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Found 319 with Last Name = 'dressman' and Initial = 'ba'
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50202918((S)-N-(2-fluoro-3-(trifluoromethyl)benzyl)-5-(4-cy...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50202900((S)-N-(3-(trifluoromethyl)benzyl)-5-(4-cyclohexylp...)
Affinity DataKi:  0.270nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50202920(2(R)-[[4-(piperidin-1-yl)piperidin-1-yl]carbonylme...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50202882((S)-N-(2,3-dichlorobenzyl)-5-(4-cyclohexylpiperazi...)
Affinity DataKi:  0.380nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50202902((S)-N-(2-fluoro-5-(trifluoromethyl)benzyl)-5-(4-cy...)
Affinity DataKi:  0.410nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50202873((S)-N-(3-(trifluoromethyl)benzyl)-5-(4-(cyclohexyl...)
Affinity DataKi:  0.460nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50202916((S)-N-(3-fluoro-5-(trifluoromethyl)benzyl)-5-(4-cy...)
Affinity DataKi:  0.510nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50202871((S)-N-(3-chlorobenzyl)-5-(4-cyclohexylpiperazin-1-...)
Affinity DataKi:  0.660nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50202860(2(R)-[[4-(piperidin-1-yl)piperidin-1-yl]carbonylme...)
Affinity DataKi:  0.660nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50202877((S)-N-(3,5-difluorobenzyl)-5-(4-cyclohexylpiperazi...)
Affinity DataKi:  0.820nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50202869((S)-N-(2-(trifluoromethyl)benzyl)-5-(4-cyclohexylp...)
Affinity DataKi:  0.930nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50202858(2(R)-[[4-(piperidin-1-yl)piperidin-1-yl]carbonylme...)
Affinity DataKi:  1.13nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50202864(4-amino-1-benzyl-1-[(3S)-3-[(3S,4R)-2-oxo-3-[(4S)-...)
Affinity DataKi:  1.13nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50202892((S)-N-(3-(trifluoromethyl)benzyl)-5-oxo-2-((3S,4R)...)
Affinity DataKi:  1.17nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50202899(CHEMBL241826 | N-(3-(trifluoromethyl)benzyl)-3-oxo...)
Affinity DataKi:  1.17nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50202851((S)-N-(3-(trifluoromethyl)benzyl)-5-oxo-2-((3S,4R)...)
Affinity DataKi:  1.19nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50202910(2(R)-[[4-(piperidin-1-yl)piperidin-1-yl]carbonylme...)
Affinity DataKi:  1.27nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 3(Homo sapiens (Human))
Centro De Investigaci£N Lilly S.A. Avda. De La Industria

Curated by ChEMBL
LigandPNGBDBM50062522((1S,2S)-2-((S)-1-amino-1-carboxy-2-(9H-xanthen-9-y...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]-LY459477 from recombinant human mGlu3 receptor expressed in hamster AV12 cell membranes co-expressing rat EAAT1 incubated for 90...More data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50202852((S)-N-(3-(trifluoromethyl)benzyl)-5-oxo-2-((3S,4R)...)
Affinity DataKi:  1.45nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50202905(2(R)-[[4-(piperidin-1-yl)piperidin-1-yl]carbonylme...)
Affinity DataKi:  1.49nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50202922((S)-N-(3-(trifluoromethyl)benzyl)-4-oxo-2-((3S,4R)...)
Affinity DataKi:  1.89nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50202915((S)-N-(3-(trifluoromethyl)benzyl)-5-oxo-2-((3S,4R)...)
Affinity DataKi:  1.95nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Agouron Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50061306((3S,4aS,8aS)-2-[(2R,3R)-2-Hydroxy-3-(3-hydroxy-2-m...)
Affinity DataKi:  2nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 3(Homo sapiens (Human))
Centro De Investigaci£N Lilly S.A. Avda. De La Industria

Curated by ChEMBL
LigandPNGBDBM50558766(CHEMBL4751065)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]-LY459477 from recombinant human mGlu3 receptor expressed in hamster AV12 cell membranes co-expressing rat EAAT1 incubated for 90...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 3(Homo sapiens (Human))
Centro De Investigaci£N Lilly S.A. Avda. De La Industria

Curated by ChEMBL
LigandPNGBDBM50204261(CHEMBL3969063)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]-LY459477 from human mGlu3 receptor expressed in hamster AV12 cell membranes co-expressing human EAAT1 after 90 mins by liquid sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Agouron Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50061307(AG-1254 | CHEMBL128696 | N-[(1R,2R)-3-(2-tert-Buty...)
Affinity DataKi:  3nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Agouron Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50061307(AG-1254 | CHEMBL128696 | N-[(1R,2R)-3-(2-tert-Buty...)
Affinity DataKi:  3nMAssay Description:Inhibitory activity HIV-1 protease enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50202849(CHEMBL439398 | N-(3-(trifluoromethyl)benzyl)-3-oxo...)
Affinity DataKi:  3.39nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50202844((3S)-3-amino-1-benzyl-1-[(3S)-3-[(3S,4R)-2-oxo-3-[...)
Affinity DataKi:  3.60nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50202842((R)-N-(3-(trifluoromethyl)benzyl)-4-oxo-2-((3S,4R)...)
Affinity DataKi:  3.70nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Centro De Investigaci£N Lilly S.A. Avda. De La Industria

Curated by ChEMBL
LigandPNGBDBM50062522((1S,2S)-2-((S)-1-amino-1-carboxy-2-(9H-xanthen-9-y...)
Affinity DataKi:  4.30nMAssay Description:Displacement of [3H]-LY459477 from recombinant human mGlu2 receptor expressed in hamster AV12 cell membranes co-expressing rat EAAT1 incubated for 90...More data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50202909((S)-N-(3,5-bis(trifluoromethyl)benzyl)-5-(4-cycloh...)
Affinity DataKi:  4.45nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 3(Homo sapiens (Human))
Centro De Investigaci£N Lilly S.A. Avda. De La Industria

Curated by ChEMBL
LigandPNGBDBM50558768(CHEMBL4759992)
Affinity DataKi:  4.5nMAssay Description:Displacement of [3H]-LY459477 from recombinant human mGlu3 receptor expressed in hamster AV12 cell membranes co-expressing rat EAAT1 incubated for 90...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Agouron Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286713(3,5-Diamino-N-[(1R,2R)-3-(2-tert-butylcarbamoyl-ph...)
Affinity DataKi:  5nMAssay Description:Inhibitory activity HIV-1 protease enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50202906((S)-N-(3-(trifluoromethyl)benzyl)-4-(4-benzyl-1,4-...)
Affinity DataKi:  5.12nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Centro De Investigaci£N Lilly S.A. Avda. De La Industria

Curated by ChEMBL
LigandPNGBDBM50558768(CHEMBL4759992)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]-LY459477 from recombinant human mGlu2 receptor expressed in hamster AV12 cell membranes co-expressing rat EAAT1 incubated for 90...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Centro De Investigaci£N Lilly S.A. Avda. De La Industria

Curated by ChEMBL
LigandPNGBDBM50558766(CHEMBL4751065)
Affinity DataKi:  5.30nMAssay Description:Displacement of [3H]-LY459477 from recombinant human mGlu2 receptor expressed in hamster AV12 cell membranes co-expressing rat EAAT1 incubated for 90...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50202903(4-amino-1-benzyl-1-[(3R)-3-[(3S,4R)-2-oxo-3-[(4S)-...)
Affinity DataKi:  5.58nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50202881((R)-N-(3-(trifluoromethyl)benzyl)-5-(4-cyclohexylp...)
Affinity DataKi:  5.84nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 3(Homo sapiens (Human))
Centro De Investigaci£N Lilly S.A. Avda. De La Industria

Curated by ChEMBL
LigandPNGBDBM50558774(CHEMBL4780402)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]-LY459477 from recombinant human mGlu3 receptor expressed in hamster AV12 cell membranes co-expressing rat EAAT1 incubated for 90...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50202862(2(R)-[[4-(piperidin-1-yl)piperidin-1-yl]carbonylme...)
Affinity DataKi: >6nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50202914(CHEMBL395778 | N-(3-(trifluoromethyl)benzyl)-3-(4-...)
Affinity DataKi:  6.5nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 3(Homo sapiens (Human))
Centro De Investigaci£N Lilly S.A. Avda. De La Industria

Curated by ChEMBL
LigandPNGBDBM50558775(CHEMBL4776989)
Affinity DataKi:  6.80nMAssay Description:Displacement of [3H]-LY459477 from recombinant human mGlu3 receptor expressed in hamster AV12 cell membranes co-expressing rat EAAT1 incubated for 90...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Centro De Investigaci£N Lilly S.A. Avda. De La Industria

Curated by ChEMBL
LigandPNGBDBM50204261(CHEMBL3969063)
Affinity DataKi:  7.40nMAssay Description:Displacement of [3H]-LY459477 from human mGlu2 receptor expressed in hamster AV12 cell membranes co-expressing human EAAT1 after 90 mins by liquid sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 3(Homo sapiens (Human))
Centro De Investigaci£N Lilly S.A. Avda. De La Industria

Curated by ChEMBL
LigandPNGBDBM50558769(CHEMBL4746125)
Affinity DataKi:  7.70nMAssay Description:Displacement of [3H]-LY459477 from recombinant human mGlu3 receptor expressed in hamster AV12 cell membranes co-expressing rat EAAT1 incubated for 90...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50202879((R)-N-(3-(trifluoromethyl)benzyl)-4-oxo-2-((3S,4R)...)
Affinity DataKi:  7.90nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Centro De Investigaci£N Lilly S.A. Avda. De La Industria

Curated by ChEMBL
LigandPNGBDBM50558772(CHEMBL4748699)
Affinity DataKi:  8.40nMAssay Description:Displacement of [3H]-LY459477 from recombinant human mGlu2 receptor expressed in hamster AV12 cell membranes co-expressing rat EAAT1 incubated for 90...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50202866(2(R)-[[ 4-[2-(1-piperidinyl)ethyl]piperidin-1-yl]c...)
Affinity DataKi:  8.70nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Centro De Investigaci£N Lilly S.A. Avda. De La Industria

Curated by ChEMBL
LigandPNGBDBM50558774(CHEMBL4780402)
Affinity DataKi:  8.90nMAssay Description:Displacement of [3H]-LY459477 from recombinant human mGlu2 receptor expressed in hamster AV12 cell membranes co-expressing rat EAAT1 incubated for 90...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50202872((S)-N1-(3-(trifluoromethyl)benzyl)-2-((3S,4R)-2-ox...)
Affinity DataKi:  9nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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