TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 0.690nMAssay Description:Inhibitory constant against rat prostate cytosol androgen receptor using [3H]miboleroneMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 0.710nMAssay Description:Inhibition of rat prostate cytosolic androgen receptorMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 0.710nMAssay Description:Inhibitory constant against rat prostate cytosol androgen receptor using [3H]miboleroneMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 0.75nMAssay Description:Binding affinity against rat prostate cytosolic Androgen receptor using [3H]mibolerone as radioligandMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 0.75nMAssay Description:Inhibition of rat prostate cytosolic androgen receptorMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 0.75nMAssay Description:Inhibitory constant against rat prostate cytosol androgen receptor using [3H]miboleroneMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Inhibitory constant against rat prostate cytosol androgen receptor using [3H]miboleroneMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Inhibition of rat prostate cytosolic androgen receptorMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Inhibitory constant against rat prostate cytosol androgen receptor using [3H]miboleroneMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 2.23nMAssay Description:Inhibition of rat prostate cytosolic androgen receptorMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Inhibition of rat prostate cytosolic androgen receptorMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 4.90nMAssay Description:Inhibition of rat prostate cytosolic androgen receptorMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 4.90nMAssay Description:Binding affinity against rat prostate cytosolic Androgen receptor using [3H]mibolerone as radioligandMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
University of Michigan Medical Center
Curated by ChEMBL
University of Michigan Medical Center
Curated by ChEMBL
Affinity DataKi: 7.30nMAssay Description:Binding affinity for peripheral benzodiazepine receptor of rat kidneyMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Inhibition of rat prostate cytosolic androgen receptorMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
University of Michigan Medical Center
Curated by ChEMBL
University of Michigan Medical Center
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Binding affinity for peripheral benzodiazepine receptor of rat kidneyMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Binding affinity against rat prostate cytosolic Androgen receptor using [3H]mibolerone as radioligandMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
University of Michigan Medical Center
Curated by ChEMBL
University of Michigan Medical Center
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Binding affinity for peripheral benzodiazepine receptor of rat kidneyMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Inhibition of rat prostate cytosolic androgen receptorMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 26nMAssay Description:Inhibition of rat prostate cytosolic androgen receptorMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 26nMAssay Description:Binding affinity against rat prostate cytosolic Androgen receptor using [3H]mibolerone as radioligandMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:Binding affinity against rat prostate cytosolic Androgen receptor using [3H]mibolerone as radioligandMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:Inhibition of rat prostate cytosolic androgen receptorMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 59nMAssay Description:Inhibition of rat prostate cytosolic androgen receptorMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 65nMAssay Description:Binding affinity against rat prostate cytosolic Androgen receptor using [3H]mibolerone as radioligandMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 77nMAssay Description:Inhibition of rat prostate cytosolic androgen receptorMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 117nMAssay Description:Inhibition of rat prostate cytosolic androgen receptorMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:Binding affinity against rat prostate cytosolic Androgen receptor using [3H]mibolerone as radioligandMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 123nMAssay Description:Binding affinity against rat prostate cytosolic Androgen receptor using [3H]mibolerone as radioligandMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 141nMAssay Description:Binding affinity against rat prostate cytosolic Androgen receptor using [3H]mibolerone as radioligandMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 150nMAssay Description:Binding affinity against rat prostate cytosolic Androgen receptor using [3H]mibolerone as radioligandMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 213nMAssay Description:Binding affinity against rat prostate cytosolic Androgen receptor using [3H]mibolerone as radioligandMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 219nMAssay Description:Inhibition of rat prostate cytosolic androgen receptorMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 321nMAssay Description:Binding affinity against rat prostate cytosolic Androgen receptor using [3H]mibolerone as radioligandMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 360nMAssay Description:Binding affinity against rat prostate cytosolic Androgen receptor using [3H]mibolerone as radioligandMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 400nMAssay Description:Inhibition of rat prostate cytosolic androgen receptorMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 415nMAssay Description:Binding affinity against rat prostate cytosolic Androgen receptor using [3H]mibolerone as radioligandMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 639nMAssay Description:Inhibition of rat prostate cytosolic androgen receptorMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataKi: 809nMAssay Description:Binding affinity against rat prostate cytosolic Androgen receptor using [3H]mibolerone as radioligandMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataIC50: 0.00715nMAssay Description:Inhibition of purified MEK1 (unknown origin) assessed as reduction in phosphorylation of inactive Erk2 incubated for 30 mins by Kinase-Glo luminescen...More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataIC50: 0.0150nMAssay Description:Inhibition of purified MEK1 (unknown origin) assessed as reduction in phosphorylation of inactive Erk2 incubated for 30 mins by Kinase-Glo luminescen...More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataIC50: 0.0190nMAssay Description:Inhibition of purified MEK1 (unknown origin) assessed as reduction in phosphorylation of inactive Erk2 incubated for 30 mins by Kinase-Glo luminescen...More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Mus musculus)
University of Michigan
Curated by ChEMBL
University of Michigan
Curated by ChEMBL
Affinity DataIC50: 0.330nMAssay Description:Inhibition of MEK1 in mouse colon 26 cells assessed as reduction in ERK1/2 phosphorylation after 1 hr by Western blot analysisMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
The University Of Michigan Medical School
Curated by ChEMBL
The University Of Michigan Medical School
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of purified MEK1 (unknown origin) assessed as reduction in phosphorylation of inactive Erk2 incubated for 30 mins by Kinase-Glo luminescen...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University of Michigan
Curated by ChEMBL
University of Michigan
Curated by ChEMBL
Affinity DataIC50: <0.700nMAssay Description:Inhibition of PI3K alpha (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University of Michigan
Curated by ChEMBL
University of Michigan
Curated by ChEMBL
Affinity DataIC50: <0.700nMAssay Description:Inhibition of PI3K alpha (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
University of Michigan
Curated by ChEMBL
University of Michigan
Curated by ChEMBL
Affinity DataIC50: <0.700nMAssay Description:Inhibition of PI3K delta (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
University of Michigan
Curated by ChEMBL
University of Michigan
Curated by ChEMBL
Affinity DataIC50: <0.700nMAssay Description:Inhibition of PI3K delta (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
University of Michigan
Curated by ChEMBL
University of Michigan
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Inhibition of recombinant human full length His-tagged PI3K p110delta/p85alpha expressed in baculovirus expression system coexpressing PIK3R1 by TR-F...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
University of Michigan
Curated by ChEMBL
University of Michigan
Curated by ChEMBL
Affinity DataIC50: 2.90nMAssay Description:Inhibition of recombinant human full length His-tagged PI3K p110delta/p85alpha expressed in baculovirus expression system coexpressing PIK3R1 by TR-F...More data for this Ligand-Target Pair