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Found 22 with Last Name = 'rigat' and Initial = 'kl'
TargetRNA-directed RNA polymerase(Hepacivirus C)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50484982(CHEMBL2017865)
Affinity DataIC50: >600nMAssay Description:Inhibition of Hepatitis C virus NS5B RNA-dependent RNA polymerase P495L mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRNA-directed RNA polymerase(Hepacivirus C)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50484986(CHEMBL2017863)
Affinity DataIC50:  1.73E+3nMAssay Description:Inhibition of Hepatitis C virus NS5B RNA-dependent RNA polymerase P495L mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRNA-directed RNA polymerase(Hepacivirus C)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50484981(CHEMBL2017862)
Affinity DataIC50:  2.28E+3nMAssay Description:Inhibition of Hepatitis C virus NS5B RNA-dependent RNA polymerase P495L mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRNA-directed RNA polymerase(Hepacivirus C)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50484983(CHEMBL2017866)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of Hepatitis C virus NS5B RNA-dependent RNA polymerase P495L mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRNA-directed RNA polymerase(Hepacivirus C)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50484985(CHEMBL2017864)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of Hepatitis C virus NS5B RNA-dependent RNA polymerase P495L mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRNA-directed RNA polymerase(Hepacivirus C)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50484977(CHEMBL2017856)
Affinity DataIC50:  3.39E+3nMAssay Description:Inhibition of Hepatitis C virus NS5B RNA-dependent RNA polymerase P495L mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRNA-directed RNA polymerase(Hepacivirus C)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50484984(CHEMBL2017858)
Affinity DataIC50:  3.72E+3nMAssay Description:Inhibition of Hepatitis C virus NS5B RNA-dependent RNA polymerase P495L mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRNA-directed RNA polymerase(Hepacivirus C)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50484980(CHEMBL2017861)
Affinity DataIC50:  4.84E+3nMAssay Description:Inhibition of Hepatitis C virus NS5B RNA-dependent RNA polymerase P495L mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRNA-directed RNA polymerase(Hepacivirus C)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50484979(CHEMBL2017860)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibition of Hepatitis C virus NS5B RNA-dependent RNA polymerase P495L mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRNA-directed RNA polymerase(Hepacivirus C)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50484978(CHEMBL2017857)
Affinity DataIC50:  5.85E+3nMAssay Description:Inhibition of Hepatitis C virus NS5B RNA-dependent RNA polymerase P495L mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50142902(CHEMBL3760108)
Affinity DataIC50:  1.66E+4nMAssay Description:Inhibition of human ERG by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50268397(CHEMBL4067852)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of human DNA polymerase betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase alpha catalytic subunit(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50268397(CHEMBL4067852)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of human DNA polymerase alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50448498(BMS-791325 | Beclabuvir)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of human ERG by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50142900(CHEMBL3759768)
Affinity DataIC50:  3.81E+4nMAssay Description:Inhibition of human ERG by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50142901(CHEMBL3758288)
Affinity DataIC50:  4.09E+4nMAssay Description:Inhibition of human ERG by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50268401(CHEMBL4105584)
Affinity DataEC50: >5.00E+4nMAssay Description:Activation of PXR in human hepatocytes assessed as induction of CYP450 expressionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50268400(CHEMBL4081189)
Affinity DataEC50:  8.33E+3nMAssay Description:Activation of PXR in human hepatocytes assessed as induction of CYP450 expressionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50268399(CHEMBL4094467)
Affinity DataEC50:  2.78E+3nMAssay Description:Activation of PXR in human hepatocytes assessed as induction of CYP450 expressionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50268398(CHEMBL4061940)
Affinity DataEC50:  1.67E+4nMAssay Description:Activation of PXR in human hepatocytes assessed as induction of CYP450 expressionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50268397(CHEMBL4067852)
Affinity DataEC50:  1.67E+4nMAssay Description:Activation of PXR in human hepatocytes assessed as induction of CYP450 expressionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50142901(CHEMBL3758288)
Affinity DataEC50: >5.00E+4nMAssay Description:Activation of PXR in human hepatocytes assessed as induction of CYP450 expressionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed