Affinity DataKi: 0.5nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 2More data for this Ligand-Target Pair
Affinity DataKi: 0.560nMAssay Description:Inhibition of Plasmodium falciparum recombinant plasmepsin 2 expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
Affinity DataKi: 35.7nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 2 expressed in Escherichia coli BL21 (DE3) after 40 mins by Kitz-Wilson plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 121nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 2More data for this Ligand-Target Pair
Affinity DataKi: 333nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 2 expressed in Escherichia coli BL21 (DE3) after 40 mins by Kitz-Wilson plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 357nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 2More data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Inhibition of HIV-1 NL4-3 wild type protease expressed in Escherichia coli preincubated for 20 mins by FRET analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Inhibition of HIV-1 NL4-3 wild type protease expressed in Escherichia coli preincubated for 20 mins by FRET analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Inhibition of HIV-1 NL4-3 wild type protease expressed in Escherichia coli preincubated for 20 mins by FRET analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Competitive inhibition of Plasmodium falciparum plasmepsin 2 expressed in Escherichia coli BL21 (DE3) after 30 mins by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Competitive inhibition of Plasmodium falciparum plasmepsin 2 expressed in Escherichia coli BL21 (DE3) after 30 mins by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Inhibition of HIV-1 NL4-3 wild type protease expressed in Escherichia coli preincubated for 20 mins by FRET analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibition of Norovirus prototypic GI.1 3CL protease using HiLyte Fluor 488-labelled DFELQGPK as substrate incubated for 90 mins measured every mins ...More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of human cathepsin D after 30 mins by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of human cathepsin D after 30 mins by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of human cathepsin D after 30 mins by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of human cathepsin D after 30 mins by FRET assayMore data for this Ligand-Target Pair
TargetGenome polyprotein(Norovirus Hu/GII.4-2002/WeertE022/2002/NL)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of Norovirus prototypic GII.4 3CL protease using HiLyte Fluor 488-labelled DFELQGPK as substrate incubated for 90 mins measured every mins...More data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibition of Norovirus prototypic GI.1 3CL protease using HiLyte Fluor 488-labelled DFELQGPK as substrate incubated for 90 mins measured every mins ...More data for this Ligand-Target Pair
Affinity DataIC50: 141nMAssay Description:Competitive inhibition of Plasmodium falciparum plasmepsin 2 expressed in Escherichia coli BL21 (DE3) after 30 mins by FRET assayMore data for this Ligand-Target Pair
TargetGenome polyprotein(Norovirus Hu/GII.4-2002/WeertE022/2002/NL)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of Norovirus prototypic GII.4 3CL protease using HiLyte Fluor 488-labelled DFELQGPK as substrate incubated for 90 mins measured every mins...More data for this Ligand-Target Pair
Affinity DataIC50: 333nMAssay Description:Competitive inhibition of Plasmodium falciparum plasmepsin 2 expressed in Escherichia coli BL21 (DE3) after 30 mins by FRET assayMore data for this Ligand-Target Pair
TargetGenome polyprotein(Norovirus Hu/GII.4-2002/WeertE022/2002/NL)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataIC50: 502nMAssay Description:Inhibition of Norovirus prototypic GII.4 3CL protease using HiLyte Fluor 488-labelled DFELQGPK as substrate incubated for 90 mins measured every mins...More data for this Ligand-Target Pair
Affinity DataIC50: 593nMAssay Description:Inhibition of Norovirus prototypic GI.1 3CL protease using HiLyte Fluor 488-labelled DFELQGPK as substrate incubated for 90 mins measured every mins ...More data for this Ligand-Target Pair
Affinity DataIC50: 654nMAssay Description:Inhibition of Norovirus prototypic GI.1 3CL protease using HiLyte Fluor 488-labelled DFELQGPK as substrate incubated for 90 mins measured every mins ...More data for this Ligand-Target Pair
Affinity DataIC50: 654nMAssay Description:Inhibition of Norovirus prototypic GI.1 3CL protease using HiLyte Fluor 488-labelled DFELQGPK as substrate incubated for 90 mins measured every mins ...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of Norovirus prototypic GI.1 3CL protease using HiLyte Fluor 488-labelled DFELQGPK as substrate incubated for 90 mins measured every mins ...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of Norovirus prototypic GI.1 3CL protease using HiLyte Fluor 488-labelled DFELQGPK as substrate incubated for 90 mins measured every mins ...More data for this Ligand-Target Pair
TargetGenome polyprotein(Norovirus Hu/GII.4-2002/WeertE022/2002/NL)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataIC50: 1.17E+3nMAssay Description:Inhibition of Norovirus prototypic GII.4 3CL protease using HiLyte Fluor 488-labelled DFELQGPK as substrate incubated for 90 mins measured every mins...More data for this Ligand-Target Pair
TargetGenome polyprotein(Norovirus Hu/GII.4-2002/WeertE022/2002/NL)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataIC50: 2.63E+3nMAssay Description:Inhibition of Norovirus prototypic GII.4 3CL protease using HiLyte Fluor 488-labelled DFELQGPK as substrate incubated for 90 mins measured every mins...More data for this Ligand-Target Pair
TargetGenome polyprotein(Norovirus Hu/GII.4-2002/WeertE022/2002/NL)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataIC50: 2.63E+3nMAssay Description:Inhibition of Norovirus prototypic GII.4 3CL protease using HiLyte Fluor 488-labelled DFELQGPK as substrate incubated for 90 mins measured every mins...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Norovirus prototypic GI.1 3CL protease using HiLyte Fluor 488-labelled DFELQGPK as substrate incubated for 90 mins measured every mins ...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Norovirus prototypic GI.1 3CL protease using HiLyte Fluor 488-labelled DFELQGPK as substrate incubated for 90 mins measured every mins ...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Norovirus prototypic GI.1 3CL protease using HiLyte Fluor 488-labelled DFELQGPK as substrate incubated for 90 mins measured every mins ...More data for this Ligand-Target Pair
TargetGenome polyprotein(Norovirus Hu/GII.4-2002/WeertE022/2002/NL)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Norovirus prototypic GII.4 3CL protease using HiLyte Fluor 488-labelled DFELQGPK as substrate incubated for 90 mins measured every mins...More data for this Ligand-Target Pair
TargetGenome polyprotein(Norovirus Hu/GII.4-2002/WeertE022/2002/NL)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Norovirus prototypic GII.4 3CL protease using HiLyte Fluor 488-labelled DFELQGPK as substrate incubated for 90 mins measured every mins...More data for this Ligand-Target Pair
TargetGenome polyprotein(Norovirus Hu/GII.4-2002/WeertE022/2002/NL)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of Norovirus prototypic GII.4 3CL protease using HiLyte Fluor 488-labelled DFELQGPK as substrate incubated for 90 mins measured every mins...More data for this Ligand-Target Pair
TargetGenome polyprotein(Norovirus Hu/GII.4-2002/WeertE022/2002/NL)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Norovirus prototypic GII.4 3CL protease using HiLyte Fluor 488-labelled DFELQGPK as substrate incubated for 90 mins measured every mins...More data for this Ligand-Target Pair
TargetGenome polyprotein(Norovirus Hu/GII.4-2002/WeertE022/2002/NL)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Norovirus prototypic GII.4 3CL protease using HiLyte Fluor 488-labelled DFELQGPK as substrate incubated for 90 mins measured every mins...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Norovirus prototypic GI.1 3CL protease using HiLyte Fluor 488-labelled DFELQGPK as substrate incubated for 90 mins measured every mins ...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Norovirus prototypic GI.1 3CL protease using HiLyte Fluor 488-labelled DFELQGPK as substrate incubated for 90 mins measured every mins ...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Norovirus prototypic GI.1 3CL protease using HiLyte Fluor 488-labelled DFELQGPK as substrate incubated for 90 mins measured every mins ...More data for this Ligand-Target Pair
TargetGenome polyprotein(Norovirus Hu/GII.4-2002/WeertE022/2002/NL)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Norovirus prototypic GII.4 3CL protease using HiLyte Fluor 488-labelled DFELQGPK as substrate incubated for 90 mins measured every mins...More data for this Ligand-Target Pair
TargetGenome polyprotein(Norovirus Hu/GII.4-2002/WeertE022/2002/NL)
Emory University
Curated by ChEMBL
Emory University
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Norovirus prototypic GII.4 3CL protease using HiLyte Fluor 488-labelled DFELQGPK as substrate incubated for 90 mins measured every mins...More data for this Ligand-Target Pair