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Found 21 with Last Name = 'kumirov' and Initial = 'vk'
TargetSubstance-P receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50355375(CHEMBL1835844)
Affinity DataKi:  6.80nMAssay Description:Displacement of [3H]substance P from human NK1 receptor expressed in CHO cells after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50355374(CHEMBL1835843)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]substance P from human NK1 receptor expressed in CHO cells after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50355377(CHEMBL1835845)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]substance P from human NK1 receptor expressed in CHO cells after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50355375(CHEMBL1835844)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in HN9.10 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50355374(CHEMBL1835843)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in HN9.10 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50355377(CHEMBL1835845)
Affinity DataKi:  400nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in HN9.10 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50008984(4-(4-Chloro-benzyl)-2-(1-methyl-azepan-4-yl)-2H-ph...)
Affinity DataIC50:  1.90nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig ileum/longitudinal muscle with myenteric plexus assessed as inhibition of PL-017-induced...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50008984(4-(4-Chloro-benzyl)-2-(1-methyl-azepan-4-yl)-2H-ph...)
Affinity DataIC50:  7.20nMAssay Description:Agonist activity at delta opioid receptor in ICR mouse vas deferens assessed as inhibition of MVD contraction heightMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50355375(CHEMBL1835844)
Affinity DataIC50:  55nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig ileum/longitudinal muscle with myenteric plexus assessed as inhibition of PL-017-induced...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50355374(CHEMBL1835843)
Affinity DataIC50:  410nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig ileum/longitudinal muscle with myenteric plexus assessed as inhibition of PL-017-induced...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50044777(Arginine Vasopressin | Beta-Hypophamine | CHEBI:34...)
Affinity DataEC50:  32nMAssay Description:Biological activity against Oxytocin receptor in ratMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOxytocin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50406331(CHEMBL5286119)
Affinity DataEC50:  0.0600nMAssay Description:Biological activity against Oxytocin receptor in ratMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOxytocin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50406330(CHEMBL5271164)
Affinity DataEC50:  220nMAssay Description:Antagonism against Tachykinin receptor 2 in rat vas deferens(RVD)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOxytocin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50406329(CHEMBL5273426)
Affinity DataEC50:  0.540nMAssay Description:Antagonism against Tachykinin receptor 2 in rat vas deferens(RVD)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOxytocin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50406328(CHEMBL5266871)
Affinity DataEC50:  7.00E+3nMAssay Description:Antagonism against Tachykinin receptor 2 in rat vas deferens(RVD)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOxytocin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50406327(CHEMBL5281925)
Affinity DataEC50:  3.80E+3nMAssay Description:Antagonism against Tachykinin receptor 2 in rat vas deferens(RVD)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOxytocin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataEC50:  2.30nMAssay Description:Biological activity against Oxytocin receptor in ratMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOxytocin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50406326(CHEMBL5280014)
Affinity DataEC50:  0.280nMAssay Description:Antagonism against Tachykinin receptor 2 in rat vas deferens(RVD)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOxytocin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50406325(CHEMBL5279634)
Affinity DataEC50:  160nMAssay Description:Antagonism against Tachykinin receptor 2 in rat vas deferens(RVD)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50044777(Arginine Vasopressin | Beta-Hypophamine | CHEBI:34...)
Affinity DataEC50:  11nMAssay Description:Antagonism against Tachykinin receptor 2 in rat vas deferens(RVD)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOxytocin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50406324(CHEMBL5275543)
Affinity DataEC50:  0.730nMAssay Description:Biological activity against Oxytocin receptor in ratMore data for this Ligand-Target Pair
In DepthDetails PubMed