TargetCysteinyl leukotriene receptor 1(Homo sapiens (Human))
University Of Naples "Federico Ii
Curated by ChEMBL
University Of Naples "Federico Ii
Curated by ChEMBL
Affinity DataIC50: 0.260nMAssay Description:Antagonist activity at human CysLT1 receptorMore data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 1(Homo sapiens (Human))
University Of Naples "Federico Ii
Curated by ChEMBL
University Of Naples "Federico Ii
Curated by ChEMBL
Affinity DataIC50: 2.30nMAssay Description:Antagonist activity at human CysLT1 receptorMore data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 1(Homo sapiens (Human))
University Of Naples "Federico Ii
Curated by ChEMBL
University Of Naples "Federico Ii
Curated by ChEMBL
Affinity DataIC50: 4.30nMAssay Description:Antagonist activity at human CysLT1 receptorMore data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University Of Naples "Federico Ii
Curated by ChEMBL
University Of Naples "Federico Ii
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Antagonist activity at human CysLT2 receptorMore data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 1(Homo sapiens (Human))
University Of Naples "Federico Ii
Curated by ChEMBL
University Of Naples "Federico Ii
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity at human CysLT1 receptorMore data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 1(Homo sapiens (Human))
University Of Naples "Federico Ii
Curated by ChEMBL
University Of Naples "Federico Ii
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity against human CysLT1 expressed in CHO cells assessed as inhibition of LTD4 induced cytosolic Calcium ion mobilization measured af...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 1(Homo sapiens (Human))
University Of Naples "Federico Ii
Curated by ChEMBL
University Of Naples "Federico Ii
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Antagonist activity against human CysLT1 expressed in CHO cells assessed as inhibition of LTD4 induced cytosolic Calcium ion mobilization measured af...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 1(Homo sapiens (Human))
University Of Naples "Federico Ii
Curated by ChEMBL
University Of Naples "Federico Ii
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Antagonist activity against human CysLT1 expressed in CHO cells assessed as inhibition of LTD4 induced cytosolic Calcium ion mobilization measured af...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 1(Homo sapiens (Human))
University Of Naples "Federico Ii
Curated by ChEMBL
University Of Naples "Federico Ii
Curated by ChEMBL
Affinity DataIC50: 2.80E+3nMAssay Description:Antagonist activity against human CysLT1 expressed in CHO cells assessed as inhibition of LTD4 induced cytosolic Calcium ion mobilization measured af...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University Of Naples "Federico Ii
Curated by ChEMBL
University Of Naples "Federico Ii
Curated by ChEMBL
Affinity DataIC50: >3.00E+3nMAssay Description:Antagonist activity at human CysLT2 receptorMore data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 1(Homo sapiens (Human))
University Of Naples "Federico Ii
Curated by ChEMBL
University Of Naples "Federico Ii
Curated by ChEMBL
Affinity DataIC50: 3.90E+3nMAssay Description:Antagonist activity against human CysLT1 expressed in CHO cells assessed as inhibition of LTD4 induced cytosolic Calcium ion mobilization measured af...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University Of Naples "Federico Ii
Curated by ChEMBL
University Of Naples "Federico Ii
Curated by ChEMBL
Affinity DataIC50: >5.00E+3nMAssay Description:Antagonist activity at human CysLT2 receptorMore data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 1(Homo sapiens (Human))
University Of Naples "Federico Ii
Curated by ChEMBL
University Of Naples "Federico Ii
Curated by ChEMBL
Affinity DataIC50: 5.11E+3nMAssay Description:Antagonist activity against human CysLT1 expressed in CHO cells assessed as inhibition of LTD4 induced cytosolic Calcium ion mobilization measured af...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 1(Homo sapiens (Human))
University Of Naples "Federico Ii
Curated by ChEMBL
University Of Naples "Federico Ii
Curated by ChEMBL
Affinity DataIC50: 9.63E+3nMAssay Description:Antagonist activity against human CysLT1 expressed in CHO cells assessed as inhibition of LTD4 induced cytosolic Calcium ion mobilization measured af...More data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
University Of Naples "Federico Ii
Curated by ChEMBL
University Of Naples "Federico Ii
Curated by ChEMBL
Affinity DataEC50: 7.40E+3nMAssay Description:Agonist activity against human GPBAR1 expressed in HEK293T cells assessed as transactivation of cAMP-responsive element incubated for 18 hrs by Dual-...More data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
University Of Naples "Federico Ii
Curated by ChEMBL
University Of Naples "Federico Ii
Curated by ChEMBL
