc(c2nn(C)c3c(C#CC1CCNCC1)cnc(N)c23)ccc4NS(=O)(=O)C(F)F)c5ccc(F)cc5
C[C@H](Oc4cc(c2nn(C)c3c(C#CC1CCN(C)CC1)cnc(N)c23)ccc4NS(=O)(=O)C(F)F)c5ccc(F)cc5
CC(C)N(C)C(=O)C(C)n1cc(-c2cnc(N)c3c(-c4ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c5ccc(F)cc5)c4)nn(C)c23)cn1
CNCCn1cc(-c2cnc(N)c3c(-c4ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c5ccc(F)cc5)c4)nn(C)c23)cn1
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C[C@H](Oc1cc(-c2nn(C)c3c(-c4cccc(Cl)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4ccccc4Cl)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4ccccc4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4ccc(Cl)cc4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CNc1c(-c2cnn(CC3CCCN3)c2)cnc(N)c1C(=N)c1ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c2ccc(F)cc2)c1
C[C@H](Oc5cc(c3nn(C)c4c(c2cnn(C1(CN)CC1)c2)cnc(N)c34)ccc5NS(=O)(=O)C(F)F)c6ccc(F)cc6
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn5c4CNCC5)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc5cc(c3nn(C)c4c(c1cnn2CCN(C)Cc12)cnc(N)c34)ccc5NS(=O)(=O)C(F)F)c6ccc(F)cc6
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CN(C)C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCN(C)C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CNC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CC1CNCC(n2cc(-c3cnc(N)c4c(-c5ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c6ccc(F)cc6)c5)nn(C)c34)cn2)C1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5(C#N)CC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C(C)(C)CO)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc5cc(c3nn(C)c4c(c2cnn(C1(CC#N)COC1)c2)cnc(N)c34)ccc5NS(=O)(=O)C(F)F)c6ccc(F)cc6
CNc1c(-c2cnn(C3CC4(C3)CN(C)C4)c2)cnc(N)c1C(=N)c1ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c2ccc(F)cc2)c1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(CCN(C)C)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CC(C)N(C)CC(C)n1cc(-c2cnc(N)c3c(-c4ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c5ccc(F)cc5)c4)nn(C)c23)cn1
COCC(Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCOCC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
[2H]C([2H])([2H])N6CCC(n5cc(c3cnc(N)c4c(c2ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c1ccc(F)cc1)c2)nn(C)c34)cn5)CC6
C[C@H](Oc5cc(c3nn(C)c4c(c2cnn(C1CCC(C)(C)N(C)C1)c2)cnc(N)c34)ccc5NS(=O)(=O)C(F)F)c6ccc(F)cc6
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnc(N5CCN(C)CC5)nc4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnc(N(C)C)nc4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@@H](Oc1cc(-c2nn(C)c3c(-c4ccc(N5CCN(C)CC5)nc4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4ccc(N5CCN(C)CC5)nc4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CC(=O)N6CCC(n5cc(c3cnc(N)c4c(c2ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c1ccc(F)cc1)c2)nn(C)c34)cn5)CC6
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnc(N5CCOCC5)nc4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
COC[C@H](Oc5cc(c3nn(C)c4c(c2cnn(C1CCOCC1)c2)cnc(N)c34)ccc5NS(=O)(=O)C(F)F)c6ccc(F)cc6
COC[C@@H](Oc5cc(c3nn(C)c4c(c2cnn(C1CCOCC1)c2)cnc(N)c34)ccc5NS(=O)(=O)C(F)F)c6ccc(F)cc6
C[C@H](Oc5cc(c3nn(C)c4c(c2cnn(C1CCN(C)C(C)(C)C1)c2)cnc(N)c34)ccc5NS(=O)(=O)C(F)F)c6ccc(F)cc6
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnc(N5CCCC5)nc4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4ccc(N5CCOCC5)nc4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(CC(F)(F)F)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
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C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCOCC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccccc1F
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCOCC5)c4)cnc(N)c23)ccc1NS(C)(=O)=O)c1ccc(F)cc1
C[C@H](Oc5cc(c3nn(C)c4c(c2cnn(C1CCC(F)(F)C1)c2)cnc(N)c34)ccc5NS(=O)(=O)C(F)F)c6ccc(F)cc6
C[C@@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCOCC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCOCC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1cccc(Cl)c1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C(F)F)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCOCC5)c4)cnc(N)c23)ccc1NS(=O)(=O)N(C)C)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCOCC5)c4)cnc(N)c23)ccc1NS(=O)(=O)Cc1ccccc1)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4ccn(C)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCOCC5)c4)cnc(N)c23)ccc1NS(=O)(=O)Cc1ccccc1)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(C#CC4CCN(CC(F)(F)F)CC4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
COc1ccc([C@H](C)Oc2cc(-c3nn(C)c4c(-c5cnn(C6CCOCC6)c5)cnc(N)c34)ccc2NS(=O)(=O)C(F)F)cc1
Cn1nc(-c2ccc(NS(=O)(=O)C(F)F)c(OCc3cccc(Cl)c3)c2)c2c(N)ncc(-c3cnn(C4CCOCC4)c3)c21
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(CCC(F)(F)F)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
Cn1nc(-c2ccc(NS(=O)(=O)C(F)F)c(OCc3ccc(Cl)c(F)c3)c2)c2c(N)ncc(-c3cnn(C4CCOCC4)c3)c21
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C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C(F)(F)F)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
Cn1nc(-c2ccc(NS(=O)(=O)C(F)F)cc2OCc2cccc(F)c2)c2c(N)ncc(-c3cnn(C4CCOCC4)c3)c21
CNc1ncc(-c2cnc(N)c3c(-c4ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c5ccc(F)cc5)c4)nn(C)c23)cn1
COCC(Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCN(C)CC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
Cn1nc(-c2ccc(NS(=O)(=O)C(F)F)c(OC3(c4ccc(F)cc4)CC3)c2)c2c(N)ncc(-c3cnn(C4CCOCC4)c3)c21
C[C@H](Oc4cc(c2nn(C)c3c(N1CCOCC1)cnc(N)c23)ccc4NS(=O)(=O)C(F)F)c5ccc(F)cc5
CC(n1cc(-c2cnc(N)c3c(-c4ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c5ccc(F)cc5)c4)nn(C)c23)cn1)C(F)(F)F
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C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCN(C)C6(CC6)C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCC(F)(F)CC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
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C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CC6CCC(C5)N6CC(F)(F)F)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
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C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCN(C)C(C)(C)C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(Cl)cc1
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C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5C[C@H]6CNC[C@H]6C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5C[C@@H]6CN(C)C[C@@H]6C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4ccc5c(c4)CC(=O)N5C)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
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C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCN(CC(F)(F)F)C(C)(C)C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCC(N(C)C)C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCN(C)C6(CC6)C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCN(C)C6(CC6)C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CC1CN(C)CC(C)C1n1cc(-c2cnc(N)c3c(-c4ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c5ccc(F)cc5)c4)nn(C)c23)cn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1ccc(F)c(F)c1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1ccccc1F
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)cc1OCc1cccc(Cl)c1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)cc1OCc1ccc(Cl)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc3ccc(F)cc3)c2)n[nH]c1Nc1cccc(C(F)(F)F)n1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccnc3)c2C(N)=O)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCC1CCN(C(C)=O)CC1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)cc1OCc1ccc(F)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)Cc3cccc(Cl)c3)cc2)n[nH]c1Nc1cccc(C(F)(F)F)n1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)cc1OCC1CCCC1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(OC)n3)c2C(N)=O)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)cc1OCC(C)C
CCS(=O)(=O)Cc1ccc(-c2nn(C(C)(C)C)c(Cc3ccccn3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnc(OC)cn3)c2C(N)=O)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cncc(OC)n3)c2C(N)=O)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)cc1OCc1ccncc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cncc(C(F)(F)F)n3)c2C(N)=O)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccnc(OC)c3)c2C(N)=O)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Cc1ccc(-c2nn(COCC[Si](C)(C)C)c(Nc3cnccn3)c2C(N)=O)cc1Oc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccccn3)c2C(N)=O)cc1OCc1ccccc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)c(OCc2ccc(F)cc2)c1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Cc3cnc(C)cn3)c2C(N)=O)cc1OCc1ccc(F)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CCC(F)F)cc2)n[nH]c1Nc1cnccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1ccccc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1cccc(F)c1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccccn3)c2C(N)=O)cc1OCc1ccncc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1ccncc1
N#CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccccn3)c2C(N)=O)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccccn3)c2C(N)=O)cc1OCc1cccnc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1cccnc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)cc1OCc1cccnc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnc(C(C)C)cn3)c2C(N)=O)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccccn3)c2C(N)=O)cc1OCC1CCCCC1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccccn3)c2C(N)=O)cc1OCC1CCCC1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccccn3)c2C(N)=O)cc1OCC(C)C
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccccn3)c2C(N)=O)cc1OCc1cccc(Cl)c1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccccn3)c2C(N)=O)cc1OCc1ccc(Cl)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCC1CCCC1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1cccc(Cl)c1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1ccc(Cl)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)cc2)n[nH]c1Nc1cccc(C(F)(F)F)n1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cncc(C(F)(F)F)n3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCC(C)C
CCS(=O)(=O)Nc1ccc(-c2nn(C(C)(C)C)c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)cc1OCc1ccccc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCC1CCCCC1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)F)cc2)n[nH]c1Nc1ccccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)F)cc2)n[nH]c1Nc1cccc(C(F)(F)F)n1
COCCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)cc1
CN(C)CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C3CC3)cc2)n[nH]c1Nc1cccc(C(F)(F)F)n1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)F)cc2)n[nH]c1Nc1cccc(C(F)(F)F)n1
CC(C)S(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)Cc3ccc(F)cc3)cc2)n[nH]c1Nc1cccc(C(F)(F)F)n1
NC(=O)c1c(-c2ccc(NS(=O)(=O)Cc3ccc(Cl)c(Cl)c3)cc2)n[nH]c1Nc1cccc(C(F)(F)F)n1
Cc1ccc(CS(=O)(=O)Nc2ccc(-c3n[nH]c(Nc4cccc(C(F)(F)F)n4)c3C(N)=O)cc2)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)Cc3ccccc3Cl)cc2)n[nH]c1Nc1cccc(C(F)(F)F)n1
Cc1cccc(CS(=O)(=O)Nc2ccc(-c3n[nH]c(Nc4cccc(C(F)(F)F)n4)c3C(N)=O)cc2)c1Cl
NC(=O)c1c(-c2ccc(NS(=O)(=O)Cc3ccc(Cl)cc3)cc2)n[nH]c1Nc1cccc(C(F)(F)F)n1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OC
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1ccc(F)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)F)cc2)n[nH]c1Nc1cnccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccnn3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnc4cc(Cl)ccc4n3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnc(C(C)C)cn3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnc4ccccc4n3)c2C(N)=O)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C3CC3)cc2)n[nH]c1Nc1cnccn1
CC(C)(C)S(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)Cc3ccc(Cl)cc3)cc2)n[nH]c1Nc1cnccn1
CC(C)S(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1
CCCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1
Cc1cccc(S(=O)(=O)Nc2ccc(-c3n[nH]c(Nc4cnccn4)c3C(N)=O)cc2)c1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C3CCCCC3)cc2)n[nH]c1Nc1cnccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnc(C(F)(F)F)cn3)c2C(N)=O)cc1
Cc1ccc(CS(=O)(=O)Nc2ccc(-c3n[nH]c(Nc4cnccn4)c3C(N)=O)cc2)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)Cc3ccccc3)cc2)n[nH]c1Nc1cnccn1
Cc1ccc(S(=O)(=O)Nc2ccc(-c3n[nH]c(Nc4cnccn4)c3C(N)=O)cc2)cc1
Cc1ccc(S(=O)(=O)Nc2ccc(-c3n[nH]c(Nc4cnccn4)c3C(N)=O)cc2)cc1
Cc1ccc(CS(=O)(=O)Nc2ccc(-c3n[nH]c(Nc4cnccn4)c3C(N)=O)cc2)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC3CCC3)cc2)n[nH]c1Nc1cnccn1
COc1ccc(S(=O)(=O)Nc2ccc(-c3n[nH]c(Nc4cnccn4)c3C(N)=O)cc2)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)Cc3cccc(C(F)(F)F)c3)cc2)n[nH]c1Nc1cnccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cncc(C)n3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cc(C(F)(F)F)ccn3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccc4ccccc4c3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cc4ccccc4cn3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccc(OC)cn3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccc4ccccc4n3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnc(OC)cn3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccn(C)n3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)F)n3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccc(C(F)(F)F)cn3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C)n3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cc(C)ccn3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccccn3)c2C(N)=O)cc1
CCCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1
CCOc1nccc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)CC)cc3)c2C(N)=O)n1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cncc(OC)n3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnn(C)c3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnc(C)cn3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccc(C#N)cc3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccnc(C(F)(F)F)c3)c2C(N)=O)cc1
CCOc1cc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)CC)cc3)c2C(N)=O)ccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccnc(OCC(F)F)c3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(OC)n3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1
C#CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccnc(OCCOC)c3)c2C(N)=O)cc1
N#CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccnc(OCCOC)c3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cc(C)ncc3F)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cc(C)nc(C)c3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccnc(C)c3)c2C(N)=O)cc1
COCCOc1cc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)C(F)(F)F)cc3)c2C(N)=O)ccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccc(OC)nc3)c2C#N)cc1
COCCOc1cc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)CCN(C)C)cc3)c2C(N)=O)ccn1
CCS(=O)(=O)N(C)c1ccc(-c2n[nH]c(Nc3ccnc(OCCOC)c3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2nn(C(C)(C)C)c(Nc3cc(OC)ncc3C)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(NC)c2C(N)=O)cc1
COCCOc1cc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)COC)cc3)c2C(N)=O)ccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccnc(OC)c3)c2C(N)=O)cc1
COCCOc1cc(Nc2[nH]nc(-c3ccc(NS(C)(=O)=O)cc3)c2C(N)=O)ccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccnc(OC)n3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccccc3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccnc(C)n3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(C2=NN=C(Nc3ccnc(OCCOC)c3)C2C(N)=O)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(OCCOC)n3)c2C(N)=O)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)Cc3cccc(Cl)c3)cc2)n[nH]c1Nc1ccccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CCc3ccccc3)cc2)n[nH]c1Nc1ccccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccccn3)c2C(N)=O)cc1
Cc1ccc(CS(=O)(=O)Nc2ccc(-c3n[nH]c(Nc4ccccn4)c3C(N)=O)cc2)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)c3ccccc3)cc2)n[nH]c1Nc1ccccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC3CCC3)cc2)n[nH]c1Nc1ccccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)cc2)n[nH]c1Nc1cnccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccc4ccc(Cl)cc4n3)c2C(N)=O)cc1OCc1ccc(F)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)cc2OCc2ccc(F)cc2)n[nH]c1Nc1cnccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)cc2OCc2ccc(F)cc2)n[nH]c1Nc1cccc(C(F)(F)F)n1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)c(OCc2ccc(F)cc2)c1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1c(C)cc(F)cc1C
COc1cnc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)CC(F)(F)F)c(OCc4ccc(F)cc4)c3)c2C(N)=O)cn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OC3(c4ccc(F)cc4)CC3)c2)n[nH]c1Nc1cnccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)F)cc2)n[nH]c1Nc1ccc(C(F)(F)F)cn1
Cc1cnc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)CC(F)(F)F)c(OCc4ccc(Cl)c(F)c4)c3)c2C(N)=O)cn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)F)c(Oc3ccc(F)cc3)c2)n[nH]c1Nc1cccc(C(F)(F)F)n1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(Oc3ccc(F)cc3)c2)n[nH]c1Nc1cccc(C(F)(F)F)n1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)cc1Oc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnc(C)cn3)c2C(N)=O)cc1OCc1ccc(F)c(Cl)c1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)F)c(OCc3ccc(F)c(F)c3)c2)n[nH]c1Nc1cccc(C(F)(F)F)n1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OC1(c2ccccc2)CC1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)cc2)n[nH]c1Nc1ccc(C(F)(F)F)cn1
C[C@H](Oc1cc(-c2n[nH]c(Nc3ccccn3)c2C(N)=O)ccc1NS(=O)(=O)CC(F)(F)F)c1ccc(F)cc1
Cc1cnc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)CC(F)(F)F)c(OCc4ccc(F)c(Cl)c4)c3)c2C(N)=O)cn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1ccc(F)cn1
COc1cnc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)CC(F)(F)F)c(OCc4ccc(Cl)cc4)c3)c2C(N)=O)cn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnc(C4CC4)cn3)c2C(N)=O)cc1
COc1ccc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)CC(F)(F)F)c(OCc4ccc(F)cc4)c3)c2C(N)=O)cn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc3ccc(F)c(F)c3)c2)n[nH]c1Nc1ccccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OC3(c4ccccc4)CC3)c2)n[nH]c1Nc1cnccn1
Cc1cnc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)CC(F)(F)F)c(OCc4ccc(Cl)cc4)c3)c2C(N)=O)cn1
Cc1cnc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)CC(F)(F)F)c(OCc4ccc(F)cc4)c3)c2C(N)=O)cn1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)ccc1NS(=O)(=O)CC(F)(F)F)c1ccc(F)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc3ccc(Cl)c(F)c3)c2)n[nH]c1Nc1cnccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1ccc(Cl)c(F)c1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(Oc3cccc(F)c3)c2)n[nH]c1Nc1cnccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(Oc3ccc(Cl)cc3)c2)n[nH]c1Nc1cnccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C3CC3)c(OCc3ccc(F)cc3)c2)n[nH]c1Nc1cnccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc3ccc(F)cc3)c2)n[nH]c1Nc1cnccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1ccc(F)cc1C
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(CC(F)(F)F)n3)c2C(N)=O)cc1OCc1ccc(F)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc3ccc(F)cc3)c2)n[nH]c1Nc1cccc(C(F)F)n1
CCS(=O)(=O)Cc1ccc(-c2n[nH]c(Nc3cccc(OCCOC)n3)c2C(N)=O)cc1OCc1ccc(F)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc3ccc(F)c(F)c3)c2)n[nH]c1Nc1cnccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc3ccc(F)cc3)c2)n[nH]c1Nc1ccc(C(F)(F)F)nc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)F)c(Oc3ccc(F)cc3)c2)n[nH]c1Nc1cnccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)F)c(OCc3ccc(F)cc3)c2)n[nH]c1Nc1cccc(C(F)(F)F)n1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)F)n3)c2C(N)=O)cc1OCc1ccc(F)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)F)c(OCc3ccc(F)cc3)c2)n[nH]c1Nc1cnccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnc(C(C)(C)C)cn3)c2C(N)=O)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CCC(F)(F)F)c(OCc3ccc(F)cc3)c2)n[nH]c1Nc1cccc(C(F)(F)F)n1
Cc1cnc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)CCC(F)(F)F)c(OCc4ccc(F)cc4)c3)c2C(N)=O)cn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CCC(F)(F)F)c(OCc3ccc(F)cc3)c2)n[nH]c1Nc1cnccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1Oc1ccc(Cl)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc3ccc(F)cc3)c2)n[nH]c1Nc1ccnc(C(F)(F)F)n1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCC1CCCN(C)C1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)F)c(OCc3ccc(F)cc3)c2)n[nH]c1Nc1ccc(C(F)(F)F)nc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CCC(F)(F)F)cc2)n[nH]c1Nc1cccc(C(F)(F)F)n1
COc1cnc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)C(F)F)c(OCc4ccc(Cl)cc4)c3)c2C(N)=O)cn1
COc1cnc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)C(F)F)c(OCc4ccc(F)cc4)c3)c2C(N)=O)cn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccnc3C(F)(F)F)c2C(N)=O)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1O[C@H](C)c1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccc(C(F)(F)F)nc3)c2C(N)=O)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccnc(C(F)(F)F)n3)c2C(N)=O)cc1OCc1ccc(F)cc1
COc1ccc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)C(F)F)c(OCc4ccc(F)cc4)c3)c2C(N)=O)nc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccc(OC)nc3)c2C(N)=O)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)c(OCc2ccc(Cl)cc2)c1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1O[C@@H](C)c1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)cc1OCC1CCCCC1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccccn3)c2C(N)=O)c(OCc2ccc(F)cc2)c1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)F)c(OCc3ccc(F)cc3)c2)n[nH]c1Nc1cnccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCC1CCN(C)CC1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1Oc1cccc(F)c1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)(F)F)cc2)n[nH]c1Nc1cccc(C(F)(F)F)n1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCCc1ccccc1Cl
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccc(C(F)(F)F)cn3)c2C(N)=O)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)c(OCc2cccc(F)c2)c1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)c(OC)c1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCCc1ccccc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCCc1ccccc1F
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCCc1cccc(Cl)c1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cc(C(F)(F)F)ccn3)c2C(N)=O)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1cccc(OC(F)(F)F)c1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1ccc(OC(F)(F)F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1ccc(C(F)(F)F)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)F)c(OCc3ccc(F)cc3)c2)n[nH]c1Nc1cccc(C(F)(F)F)n1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1cccc(C(F)(F)F)c1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCCc1cccc(F)c1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccc4cc(Cl)ccc4n3)c2C(N)=O)cc1OCc1ccc(F)cc1
COCCOc1cc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)N(C)C)cc3)c2C(N)=O)ccn1
CCS(=O)(=O)Nc1ccc(-c2c(C(N)=O)c(Nc3cnccn3)nn2C)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OC1CCCc2cc(F)ccc21
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc3ccc(F)c(Cl)c3)c2)n[nH]c1Nc1cnccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)F)c(OCc3ccc(F)c(F)c3)c2)n[nH]c1Nc1ccccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc3ccccn3)c2)n[nH]c1Nc1cnccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OC(C)(C)c1ccc(F)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1O[C@@H](C)c1ccccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc3ccc(F)cn3)c2)n[nH]c1Nc1cnccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OC1CCCc2ccccc21
CCC(Oc1cc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc3ccc(Cl)cc3)c2)n[nH]c1Nc1cnc(C(F)(F)F)cn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)F)c(OCc3ccc(Cl)cc3)c2)n[nH]c1Nc1cnc(C(F)(F)F)cn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)F)c(OC(c3ccc(F)cc3)C3CCC3)c2)n[nH]c1Nc1cnccn1
N#Cc1cccc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)CC(F)(F)F)cc3)c2C(N)=O)n1
NC(=O)c1c(-c2ccc(CS(=O)(=O)CC(F)(F)F)c(OCc3ccc(F)cc3)c2)n[nH]c1Nc1cnc(C(F)(F)F)cn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc3ccc(F)cc3)c2)n[nH]c1Nc1ccccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc3ccc(F)cn3)c2)n[nH]c1Nc1ccccn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccccn3)c2C(N)=O)cc1OCc1ccc(F)cn1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1ccc(Cl)cn1
C[C@H](Oc1cc(NS(=O)(=O)C(F)F)ccc1-c1n[nH]c(Nc2cnccn2)c1C(N)=O)c1ccc(F)cc1
C[C@H](Oc1cc(NS(=O)(=O)CC(F)(F)F)ccc1-c1n[nH]c(Nc2cnccn2)c1C(N)=O)c1ccc(F)cc1
Cc1cnc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c4ccc(F)cc4)c3)c2C(N)=O)cn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)F)c(OCc3ccc(F)cc3)c2)n[nH]c1Nc1cnc(C(F)(F)F)cn1
CCS(=O)(=O)Nc3ccc(c2n[nH]c(Nc1cnccn1)c2C#N)cc3OC5(c4ccc(F)c(C)c4)CC5
CCS(=O)(=O)Nc3ccc(c2n[nH]c(Nc1cnccn1)c2C#N)cc3OC5(c4ccc(F)cc4)CC5
C[C@H](Oc1cc(-c2n[nH]c(Nc3cccc(C(F)(F)F)n3)c2C(N)=O)ccc1NS(=O)(=O)CC(F)(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(Cl)cc1
C[C@H](Oc1cc(-c2c(C(N)=O)c(Nc3cnccn3)nn2C)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@@H](Oc1cc(NS(=O)(=O)CC(F)(F)F)ccc1-c1n[nH]c(Nc2cnccn2)c1C(N)=O)c1ccc(F)cc1
C[C@@H](Oc1cc(NS(=O)(=O)C(F)F)ccc1-c1n[nH]c(Nc2cnccn2)c1C(N)=O)c1ccc(F)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)ccc1NS(=O)(=O)CC(F)(F)F)c1cccc(Cl)c1
NC(=O)c1cccc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)C(F)F)cc3)c2C(N)=O)n1
N#Cc1cccc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)C(F)F)cc3)c2C(N)=O)n1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)ccc1NS(=O)(=O)CC(F)(F)F)c1ccc(Cl)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3ccccn3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1OCc1ccccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc3ccc(Cl)cn3)c2)n[nH]c1Nc1cnccn1
CCC(Oc1cc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)ccc1NS(=O)(=O)CC)c1ccc(F)cc1
Cc1cnc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)CC(F)(F)F)c(O[C@@H](C)c4ccc(F)cc4)c3)c2C(N)=O)cn1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)ccc1NS(=O)(=O)CC(F)(F)F)c1cccc(F)c1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OC(c3ccc(F)cc3)C3CCC3)c2)n[nH]c1Nc1cnccn1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)ccc1NS(=O)(=O)CC(F)(F)F)c1ccccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)cc2)n[nH]c1Nc1ccccn1
NC(=O)c1c(-c2ccc(NS(=O)(=O)CC(F)(F)F)c(OCc3ccc(Cl)cc3)c2)n[nH]c1Nc1ccccn1
Cc1nn(C)cc1Nc1[nH]nc(-c2ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c3ccc(F)cc3)c2)c1C(N)=O
C[C@@H](Oc1cc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1O[C@@H](COC)c1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)cc1O[C@H](COC)c1ccc(F)cc1
CCc1cc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c4ccc(F)cc4)c3)c2C(N)=O)no1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)F)c(OCc3nccs3)c2)n[nH]c1Nc1cnccn1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cc(C4(C)CC4)on3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cc(C(F)(F)F)n(C)n3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3ccc(C4CCOCC4)cn3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@@H](Oc1cc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)ccc1CS(=O)(=O)C(F)F)c1ncco1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)ccc1CS(=O)(=O)C(F)F)c1ncco1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cc(C4CCC4)on3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cc(C(C)(C)C)on3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3ncn(C)n3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
Cc1nc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c4ccc(F)cc4)c3)c2C(N)=O)sc1C
Cc1cc(Nc2[nH]nc(-c3ccc(CS(=O)(=O)C(F)F)c(O[C@@H](C)c4ccc(F)cc4)c3)c2C(N)=O)nn1C
Cc1cn(C)nc1Nc1[nH]nc(-c2ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c3ccc(F)cc3)c2)c1C(N)=O
C[C@H](Oc1cc(-c2n[nH]c(Nc3cc(C4CCOCC4)ccn3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
COCC(C)(C)c1cc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c4ccc(F)cc4)c3)c2C(N)=O)no1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cc(C4(C(F)(F)F)CC4)on3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
Cc1cnc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)C(F)F)c(OC4(c5ccc(F)cc5)CC4)c3)c2C(N)=O)cn1
Cc1ccc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)C(F)F)c(OCc4ccc(F)c(F)c4)c3)c2C(N)=O)nc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cc(C4(C)COC4)on3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CC(Oc1cc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ncco1
COc1cc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c4ccc(F)cc4)c3)c2C(N)=O)nn1C
C[C@H](Oc1cc(-c2n[nH]c(Nc3cc(C(C)(C)C)no3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cnc(C4CCOCC4)cn3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cc(C(C)(C)F)on3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
COCC(Oc1cc(-c2n[nH]c(Nc3cc(C)on3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CCS(=O)(=O)Cc1ccc(-c2n[nH]c(Nc3cc(C)on3)c2C(N)=O)cc1O[C@@H](COC)c1ccc(F)cc1
CCS(=O)(=O)Cc1ccc(-c2n[nH]c(Nc3cc(C)on3)c2C(N)=O)cc1O[C@H](COC)c1ccc(F)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cc(C4(C)CCOCC4)on3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
Cc1cc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c4ccc(F)cc4)c3)c2C(N)=O)on1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cc(C4CCOCC4)on3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cc(C45CC6CC(CC(C6)C4)C5)on3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cc(C4CCOC4)on3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cnn(C4CCOCC4)c3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)F)c(OC3(c4ccc(F)cc4)CC3)c2)n[nH]c1Nc1cnccn1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cc4n(n3)CCOC4)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
