TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University Of Melbourne
Curated by PDSP Ki Database
The University Of Melbourne
Curated by PDSP Ki Database
Affinity DataKi: 4nMAssay Description:Inhibition of [3H]-U-69,593 binding to rat opioid receptor kappa 1 expressed in HEK 293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:Inhibition constant against human 5-hydroxytryptamine 2C receptor [INI isoforms] using [3H]-mesulergine as radioligand with the compound (10 uM) diss...More data for this Ligand-Target Pair
Affinity DataKi: 5.80nMAssay Description:Inhibition constant against human 5-hydroxytryptamine 2B receptor using [3H]-LSD as radioligand with the compound (10 uM) dissolved in DMSOMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University Of Melbourne
Curated by PDSP Ki Database
The University Of Melbourne
Curated by PDSP Ki Database
Affinity DataKi: 6nMAssay Description:Inhibition of [3H]-U-69,593 binding to rat opioid receptor kappa 1 expressed in HEK 293 cellsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University Of Melbourne
Curated by PDSP Ki Database
The University Of Melbourne
Curated by PDSP Ki Database
Affinity DataKi: 6nMAssay Description:Inhibition of [3H]-U-69,593 binding to rat opioid receptor kappa 1 expressed in HEK 293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Inhibition constant against human 5-hydroxytryptamine 2C receptor [INI isoforms] using [3H]-mesulergine as radioligand with the compound (10 uM) diss...More data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
Affinity DataKi: 8.39nMAssay Description:Inhibition constant against human 5-hydroxytryptamine 2B receptor using [3H]-LSD as radioligand with the compound (10 uM) dissolved in DMSOMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
Affinity DataKi: 12.6nMAssay Description:Inhibition constant against human 5-hydroxytryptamine 2C receptor [VGI isoforms] using [3H]-mesulergine as radioligand with the compound (10 uM) diss...More data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
Affinity DataKi: 14nMAssay Description:Inhibition constant against human 5-hydroxytryptamine 2C receptor [VGI isoforms] using [3H]-mesulergine as radioligand with the compound (10 uM) diss...More data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
Affinity DataKi: 15.7nMAssay Description:Inhibition constant against rat 5-hydroxytryptamine 2C receptor using [3H]-mesulergine as radioligand with the compound (10 uM) dissolved in DMSOMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University Of Melbourne
Curated by PDSP Ki Database
The University Of Melbourne
Curated by PDSP Ki Database
Affinity DataKi: 18nMAssay Description:Inhibition of [3H]-U-69,593 binding to rat opioid receptor kappa 1 expressed in HEK 293 cellsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University Of Melbourne
Curated by PDSP Ki Database
The University Of Melbourne
Curated by PDSP Ki Database
Affinity DataKi: 18nMAssay Description:Inhibition of [3H]-U-69,593 binding to rat opioid receptor kappa 1 expressed in HEK 293 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
Affinity DataKi: 24nMAssay Description:Inhibition constant against human 5-hydroxytryptamine 2C receptor [INI isoforms] using [3H]-mesulergine as radioligand with the compound (10 uM) diss...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
Affinity DataKi: 33nMAssay Description:Inhibition constant against human 5-hydroxytryptamine 2C receptor [VGI isoforms] using [3H]-mesulergine as radioligand with the compound (10 uM) diss...More data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Inhibition constant against human 5-hydroxytryptamine 2B receptor using [3H]-LSD as radioligand with the compound (10 uM) dissolved in DMSOMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
Affinity DataKi: 48nMAssay Description:Inhibition constant against rat 5-hydroxytryptamine 2C receptor using [3H]-mesulergine as radioligand with the compound (10 uM) dissolved in DMSOMore data for this Ligand-Target Pair
Affinity DataKi: 49nMAssay Description:Inhibition constant against rat 5-hydroxytryptamine 2C receptor using [3H]-mesulergine as radioligand with the compound (10 uM) dissolved in DMSOMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University Of Melbourne
Curated by PDSP Ki Database
The University Of Melbourne
Curated by PDSP Ki Database
Affinity DataKi: 59nMAssay Description:Inhibition of [3H]-U-69,593 binding to rat opioid receptor kappa 1 expressed in HEK 293 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
Affinity DataKi: 73nMAssay Description:Inhibition constant against human 5-hydroxytryptamine 2C receptor [INI isoforms] using [3H]-mesulergine as radioligand with the compound (10 uM) diss...More data for this Ligand-Target Pair
Affinity DataKi: 82nMAssay Description:Inhibition constant against human 5-hydroxytryptamine 2C receptor [INI isoforms] using [3H]-mesulergine as radioligand with the compound (10 uM) diss...More data for this Ligand-Target Pair
Affinity DataKi: 84nMAssay Description:Inhibition constant against human 5-hydroxytryptamine 2C receptor [VGI isoforms] using [3H]-mesulergine as radioligand with the compound (10 uM) diss...More data for this Ligand-Target Pair
Affinity DataKi: 84nMAssay Description:Inhibition constant against human 5-hydroxytryptamine 2C receptor [VGI isoforms] using [3H]-mesulergine as radioligand with the compound (10 uM) diss...More data for this Ligand-Target Pair
Affinity DataKi: 87nMAssay Description:Inhibition constant against human 5-hydroxytryptamine 2C receptor [INI isoforms] using [3H]-mesulergine as radioligand with the compound (10 uM) diss...More data for this Ligand-Target Pair
Affinity DataKi: 98nMAssay Description:Inhibition constant against human 5-hydroxytryptamine 2B receptor using [3H]-LSD as radioligand with the compound (10 uM) dissolved in DMSOMore data for this Ligand-Target Pair
Affinity DataKi: 103nMAssay Description:Inhibition constant against human 5-hydroxytryptamine 2C receptor [INI isoforms] using [3H]-mesulergine as radioligand with the compound (10 uM) diss...More data for this Ligand-Target Pair
Affinity DataKi: 116nMAssay Description:Inhibition constant against human 5-hydroxytryptamine 2B receptor using [3H]-LSD as radioligand with the compound (10 uM) dissolved in DMSOMore data for this Ligand-Target Pair
Affinity DataKi: 122nMAssay Description:Inhibition constant against human 5-hydroxytryptamine 2A receptor using [3H]-ketanserin as radioligand with the compound (10 uM) dissolved in DMSOMore data for this Ligand-Target Pair
Affinity DataKi: 125nMAssay Description:Inhibition constant against human 5-hydroxytryptamine 2C receptor [VGI isoforms] using [3H]-mesulergine as radioligand with the compound (10 uM) diss...More data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Inhibition constant against human 5-hydroxytryptamine 2C receptor [INI isoforms] using [3H]-mesulergine as radioligand with the compound (10 uM) diss...More data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University Of Melbourne
Curated by PDSP Ki Database
The University Of Melbourne
Curated by PDSP Ki Database
Affinity DataKi: 156nMAssay Description:Inhibition of [3H]-U-69,593 binding to rat opioid receptor kappa 1 expressed in HEK 293 cellsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University Of Melbourne
Curated by PDSP Ki Database
The University Of Melbourne
Curated by PDSP Ki Database
Affinity DataKi: 163nMAssay Description:Inhibition of [3H]-U-69,593 binding to rat opioid receptor kappa 1 expressed in HEK 293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Inhibition constant against human 5-hydroxytryptamine 2B receptor using [3H]-LSD as radioligand with the compound (10 uM) dissolved in DMSOMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Inhibition constant against rat 5-hydroxytryptamine 2A receptor using [3H]-ketanserin as radioligand with the compound (10 uM) dissolved in DMSOMore data for this Ligand-Target Pair