Affinity DataEC50: 3.00E+3nMAssay Description:Agonist activity against human GPBAR1 expressed in HEK293T cells assessed as transactivation of cAMP-responsive element incubated for 18 hrs by Dual-...More data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
University Of Naples "Federico Ii
Curated by ChEMBL
University Of Naples "Federico Ii
Curated by ChEMBL
Affinity DataEC50: 1.65E+4nMAssay Description:Agonist activity against human GPBAR1 expressed in HEK293T cells assessed as transactivation of cAMP-responsive element incubated for 18 hrs by Dual-...More data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
University Of Naples "Federico Ii
Curated by ChEMBL
University Of Naples "Federico Ii
Curated by ChEMBL
Affinity DataEC50: 2.50E+3nMAssay Description:Agonist activity against human GPBAR1 expressed in HEK293T cells assessed as transactivation of cAMP-responsive element incubated for 18 hrs by Dual-...More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University Of Naples "Federico Ii
Curated by ChEMBL
University Of Naples "Federico Ii
Curated by ChEMBL
Affinity DataEC50: 293nMAssay Description:Agonist activity at human CysLT2 receptorMore data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University Of Naples "Federico Ii
Curated by ChEMBL
University Of Naples "Federico Ii
Curated by ChEMBL
Affinity DataEC50: 4.40nMAssay Description:Agonist activity at human CysLT2 receptorMore data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 2(Homo sapiens (Human))
University Of Naples "Federico Ii
Curated by ChEMBL
University Of Naples "Federico Ii
Curated by ChEMBL
Affinity DataEC50: 8.90nMAssay Description:Agonist activity at human CysLT2 receptorMore data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 1(Homo sapiens (Human))
University Of Naples "Federico Ii
Curated by ChEMBL
University Of Naples "Federico Ii
Curated by ChEMBL
Affinity DataEC50: 104nMAssay Description:Agonist activity at human CysLT1 receptorMore data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 1(Homo sapiens (Human))
University Of Naples "Federico Ii
Curated by ChEMBL
University Of Naples "Federico Ii
Curated by ChEMBL
Affinity DataEC50: 0.900nMAssay Description:Agonist activity at human CysLT1 receptorMore data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 1(Homo sapiens (Human))
University Of Naples "Federico Ii
Curated by ChEMBL
University Of Naples "Federico Ii
Curated by ChEMBL
Affinity DataEC50: 43nMAssay Description:Agonist activity at human CysLT1 receptorMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
University Of Naples "Federico Ii
Curated by ChEMBL
University Of Naples "Federico Ii
Curated by ChEMBL
Affinity DataEC50: 1.80E+3nMAssay Description:Agonist activity against human GPBAR1 expressed in HEK293T cells assessed as transactivation of cAMP-responsive element incubated for 18 hrs by Dual-...More data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
University Of Naples "Federico Ii
Curated by ChEMBL
University Of Naples "Federico Ii
Curated by ChEMBL
Affinity DataEC50: 170nMAssay Description:Agonist activity against human GPBAR1 expressed in HEK293T cells assessed as transactivation of cAMP-responsive element incubated for 18 hrs by Dual-...More data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
University Of Naples "Federico Ii
Curated by ChEMBL
University Of Naples "Federico Ii
Curated by ChEMBL
Affinity DataEC50: 500nMAssay Description:Agonist activity against human GPBAR1 expressed in HEK293T cells assessed as transactivation of cAMP-responsive element incubated for 18 hrs by Dual-...More data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
University Of Naples "Federico Ii
Curated by ChEMBL
University Of Naples "Federico Ii
Curated by ChEMBL
Affinity DataEC50: 100nMAssay Description:Agonist activity against human GPBAR1 expressed in HEK293T cells assessed as transactivation of cAMP-responsive element incubated for 18 hrs by Dual-...More data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
University Of Naples "Federico Ii
Curated by ChEMBL
University Of Naples "Federico Ii
Curated by ChEMBL
Affinity DataEC50: 2.30E+4nMAssay Description:Agonist activity against human GPBAR1 expressed in HEK293T cells assessed as transactivation of cAMP-responsive element incubated for 18 hrs by Dual-...More data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
University Of Naples "Federico Ii
Curated by ChEMBL
University Of Naples "Federico Ii
Curated by ChEMBL
Affinity DataEC50: 2.00E+4nMAssay Description:Agonist activity against human GPBAR1 expressed in HEK293T cells assessed as transactivation of cAMP-responsive element incubated for 18 hrs by Dual-...More data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
University Of Naples "Federico Ii
Curated by ChEMBL
University Of Naples "Federico Ii
Curated by ChEMBL
Affinity DataEC50: 1.00E+3nMAssay Description:Agonist activity against human GPBAR1 expressed in HEK293T cells assessed as transactivation of cAMP-responsive element incubated for 18 hrs by Dual-...More data for this Ligand-Target Pair