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Found 66 with Last Name = 'osborne' and Initial = 'm'
TargetAdenosine receptor A2a(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50330987(2-amino-4-phenyl-8-(pyrrolidin-1-ylmethyl)-5H-inde...)
Affinity DataKi:  4.10nMAssay Description:Antagonist activity at adenosine A2A receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50330987(2-amino-4-phenyl-8-(pyrrolidin-1-ylmethyl)-5H-inde...)
Affinity DataKi:  17nMAssay Description:Antagonist activity at adenosine A1 receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM50125052(CHEMBL3623004 | US10130617, Example 1 | US20240043...)
Affinity DataIC50:  140nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM292004((E)-3-(3,5-difluoro-4-(2-((S)-3-fluoro-2-methylpro...)
Affinity DataIC50:  200nMAssay Description:The ability of compounds to bind to isolated Estrogen Receptor Alpha Ligand binding domain (ER alpha LBD (GST)) was assessed in competition assays us...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM289785((E)-3-(3,5-Difluoro-4-((1R,3R)-2-((S)-3-fluoro-2-m...)
Affinity DataIC50:  400nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM292005((E)-3-(3,5-difluoro-4-(2-(2-fluoro-2-methylpropyl)...)
Affinity DataIC50:  440nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM292004((E)-3-(3,5-difluoro-4-(2-((S)-3-fluoro-2-methylpro...)
Affinity DataIC50:  570nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM50125052(CHEMBL3623004 | US10130617, Example 1 | US20240043...)
Affinity DataIC50: <640nMAssay Description:The ability of compounds to bind to isolated Estrogen Receptor Alpha Ligand binding domain (ER alpha LBD (GST)) was assessed in competition assays us...More data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM50125054(CHEMBL3623003 | US10130617, Example 2 | WO-2014/19...)
Affinity DataIC50:  850nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM292003((E)-3-(4-((1R,3R)-2-((S)-3-fluoro-2-methylpropyl)-...)
Affinity DataIC50:  990nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM289785((E)-3-(3,5-Difluoro-4-((1R,3R)-2-((S)-3-fluoro-2-m...)
Affinity DataIC50:  1.00E+3nMAssay Description:The ability of compounds to bind to isolated Estrogen Receptor Alpha Ligand binding domain (ER alpha LBD (GST)) was assessed in competition assays us...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM50125054(CHEMBL3623003 | US10130617, Example 2 | WO-2014/19...)
Affinity DataIC50:  1.00E+3nMAssay Description:The ability of compounds to bind to isolated Estrogen Receptor Alpha Ligand binding domain (ER alpha LBD (GST)) was assessed in competition assays us...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM299742((E)-3-(3-fluoro-4-(2-((S)-3-fluoro-2-methylpropyl)...)
Affinity DataIC50: <1.20E+3nMAssay Description:The ability of compounds to bind to isolated Estrogen Receptor Alpha Ligand binding domain (ER alpha LBD (GST)) was assessed in competition assays us...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM292005((E)-3-(3,5-difluoro-4-(2-(2-fluoro-2-methylpropyl)...)
Affinity DataIC50: <1.30E+3nMAssay Description:The ability of compounds to bind to isolated Estrogen Receptor Alpha Ligand binding domain (ER alpha LBD (GST)) was assessed in competition assays us...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM299742((E)-3-(3-fluoro-4-(2-((S)-3-fluoro-2-methylpropyl)...)
Affinity DataIC50:  1.50E+3nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM292003((E)-3-(4-((1R,3R)-2-((S)-3-fluoro-2-methylpropyl)-...)
Affinity DataIC50:  1.60E+3nMAssay Description:The ability of compounds to bind to isolated Estrogen Receptor Alpha Ligand binding domain (ER alpha LBD (GST)) was assessed in competition assays us...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM298313((E)-3-(4-(2-((S)-3-fluoro-2-methylpropyl)-3,3-dime...)
Affinity DataIC50:  1.70E+3nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM298314((E)-3-(4-(2-(2-fluoro-2-methylpropyl)-3,3-dimethyl...)
Affinity DataIC50:  2.20E+3nMAssay Description:The ability of compounds to bind to isolated Estrogen Receptor Alpha Ligand binding domain (ER alpha LBD (GST)) was assessed in competition assays us...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM298314((E)-3-(4-(2-(2-fluoro-2-methylpropyl)-3,3-dimethyl...)