Cc1nccc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c4ccc(F)cc4)c3)c2C(N)=O)n1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cc(C4CC4)on3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cc(C)on3)c2C(N)=O)cc1O[C@@H](C)c1ccc(F)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cnc(C(C)(C)C)cn3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
NC(=O)c1c(-c2ccc(NS(=O)(=O)C(F)F)c(OCc3ncco3)c2)n[nH]c1Nc1cnccn1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cc(C(F)F)on3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccc(C(=O)O)cn3)c2C(N)=O)cc1O[C@@H](C)c1ccc(F)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cnc(C4CC4)cn3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3cc(C)on3)c2C(N)=O)cc1O[C@@H](C)c1ccc(F)cc1
C[C@H](Oc1cc(-c2n[nH]c(Nc3cc4n(n3)CCCN(C)C4)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
COCC(Oc1cc(-c2n[nH]c(Nc3cnccn3)c2C(N)=O)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
Cc1cc(Nc2c(C(N)=O)c(-c3ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c4ccc(F)cc4)c3)nn2C)no1
Cn1nc(-c2ccc(NS(=O)(=O)C(F)F)c(OCc3ccc(F)cc3)c2)c2c(N)nccc21
C[C@H](Oc1cc(-c2cnn3ccnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4ccncn4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(C4CCN(C)CC4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(C4=CCOCC4)cnc(N)c23)ccc1NS(=O)(=O)CC(F)(F)F)c1ccc(F)cc1
CC(C)n1nc(-c2ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c3ccc(F)cc3)c2)c2c(N)nccc21
CC(C)n1nc(-c2ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c3ccc(F)cc3)c2)c2c(N)ncc(C3=CCCNC3)c21
C[C@H](Oc1cc(-c2nn(C)c3c(C4=CCCN(C)C4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2cccc3[nH]nc(N)c23)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2ncn3ccnc(N)c23)cc1OCc1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(-c2cnn3ccnc(N)c23)cc1OCc1ccc(F)cc1
Nc1n[nH]c2ccnc(-c3ccc(NS(=O)(=O)CC(F)(F)F)c(OCc4ccc(F)cc4)c3)c12
Nc1n[nH]c2nccc(-c3ccc(NS(=O)(=O)C(F)F)c(OCc4ccc(F)cc4)c3)c12
Nc1n[nH]c2nccc(-c3ccc(NS(=O)(=O)CC(F)(F)F)c(OCc4ccc(F)cc4)c3)c12
Nc1n[nH]c2ccnc(-c3ccc(NS(=O)(=O)C(F)F)c(OCc4ccc(F)cc4)c3)c12
Nc1n[nH]c2ncnc(-c3ccc(NS(=O)(=O)C(F)F)c(OCc4ccc(F)cc4)c3)c12
Cc1cc(-c2ccc(NS(=O)(=O)C(F)F)c(OCc3ccc(F)cc3)c2)c2c(N)n[nH]c2n1
Nc1n[nH]c2nc(-c3ccccc3)cc(-c3ccc(NS(=O)(=O)C(F)F)c(OCc4ccc(F)cc4)c3)c12
C[C@H](Oc1cc(-c2ccnc3[nH]nc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCCNCC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CN(CC(F)(F)F)C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(C#CC4CCNCC4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(C#CC4CCN(C)CC4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(CC5CCCN5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5(CN)CC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn5c4CN(C)CC5)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5(CC#N)COC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CC6(C5)CN(C)C6)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCC(C)(C)N(C)C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4ccc(N5CCNCC5)nc4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
CC(=O)N1CCC(n2cc(-c3cnc(N)c4c(-c5ccc(NS(=O)(=O)C(F)F)c(O[C@@H](C)c6ccc(F)cc6)c5)nn(C)c34)cn2)CC1
COC[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCOCC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
COC[C@@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCOCC5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCC(F)(F)C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
Nc1ncc(-c2cnn(C3CCOCC3)c2)c2[nH]nc(-c3ccc(NS(=O)(=O)C(F)F)c(OCc4cccc(Cl)c4)c3)c12
C[C@H](Oc1cc(-c2nn(C)c3c(N4CCOCC4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn(C5CCN(C)C(C(F)(F)F)C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
C[C@H](Oc1cc(-c2nn(C)c3c(-c4cnn([C@@H]5CCN(C)C(C)(C)C5)c4)cnc(N)c23)ccc1NS(=O)(=O)C(F)F)c1ccc(F)cc1
Cn1c2nc(Nc3ccc4[nH]ccc4c3)ncc2cc(c1=O)S(=O)(=O)c1ccc(F)cc1F
CC(C)(C)S(=O)(=O)c1ccc2nccc(Nc3n[nH]c4ccc(F)cc34)c2c1
CC(C)(C)NS(=O)(=O)c1cncc(c1)-c1ccn2nc(N)nc2c1
CCOC1=CS(=O)(=O)c2cc3c(Nc4ccc5scnc5c4)ncnc3cc12 |t:3|
CC(C)n1cc(C2=C(C(=O)N(O)C2=O)c2c[nH]c3ccccc23)c2ccccc12 |t:6|
O=C1NC(=O)C(=C1c1cn(CCCCCC#N)c2ccccc12)c1cn(CCCCCC#N)c2ccccc12 |c:5|
CCn1cc(C2=C(C(=O)N(O)C2=O)c2cn(C(C)C)c3ccccc23)c2ccccc12 |t:5|
Cn1cc(C2=C(C(=O)N(O)C2=O)c2c[nH]c3ccccc23)c2ccccc12 |t:4|
Cn1cc(C2=C(C(=O)N(O)C2=O)c2cn(C)c3ccccc23)c2ccccc12 |t:4|
ON1C(=O)C(=C(C1=O)c1cn(CCCCCC#N)c2ccccc12)c1cn(CCCCCC#N)c2ccccc12 |c:4|
ON1C(=O)C2=C(C1=O)c1cn(CCCCCCn3cc2c2ccccc32)c2ccccc12 |c:4|
CC(C)n1cc(C2=C(C(=O)N(O)C2=O)c2cn(C)c3ccccc23)c2ccccc12 |t:6|
Cn1cc(C2=C(C(=O)N(O)C2=O)c2cn(CCCCCC(O)=O)c3ccccc23)c2ccccc12 |t:4|
Cn1cc(C2=C(C(=O)N(O)C2=O)c2cn(CCCCCC#N)c3ccccc23)c2ccccc12 |t:4|
ON1C(=O)C(=C(C1=O)c1c[nH]c2ncccc12)c1c[nH]c2ccccc12 |c:4|
Cn1cc(C2=C(C(=O)NC2=O)c2cn(C)c3ncccc23)c2ccccc12 |t:4|
ON1C(=O)C(=C(C1=O)c1cn(CCCCCC(O)=O)c2ccccc12)c1c[nH]c2ccccc12 |c:4|
CCn1cc(C2=C(C(=O)N(O)C2=O)c2cn(C)c3ccccc23)c2ccccc12 |t:5|
CCn1cc(-c2ccc3N(CCc3c2)C(=O)Cc2cccc(OC(F)(F)F)c2)c2c(N)ncnc12
CN1CCN(CC1)c1ccc2nc(c(-c3ccncc3)n2n1)-c1cccc(c1)-c1ccccc1
CN1CCN(CC1)c1ccc2nc(c(-c3ccncc3)n2n1)-c1cccc(c1)C(=O)N1CCOCC1
CN1CCN(CC1)c1ccc2nc(c(-c3ccncc3)n2c1)-c1cccc2OCOc12
CN1CCN(CC1)c1ccc2nc(c(-c3cccnc3)n2n1)-c1cccc2OCOc12
CN1CCN(CC1)c1ccc2nc(c(-c3ccncc3)n2n1)-c1cccc(c1)-c1cccs1
CCOc1ccc2c(cccc2c1)-c1nc2ccc(nn2c1-c1ccncc1)N1CCN(C)CC1
CN1CCN(CC1)c1ccc2nc(c(-c3ccncc3)n2n1)-c1ccc2OCCOc2c1
CN1CCN(CC1)c1ccc2nc(c(-c3ccncc3)n2n1)-c1cccc2OCOc12
CN1CCN(CC1)c1ccc2nc(-c3ccc(s3)-c3ccccc3)c(-c3ccncc3)n2n1
CN1CCN(CC1)c1ccc2nc(c(-c3ccncc3)n2n1)-c1cccc2OCCOc12
C1Oc2cccc(c2O1)-c1nc2cccnn2c1-c1ccncc1
CN1CCN(CC1)c1ccc2nc(c(-c3ccncc3)n2n1)-c1ccc(cc1)-c1ccccc1
CN1CCN(CC1)c1ccc2nc(c(-c3ccncc3)n2n1)-c1ccc2ncsc2c1
COc1ccc2c(cccc2c1)-c1nc2ccc(nn2c1-c1ccncc1)N1CCN(C)CC1
CN1CCN(CC1)c1ccc2nc(c(-c3ccccc3)n2n1)-c1cccc2OCOc12
CN1CCN(CC1)c1ccc2nc(c(-c3ccncc3)n2n1)-c1cccc(c1)-c1ccsc1
CN1CCN(CC1)c1ccc2nc(c(-c3ccncc3)n2n1)-c1cccc2ccccc12
CN1CCN(CC1)c1ccc2nc(c(-c3ccncc3)n2n1)-c1ccc(cc1)C(=O)N1CCOCC1
CN1CCN(CC1)c1ccc2nc(c(-c3ccncc3)n2n1)-c1ccc2OCOc2c1
Oc1c(Br)cc(\C=C2/C(=O)Nc3ccc(I)cc23)cc1Br
Fc1ccc(cc1)-n1cccc(C(=O)Nc2ccc(Oc3ccncc3)c3ccccc23)c1=O
Cc1ccc(COC(=O)Nc2cc(ccn2)-c2cc3c(CCNC3=O)[nH]2)cc1
Fc1ccc(cc1)-n1cccc(C(=O)Nc2ccc(Oc3ccnc4[nH]ccc34)c(F)c2)c1=O
c1cc(ccc1N2C=CC=C(C2=O)C(=O)Nc3ccc(c(c3)F)Oc4ccnc(c4)NC(=O)C5CC5)F
Fc1ccc(cc1)-n1cccc(C(=O)Nc2ccc(Oc3ccncc3)c(F)c2)c1=O
Cc1cc(NC(=O)c2cccn(-c3ccc(F)cc3)c2=O)ccc1Oc1ccnc(NC(=O)C2CC2)c1
Cc1cc(NC(=O)c2cccn(-c3ccc(F)cc3)c2=O)cc(C)c1Oc1ccnc(NC(=O)C2CC2)c1
Cc1cc(NC(=O)c2cccn(-c3ccc(F)cc3)c2=O)cc(C)c1Oc1ccncc1
Fc1ccc(cc1)-c1cccc(c1)C(=O)Nc1ccc(Oc2ccncc2)c(F)c1
Nc1ccc(nc1)C#Cc1c(N)nccc1Oc1ccc(NC(=O)c2cccn(-c3ccc(F)cc3)c2=O)cc1F
CC#Cc1c(N)nccc1Oc1ccc(NC(=O)c2cccn(-c3ccc(F)cc3)c2=O)cc1F
Cc1c(C)c(Oc2ccncc2)ccc1NC(=O)c1cccn(-c2ccc(F)cc2)c1=O
Cc1c(c(ccc1NC(=O)C2=CC=CN(C2=O)c3ccc(cc3)F)Oc4ccnc(c4)NC(=O)C5CC5)C
[H][C@@]12CCC(=O)[C@]3(C)[C@@H](CCC(C)(C)[C@@]3([H])C[C@@H](O)C(=C1)C(=O)[C@H]2C)OC(C)=O |r,t:20|
Cc1ccc(cc1C#Cc2cnc3n2nccc3)C(=O)Nc4ccc(c(c4)C(F)(F)F)CN5CCN(CC5)C
CNC(=O)c1cc(ccn1)Oc2ccc(cc2)NC(=O)Nc3ccc(c(c3)C(F)(F)F)Cl
CC(C)(C)c1nc(c(s1)c2ccnc(n2)N)c3cccc(c3F)NS(=O)(=O)c4c(cccc4F)F
C[C@@H](Oc1cc(cnc1N)-c1cnn(c1)C1CCNCC1)c1c(Cl)ccc(F)c1Cl |r|
CC(=O)Nc1nc2ccc(cc2s1)-c1cnc(Cl)c(CC(=O)Cc2ccccc2)c1
CC(=O)Nc1nc2ccc(cc2s1)-c1cnc(C)c(CC(=O)OC2CCCCC2)c1
Cc1ccc(CCCCN2C(=O)N[C@H](Cc3c[nH]c4c(Cl)cccc34)C2=O)cc1C#Cc1cnc2cccnn12 |r|
c1ccc(cc1)[C@H](C(=O)Nc2ccc(cc2)F)OC(=O)c3c(nccn3)N
Fc1ccc(Oc2ccc3nc(NC(=O)C4CC4)sc3c2)cc1NC(=O)Cc1ccc2OCOc2c1
CC(=O)c1cccc(NC(=O)Nc2cc(Oc3ccc4nc(NC(=O)C5CC5)sc4c3)ccc2F)c1
c1cc(cc(c1)C(F)(F)F)CC(=O)Nc2cc(ccc2F)Oc3ccc4c(c3C#N)sc(n4)NC(=O)C5CC5
Fc1ccc(Oc2ccc3nc(NC(=O)C4CC4)sc3c2)cc1NC(=O)Cc1cccc(c1)C(F)(F)F
Fc1ccc(Oc2ccc3nc(NC(=O)C4CC4)sc3c2)cc1NC(=O)Cc1cccc(c1F)C(F)(F)F
Fc1ccc(Oc2ccc3nc(NC(=O)C4CC4)sc3c2)cc1NC(=O)Cc1ccc(F)c(c1)C(F)(F)F
[O-][N+](=O)c1cccc(CC(=O)Nc2cc(Oc3ccc4nc(NC(=O)C5CC5)sc4c3)ccc2F)c1
COc1cccc(CC(=O)Nc2cc(Oc3ccc4nc(NC(=O)C5CC5)sc4c3)ccc2F)c1
Fc1ccc(Oc2ccc3nc(NC(=O)C4CC4)sc3c2)cc1NC(=O)Cc1cccc(n1)C(F)(F)F
Fc1ccc(Oc2ccc3nc(NC(=O)C4CC4)sc3c2)cc1NC(=O)CCc1cccc(c1)C(F)(F)F
Cc1cccc(NC(=O)Nc2cc(Oc3ccc4nc(NC(=O)C5CC5)sc4c3)ccc2F)c1
Fc1ccc(Oc2ccc3nc(NC(=O)C4CC4)sc3c2)cc1NC(=O)Nc1cccc(Br)c1
Cc1cccc(CC(=O)Nc2cc(Oc3ccc4nc(NC(=O)C5CC5)sc4c3)ccc2F)c1
Cn1cc(CC(=O)Nc2cc(Oc3ccc4nc(NC(=O)C5CC5)sc4c3)ccc2F)c2ccccc12
COc1cccc(NC(=O)Nc2cc(Oc3ccc4nc(NC(=O)C5CC5)sc4c3)ccc2F)c1
Fc1ccc(Oc2ccc3nc(NC(=O)C4CC4)sc3c2)cc1NC(=O)Cc1cccc(OC(F)(F)F)c1
Cc1ccc(CC(=O)Nc2cc(Oc3ccc4nc(NC(=O)C5CC5)sc4c3)ccc2F)cc1C
Fc1ccc(Oc2ccc3nc(NC(=O)C4CC4)sc3c2)cc1NC(=O)Cc1cccc(c1)C#N
CCOC(=O)c1cccc(NC(=O)Nc2cc(Oc3ccc4nc(NC(=O)C5CC5)sc4c3)ccc2F)c1
CNC(=O)c1ccc2n(cnc2c1)-c1ccc(CC(=O)OC(C)(C)C)cc1
CCCCNc1nc2ccc(cc2[nH]1)[N+]([O-])=O
CCCCNc1nc2cc(ccc2s1)[N+]([O-])=O
O=S1(=O)CC2(OCCO2)c2cc3nccc(Nc4ccc5scnc5c4)c3cc12
CC1(C)CC1C(=O)Nc1nc2ccc(Oc3ccc(F)c(NC(=O)Cc4cccc(c4)C(F)(F)F)c3)cc2s1
CC1(C)C[C@H]1C(=O)Nc1nc2ccc(Oc3ccc(F)c(NC(=O)Cc4cccc(c4)C(F)(F)F)c3)cc2s1 |r|
CC1(C)C[C@@H]1C(=O)Nc1nc2ccc(Oc3ccc(F)c(NC(=O)Cc4cccc(c4)C(F)(F)F)c3)cc2s1 |r|
Fc1ccc(Oc2cc3nc(NC(=O)C4CC4)sc3cc2F)cc1NC(=O)Cc1cccc(c1)C(F)(F)F
Fc1ccc(Oc2cc3nc(NC(=O)C4CC4)sc3cc2F)cc1NC(=O)Cc1cccc(OC(F)(F)F)c1
Fc1ccc(Oc2cc3nc(NC(=O)C4CCOC4)sc3cc2F)cc1NC(=O)Cc1cccc(OC(F)(F)F)c1
Fc1ccc(Oc2cc3nc(NC(=O)C4CC(=O)C4)sc3cc2F)cc1NC(=O)Cc1cccc(OC(F)(F)F)c1
Fc1ccc(Oc2cc3nc(NC(=O)C4CCC(=O)C4)sc3cc2F)cc1NC(=O)Cc1cccc(OC(F)(F)F)c1
Fc1ccc(Oc2cc3nc(NC(=O)C4CCC(=O)CC4)sc3cc2F)cc1NC(=O)Cc1cccc(OC(F)(F)F)c1
CC1(C)CC1C(=O)Nc1nc2cc(Oc3ccc(F)c(NC(=O)Cc4cccc(OC(F)(F)F)c4)c3)c(F)cc2s1
FC1CC1C(=O)Nc1nc2cc(Oc3ccc(F)c(NC(=O)Cc4cccc(OC(F)(F)F)c4)c3)c(F)cc2s1
Cc1ccc(-c2cn([C@@H]3CC[C@H](N)CC3)c3ncnc(N)c23)c(F)c1 |r,wU:8.7,11.11,(2.17,7.19,;1.77,5.71,;.28,5.31,;-.11,3.82,;.97,2.74,;.58,1.25,;1.48,0,;.58,-1.24,;.97,-2.73,;-.11,-3.82,;.28,-5.31,;1.77,-5.71,;2.17,-7.19,;2.86,-4.62,;2.46,-3.13,;-.89,-.77,;-2.22,-1.54,;-3.56,-.77,;-3.56,.77,;-2.22,1.54,;-2.22,3.08,;-.89,.77,;2.47,3.14,;3.56,2.05,;2.86,4.62,)|
CN(c1ccc(cc1)NC(=O)Nc2ccc(cc2)OC(F)(F)F)c3ccnc(n3)Nc4cccc(c4)S(=O)(=O)N
CN(c1ccc(cc1)NC(=O)Nc2cc(ccc2F)C(F)(F)F)c3ccnc(n3)Nc4cccc(c4)S(=O)(=O)N
Fc1ccc(Oc2ccc3nc(NC(=O)C4CC4)sc3c2)cc1NC(=O)Cc1cccc(Br)c1
Fc1ccc(Oc2cc3sc(NC(=O)C4CC4)nc3cc2F)cc1NC(=O)Cc1cccc(c1)C(F)(F)F
CN1c2ccccc2OC[C@H](NC(=O)c2cc3cccc(-c4ccccc4)c3[nH]2)C1=O |r|
Cc1cc(-c2cnc(N)c3c(csc23)-c2ccc3scnc3c2)n(C)n1
CC(C)S(=O)(=O)c1ccc2c(c1)c(ccn2)Nc3ccc4c(c3)ncs4
O=S1(=O)C=C(C2CC2)c2cc3nccc(Nc4ccc5scnc5c4)c3cc12
Cc1ccc(Oc2ccnc3cc(ccc23)-c2cnn(c2)C2CCNCC2)cc1
Cc1ccc(O)cc1Nc1ccnc2cc(ccc12)-c1ccccn1
Fc1ccc(cc1NC(=O)Cc1cccc(OC(F)(F)F)c1)-c1ccc2nc(NC(=O)C3CC3)sc2c1
Fc1c(NC(=O)Cc2cccc(OC(F)(F)F)c2)cccc1-c1ccc2nc(NC(=O)C3CC3)sc2c1
CC(C)C(=O)NC1CCC(CC1)C(=O)Nc1nc2cc(F)c(Oc3ccc(F)c(NC(=O)Cc4cccc(c4)C(F)(F)F)c3)cc2s1 |(-12.06,-2.87,;-13.6,-2.87,;-14.37,-4.21,;-14.37,-1.54,;-15.91,-1.54,;-13.6,-.21,;-12.06,-.21,;-11.29,1.13,;-9.75,1.13,;-8.98,-.21,;-9.75,-1.54,;-11.29,-1.54,;-7.44,-.21,;-6.67,-1.54,;-6.67,1.13,;-5.13,1.13,;-4.23,-.12,;-2.76,.36,;-1.43,-.41,;-.09,.36,;1.24,-.41,;-.09,1.9,;1.24,2.67,;2.57,1.9,;2.57,.36,;3.91,-.41,;5.24,.36,;6.57,-.41,;5.24,1.9,;6.57,2.67,;7.91,1.9,;7.91,.36,;9.24,2.67,;10.58,1.9,;10.58,.36,;11.91,-.41,;13.24,.36,;13.24,1.9,;11.91,2.67,;14.58,2.67,;15.91,3.44,;15.91,1.9,;14.58,4.21,;3.91,2.67,;-1.43,2.67,;-2.76,1.9,;-4.23,2.37,)|
CCCCC(=O)NC1CCC(CC1)C(=O)Nc1nc2cc(F)c(Oc3ccc(F)c(NC(=O)Cc4cccc(c4)C(F)(F)F)c3)cc2s1 |(-9.75,-4.21,;-11.29,-4.21,;-12.06,-2.87,;-13.6,-2.87,;-14.37,-1.54,;-15.91,-1.54,;-13.6,-.21,;-12.06,-.21,;-11.29,1.13,;-9.75,1.13,;-8.98,-.21,;-9.75,-1.54,;-11.29,-1.54,;-7.44,-.21,;-6.67,-1.54,;-6.67,1.13,;-5.13,1.13,;-4.23,-.12,;-2.76,.36,;-1.43,-.41,;-.09,.36,;1.24,-.41,;-.09,1.9,;1.24,2.67,;2.57,1.9,;2.57,.36,;3.91,-.41,;5.24,.36,;6.57,-.41,;5.24,1.9,;6.57,2.67,;7.91,1.9,;7.91,.36,;9.24,2.67,;10.58,1.9,;10.58,.36,;11.91,-.41,;13.24,.36,;13.24,1.9,;11.91,2.67,;14.58,2.67,;15.91,3.44,;15.91,1.9,;14.58,4.21,;3.91,2.67,;-1.43,2.67,;-2.76,1.9,;-4.23,2.37,)|
Fc1ccc(Oc2cc3sc(NC(=O)C4CCC(CC4)NC(=O)CCCl)nc3cc2F)cc1NC(=O)Cc1cccc(c1)C(F)(F)F |(6.57,-.41,;5.24,.36,;3.91,-.41,;2.57,.36,;2.57,1.9,;1.24,2.67,;-.09,1.9,;-1.43,2.67,;-2.76,1.9,;-4.23,2.37,;-5.13,1.13,;-6.67,1.13,;-7.44,-.21,;-6.67,-1.54,;-8.98,-.21,;-9.75,1.13,;-11.29,1.13,;-12.06,-.21,;-11.29,-1.54,;-9.75,-1.54,;-13.6,-.21,;-14.37,-1.54,;-15.91,-1.54,;-13.6,-2.87,;-12.06,-2.87,;-11.29,-4.21,;-4.23,-.12,;-2.76,.36,;-1.43,-.41,;-.09,.36,;1.24,-.41,;3.91,2.67,;5.24,1.9,;6.57,2.67,;7.91,1.9,;7.91,.36,;9.24,2.67,;10.58,1.9,;10.58,.36,;11.91,-.41,;13.24,.36,;13.24,1.9,;11.91,2.67,;14.58,2.67,;15.91,3.44,;15.91,1.9,;14.58,4.21,)|
COCC(=O)NC1CCC(CC1)C(=O)Nc1nc2cc(F)c(Oc3ccc(F)c(NC(=O)Cc4cccc(c4)C(F)(F)F)c3)cc2s1 |(-11.29,-4.21,;-12.06,-2.87,;-13.6,-2.87,;-14.37,-1.54,;-15.91,-1.54,;-13.6,-.21,;-12.06,-.21,;-11.29,1.13,;-9.75,1.13,;-8.98,-.21,;-9.75,-1.54,;-11.29,-1.54,;-7.44,-.21,;-6.67,-1.54,;-6.67,1.13,;-5.13,1.13,;-4.23,-.12,;-2.76,.36,;-1.43,-.41,;-.09,.36,;1.24,-.41,;-.09,1.9,;1.24,2.67,;2.57,1.9,;2.57,.36,;3.91,-.41,;5.24,.36,;6.57,-.41,;5.24,1.9,;6.57,2.67,;7.91,1.9,;7.91,.36,;9.24,2.67,;10.58,1.9,;10.58,.36,;11.91,-.41,;13.24,.36,;13.24,1.9,;11.91,2.67,;14.58,2.67,;15.91,3.44,;15.91,1.9,;14.58,4.21,;3.91,2.67,;-1.43,2.67,;-2.76,1.9,;-4.23,2.37,)|
CCOCC(=O)NC1CCC(CC1)C(=O)Nc1nc2cc(F)c(Oc3ccc(F)c(NC(=O)Cc4cccc(c4)C(F)(F)F)c3)cc2s1 |(-9.75,-4.21,;-11.29,-4.21,;-12.06,-2.87,;-13.6,-2.87,;-14.37,-1.54,;-15.91,-1.54,;-13.6,-.21,;-12.06,-.21,;-11.29,1.13,;-9.75,1.13,;-8.98,-.21,;-9.75,-1.54,;-11.29,-1.54,;-7.44,-.21,;-6.67,-1.54,;-6.67,1.13,;-5.13,1.13,;-4.23,-.12,;-2.76,.36,;-1.43,-.41,;-.09,.36,;1.24,-.41,;-.09,1.9,;1.24,2.67,;2.57,1.9,;2.57,.36,;3.91,-.41,;5.24,.36,;6.57,-.41,;5.24,1.9,;6.57,2.67,;7.91,1.9,;7.91,.36,;9.24,2.67,;10.58,1.9,;10.58,.36,;11.91,-.41,;13.24,.36,;13.24,1.9,;11.91,2.67,;14.58,2.67,;15.91,3.44,;15.91,1.9,;14.58,4.21,;3.91,2.67,;-1.43,2.67,;-2.76,1.9,;-4.23,2.37,)|
Fc1ccc(Oc2cc3sc(NC(=O)C4CCC(CC4)NC(=O)c4cccs4)nc3cc2F)cc1NC(=O)Cc1cccc(c1)C(F)(F)F |(6.57,.14,;5.24,.91,;3.91,.14,;2.57,.91,;2.57,2.45,;1.24,3.22,;-.09,2.45,;-1.43,3.22,;-2.76,2.45,;-4.23,2.92,;-5.13,1.68,;-6.67,1.68,;-7.44,.34,;-6.67,-.99,;-8.98,.34,;-9.75,1.68,;-11.29,1.68,;-12.06,.34,;-11.29,-.99,;-9.75,-.99,;-13.6,.34,;-14.37,-.99,;-15.91,-.99,;-13.6,-2.32,;-12.07,-2.48,;-11.75,-3.99,;-13.08,-4.76,;-14.23,-3.73,;-4.23,.43,;-2.76,.91,;-1.43,.14,;-.09,.91,;1.24,.14,;3.91,3.22,;5.24,2.45,;6.57,3.22,;7.91,2.45,;7.91,.91,;9.24,3.22,;10.58,2.45,;10.58,.91,;11.91,.14,;13.24,.91,;13.24,2.45,;11.91,3.22,;14.58,3.22,;15.91,3.99,;15.91,2.45,;14.58,4.76,)|
CCS(=O)(=O)NC1CCC(CC1)C(=O)Nc1nc2cc(F)c(Oc3ccc(F)c(NC(=O)Cc4cccc(c4)C(F)(F)F)c3)cc2s1 |(-14.4,-4.21,;-13.63,-2.87,;-14.4,-1.54,;-15.49,-.45,;-15.88,-1.94,;-13.63,-.21,;-12.09,-.21,;-11.32,1.13,;-9.78,1.13,;-9.01,-.21,;-9.78,-1.54,;-11.32,-1.54,;-7.47,-.21,;-6.7,-1.54,;-6.7,1.13,;-5.16,1.13,;-4.25,-.12,;-2.79,.36,;-1.45,-.41,;-.12,.36,;1.21,-.41,;-.12,1.9,;1.21,2.67,;2.55,1.9,;2.55,.36,;3.88,-.41,;5.21,.36,;6.55,-.41,;5.21,1.9,;6.55,2.67,;7.88,1.9,;7.88,.36,;9.22,2.67,;10.55,1.9,;10.55,.36,;11.88,-.41,;13.22,.36,;13.22,1.9,;11.88,2.67,;14.55,2.67,;15.88,3.44,;15.88,1.9,;14.55,4.21,;3.88,2.67,;-1.45,2.67,;-2.79,1.9,;-4.25,2.37,)|
CN1c2ccccc2OC[C@H](NC(=O)c2n[nH]c(Cc3ccccc3)n2)C1=O |r|
CN1C(=O)[C@@H](NC(=O)c2ccc3[nH]cc(-c4ccccc4)c3c2)COc2ccccc21
CN1C(=O)[C@@H](NC(=O)c2ccc3[nH]cc(-c4ccccc4F)c3c2)COc2ccccc21
CN1C(=O)[C@@H](NC(=O)c2ccc3[nH]cc(-c4cccc(F)c4)c3c2)COc2ccccc21
Cc1ccccc1-c1c[nH]c2ccc(C(=O)N[C@H]3COc4ccccc4N(C)C3=O)cc12
Cc1ccc(-c2c[nH]c3ccc(C(=O)N[C@H]4COc5ccccc5N(C)C4=O)cc23)cc1
CN1C(=O)[C@@H](NC(=O)c2ccc3[nH]cc(-c4ccccc4C(F)(F)F)c3c2)COc2ccccc21
COc1cccc(-c2c[nH]c3ccc(C(=O)N[C@H]4COc5ccccc5N(C)C4=O)cc23)c1
CN1C(=O)[C@@H](NC(=O)c2ccc3[nH]cc(-c4ccc(-c5ccccc5)cc4)c3c2)COc2ccccc21
CN1C(=O)[C@@H](NC(=O)c2ccc3[nH]cc(-c4cccc(F)c4F)c3c2)COc2ccccc21
CN1C(=O)[C@@H](NC(=O)c2ccc3[nH]cc(-c4ccc(F)cc4F)c3c2)COc2ccccc21
CN1C(=O)[C@@H](NC(=O)c2ccc3[nH]cc(-c4cc(F)ccc4F)c3c2)COc2ccccc21
CN1C(=O)[C@@H](NC(=O)c2ccc3[nH]cc(-c4c(F)cccc4F)c3c2)COc2ccccc21
Cc1cccc(-c2c[nH]c3ccc(C(=O)N[C@H]4COc5ccccc5N(C)C4=O)cc23)c1C
Cc1ccc(-c2c[nH]c3ccc(C(=O)N[C@H]4COc5ccccc5N(C)C4=O)cc23)c(C)c1
Cc1ccc(C)c(-c2c[nH]c3ccc(C(=O)N[C@H]4COc5ccccc5N(C)C4=O)cc23)c1
Cc1ccc(-c2c[nH]c3ccc(C(=O)N[C@H]4COc5ccccc5N(C)C4=O)cc23)cc1C
COc1ccc(-c2c[nH]c3ccc(C(=O)N[C@H]4COc5ccccc5N(C)C4=O)cc23)c(OC)c1
COc1ccc(-c2c[nH]c3ccc(C(=O)N[C@H]4COc5ccccc5N(C)C4=O)cc23)cc1OC
CN1C(=O)[C@@H](NC(=O)c2ccc3[nH]cc(-c4cccc5ccccc45)c3c2)COc2ccccc21
Cc1ccc(C(=O)Nc2ccccc2)cc1-c1ccc2nc(NCCN3CCOCC3)ncc2c1
CNC(=O)c1cc(Oc2ccc(NC(=O)Nc3cc(nn3-c3ccc4ncccc4c3)C(C)(C)C)c(F)c2)ccn1
Cc1ccc(F)c(NC(=O)Nc2ccc(cc2)-c2cccc3[nH]nc(N)c23)c1
CN1C(=O)N(Cc2cnc(Nc3ccc(C)nc3)nc12)c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C
COc1cc(CCc2cc(NC(=O)c3ccc(cc3)N3C[C@H](C)N[C@H](C)C3)n[nH]2)cc(OC)c1
Cc1ccc(CCCCN2C(=O)NC(Cc3c[nH]c4c(Cl)cccc34)C2=O)cc1C#Cc1cnc2cccnn12
CN1C(=O)[C@@H](Cc2c[nH]c3c(Cl)c(F)ccc23)N(C=O)C1=O
CC(C)(C)c1cc(NC(=O)Nc2ccc(cc2)-c2cn3c(n2)sc2cc(OCCN4CCOCC4)ccc32)no1
CC1(Cn2cc(-c3ccc4c(c3)CCN4C(=O)Cc3cccc(OC(F)(F)F)c3)c3c(N)n[nH]c(=O)c32)COC1
C[C@H](NC(=O)c1cn(C)c2ccc(cc12)-c1ccn2nc(NC(=O)C3CC3)nc2c1)c1cccc(F)c1 |r|
CNC(=O)c1ncn2cc(ncc12)-c1c(F)ccc(NS(=O)(=O)c2cc(Cl)cnc2OC)c1F
CN1C(=S)NC(Cc2c[nH]c3ccccc23)C1=O
C=Cc1cc2c(Nc3ccc4scnc4c3)ncnc2cn1
Clc1ccc(/C=C/c2cc3c(Nc4ccc5scnc5c4)ncnc3cn2)cc1
Cc1ccc(Nc2ncnc3cnc(/C=C/c4ccc(Cl)cc4)cc23)cn1
Cn1nccc1-c1cc2c(Nc3ccc4scnc4c3)ncnc2cc1Cl
Cn1nc(C(F)(F)F)cc1-c1cc2c(Nc3ccc4scnc4c3)ncnc2cc1Cl
c1csc(-c2ccc3ncnc(Nc4ccc5scnc5c4)c3c2)c1
Cc1ncc(-c2ccc3ncnc(Nc4ccc5scnc5c4)c3c2)s1
Cn1cccc1-c1ccc2ncnc(Nc3ccc4scnc4c3)c2c1
Cc1csc(-c2ccc3ncnc(Nc4ccc5scnc5c4)c3c2)n1
Cn1cc(-c2ccc3ncnc(Nc4ccc5scnc5c4)c3c2)cn1
Cc1ccsc1-c1ccc2ncnc(Nc3ccc4scnc4c3)c2c1
c1nc(Nc2ccc3scnc3c2)c2cc(-c3cc[nH]n3)ccc2n1
c1ccc(-c2ccc3ncnc(Nc4ccc5scnc5c4)c3c2)cc1
Cc1cscc1-c1ccc2ncnc(Nc3ccc4scnc4c3)c2c1
OCc1cccc(-c2cc3ncnc(Nc4ccc5scnc5c4)c3cc2-c2cccs2)c1
Cn1cccc1-c1cc2c(Nc3ccc4scnc4c3)ncnc2cc1-c1cccc(CO)c1
Cc1ccsc1-c1cc2c(Nc3ccc4scnc4c3)ncnc2cc1-c1cccc(CO)c1
OCc1ccc(-c2cc3ncnc(Nc4ccc5scnc5c4)c3cc2-c2cccs2)o1
C1=C(c2cc3ncnc(Nc4ccc5scnc5c4)c3cc2-c2cccs2)COC1
O=C(N1CCOCC1)c1ccc(cc1)-c1cc2cccnc2[nH]1
Cc1ccc(C(=O)Nc2cccc(C(F)(F)F)c2)cc1Nc1nc(-c2cccnc2)nc2nn(C)cc12
Cc1ccc(C(=O)Nc2cccc(C(F)(F)F)c2)cc1Nc1nc(-c2cccnc2)nc2c1cnn2C