TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataKi: 104nMAssay Description:Inhibition of DYRK1A (unknown origin) using DYRKtide as substrate by ATP regenerative NADH consuming assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataKi: 158nMAssay Description:Inhibition of DYRK1A (unknown origin) using DYRKtide as substrate by ATP regenerative NADH consuming assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataKi: 252nMAssay Description:Inhibition of DYRK1A (unknown origin) using DYRKtide as substrate by ATP regenerative NADH consuming assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataKi: 383nMAssay Description:Inhibition of DYRK1A (unknown origin) using DYRKtide as substrate by ATP regenerative NADH consuming assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataKi: 575nMAssay Description:Inhibition of DYRK1A (unknown origin) using DYRKtide as substrate by ATP regenerative NADH consuming assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataKi: 1.68E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) using DYRKtide as substrate by ATP regenerative NADH consuming assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataKi: 2.02E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) using DYRKtide as substrate by ATP regenerative NADH consuming assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataKi: >2.80E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) using DYRKtide as substrate by ATP regenerative NADH consuming assayMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Binding affinity to CDK2More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 216nMAssay Description:Inhibition of DYRK1A (unknown origin) using DYRKtide as substrate by ATP regenerative NADH consuming assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 329nMAssay Description:Inhibition of DYRK1A (unknown origin) using DYRKtide as substrate by ATP regenerative NADH consuming assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of DYRK1A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 532nMAssay Description:Inhibition of DYRK1A (unknown origin) using DYRKtide as substrate by ATP regenerative NADH consuming assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of DYRK1A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of DYRK1A (unknown origin) using DYRKtide as substrate by ATP regenerative NADH consuming assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of DYRK1A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) using DYRKtide as substrate by ATP regenerative NADH consuming assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) using DYRKtide as substrate by ATP regenerative NADH consuming assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) using DYRKtide as substrate by ATP regenerative NADH consuming assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: >6.00E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) using DYRKtide as substrate by ATP regenerative NADH consuming assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibition of DYRK1A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 1.23E+4nMAssay Description:Inhibition of DYRK1A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 1.57E+4nMAssay Description:Inhibition of DYRK1A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Institute For Biochemistry
Curated by ChEMBL
Institute For Biochemistry
Curated by ChEMBL
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 2.36E+4nMAssay Description:Inhibition of DYRK1A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 2.65E+4nMAssay Description:Inhibition of DYRK1A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 2.81E+4nMAssay Description:Inhibition of DYRK1A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 2.93E+4nMAssay Description:Inhibition of DYRK1A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of DYRK1A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 3.60E+4nMAssay Description:Inhibition of DYRK1A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institute For Biochemistry
Curated by ChEMBL
Institute For Biochemistry
Curated by ChEMBL
Affinity DataIC50: 6.50E+4nMAssay Description:Inhibition of p60 c-SrcMore data for this Ligand-Target Pair
Affinity DataKd: 1.00E+5nMAssay Description:Binding affinity to CDK2More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Institute For Biochemistry
Curated by ChEMBL
Institute For Biochemistry
Curated by ChEMBL
Affinity DataKd: 8.00E+3nMAssay Description:Binding affinity to human wild type Mdm2 by NMR ligand-protein binary titrationMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Institute For Biochemistry
Curated by ChEMBL
Institute For Biochemistry
Curated by ChEMBL
Affinity DataKd: 700nMAssay Description:Binding affinity to human wild type Mdm2 by isothermal titration calorimetryMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Institute For Biochemistry
Curated by ChEMBL
Institute For Biochemistry
Curated by ChEMBL
Affinity DataKd: 2.00E+3nMAssay Description:Binding affinity to human wild type Mdm2 by isothermal titration calorimetryMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Institute For Biochemistry
Curated by ChEMBL
Institute For Biochemistry
Curated by ChEMBL
Affinity DataKd: 8.00E+3nMAssay Description:Binding affinity to human wild type Mdm2 by NMR ligand-protein binary titrationMore data for this Ligand-Target Pair