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Found 20 with Last Name = 'sakurai' and Initial = 'h'
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50256010(3-{2,4-dimethyl-5-[2-oxo-5-(N'-phenylhydrazinocarb...)
Affinity DataIC50:  40nMAssay Description:Inhibition of PDGFRbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM4811((Z)-3-[2,4-dimethyl-5-(2-oxo-1,2-dihydro-indol-3-y...)
Affinity DataIC50:  50nMAssay Description:Inhibition of PDGFRbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50256010(3-{2,4-dimethyl-5-[2-oxo-5-(N'-phenylhydrazinocarb...)
Affinity DataIC50:  70nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50256010(3-{2,4-dimethyl-5-[2-oxo-5-(N'-phenylhydrazinocarb...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human FGFR1 expressed in insect cells by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50217602((Z)-3-(5-((6-(3,5-dimethoxyphenyl)-2-oxoindolin-3-...)
Affinity DataIC50:  400nMAssay Description:Inhibition of human FGFR1 kinase expressed in insect cell by HTRF detection methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50217602((Z)-3-(5-((6-(3,5-dimethoxyphenyl)-2-oxoindolin-3-...)
Affinity DataIC50:  520nMAssay Description:Inhibition of human FGFR1 expressed in insect cells by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM4811((Z)-3-[2,4-dimethyl-5-(2-oxo-1,2-dihydro-indol-3-y...)
Affinity DataIC50:  680nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50217602((Z)-3-(5-((6-(3,5-dimethoxyphenyl)-2-oxoindolin-3-...)
Affinity DataIC50:  780nMAssay Description:Inhibition of PDGFRbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50217602((Z)-3-(5-((6-(3,5-dimethoxyphenyl)-2-oxoindolin-3-...)
Affinity DataIC50:  930nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Toyama Prefectural University

Curated by ChEMBL
LigandPNGBDBM50481798(Amo-01 | BU-4664L | Diazepinomicin | ECO-4601 | TL...)
Affinity DataIC50:  994nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM4901(3-(5-{[(3Z)-6-(3-methoxyphenyl)-2-oxo-2,3-dihydro-...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of human FGFR1 kinase expressed in insect cell by HTRF detection methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Toyama Prefectural University

Curated by ChEMBL
LigandPNGBDBM50481798(Amo-01 | BU-4664L | Diazepinomicin | ECO-4601 | TL...)
Affinity DataIC50:  1.29E+3nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM4811((Z)-3-[2,4-dimethyl-5-(2-oxo-1,2-dihydro-indol-3-y...)
Affinity DataIC50:  1.81E+3nMAssay Description:Inhibition of human FGFR1 expressed in insect cells by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50256010(3-{2,4-dimethyl-5-[2-oxo-5-(N'-phenylhydrazinocarb...)
Affinity DataIC50:  3.48E+3nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM4901(3-(5-{[(3Z)-6-(3-methoxyphenyl)-2-oxo-2,3-dihydro-...)
Affinity DataIC50:  1.79E+4nMAssay Description:Inhibition of rhFGF2-induced cellular proliferation of HUVECMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50217602((Z)-3-(5-((6-(3,5-dimethoxyphenyl)-2-oxoindolin-3-...)
Affinity DataIC50:  1.82E+4nMAssay Description:Inhibition of rhFGF2-induced cellular proliferation of HUVECMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM4900(3-(2,4-dimethyl-5-{[(3Z)-2-oxo-6-phenyl-2,3-dihydr...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of rhFGF2-induced cellular proliferation of HUVECMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM4811((Z)-3-[2,4-dimethyl-5-(2-oxo-1,2-dihydro-indol-3-y...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of rhFGF2-induced cellular proliferation of HUVECMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM4811((Z)-3-[2,4-dimethyl-5-(2-oxo-1,2-dihydro-indol-3-y...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50217602((Z)-3-(5-((6-(3,5-dimethoxyphenyl)-2-oxoindolin-3-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed