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Found 101 with Last Name = 'mosset' and Initial = 'p'
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50592423(CHEMBL4434865)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]-(+)-pentazocine from human sigma1 receptor measured after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50592424(CHEMBL4567314)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]-(+)-pentazocine from human sigma1 receptor measured after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50592426(CHEMBL4547253)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-(+)-pentazocine from human sigma1 receptor measured after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50592427(CHEMBL4444356)
Affinity DataKi:  3.30nMAssay Description:Displacement of [3H]-(+)-pentazocine from human sigma1 receptor measured after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50064947(CHEMBL76895 | N-(1-Benzyl-piperidin-4-yl)-2-phenyl...)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50592424(CHEMBL4567314)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D4.4 receptor measured after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50592426(CHEMBL4547253)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D4.4 receptor measured after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50030474(Avandamet | Avandaryl | Avandia | BRL-49653 | CHEB...)
Affinity DataKi:  8nM ΔG°:  -43.0kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)
Affinity DataKi:  8nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50059227(1-Benzyl-4-(5-phenyl-1H-pyrazol-3-yl)-piperidine |...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]spiperone from recombinant human D4 receptor stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50592425(CHEMBL4435399)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D4.4 receptor measured after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50592425(CHEMBL4435399)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-(+)-pentazocine from human sigma1 receptor measured after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50592427(CHEMBL4444356)
Affinity DataKi:  144nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D4.4 receptor measured after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50592423(CHEMBL4434865)
Affinity DataKi:  260nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D4.4 receptor measured after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM233176(Sodium 8-hydroxy-8-(2-octyloxy-quinolin-3-yl)-oct-...)
Affinity DataKi:  378nM ΔG°:  -34.1kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50172823(8-Hydroxy-8-(2-pentyloxy-phenyl)-octanoic acid met...)
Affinity DataKi:  515nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50172805(9-Hydroxy-9-(3-pentyloxy-naphthalen-2-yl)-nonanoic...)
Affinity DataKi:  579nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM233183(Sodium 8-hydroxy-8-(6-methoxy-2-pentyloxy-quinolin...)
Affinity DataKi:  583nM ΔG°:  -33.1kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50172816(8-Hydroxy-8-(3-pentyloxy-naphthalen-2-yl)-oct-5-yn...)
Affinity DataKi:  695nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50172806((E)-8-Hydroxy-8-(3-pentyloxy-naphthalen-2-yl)-oct-...)
Affinity DataKi:  718nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50172802(CHEMBL383607 | Sodium 8-hydroxy-8-(2-pentyloxy-qui...)
Affinity DataKi:  947nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50172802(CHEMBL383607 | Sodium 8-hydroxy-8-(2-pentyloxy-qui...)
Affinity DataKi:  947nM ΔG°:  -32.0kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50172810(CHEMBL199121 | Sodium; 8-hydroxy-8-(3-pentyloxy-na...)
Affinity DataKi:  969nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50172817(8-Hydroxy-8-(2-pentyloxy-phenyl)-oct-5-ynoic acid ...)
Affinity DataKi:  1.05E+3nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM233180(Sodium [5-hydroxy-5-(2-pentyloxy-quinolin-3-yl)-pe...)
Affinity DataKi:  1.93E+3nM ΔG°:  -30.3kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM233181(Sodium [5-hydroxy-5-(2-methoxy-quinolin-3-yl)-pent...)
Affinity DataKi:  3.81E+3nM ΔG°:  -28.8kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50172822(CHEMBL198163 | Sodium; 8-hydroxy-8-(3-pentyloxy-na...)
Affinity DataKi:  4.39E+3nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50592423(CHEMBL4434865)
Affinity DataKi:  4.60E+3nMAssay Description:Displacement of [3H]dofetilide from recombinant human ERG stably expressed in HEK293 cell membranes measured after 60 mins by scintillation counting ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50592423(CHEMBL4434865)
Affinity DataKi:  6.30E+3nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D2S receptor measured after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50172818(CHEMBL196261 | Sodium; 8-hydroxy-8-(2-pentyloxy-ph...)
Affinity DataKi:  6.69E+3nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM233173(8-Hydroxy-8-[2-(3-methoxy-propoxy)-quinolin-3-yl]-...)
Affinity DataKi: >1.00E+4nM ΔG°: >-26.5kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM233174(8-Hydroxy-8-[2-(4,4,4-trifluoro-butoxy)-quinolin-3...)
Affinity DataKi: >1.00E+4nM ΔG°: >-26.5kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM233175(Sodium 8-hydroxy-8-(2-methoxy-quinolin-3-yl)-oct-5...)
Affinity DataKi: >1.00E+4nM ΔG°: >-26.5kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM233177(Sodium 8-hydroxy-8-[2-(3-methoxy-propoxy)-quinolin...)
Affinity DataKi: >1.00E+4nM ΔG°: >-26.5kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM233178(Sodium 8-hydroxy-8-[2-(4,4,4-trifluoro-butoxy)-qui...)
Affinity DataKi: >1.00E+4nM ΔG°: >-26.5kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM233179(8-Hydroxy-8-(2-pentyloxy-quinolin-3-yl)-oct-5-ynoi...)
Affinity DataKi: >1.00E+4nM ΔG°: >-26.5kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM233182(8-Hydroxy-8-(2-pentyloxy-benzo[h]quinolin-3-yl)-oc...)
Affinity DataKi: >1.00E+4nM ΔG°: >-26.5kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM233184(Sodium 8-hydroxy-8-(2-pentyloxy-benzo[h]quinolin-3...)
Affinity DataKi: >1.00E+4nM ΔG°: >-26.5kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50172808(8-Hydroxy-8-(2-pentyloxy-pyridin-3-yl)-octanoic ac...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50172814(8-Hydroxy-8-(2-pentyloxy-pyridin-3-yl)-oct-5-ynoic...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50172809(CHEMBL199172 | Sodium; 8-hydroxy-8-(2-pentyloxy-py...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50172813(8-Hydroxy-8-(2-pentyloxy-quinolin-3-yl)-oct-5-ynoi...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50172804(CHEMBL198034 | Sodium; 8-hydroxy-8-(2-pentyloxy-py...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50172820(CHEMBL196260 | Sodium; (E)-8-hydroxy-8-(2-pentylox...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50172815(CHEMBL370374 | Sodium; 8-hydroxy-8-(2-pentyloxy-ph...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50172824(9-Hydroxy-9-(2-pentyloxy-quinolin-3-yl)-nonanoic a...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50172803((E)-8-Hydroxy-8-(2-pentyloxy-pyridin-3-yl)-oct-5-e...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens)
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50592423(CHEMBL4434865)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor measured after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50172813(8-Hydroxy-8-(2-pentyloxy-quinolin-3-yl)-oct-5-ynoi...)
Affinity DataKi: >1.00E+4nM ΔG°: >-26.5kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM233172(8-Hydroxy-8-(2-octyloxy-quinolin-3-yl)-oct-5-ynoic...)
Affinity DataKi: >1.00E+4nM ΔG°: >-26.5kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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