Affinity DataKi: 6.80nMAssay Description:Displacement of [3H]substance P from human NK1 receptor expressed in CHO cells after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of [3H]substance P from human NK1 receptor expressed in CHO cells after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Displacement of [3H]substance P from human NK1 receptor expressed in CHO cells after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in HN9.10 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in HN9.10 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in HN9.10 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig ileum/longitudinal muscle with myenteric plexus assessed as inhibition of PL-017-induced...More data for this Ligand-Target Pair
Affinity DataIC50: 7.20nMAssay Description:Agonist activity at delta opioid receptor in ICR mouse vas deferens assessed as inhibition of MVD contraction heightMore data for this Ligand-Target Pair
Affinity DataIC50: 55nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig ileum/longitudinal muscle with myenteric plexus assessed as inhibition of PL-017-induced...More data for this Ligand-Target Pair
Affinity DataIC50: 410nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig ileum/longitudinal muscle with myenteric plexus assessed as inhibition of PL-017-induced...More data for this Ligand-Target Pair
Affinity DataEC50: 32nMAssay Description:Biological activity against Oxytocin receptor in ratMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0600nMAssay Description:Biological activity against Oxytocin receptor in ratMore data for this Ligand-Target Pair
Affinity DataEC50: 220nMAssay Description:Antagonism against Tachykinin receptor 2 in rat vas deferens(RVD)More data for this Ligand-Target Pair
Affinity DataEC50: 0.540nMAssay Description:Antagonism against Tachykinin receptor 2 in rat vas deferens(RVD)More data for this Ligand-Target Pair
Affinity DataEC50: 7.00E+3nMAssay Description:Antagonism against Tachykinin receptor 2 in rat vas deferens(RVD)More data for this Ligand-Target Pair
Affinity DataEC50: 3.80E+3nMAssay Description:Antagonism against Tachykinin receptor 2 in rat vas deferens(RVD)More data for this Ligand-Target Pair
Affinity DataEC50: 2.30nMAssay Description:Biological activity against Oxytocin receptor in ratMore data for this Ligand-Target Pair
Affinity DataEC50: 0.280nMAssay Description:Antagonism against Tachykinin receptor 2 in rat vas deferens(RVD)More data for this Ligand-Target Pair
Affinity DataEC50: 160nMAssay Description:Antagonism against Tachykinin receptor 2 in rat vas deferens(RVD)More data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:Antagonism against Tachykinin receptor 2 in rat vas deferens(RVD)More data for this Ligand-Target Pair
Affinity DataEC50: 0.730nMAssay Description:Biological activity against Oxytocin receptor in ratMore data for this Ligand-Target Pair