Affinity DataIC50:  3.00E+3nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM298313((E)-3-(4-(2-((S)-3-fluoro-2-methylpropyl)-3,3-dime...)
Affinity DataIC50:  5.00E+3nMAssay Description:The ability of compounds to bind to isolated Estrogen Receptor Alpha Ligand binding domain (ER alpha LBD (GST)) was assessed in competition assays us...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50138056((2-{2-[4-(5-Hydroxyimino-hexyl)-3-oxo-3,4-dihydro-...)
Affinity DataEC50:  10nMAssay Description:Agonistic activity against PPAR (peroxisome proliferator activated receptor gamma) in Suarus chinesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50138059((2-{2-[(R)-4-(4-Methoxy-butyl)-3-oxo-3,4-dihydro-2...)
Affinity DataEC50:  274nMAssay Description:Agonistic activity against PPAR (peroxisome proliferator activated receptor gamma) in Suarus chinesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50138057((2-{2-[4-(5-Hydroxy-pentyl)-3-oxo-3,4-dihydro-2H-b...)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonistic activity against PPAR (peroxisome proliferator activated receptor gamma) in Suarus chinesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50138058(CHEMBL427478 | {2-[2-(4-Ethyl-3-oxo-3,4-dihydro-2H...)
Affinity DataEC50: >5.00E+3nMAssay Description:Agonistic activity against PPAR (peroxisome proliferator activated receptor gamma) in Suarus chinesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50138062((2-{2-[(S)-4-(6-Fluoro-hexyl)-3-oxo-3,4-dihydro-2H...)
Affinity DataEC50:  570nMAssay Description:Agonistic activity against PPAR (peroxisome proliferator activated receptor gamma) in Suarus chinesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50138063((2-{2-[4-(7-Fluoro-heptyl)-3-oxo-3,4-dihydro-2H-be...)
Affinity DataEC50:  718nMAssay Description:Agonistic activity against PPAR (peroxisome proliferator activated receptor gamma) in Suarus chinesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50138061((2-{2-[4-(3-Cyclopentyl-propyl)-3-oxo-3,4-dihydro-...)
Affinity DataEC50:  2.70E+3nMAssay Description:Agonistic activity against PPAR (peroxisome proliferator activated receptor gamma) in Suarus chinesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50138060(5-{2-[2-(2-Carboxymethyl-phenoxy)-ethyl]-3-oxo-2,3...)
Affinity DataEC50: >5.00E+3nMAssay Description:Agonistic activity against PPAR (peroxisome proliferator activated receptor gamma) in Suarus chinesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50138065((2-{2-[4-(2-Hydroxy-ethyl)-3-oxo-3,4-dihydro-2H-be...)
Affinity DataEC50: >5.00E+3nMAssay Description:Agonistic activity against PPAR (peroxisome proliferator activated receptor gamma) in Suarus chinesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50138064(CHEMBL178536 | {2-[2-(4-Octyl-3-oxo-3,4-dihydro-2H...)
Affinity DataEC50:  300nMAssay Description:Agonistic activity against PPAR (peroxisome proliferator activated receptor gamma) in Suarus chinesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50138066((2-{2-[4-(5,5-Difluoro-hexyl)-3-oxo-3,4-dihydro-2H...)
Affinity DataEC50:  179nMAssay Description:Agonistic activity against PPAR (peroxisome proliferator activated receptor gamma) in Suarus chinesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50138067((2-{2-[4-(4-Methoxy-butyl)-3-oxo-3,4-dihydro-2H-be...)
Affinity DataEC50:  274nMAssay Description:Agonistic activity against PPAR (peroxisome proliferator activated receptor gamma) in Suarus chinesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50138068(CHEMBL174167 | {2-[2-(4-Methyl-3-oxo-3,4-dihydro-2...)
Affinity DataEC50: >5.00E+3nMAssay Description:Agonistic activity against PPAR (peroxisome proliferator activated receptor gamma) in Suarus chinesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50138069((2-{2-[4-(5-Hydroxy-hexyl)-3-oxo-3,4-dihydro-2H-be...)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonistic activity against PPAR (peroxisome proliferator activated receptor gamma) in Suarus chinesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50138071((2-{2-[(S)-4-(5,5-Difluoro-hexyl)-3-oxo-3,4-dihydr...)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonistic activity against PPAR (peroxisome proliferator activated receptor gamma) in Suarus chinesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50138070((2-{2-[(R)-4-(6-Fluoro-hexyl)-3-oxo-3,4-dihydro-2H...)
Affinity DataEC50:  152nMAssay Description:Agonistic activity against PPAR (peroxisome proliferator activated receptor gamma) in Suarus chinesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50138072(CHEMBL176770 | {2-[2-(4-Heptyl-3-oxo-3,4-dihydro-2...)
Affinity DataEC50:  234nMAssay Description:Agonistic activity against PPAR (peroxisome proliferator activated receptor gamma) in Suarus chinesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50138073((2-{2-[(R)-4-(5,5-Difluoro-hexyl)-3-oxo-3,4-dihydr...)
Affinity DataEC50:  295nMAssay Description:Agonistic activity against PPAR (peroxisome proliferator activated receptor gamma) in Suarus chinesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50138076((2-{2-[4-(4-Carbamoyl-butyl)-3-oxo-3,4-dihydro-2H-...)
Affinity DataEC50: >5.00E+3nMAssay Description:Agonistic activity against PPAR (peroxisome proliferator activated receptor gamma) in Suarus chinesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50138077(6-{2-[2-(2-Carboxymethyl-phenoxy)-ethyl]-3-oxo-2,3...)
Affinity DataEC50: >5.00E+3nMAssay Description:Agonistic activity against PPAR (peroxisome proliferator activated receptor gamma) in Suarus chinesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50138074((2-{2-[4-(6-Fluoro-hexyl)-3-oxo-3,4-dihydro-2H-ben...)
Affinity DataEC50:  117nMAssay Description:Agonistic activity against PPAR (peroxisome proliferator activated receptor gamma) in Suarus chinesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50138075(CHEMBL174644 | {2-[2-(4-Isopropyl-3-oxo-3,4-dihydr...)
Affinity DataEC50: >5.00E+3nMAssay Description:Agonistic activity against PPAR (peroxisome proliferator activated receptor gamma) in Suarus chinesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50138079(6-{2-[2-(2-Carboxymethyl-phenoxy)-ethyl]-3-oxo-2,3...)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonistic activity against PPAR (peroxisome proliferator activated receptor gamma) in Suarus chinesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50138078(CHEMBL177830 | {2-[2-(4-Hex-5-enyl-3-oxo-3,4-dihyd...)
Affinity DataEC50:  208nMAssay Description:Agonistic activity against PPAR (peroxisome proliferator activated receptor gamma) in Suarus chinesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50138082((2-{2-[4-(5-Hydroxy-5-methyl-hexyl)-3-oxo-3,4-dihy...)
Affinity DataEC50:  644nMAssay Description:Agonistic activity against PPAR (peroxisome proliferator activated receptor gamma) in Suarus chinesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50138083((2-{2-[3-Oxo-4-(5-oxo-hexyl)-3,4-dihydro-2H-benzo[...)
Affinity DataEC50:  260nMAssay Description:Agonistic activity against PPAR (peroxisome proliferator activated receptor gamma) in Suarus chinesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50138085(CHEMBL369054 | {2-[2-(4-Decyl-3-oxo-3,4-dihydro-2H...)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonistic activity against PPAR (peroxisome proliferator activated receptor gamma) in Suarus chinesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50138080(CHEMBL176035 | {2-[2-(3-Oxo-4-propylcarbamoylmethy...)
Affinity DataEC50: >5.00E+3nMAssay Description:Agonistic activity against PPAR (peroxisome proliferator activated receptor gamma) in Suarus chinesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50138081((2-{2-[4-(3-Methylcarbamoyl-propyl)-3-oxo-3,4-dihy...)
Affinity DataEC50: >5.00E+3nMAssay Description:Agonistic activity against PPAR (peroxisome proliferator activated receptor gamma) in Suarus chinesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50138084(CHEMBL177439 | {2-[2-(2-Carboxymethyl-phenoxy)-eth...)
Affinity DataEC50: >5.00E+3nMAssay Description:Agonistic activity against PPAR (peroxisome proliferator activated receptor gamma) in Suarus chinesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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