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Found 137 with Last Name = 'gundla' and Initial = 'r'
TargetAdenomatous polyposis coli protein(Homo sapiens (Human))TBA
LigandPNGBDBM50407493(CHEMBL5288446)
Affinity DataKi:  15nMAssay Description:Relative potency against Histamine H1 receptor in rat aortaMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenomatous polyposis coli protein(Homo sapiens (Human))TBA
LigandPNGBDBM50407492(CHEMBL5280732)
Affinity DataKi:  120nMAssay Description:Apparent pA2 value of compound at 50 nM concentration of mepyramine in rat aortaMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenomatous polyposis coli protein(Homo sapiens (Human))TBA
LigandPNGBDBM50407464(CHEMBL5289275)
Affinity DataKi:  2.41E+3nMAssay Description:Apparent pA2 value of compound at 10 nM concentration of mepyramine in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenomatous polyposis coli protein(Homo sapiens (Human))TBA
LigandPNGBDBM50407467(CHEMBL5289169)
Affinity DataKi:  3.12E+3nMAssay Description:Antagonistic activity for carbachol induced contractions in guinea pig ileum against Muscarinic acetylcholine receptor M3 in the presence of mepyrami...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenomatous polyposis coli protein(Homo sapiens (Human))TBA
LigandPNGBDBM50407491(CHEMBL5282293)
Affinity DataKi:  3.80E+3nMAssay Description:Antagonistic activity for carbachol induced contractions in guinea pig ileum against Muscarinic acetylcholine receptor M3 in the presence of mepyrami...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenomatous polyposis coli protein(Homo sapiens (Human))TBA
LigandPNGBDBM50407461(CHEMBL5274458)
Affinity DataKi:  4.46E+4nMAssay Description:Tetsed for Antagonistic activity at histamine H3 receptor in guinea pig ileal longitudinal muscle in the presence of mepyramine at a concentration of...More data for this Ligand-Target Pair
In DepthDetails PubMed
Target7-dehydrocholesterol reductase(Homo sapiens (Human))TBA
LigandPNGBDBM50407454(CHEMBL5281526)
Affinity DataIC50:  0.100nMAssay Description:Antagonistic activity for carbachol induced contractions in guinea pig ileum against Muscarinic acetylcholine receptor M3 in the presence of mepyrami...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483581(CHEMBL1689301)
Affinity DataIC50:  0.520nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50271271((R)-N-(3-chloro-4-(pyrazin-2-ylmethoxy)phenyl)-5-(...)
Affinity DataIC50:  1nMAssay Description:Inhibition of HER2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50271272(CHEMBL490062 | N-(1-benzyl-1H-indazol-5-yl)-6-(5-(...)
Affinity DataIC50:  1nMAssay Description:Inhibition of HER2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483589(CHEMBL1689302)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50270524(2-(4-(3-chloro-4-(pyridin-2-ylmethoxy)phenylamino)...)
Affinity DataIC50:  2nMAssay Description:Inhibition of HER2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483582(CHEMBL1689303)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50407449(CHEMBL5285995)
Affinity DataIC50:  3nMAssay Description:Antagonistic affinity tested against isolated Rat Thoracic Aorta Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483597(CHEMBL1689304)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483583(CHEMBL1689305)
Affinity DataIC50:  4nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50270525((5-(4-(4-(benzyloxy)phenylamino)pyrido[3,4-d]pyrim...)
Affinity DataIC50:  4nMAssay Description:Inhibition of HER2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))TBA
LigandPNGBDBM50407495(CHEMBL5286471)
Affinity DataIC50:  4nMAssay Description:Tetsed for Antagonistic activity at histamine H3 receptor in guinea pig ileal longitudinal muscle in the presence of mepyramine at a concentration of...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDNA polymerase beta(Homo sapiens (Human))TBA
LigandPNGBDBM50407496(CHEMBL5284382)
Affinity DataIC50:  5nMAssay Description:Tetsed for Antagonistic activity at histamine H3 receptor in guinea pig ileal longitudinal muscle in the presence of mepyramine at a concentration of...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483595(CHEMBL1689306)
Affinity DataIC50:  5.40nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483584(CHEMBL1689307)
Affinity DataIC50:  6.90nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50271239(((1S,5R,6s)-3-((4-(4-(3-methoxy-4-phenoxyphenylami...)
Affinity DataIC50:  8nMAssay Description:Inhibition of HER2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50161879(4-Dimethylamino-but-2-enoic acid {4-[3-chloro-4-(3...)
Affinity DataIC50:  8nMAssay Description:Inhibition of HER2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM4581(4-anilinoquinazoline deriv. 10n | CHEMBL93049 | N-...)
Affinity DataIC50:  9nMAssay Description:Inhibition of HER2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM5445(CHEMBL554 | GW572016 | LAPATINIB DITOSYLATE | Lapa...)
Affinity DataIC50:  9nMAssay Description:Inhibition of HER2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50407448(CHEMBL4454956)
Affinity DataIC50:  9.40nMAssay Description:Antagonistic affinity tested against isolated Rat Thoracic Aorta Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM5444(6-Thiazolylquinazoline 6 | CHEMBL453376 | N-{3-chl...)
Affinity DataIC50:  10nMAssay Description:Inhibition of HER2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50407495(CHEMBL5286471)
Affinity DataIC50:  11nMAssay Description:Tetsed for Antagonistic activity at histamine H3 receptor in guinea pig ileal longitudinal muscle in the presence of mepyramine at a concentration of...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM31340(2-methoxy-N-[(E)-3-[4-[3-methyl-4-(6-methylpyridin...)
Affinity DataIC50:  12nMAssay Description:Inhibition of HER2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50270583(CHEMBL488350 | methyl 2-((5-(4-(4-(benzyloxy)pheny...)
Affinity DataIC50:  13nMAssay Description:Inhibition of HER2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50161956(4-Dimethylamino-but-2-enoic acid {4-[3-chloro-4-(4...)
Affinity DataIC50:  13nMAssay Description:Inhibition of HER2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50270523(2-((5-(4-(4-(benzyloxy)phenylamino)pyrido[3,4-d]py...)
Affinity DataIC50:  19nMAssay Description:Inhibition of HER2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483593(CHEMBL1687958)
Affinity DataIC50:  20nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Syntrix Biosystems

Curated by ChEMBL
LigandPNGBDBM150812(US8981106, 2 (SX-576) | USRE47267, Compound 2)
Affinity DataIC50:  21nMAssay Description:Inhibition of CXCR2 (unknown origin) transfected with RBL cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483585(CHEMBL1689308)
Affinity DataIC50:  24nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))TBA
LigandPNGBDBM50407494(CHEMBL5276118)
Affinity DataIC50:  25nMAssay Description:Apparent pA2 value of compound at 10 nM concentration of mepyramine in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483586(CHEMBL1689309)
Affinity DataIC50:  27nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target7-dehydrocholesterol reductase(Homo sapiens (Human))TBA
LigandPNGBDBM50407452(CHEMBL5284923)
Affinity DataIC50:  30nMAssay Description:Tetsed for Antagonistic activity at histamine H3 receptor in guinea pig ileal longitudinal muscle in the presence of mepyramine at a concentration of...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Syntrix Biosystems

Curated by ChEMBL
LigandPNGBDBM150812(US8981106, 2 (SX-576) | USRE47267, Compound 2)
Affinity DataIC50:  31nMAssay Description:Inhibition of CXCR1 (unknown origin) transfected with RBL cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483574(CHEMBL1689310)
Affinity DataIC50:  31nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50407494(CHEMBL5276118)
Affinity DataIC50:  46nMAssay Description:Antagonistic activity for carbachol induced contractions in guinea pig ileum against Muscarinic acetylcholine receptor M3 in the presence of mepyrami...More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50407454(CHEMBL5281526)
Affinity DataIC50:  49nMAssay Description:Histamine-induced inhibition of forskolin- stimulated cAMP accumulation in SK-N-MC cells overexpressing the human Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483587(CHEMBL1689312)
Affinity DataIC50:  54nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483590(CHEMBL1689311)
Affinity DataIC50:  80nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50407450(CHEMBL4544901)
Affinity DataIC50:  97nMAssay Description:Antagonistic affinity tested against isolated Rat Thoracic Aorta Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483596(CHEMBL1689314)
Affinity DataIC50:  100nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483575(CHEMBL1689313)
Affinity DataIC50:  111nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Syntrix Biosystems

Curated by ChEMBL
LigandPNGBDBM150812(US8981106, 2 (SX-576) | USRE47267, Compound 2)
Affinity DataIC50:  130nMAssay Description:Inhibition of CXCR2 (unknown origin) expressed in PathHunter celline by beta-arrestin assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483591(CHEMBL1689315)
Affinity DataIC50:  137nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50407451(CHEMBL5270628)
Affinity DataIC50:  188nMAssay Description:In vitro relative antagonist potency towards guinea pig Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails PubMed
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