TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARgamma after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 2.10E+3nMAssay Description:Agonist activity at human PPARalpha after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 2.30nMAssay Description:Agonist activity at GAL4-fused human PPARalpha LBDMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 5.60E+3nMAssay Description:Agonist activity at human PPARgamma after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARdelta after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 5.10E+3nMAssay Description:Agonist activity at human PPARalpha after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 5.60E+3nMAssay Description:Agonist activity at human PPARalpha after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARdelta after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 2nMAssay Description:Agonist activity at human PPARdelta after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARgamma after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 1.83E+4nMAssay Description:Agonist activity at human PPARgamma after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 0.280nMAssay Description:Agonist activity at GAL4-fused human PPARgamma LBDMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 2.50E+4nMAssay Description:Agonist activity at PPARalpha (unknown origin) expressed in reporter combo cells after 36 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 5.24E+4nMAssay Description:Agonist activity at human PPARalpha after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 2.53E+4nMAssay Description:Agonist activity at human PPARalpha after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 12nMAssay Description:Agonist activity at human PPARalpha after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 8.90E+3nMAssay Description:Agonist activity at human PPARdelta after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 83nMAssay Description:Agonist activity at human PPARgamma after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 3.86E+4nMAssay Description:Agonist activity at human PPARdelta after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 900nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 8.52E+3nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 29nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 27nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 18nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 67nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 52nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARgamma expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARgamma expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 280nMAssay Description:Agonist activity at human PPARgamma expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARgamma expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARdelta expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 1.90nMAssay Description:Agonist activity at human PPARdelta expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 300nMAssay Description:Binding affinity to PPARalpha in human MIO-M1 cells assessed as increase in thermal stability preincubated for 3 hrs followed by exposure to 45.5 deg...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 93nMAssay Description:Binding affinity to PPARalpha in human MIO-M1 cells assessed as increase in thermal stability preincubated for 3 hrs followed by exposure to 45.5 deg...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataKd: 170nMAssay Description:Binding affinity to His-tagged PPARalpha LBD (unknown origin) expressed in Escherichia coli Rosetta (DE3) at 25 degree C by isothermal titration calo...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataKd: 140nMAssay Description:Binding affinity to His-tagged PPARalpha LBD (unknown origin) expressed in Escherichia coli Rosetta (DE3) at 25 degree C by isothermal titration calo...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARdelta expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataKd: 1.69E+4nMAssay Description:Binding affinity to His-tagged PPARalpha LBD (unknown origin) expressed in Escherichia coli Rosetta (DE3) at 25 degree C by isothermal titration calo...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 2.53E+4nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 1.45E+3nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 540nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 1.45E+3nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 2.56E+4nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 56nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 40nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARgamma expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARgamma expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARdelta expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataKd: 5.32E+3nMAssay Description:Binding affinity to His-tagged PPARalpha LBD (unknown origin) expressed in Escherichia coli Rosetta (DE3) at 25 degree C by isothermal titration calo...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 1.12E+3nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
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