Affinity DataKi: 0.0190nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0466nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0500nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
Affinity DataKi: 0.0558nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0596nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
King'S College London
Curated by PDSP Ki Database
King'S College London
Curated by PDSP Ki Database
Affinity DataKi: 0.120nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
King'S College London
Curated by PDSP Ki Database
King'S College London
Curated by PDSP Ki Database
Affinity DataKi: 0.160nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
Affinity DataKi: 0.170nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
King'S College London
Curated by PDSP Ki Database
King'S College London
Curated by PDSP Ki Database
Affinity DataKi: 0.190nMAssay Description:Binding affinity towards melatonin receptor in chicken brain.More data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
King'S College London
Curated by PDSP Ki Database
King'S College London
Curated by PDSP Ki Database
Affinity DataKi: 0.200nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
Affinity DataKi: 0.210nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
Affinity DataKi: 0.260nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
King'S College London
Curated by PDSP Ki Database
King'S College London
Curated by PDSP Ki Database
TargetMelatonin receptor type 1A(Homo sapiens (Human))
King'S College London
Curated by PDSP Ki Database
King'S College London
Curated by PDSP Ki Database
Affinity DataKi: 0.263nMAssay Description:Displacement of 2[125I]iodomelatonin from human recombinant MT1 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.270nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.305nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.330nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
Affinity DataKi: 0.339nMAssay Description:Displacement of 2[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.350nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.355nMAssay Description:Displacement of 2[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.378nMAssay Description:Binding affinity towards melatonin receptor, determined in chicken brain membranes using [2-125I]melatoninMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
King'S College London
Curated by PDSP Ki Database
King'S College London
Curated by PDSP Ki Database
Affinity DataKi: 0.390nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT1 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.410nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
King'S College London
Curated by PDSP Ki Database
King'S College London
Curated by PDSP Ki Database
Affinity DataKi: 0.470nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
Affinity DataKi: 0.510nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
Affinity DataKi: 0.537nMAssay Description:Displacement of 2[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
King'S College London
Curated by PDSP Ki Database
King'S College London
Curated by PDSP Ki Database
Affinity DataKi: 0.590nMAssay Description:Binding affinity towards melatonin receptor in chicken brain.More data for this Ligand-Target Pair
Affinity DataKi: 0.590nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.590nMAssay Description:Binding affinity towards melatonin receptor, determined in chicken brain membranes using [2-125I]melatoninMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
King'S College London
Curated by PDSP Ki Database
King'S College London
Curated by PDSP Ki Database
TargetMelatonin receptor type 1A(Homo sapiens (Human))
King'S College London
Curated by PDSP Ki Database
King'S College London
Curated by PDSP Ki Database
Affinity DataKi: 0.660nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1A expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair