Affinity DataKi: 25nMAssay Description:Binding affinity against cytidine deaminase of human liverMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Binding affinity against cytidine deaminase of human liverMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Binding affinity against cytidine deaminase of mouse kidneyMore data for this Ligand-Target Pair
Affinity DataKi: 230nMAssay Description:Compound was tested for inhibitory activity against Inosine-5'-monophosphate dehydrogenase, the type of inhibition in not competitiveMore data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:Compound was tested for inhibitory activity against Inosine-5'-monophosphate dehydrogenase, the type of inhibition in not competitiveMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Binding affinity against cytidine deaminase of mouse kidneyMore data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Binding affinity against cytidine deaminase of human liverMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Eli Lilly
Curated by PDSP Ki Database
Eli Lilly
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Eli Lilly
Curated by PDSP Ki Database
Eli Lilly
Curated by PDSP Ki Database
Affinity DataKi: 1.97E+3nMAssay Description:Compound was tested for inhibitory activity against Inosine-5'-monophosphate dehydrogenase, the type of inhibition in not competitiveMore data for this Ligand-Target Pair
Affinity DataKi: 2.80E+3nMAssay Description:Binding affinity against cytidine deaminase of human liverMore data for this Ligand-Target Pair
Affinity DataKi: 4.00E+3nMAssay Description:Binding affinity against cytidine deaminase of mouse kidneyMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+4nMAssay Description:Binding affinity against cytidine deaminase of human liverMore data for this Ligand-Target Pair
Affinity DataKi: 1.70E+4nMAssay Description:Compound was tested for inhibitory activity against Inosine-5'-monophosphate dehydrogenase, the type of inhibition in not competitiveMore data for this Ligand-Target Pair
Affinity DataKi: 3.40E+4nMAssay Description:Binding affinity against cytidine deaminase of mouse kidneyMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+5nMAssay Description:Binding affinity against cytidine deaminase of mouse kidneyMore data for this Ligand-Target Pair
Affinity DataKi: 3.00E+5nMAssay Description:Binding affinity against cytidine deaminase of human liverMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Inhibitory activity against Dopamine receptor D2 in rat corpus striatum using [3H]-Apomorphine as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Inhibition of [3H]apomorphine binding to dopamine receptor of rat corpus striatumMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Tested for its binding affinity towards 5-hydroxytryptamine 1 receptor in rat cortical membrane homogenates using radioligand ([3H]5-HT) binding assa...More data for this Ligand-Target Pair
Affinity DataIC50: 4.10nMAssay Description:Inhibition of [3H]dopamine binding to dopamine receptor of rat corpus striatumMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Tested for its binding affinity towards 5-hydroxytryptamine 1 receptor in rat cortical membrane homogenates using radioligand ([3H]5-HT) binding assa...More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Tested for its binding affinity towards 5-hydroxytryptamine 1 receptor in rat cortical membrane homogenates using radioligand ([3H]5-HT) binding assa...More data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Tested for its binding affinity towards 5-hydroxytryptamine 1 receptor in rat cortical membrane homogenates using radioligand ([3H]5-HT) binding assa...More data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1 receptor using [3H]5-HT as a radioligand from rat frontal cortex homogenatesMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Tested for its binding affinity towards 5-hydroxytryptamine 1 receptor in rat cortical membrane homogenates using radioligand ([3H]5-HT) binding assa...More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1 receptor using [3H]5-HT as a radioligand from rat frontal cortex homogenatesMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1 receptor using [3H]5-HT as a radioligand from rat frontal cortex homogenatesMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Tested for its binding affinity towards 5-hydroxytryptamine 1 receptor in rat cortical membrane homogenates using radioligand ([3H]5-HT) binding assa...More data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1 receptor using [3H]5-HT as a radioligand from rat frontal cortex homogenatesMore data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:Ability to inhibit binding of titreated serotonin to the 5-hydroxytryptamine 1 receptor in rat brain frontal cortex membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Tested for its binding affinity towards 5-hydroxytryptamine 1 receptor in rat cortical membrane homogenates using radioligand ([3H]5-HT) binding assa...More data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Inhibitory activity against Dopamine receptor D2 in calf corpus striatum using [3H]-Spiperone as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Inhibition of [3H]spiperone binding to dopamine receptor of rat corpus striatumMore data for this Ligand-Target Pair
Affinity DataIC50: 65nMAssay Description:Inhibitory activity against dopamine receptor D2 in rat corpus striatum using [3H]-Apomorphine as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Tested for its binding affinity towards 5-hydroxytryptamine 1 receptor in rat cortical membrane homogenates using radioligand ([3H]5-HT) binding assa...More data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1 receptor using [3H]5-HT as a radioligand from rat frontal cortex homogenatesMore data for this Ligand-Target Pair
Affinity DataIC50: 83nMAssay Description:Ability to inhibit binding of titreated serotonin to the 5-hydroxytryptamine 1 receptor in rat brain frontal cortex membranesMore data for this Ligand-Target Pair