Affinity DataKi: 0.0500nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
Affinity DataKi: 0.170nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Binding affinity towards melatonin receptor in chicken brain.More data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
Affinity DataKi: 0.210nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
Affinity DataKi: 0.260nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
Affinity DataKi: 0.270nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.330nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
Affinity DataKi: 0.350nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.390nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT1 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.410nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.470nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
National Hellenic Research Foundation
Curated by ChEMBL
National Hellenic Research Foundation
Curated by ChEMBL
Affinity DataKi: 0.480nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in rat brain synaptosomal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
Affinity DataKi: 0.510nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
Affinity DataKi: 0.590nMAssay Description:Binding affinity towards melatonin receptor in chicken brain.More data for this Ligand-Target Pair
Affinity DataKi: 0.660nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1A expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
National Hellenic Research Foundation
Curated by ChEMBL
National Hellenic Research Foundation
Curated by ChEMBL
Affinity DataKi: 0.720nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in rat brain synaptosomal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.740nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.860nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
National Hellenic Research Foundation
Curated by ChEMBL
National Hellenic Research Foundation
Curated by ChEMBL
Affinity DataKi: 0.930nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in rat brain synaptosomal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.950nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
Affinity DataKi: 0.970nMAssay Description:Binding affinity towards melatonin receptor in chicken brain.More data for this Ligand-Target Pair
Affinity DataKi: 1.02nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.12nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT1 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.15nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]CP55940 from CB2 receptor in mouse spleen membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.22nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT1 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.29nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.41nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
National Hellenic Research Foundation
Curated by ChEMBL
National Hellenic Research Foundation
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in rat brain synaptosomal membraneMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
National Hellenic Research Foundation
Curated by ChEMBL
National Hellenic Research Foundation
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in rat brain synaptosomal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.67nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT1 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]CP55940 from CB2 receptor in mouse spleen membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]CP55940 from CB2 receptor in mouse spleen membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.82nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1A expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
National Hellenic Research Foundation
Curated by ChEMBL
National Hellenic Research Foundation
Curated by ChEMBL
Affinity DataKi: 2.70nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in rat brain synaptosomal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2.75nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.94nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
National Hellenic Research Foundation
Curated by ChEMBL
National Hellenic Research Foundation
Curated by ChEMBL
Affinity DataKi: 3.90nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in rat brain synaptosomal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 4.07nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1A expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Displacement of [3H]CP55940 from CB2 receptor in mouse spleen membraneMore data for this Ligand-Target Pair
Affinity DataKi: 4.27nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT1 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.37nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1A expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair