Affinity DataKi: 0.120nMAssay Description:Compound was evaluated for binding affinity towards DA D-2 receptor using radioligand [3H]SPIMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
Lund University
Curated by ChEMBL
Lund University
Curated by ChEMBL
Affinity DataKi: 0.270nMAssay Description:Displacement of [3H]Flumazenil from human GABA-Aalpha1 receptor plus beta-2-gamma-2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Binding affinity to displace [3H]- SCH 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Compound was tested for the displacement of [3H]-SCH- 23390 from dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Binding affinity to displace [3H]- SCH 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Binding affinity to displace [3H]- SCH 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Binding affinity to displace [3H]- SCH 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity to displace [3H]- SCH 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Compound was tested for the displacement of [3H]-SCH- 23390 from dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Binding affinity to displace [3H]-SCH- 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Compound was evaluated for binding affinity towards DA D-2 receptor using radioligand [3H]SPIMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
Lund University
Curated by ChEMBL
Lund University
Curated by ChEMBL
Affinity DataKi: 4.10nMAssay Description:Displacement of [3H]Flumazenil from human GABA-Aalpha1 receptor plus beta-2-gamma-2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Binding affinity against Dopamine receptor D1 in rat radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Binding affinity to displace [3H]-SCH- 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Binding affinity to displace [3H]- SCH 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Compound was tested for the displacement of [3H]-SCH- 23390 from dopamine receptor D1More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Homo sapiens (Human))
Lund University
Curated by ChEMBL
Lund University
Curated by ChEMBL
Affinity DataKi: 7.20nMAssay Description:Displacement of [3H]Flumazenil from human GABA-Aalpha3 receptor plus beta-2-gamma-2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 9.5nMAssay Description:Compound was evaluated for binding affinity towards DA D-2 receptor using radioligand [3H]SPIMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
Lund University
Curated by ChEMBL
Lund University
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Displacement of [3H]Flumazenil from human GABA-Aalpha1 receptor plus beta-2-gamma-2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Homo sapiens (Human))
Lund University
Curated by ChEMBL
Lund University
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Displacement of [3H]Flumazenil from human GABA-Aalpha3 receptor plus beta-2-gamma-2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
Lund University
Curated by ChEMBL
Lund University
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Displacement of [3H]Flumazenil from human GABA-Aalpha1 receptor plus beta-2-gamma-2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Binding affinity against Dopamine receptor D1 in rat radioligandMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Homo sapiens (Human))
Lund University
Curated by ChEMBL
Lund University
Curated by ChEMBL
Affinity DataKi: 26nMAssay Description:Displacement of [3H]Flumazenil from human GABA-Aalpha3 receptor plus beta-2-gamma-2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Compound was evaluated for binding affinity towards Dopamine receptor D2 using radioligand [3H]SPIMore data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Inhibitory concentration required for displacing radioligand [3H]SPI from DA D-2 receptorMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
Lund University
Curated by ChEMBL
Lund University
Curated by ChEMBL
Affinity DataKi: 53nMAssay Description:Displacement of [3H]Flumazenil from human GABA-Aalpha1 receptor plus beta-2-gamma-2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Homo sapiens (Human))
Lund University
Curated by ChEMBL
Lund University
Curated by ChEMBL
Affinity DataKi: 89nMAssay Description:Displacement of [3H]Flumazenil from human GABA-Aalpha3 receptor plus beta-2-gamma-2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 104nMAssay Description:Inhibitory concentration required for displacing radioligand [3H]SPI from DA D-2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 104nMAssay Description:Compound was evaluated for binding affinity towards DA D-2 receptor using radioligand [3H]SPIMore data for this Ligand-Target Pair
Affinity DataKi: 192nMAssay Description:Binding affinity to displace [3H]- SCH 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 192nMAssay Description:Compound was tested for the displacement of [3H]-SCH- 23390 from dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 513nMAssay Description:Binding affinity to displace [3H]-SCH- 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 531nMAssay Description:Binding affinity to displace [3H]-SCH- 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 898nMAssay Description:Binding affinity to displace [3H]-SCH- 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 1.22E+3nMAssay Description:Binding affinity against Dopamine receptor D1 in rat radioligandMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Homo sapiens (Human))
Lund University
Curated by ChEMBL
Lund University
Curated by ChEMBL
Affinity DataKi: 1.85E+3nMAssay Description:Displacement of [3H]Flumazenil from human GABA-Aalpha3 receptor plus beta-2-gamma-2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0300nMAssay Description:Displacement of [125I]-GLP1 from human GLP1 receptor expressed in BHK cells after 2 hrs in absence of human serum albuminMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0400nMAssay Description:Displacement of [125I]-GLP1 from human GLP1 receptor expressed in BHK cells after 2 hrs in absence of human serum albuminMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0600nMAssay Description:Displacement of [125I]-GLP1 from human GLP1 receptor expressed in BHK cells after 2 hrs in absence of human serum albuminMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0600nMAssay Description:Displacement of [125I]-GLP1 from human GLP1 receptor expressed in BHK cells after 2 hrs in absence of human serum albuminMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0800nMAssay Description:Displacement of [125I]-GLP1 from human GLP1 receptor expressed in BHK cells after 2 hrs in presence of 2% human serum albuminMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0900nMAssay Description:Displacement of [125I]-GLP1 from human GLP1 receptor expressed in BHK cells after 2 hrs in absence of human serum albuminMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Displacement of [125I]-GLP1 from human GLP1 receptor expressed in BHK cells after 2 hrs in presence of 2% human serum albuminMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Displacement of [125I]-GLP1 from human GLP1 receptor expressed in BHK cells after 2 hrs in absence of human serum albuminMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Displacement of [125I]-GLP1 from human GLP1 receptor expressed in BHK cells after 2 hrs in absence of human serum albuminMore data for this Ligand-Target Pair
Affinity DataIC50: 0.110nMAssay Description:Displacement of [125I]-GLP1 from human GLP1 receptor expressed in BHK cells after 2 hrs in absence of human serum albuminMore data for this Ligand-Target Pair
Affinity DataIC50: 0.110nMAssay Description:Displacement of [125I]-GLP1 from human GLP1 receptor expressed in BHK cells after 2 hrs in absence of human serum albuminMore data for this Ligand-Target Pair
Affinity DataIC50: 0.120nMAssay Description:Displacement of [125I]-GLP1 from human GLP1 receptor expressed in BHK cells after 2 hrs in absence of human serum albuminMore data for this Ligand-Target Pair
Affinity DataIC50: 0.130nMAssay Description:Displacement of [125I]-GLP1 from human GLP1 receptor expressed in BHK cells after 2 hrs in absence of human serum albuminMore data for this Ligand-Target Pair
Affinity DataIC50: 0.140nMAssay Description:Displacement of [125I]-GLP1 from human GLP1 receptor expressed in BHK cells after 2 hrs in presence of 2% human serum albuminMore data for this Ligand-Target Pair