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Found 149 with Last Name = 'hill' and Initial = 'dt'
TargetType-2 angiotensin II receptor(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50011972(CHEMBL385189 | Sar-Arg-Val-Tyr-Ile-His-Pro-Thi-OH)
Affinity DataIC50:  0.110nMAssay Description:In vitro inhibition of [125I]-AII specific binding towards angiotensin II receptor in rat mesenteric membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230790(CHEMBL292892)
Affinity DataIC50:  0.150nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50282363(4-[2-Butyl-5-((E)-2-carboxy-3-thiophen-2-yl-propen...)
Affinity DataIC50:  0.160nMAssay Description:Tested for inhibition of [125I]- AII specific binding to rat mesenteric arteries, expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50230779(CHEMBL294686)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230811(CHEMBL293091)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230778(CHEMBL56211)
Affinity DataIC50:  0.560nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230771(CHEMBL55510)
Affinity DataIC50:  0.590nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230806(CHEMBL294415)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50048078(4-[2-Butyl-5-((E)-2-carboxy-3-thiophen-2-yl-propen...)
Affinity DataIC50:  1nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50011977((E)-2-butyl-1-(p-carboxybenzyl)-alpha-2-thenylimid...)
Affinity DataIC50:  1nMAssay Description:Tested for inhibition of [125I]- AII specific binding to rat mesenteric arteries, expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50048078(4-[2-Butyl-5-((E)-2-carboxy-3-thiophen-2-yl-propen...)
Affinity DataIC50:  1nMAssay Description:Tested for inhibition of [125I]- AII specific binding to rat mesenteric arteries, expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50011977((E)-2-butyl-1-(p-carboxybenzyl)-alpha-2-thenylimid...)
Affinity DataIC50:  1nMAssay Description:In vitro inhibition of [125I]-AII specific binding towards Angiotensin II receptor in rat mesenteric membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282362(4-[2-Butyl-5-((E)-2-carboxy-3-thiophen-2-yl-propen...)
Affinity DataIC50:  1.20nMAssay Description:Tested for Angiotensin II receptor, type 1 affinity in the absence of BSAMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50011973(CHEMBL216061 | Sar-Arg-Val-Tyr-Ile-His-Pro-Phe | S...)
Affinity DataIC50:  1.30nMAssay Description:In vitro inhibition of [125I]-AII specific binding towards Angiotensin II receptor in rat mesenteric membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50011975(4-[2-Butyl-5-((E)-2-carboxy-3-thiophen-2-yl-propen...)
Affinity DataIC50:  1.5nMAssay Description:In vitro inhibition of [125I]-AII specific binding towards angiotensin II receptor in rat mesenteric membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50011975(4-[2-Butyl-5-((E)-2-carboxy-3-thiophen-2-yl-propen...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50011975(4-[2-Butyl-5-((E)-2-carboxy-3-thiophen-2-yl-propen...)
Affinity DataIC50:  1.5nMAssay Description:Tested for inhibition of [125I]- AII specific binding to rat mesenteric arteries, expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50011977((E)-2-butyl-1-(p-carboxybenzyl)-alpha-2-thenylimid...)
Affinity DataIC50:  2nMAssay Description:Tested for Angiotensin II receptor, type 1 affinity in the absence of bovine serum albumin (BSA)More data for this Ligand-Target Pair
In DepthDetails ArticleDrugBank

LigandPNGBDBM50230787(CHEMBL54421)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284297(4-(2-Butyl-5-{[(R)-1-carboxy-2-(1H-indol-3-yl)-eth...)
Affinity DataIC50:  2.90nMAssay Description:Tested for inhibition of Angiotensin II specific binding to Angiotensin II receptor, type 1 in the recombinant human AT-1 receptor expressed in LhAT-...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50230792(CHEMBL56497)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230799(CHEMBL56333)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230774(CHEMBL291955)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230762(CHEMBL56160)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230810(CHEMBL299064)
Affinity DataIC50:  4.60nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230764(CHEMBL299954)
Affinity DataIC50:  4.80nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230767(CHEMBL56522)
Affinity DataIC50:  5nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230796(CHEMBL56690)
Affinity DataIC50:  6.60nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50011977((E)-2-butyl-1-(p-carboxybenzyl)-alpha-2-thenylimid...)
Affinity DataIC50:  7.30nMAssay Description:Tested for Angiotensin II receptor, type 1 affinity in the presence of 0.25% bovine serum albumin (BSA)More data for this Ligand-Target Pair
In DepthDetails ArticleDrugBank

LigandPNGBDBM50230772(CHEMBL59043)
Affinity DataIC50: >10nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50282362(4-[2-Butyl-5-((E)-2-carboxy-3-thiophen-2-yl-propen...)
Affinity DataIC50:  12nMAssay Description:Tested for inhibition of [125I]- AII specific binding to rat mesenteric arteries, expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50230805(CHEMBL54645)
Affinity DataIC50:  15nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50011978(3-[2-Butyl-3-(4-hydroxy-3-methyl-benzyl)-3H-imidaz...)
Affinity DataIC50:  21nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50011978(3-[2-Butyl-3-(4-hydroxy-3-methyl-benzyl)-3H-imidaz...)
Affinity DataIC50:  21nMAssay Description:In vitro inhibition of [125I]-AII specific binding towards Angiotensin II receptor in rat mesenteric membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230785(CHEMBL300566)
Affinity DataIC50:  21nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230783(CHEMBL54711)
Affinity DataIC50:  22nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230809(CHEMBL57620)
Affinity DataIC50:  23nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230791(CHEMBL55950)
Affinity DataIC50:  28nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(RAT)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50011974(3-[2-Butyl-3-(2-nitro-benzyl)-3H-imidazol-4-yl]-2-...)
Affinity DataIC50:  31nMAssay Description:In vitro inhibition of [125I]-AII specific binding towards Angiotensin II receptor in rat mesenteric membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282362(4-[2-Butyl-5-((E)-2-carboxy-3-thiophen-2-yl-propen...)
Affinity DataIC50:  31nMAssay Description:Tested for Angiotensin II receptor, type 1 affinity in the presence of 0.25% BSAMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50011974(3-[2-Butyl-3-(2-nitro-benzyl)-3H-imidazol-4-yl]-2-...)
Affinity DataIC50:  31nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230795(CHEMBL59580)
Affinity DataIC50:  34nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50011971(3-[2-Butyl-3-(2-hydroxy-benzyl)-3H-imidazol-4-yl]-...)
Affinity DataIC50:  34nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230781(CHEMBL291688)
Affinity DataIC50:  34nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50048076(4-[2-Butyl-5-((E)-2-carboxy-3-thiophen-2-yl-propen...)
Affinity DataIC50:  35nMAssay Description:Tested for inhibition of [125I]- AII specific binding to rat mesenteric arteries, expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50048076(4-[2-Butyl-5-((E)-2-carboxy-3-thiophen-2-yl-propen...)
Affinity DataIC50:  35nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230804(CHEMBL293706)
Affinity DataIC50:  39nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230770(CHEMBL55216)
Affinity DataIC50:  43nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230768(CHEMBL417752)
Affinity DataIC50:  46nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284298(4-(2-Butyl-5-{[(S)-1-carboxy-2-(1H-indol-3-yl)-eth...)
Affinity DataIC50:  48.3nMAssay Description:Tested for inhibition of Angiotensin II specific binding to Angiotensin II receptor, type 1 in the recombinant human AT-1 receptor expressed in LhAT-...More data for this Ligand-Target Pair
In DepthDetails Article
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